Información del producto
GSK837149A is a potent inhibitor of the protein target that inhibits the growth of cancer cells. GSK837149A binds to the ATP-binding site in the ATPase domain of the protein target, preventing ATP hydrolysis and inhibiting cancer cell growth. This drug is selective for tumours with a m2 phenotype and has been shown to inhibit autophagy in colorectal adenocarcinoma cells. GSK837149A also has anti-inflammatory properties, which may be due to its ability to inhibit metabolism in cancer tissues.
Propiedades químicas
Consulta técnica sobre: 3D-NAA61629 GSK837149A
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