Ethyl 3-tert-butyl-1H-pyrazole-5-carboxylate

CAS: 916791-97-4

Ref. 3D-RLB79197

Información del producto

• Nombre: Ethyl 3-tert-butyl-1H-pyrazole-5-carboxylate

Descripción

Ethyl 3-tert-butyl-1H-pyrazole-5-carboxylate (ETBP) is an orally active, water soluble prodrug of piperidine. ETBP has been shown to be safe and effective in monkeys, with low toxicity. ETBP interacts with CYP3A4 and can be metabolized by CYP2D6 to form a pharmacokinetic profile that is similar to the parent drug. The physicochemical properties of ETBP make it difficult for the drug to cross the blood brain barrier, which may limit its use as a psychotropic agent. Benzimidazole derivatives are structurally modified ETBP analogues that have been shown to have better bioavailability and reduced neurotoxicity.

• Marca: Biosynth

Propiedades químicas

• Peso molecular: 196.25 g/mol
• Fórmula: C₁₀H₁₆N₂O₂
• Pureza: Min. 95%