CymitQuimica logo
Entre las marcas de nuestros más de 25 colaboradores destaca TargetMol

Entre las marcas de nuestros más de 25 colaboradores destaca TargetMol

We have reached an agreement with TargetMol: CymitQuimica clients will benefit for a 20% discount on all TargetMol products until the end of the year.On our website you can find the products offered by this partner, which has become one of the world's most recognised compound libraries and small molecule inhibitors supplier. TargetMol offers approximately 120 compound libraries and a wide range of chemical products and kits for life sciences.

Termina el 31 dic( quedan 8 días )

productos por página.Hay 111930 productos en esta promoción.
  • 7-Methoxyisoflavone

    CAS:
    7-Methoxyisoflavone is an activator of adenosine monophosphate-activated protein kinase (AMPK).
    Fórmula:C16H12O3
    Pureza:99.93% - 99.94%
    Forma y color:Solid
    Peso molecular:252.26
  • GSK3-IN-2

    CAS:
    <p>GSK3-IN-2 is a potent GSK3 inhibitor for the treatment of diabetes and neurodegenerative diseases.</p>
    Fórmula:C17H19N3OS
    Pureza:98.8%
    Forma y color:Solid
    Peso molecular:313.42
  • MMV688845

    CAS:
    MMV688845: NTM RNA polymerase inhibitor, kills Mycobacterium abscessus, and fights TB.
    Fórmula:C24H25N3O3S
    Forma y color:Solid
    Peso molecular:435.54
  • VU6019650


    VU6019650: potent M5 mAChR antagonist, IC50=36nM. May help with OUD, crosses blood-brain barrier, affects VTA dopamine neurons.
    Fórmula:C18H22FN3O3S2
    Forma y color:Solid
    Peso molecular:411.51
  • SERT-IN-2


    SERT-IN-2, a potent SERT inhibitor (IC 50 = 0.58 nM), exhibits promising efficacy as an anti-depressant.
    Forma y color:Solid
  • CamA-IN-1


    CamA-IN-1, specific Clostridioides difficile methyltransferase inhibitor, IC50 = 0.4μM, Kd = 0.2μM, targets CDI research.
    Fórmula:C23H36N6O6
    Forma y color:Solid
    Peso molecular:492.57
  • BTK-IN-22

    CAS:
    BTK-IN-22 is a selective BTK inhibitor with IC50 of 0.9 nM; also targets BLX, BMX (IC50s: 1.4, 1.2 nM); better selectivity than Ibrutinib.
    Fórmula:C26H26N6O2
    Forma y color:Solid
    Peso molecular:454.52
  • BTK-IN-23

    CAS:
    BTK-IN-23: BTK inhibitor, IC50=12.8 nM; also blocks BLX (35.6 nM), BMX (5.7 nM); better selectivity than Ibrutinib.
    Fórmula:C27H28N6O2
    Forma y color:Solid
    Peso molecular:468.55
  • FABP-IN-2

    CAS:
    FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.
    Fórmula:C25H21ClN2O3
    Forma y color:Solid
    Peso molecular:432.9
  • MLKL-IN-5

    CAS:
    MLKL-IN-5 is a potent MLKL inhibitor that mediates necroptosis .
    Fórmula:C18H20N6O4S
    Forma y color:Solid
    Peso molecular:416.45
  • HBV-IN-29

    CAS:
    HBV-IN-29 (ex8), a flavone derivative, inhibits cccDNA in HBV research.
    Fórmula:C22H19ClO6
    Forma y color:Solid
    Peso molecular:414.84
  • HBV-IN-30

    CAS:
    <p>HBV-IN-30, a flavone derivative, inhibits cccDNA in HBV research.</p>
    Fórmula:C22H18BrClO6
    Forma y color:Solid
    Peso molecular:493.73
  • HBV-IN-31

    CAS:
    HBV-IN-31: strong cccDNA inhibitor, anti-HBV, IC50=0.13 µM HBsAg, hampers cell growth.
    Fórmula:C23H18ClNO6
    Forma y color:Solid
    Peso molecular:439.85
  • HBV-IN-32

    CAS:
    HBV-IN-32 is a strong cccDNA inhibitor with an IC50 of 0.14 µM against HBsAg, also halting cell growth.
    Fórmula:C22H19ClO5S
    Forma y color:Solid
    Peso molecular:430.9
  • Vonifimod

