Kelatorphan

CAS: 92175-57-0

Ref. 3D-SDA17557

Información del producto

• Nombre: Kelatorphan
• Sinónimos: <span class="text-smallcaps">L</span>-Alanine, N-[(2R)-4-(hydroxyamino)-1,4-dioxo-2-(phenylmethyl)butyl]-, <span class="text-smallcaps">L</span>-Alanine, N-[4-(hydroxyamino)-1,4-dioxo-2-(phenylmethyl)butyl]-, (R)-, L-alanine, N-[(2R)-4-(hydroxyamino)-1,4-dioxo-2-(phenylmethyl)butyl]-, N-[(2R)-4-(Hydroxyamino)-1,4-dioxo-2-(phenylmethyl)butyl]-<span class="text-smallcaps">L</span>-alanine

Descripción

Kelatorphan is a drug that belongs to the class of nonsteroidal anti-inflammatory drugs. It has been shown to be an inhibitor of the enzyme polymerase chain reaction (PCR) in vitro. Kelatorphan was used as a model system to study the effects of atrial natriuretic peptide (ANP) in inhibiting protein synthesis and cell division. The IC50 for kelatorphan was found to be 0.5 micrograms/mL, which is much lower than its concentration in blood plasma. The IC50 for ANP was found to be between 10-25 micrograms/mL, which is higher than its concentration in blood plasma. Kelatorphan has also been shown to inhibit toll-like receptor 4 (TLR4) and TLR2, which are involved with inflammation and immunity.

• Marca: Biosynth

Propiedades químicas

• Peso molecular: 294.3 g/mol
• Fórmula: C₁₄H₁₈N₂O₅
• Pureza: Min. 95%