CGP 52432
CAS: 139667-74-6
Ref. 3D-PFA66774
5mg | A consultar | |
10mg | A consultar | |
25mg | A consultar | |
50mg | A consultar | |
100mg | A consultar |
Información del producto
- Phosphinic acid, P-[3-[[(3,4-dichlorophenyl)methyl]amino]propyl]-P-(diethoxymethyl)-
CGP 52432 is a baclofen analog that blocks 2-adrenergic receptors, which are G protein-coupled receptors. CGP 52432 has been shown to inhibit the binding of estradiol benzoate with DNA in vitro and to have pharmacological properties similar to those of nonsteroidal anti-inflammatory drugs. The drug has been shown to be a low potency antagonist of rat 2-adrenergic receptors in vitro and is being studied for its potential as a treatment for neuropathic pain.
Propiedades químicas
Consulta técnica sobre: 3D-PFA66774 CGP 52432
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