    CAS:
    Vonifimod is an immunomodulator .
    Fórmula:C17H34N4O2
    Forma y color:Solid
    Peso molecular:326.48
  • SRI-42127

    CAS:
    SRI-42127 is a novel small molecule inhibitor of the RNA regulatory factor HuR that inhibits tumor growth and reduces neuropathic pain following nerve injury.
    Fórmula:C19H20N6O
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:348.4
  • Nek2-IN-6

    CAS:
    Nek2-IN-6 inhibitor .
    Fórmula:C33H33F3N6O4S
    Forma y color:Solid
    Peso molecular:666.71
  • DC-BPi-03

    CAS:
    DC-BPi-03 is a potent BPTF-BRD inhibitor with an IC 50 of 698.3 nM and a K d of 2.81 μM .
    Fórmula:C14H14N4O2S
    Pureza:98.96%
    Forma y color:Solid
    Peso molecular:302.35
  • mHTT-IN-1

    CAS:
    mHTT-IN-1 is a potent inhibitor of toxic mHTT, linked to Huntington's disease, with an EC50 of 46 nM.
    Fórmula:C18H19N7OS
    Forma y color:Solid
    Peso molecular:381.45
  • C-178

    CAS:
    <p>C-178 inhibits STING by binding Cys91, blocking palmitoylation and TBK1 activation in HEK293T cells.</p>
    Fórmula:C17H10N2O5
    Pureza:97.69%
    Forma y color:Solid
    Peso molecular:322.27
  • Fabimycin

    CAS:
    Fabimycin, a FabI inhibitor, combats drug-resistant gram-negative bacterial infections effectively.
    Fórmula:C23H25ClN4O3
    Forma y color:Solid
    Peso molecular:440.92
  • ZIKV-IN-3

    CAS:
    ZIKV-IN-3, an andrographolide derivative, inhibits ZIKV NS5 MTase (IC50: 18.34 μM) and replication. Used for Zika virus research.
    Fórmula:C39H41NO4
    Forma y color:Solid
    Peso molecular:587.75
  • WNK1-IN-1

    CAS:
    WNK1-IN-1, a WNK1 inhibitor (IC50: 1.6 μM), also inhibits OSR1 phosphorylation (IC50: 4.3 μM), used in blood pressure and cancer research.
    Fórmula:C13H15BrCl2N2O4S
    Pureza:98.09%
    Forma y color:Solid
    Peso molecular:446.14
  • iBRD4-BD1

    CAS:
    iBRD4-BD1 inhibits BRD4 bromodomain selectively with 12 nM IC50, useful in inflammation and cancer research.
    Fórmula:C29H30F3N5O
    Forma y color:Solid
    Peso molecular:521.58
  • TDI-11861

    CAS:
    TDI-11861 is a second-gen sAC (ADCY10) inhibitor with an IC50 of 5.5 nM and slow dissociation.
    Fórmula:C22H25ClF2N6O3
    Forma y color:Solid
    Peso molecular:494.92
  • MurA-IN-3

    CAS:
    MurA-IN-3, a reversible pyrrolidinedione-based MurA inhibitor, exhibits an IC50 of 4.5 μM against MurA and demonstrates antibacterial activity [1].
    Fórmula:C27H23ClN2O5S
    Forma y color:Solid
    Peso molecular:523
  • APE1-IN-2

    CAS:
    <p>APE1-IN-2 (AP1), a Pt(IV) proagent, targets APE1 protein, induces DNA damage, and triggers apoptosis with anticancer effects.</p>
    Fórmula:C9H12Cl2N4O5Pt
    Pureza:98%
    Forma y color:Solid
    Peso molecular:522.21
  • Nucleozin

    CAS:
    Nucleozin targets influenza A nucleoprotein (NP), a multifunctional, RNA-binding protein necessary for virus replication.
    Fórmula:C21H19ClN4O4
    Pureza:97.72%
    Forma y color:Solid
    Peso molecular:426.85
  • AXL-IN-13

    CAS:
    AXL-IN-13: potent, oral AXL inhibitor, IC50=1.6nM, Kd=0.26nM, anti-cancer, inhibits EMT, cell migration & invasion.
    Fórmula:C34H41FN6O5
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:632.72
  • ATR-IN-20


