TAPI 0
CAS: 163958-73-4
Ref. 3D-NGA95873
1mg | A consultar | ||
5mg | A consultar | ||
10mg | A consultar | ||
25mg | A consultar | ||
50mg | A consultar |
Información del producto
TAPI-0 is a novel anti-inflammatory drug that binds to calmodulin and prevents the activation of protein kinase C. This compound inhibits many inflammatory mediators, including prostaglandin E2, cytokines and nitric oxide. Tapi-0 has been shown to be effective in decreasing the expression of chemokines such as MCP-1, MIP-1α, MIP-1β, RANTES and eotaxin in models of inflammation. TAPI-0 also inhibits the growth of cancerous cells by inhibiting transcriptional regulation. The mechanism by which TAPI-0 inhibits transcriptional regulation is not yet well understood but may involve inhibition of DNA polymerase activity.
Propiedades químicas
Consulta técnica sobre: 3D-NGA95873 TAPI 0
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