    ATR-IN-20: potent ATR inhibitor, IC50=3nM; inhibits mTOR, IC50=18nM; selective vs PI3Kα, ATM, DNA-PK; good pharmacokinetics; anticancer.
    Fórmula:C29H31N5O4S
    Forma y color:Solid
    Peso molecular:545.65
  • FAAH-IN-7


    <p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>
    Fórmula:C26H29N3O4
    Forma y color:Solid
    Peso molecular:447.53
  • BTK-IN-17


    BTK-IN-17: selective, oral BTK inhibitor, IC50=13.7 nM, reduces p-BTK Y223/p-PLCγ2 Y1217, anti-inflammatory.
    Fórmula:C26H23N7O2
    Forma y color:Solid
    Peso molecular:465.51
  • ALR2-IN-2


    ALR2-IN-2 inhibits ALR2 (27 nM IC50) & ALR1 (228 nM IC50), used in diabetes complication research.
    Fórmula:C17H11FN2O2S2
    Forma y color:Solid
    Peso molecular:358.41
  • ALR2-IN-3


    ALR2-IN-2 inhibits ALR2 strongly (IC50: 22 nM) and ALR1 less (IC50: 116 nM), used in diabetes complication studies.
    Fórmula:C17H12N2O3S2
    Forma y color:Solid
    Peso molecular:356.42
  • TrkA-IN-3


    TrkA-IN-3: potent allosteric TrkA inhibitor, IC50=22.4 nM, >8000x selective over TrkB/C, for pain research.
    Fórmula:C24H17F3N4O3
    Forma y color:Solid
    Peso molecular:466.41
  • TrkA-IN-4


    TrkA-IN-4, a potent, orally active and allosteric TrkA inhibitor, is a prodrug of TrkA-IN-3 . TrkA-IN-4 exhibits potent antinociceptive effects [1] .
    Fórmula:C27H21F3N4O5
    Forma y color:Solid
    Peso molecular:538.47
  • Mps1-IN-5

    CAS:
    Mps1-IN-5: oral Mps1 inhibitor with 29 nM IC50, induces apoptosis, G2/M arrest, and has anti-tumor properties.
    Fórmula:C24H25N9
    Forma y color:Solid
    Peso molecular:439.52
  • RET-IN-20


    RET-IN-20: potent RET inhibitor (IC50 = 13.7 nM), reduces p-Ret/p-Shc, induces apoptosis, anti-tumor effects.
    Fórmula:C32H33FN6O4
    Forma y color:Solid
    Peso molecular:584.64
  • Ursocholic acid

    CAS:
    Ursocholic acid, a bile acid found predominantly in bile of mammals.
    Fórmula:C24H40O5
    Pureza:98.89% - 99.62%
    Forma y color:Solid
    Peso molecular:408.57
  • AXL-IN-14

    CAS:
    AXL-IN-14: orally active, potent AXL inhibitor (IC50=0.8 nM); hinders Gas6/AXL migration, invasion; lowers p-AXL, p-AKT; anti-tumor.
    Fórmula:C32H24F2N4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:566.55
  • DENV-IN-7

    CAS:
    DENV-IN-7, a flavone analog, inhibits dengue virus at 70 nM EC50 with low toxicity to normal cells.
    Fórmula:C24H22O8
    Forma y color:Solid
    Peso molecular:438.43
  • DENV-IN-9

    CAS:
    DENV-IN-9 is a DENV2 inhibitor with an EC 50 of 0.88 μM .
    Fórmula:C15H9BrO5
    Forma y color:Solid
    Peso molecular:349.13
  • (R)-ZG197


    (R)-ZG197: Activates Sa ClpP (EC50=1.5μM) & Hs ClpP (EC50=31.4μM); selective for Sa ClpP.
    Fórmula:C28H35F3N4O3
    Forma y color:Solid
    Peso molecular:532.6
  • (S)-ZG197


    (S)-ZG197 is a compound that acts as a highly selective activator of the Staphylococcus aureus Caseinolytic Protease P (Sa ClpP), demonstrating efficacy at a
    Fórmula:C28H35F3N4O3
    Forma y color:Solid
    Peso molecular:532.6
  • FGFR-IN-9


    FGFR-IN-9: oral FGFR inhibitor, IC50: 17.1 nM (FGFR4 WT), 29.6 (FGFR3), 30.7 (V550L), 46.7 (FGFR2), 64.3 nM (FGFR1).
    Fórmula:C25H28N6O3S
    Forma y color:Solid
    Peso molecular:492.59
  • JZP-MA-13


    JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.
    Fórmula:C14H15FN4O3S
    Forma y color:Solid
    Peso molecular:338.36
  • BTK-IN-18

    CAS:
    <p>BTK-IN-18 is a potent, reversible inhibitor of Bruton's tyrosine kinase (BTK) with an inhibitory concentration (IC50) of 0.002 µM.</p>
    Fórmula:C20H22Cl2N6O
    Forma y color:Solid
    Peso molecular:433.33
  • BTK-IN-19

    CAS:
    BTK-IN-19 is a reversible BTK inhibitor with an IC 50 of <0.001 μM .
    Fórmula:C21H22Cl2N6O
    Forma y color:Solid
    Peso molecular:445.35
  • (E)-2-Decenoic acid

    CAS:
    (E)-2-Decenoic acid (trans-2-Decenoic acid) is an unsaturated fatty acid found in royal jelly produced from the mandibular gland secretions of honeybees.
    Fórmula:C10H18O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:170.25
  • CLK1-IN-2


    <p>CLK1-IN-2: Metabolically stable, Clk1-selective inhibitor; IC50=1.7nM; useful in tumor, Duchenne MD, HIV-1, influenza research.</p>
    Fórmula:C16H12Cl2N2O2S
    Forma y color:Solid
    Peso molecular:367.25
  • TBK1-IN-1

    CAS:
    TBK1-IN-1 is a TANK-binding kinase 1 inhibitor with anticancer activity.TBK1-IN-1 inhibits the expression of TBK1 downstream target genes, cxcl10 and ifnβ.
    Fórmula:C27H37N7O2
    Pureza:99.81% - >99.99%
    Forma y color:Solid
    Peso molecular:491.63
  • RdRP-IN-5

    CAS:
    <p>RdRP-IN-5 (compound 20), a potent inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), has potential application in influenza research [1].</p>
    Fórmula:C23H21N3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:419.43
  • PARL-IN-1


    PARL-IN-1: Strong PARL blocker, IC50 28 nM, boosts PINK1/Parkin mitophagy.
    Fórmula:C40H58N6O7
    Forma y color:Solid
    Peso molecular:734.92
  • MenA-IN-1


    MenA IN-1 inhibits MTB's MenA enzyme; IC50=13µM, GIC50=8µM, helps fight tuberculosis spread.
    Fórmula:C29H36N2O2
    Forma y color:Solid
    Peso molecular:444.61
  • CB2R-IN-3


    CB2R-IN-3 selectively blocks CB2R with high affinity, enhances anti-inflammatory cytokines, and can be used with CB65.
    Fórmula:C27H42N2O
    Forma y color:Solid
    Peso molecular:410.64
  • Merigolix

    CAS:
    Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .
    Fórmula:C36H35F7N4O6
    Forma y color:Solid
    Peso molecular:752.68
  • DHFR-IN-5

    CAS:
    <p>DHFR-IN-5: potent, oral DHFR inhibitor, Ki 0.54 nM against mutant P. falciparum, anti-malarial.</p>
    Fórmula:C18H24N4O4
    Forma y color:Solid
    Peso molecular:360.41
  • P 218

    CAS:
    P 218 is a novel DHFR inhibitor with antimalarial activity and antifolate effects and can be used to study Buruli ulcer.
    Fórmula:C18H25ClN4O4
    Pureza:98.83%
    Forma y color:Soild
    Peso molecular:396.87
  • MMV676584

    CAS:
    MMV676584 has anti-tuberculosis avtivity. MMV676584 is a novel drug candidate for eumycetoma .
    Fórmula:C12H8ClFN2OS2
    Forma y color:Solid
    Peso molecular:314.79
  • Pyrvinium pamoate

    CAS:
    Pyrvinium pamoate (Pyrvinium embonate) is an old anthelminthic medicine for the treatment of enterobiasis , which re-attracts attention as an anti-cancer drug
    Fórmula:C26H28N3C23H14O6
    Pureza:99.76% - >99.99%
    Forma y color:Solid
    Peso molecular:575.71
  • JAK-IN-24

    CAS:
    JAK-IN-24: JAK inhibitor, IC50: 0.534 nM (4 μM ATP), 24 nM (1mM ATP), STAT5 phosphorylation IC50: 86.171 nM.
    Fórmula:C20H25N5O2
    Forma y color:Solid
    Peso molecular:367.44
  • GSK3-IN-3

    CAS:
    <p>GSK3-IN-3 is a mitochondrial autophagy (mitophagy) inducer and GSK-3 inhibitor (IC50: 3.01 μM) that induces parkin-dependent mitochondrial autophagy.</p>
    Fórmula:C24H35N3O4
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:429.55
  • BI-685509

    CAS:
    BI-685509: potent, oral sGC activator, boosts cGMP, enhances NO pathways, for CKD/DKD research.
    Fórmula:C34H38N4O5
    Forma y color:Solid
    Peso molecular:582.69
  • OICR12694

    CAS:
    <p>OICR12694 (JNJ-65234637) is an orally active inhibitor of B cell lymphoma 6 (BCL6) .</p>
    Fórmula:C29H28ClF3N8O4
    Forma y color:Solid
    Peso molecular:645.03
  • Larotinib

    CAS:
    Larotinib is an orally active, potent, and broad-spectrum tyrosine kinase inhibitor (TKI) with an IC50 of 0.6 nM for EGFR.
    Fórmula:C24H26ClFN4O4
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:488.94
  • P2X7-IN-2

    CAS:
    P2X7-IN-2 is a P2X7 receptor blocker, halts IL-Iβ release (IC50: 0.01 nM), researched for autoimmunity and heart issues.
    Fórmula:C22H21F4N3O2
    Forma y color:Solid
    Peso molecular:435.41
  • Ketotifen

    CAS:
    Ketotifen: Oral H1 blocker & mast cell stabilizer, inhibits 6-phosphogluconate dehydrogenase, antiviral, for EAE & asthma prevention research.
    Fórmula:C19H19NOS
    Forma y color:Solid
    Peso molecular:309.43
  • Articaine

    CAS:
    <p>Articaine (Hoe-045 free base), an amide anesthetic featuring an ester group, effectively relieves pain by reversibly binding to the α-subunit of the voltage-</p>
    Fórmula:C13H20N2O3S
    Forma y color:Solid
    Peso molecular:284.37
  • Obtusalin

    CAS:
    <p>Obtusalin, a triterpenoid initially identified in R. dauricum, exhibits UV absorption at 210 nm and possesses antibacterial properties.</p>
    Fórmula:C30H50O2
    Forma y color:Solid
    Peso molecular:442.72
  • NP118809

    CAS:
    <p>NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).</p>
    Fórmula:C32H32N2O
    Pureza:97.74% - 98.68%
    Forma y color:Solid
    Peso molecular:460.61
  • Quipazine

    CAS:
    <p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>
    Fórmula:C13H15N3
    Forma y color:Solid
    Peso molecular:213.28
  • Prenderol

    CAS:
    <p>Prenderol, a potent central-nervous-system (CNS) depressant, exhibits anticonvulsant activity.</p>
    Fórmula:C7H16O2
    Forma y color:Solid
    Peso molecular:132.2
  • BAP1-IN-1

    CAS:
    BAP1-IN-1 is an inhibitor of the catalytic activity of BRCA1-associated protein 1 (BAP1), which is related to cancer and can be used to study cancer.
    Fórmula:C18H16N2O2
    Pureza:98.11%
    Forma y color:Solid
    Peso molecular:292.33
  • AP 24149

    CAS:
    AP 24149, a potent dual inhibitor targeting Src and Abl, exhibits IC50 values of 9.1 nM for Src and 3.6 nM for Abl, respectively.
    Fórmula:C23H24N5OP
    Forma y color:Solid
    Peso molecular:417.44
  • SC 34301

    CAS:
    SC 34301 (Enisoprost), a strong oral PGE1 analog, decreases bacterial translocation and increases burned mice survival.
    Fórmula:C22H36O5
    Forma y color:Solid
    Peso molecular:380.52
  • BCX-1898

    CAS:
    BCX-1898: Oral cyclopentane-based neuraminidase inhibitor for flu A/B; EC50 <0.01-21µM; effective in mouse models.
    Fórmula:C17H32N4O3
    Forma y color:Solid
    Peso molecular:340.46
  • CCG-2046

    CAS:
    CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.
    Fórmula:C11H10N4
    Forma y color:Solid
    Peso molecular:198.22
  • TTT 3002

    CAS:
    TTT 3002: oral FLT3 inhibitor for AML research, blocks D835 mutations, potent at 0.2 nM IC50.
    Fórmula:C27H23N5O3
    Forma y color:Solid
    Peso molecular:465.50
  • 2,3-Diaminopropionic acid

    CAS:
    2,3-Diaminopropionic acid (L-2,3-Diaminopropionic acid) is an amino acid that is a precursor of antibiotics and staphyloferrin B a siderophore produced by
    Fórmula:C3H8N2O2
    Pureza:99.61% - 99.90%
    Forma y color:Solid
    Peso molecular:104.11
  • BAY-3827

    CAS:
    BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.
    Fórmula:C27H25FN6O
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:468.53
  • CAY10581

    CAS:
    CAY10581, a derivative of pyranonaphthoquinone, serves as a highly specific and reversible uncompetitive inhibitor of IDO, demonstrating potency with an IC50
    Fórmula:C22H21NO4
    Forma y color:Solid
    Peso molecular:363.41
  • A-943931

    CAS:
    A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.
    Fórmula:C17H21N5
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:295.38
  • NOS-IN-3

    CAS:
    NOS-IN-3: potent, selective iNOS inhibitor; IC50 of 4.6 µM; spares eNOS; low toxicity; potential for septic shock treatment.
    Fórmula:C10H15N3O
    Forma y color:Solid
    Peso molecular:193.25
  • TPN729MA

    CAS:
    <p>TPN729MA, a potent PDE5 inhibitor, IC50: 2.28 nM, targets erectile dysfunction research.</p>
    Fórmula:C29H40N6O8S
    Forma y color:Solid
    Peso molecular:632.73
  • Ac32Az19

    CAS:
    Ac32Az19 is a potent, non-toxic, and highly selective inhibitor of Breast Cancer Resistance Protein (BCRP), demonstrating an EC50 of 13 nM in BCRP-overexpressed
    Fórmula:C37H33N3O6
    Forma y color:Solid
    Peso molecular:615.67
  • (-)SHIN2


    <p>'(-)SHIN2 isomer of (+)SHIN2, an SHMT inhibitor with antileukemic properties; enhances Methotrexate's effect in vivo.</p>
    Fórmula:C23H26N4O3
    Forma y color:Solid
    Peso molecular:406.48
  • NYX-2925

    CAS:
    NYX-2925, an oral NMDAR modulator, enhances Src in mPFC. No CAMKII impact or addictive/sedative effects. Useful for CNS disorder studies.
    Fórmula:C14H23N3O4
    Forma y color:Solid
    Peso molecular:297.35
  • ICA-121431

    CAS:
    <p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>
    Fórmula:C23H19N3O3S2
    Pureza:98.06%
    Forma y color:Solid
    Peso molecular:449.55
  • RP101442

    CAS:
    RP101442: Ozanimod metabolite, selective S1PR1 agonist, EC50: 2.6 nM (S1PR1), 171 nM (S1PR5).
    Fórmula:C23H22N4O3
    Forma y color:Solid
    Peso molecular:402.45
  • RP101988


    RP101988, a potent Ozanimod metabolite, selectively targets S1PR1 with EC50 of 0.19 nM and S1PR5 at 32.8 nM.
    Fórmula:C23H22N4O4
    Forma y color:Solid
    Peso molecular:418.45
  • C-di-IMP

    CAS:
    Cyclic-di-IMP (C-di-IMP), a STING agonist, serves as a research tool in tumor studies.
    Fórmula:C20H22N8O14P2
    Forma y color:Solid
    Peso molecular:660.38
  • MEK-IN-5

    CAS:
    <p>MEK-IN-5: strong MEK inhibitor and NO donor, reduces pMEK/pERK dose/time-dependently, triggers apoptosis in MDA-MB-231 cells.</p>
    Fórmula:C29H27FN4O10S2
    Forma y color:Solid
    Peso molecular:674.67
  • BLK-IN-2

    CAS:
    <p>BLK-IN-2为一种高效、选择性且不可逆的B-淋巴酪氨酸激酶(BLK)抑制剂,具有5.9 nM的IC50值。该化合物亦能抑制BTK,其IC50值为202.0 nM。BLK-IN-2在多种淋巴瘤细胞中展现出显著的抗增殖作用。</p>
    Fórmula:C39H41N9O3
    Forma y color:Solid
    Peso molecular:683.8
  • Zn(BQTC)

    CAS:
    Zn(BQTC) inhibits mtDNA and nDNA, damages mitochondria/nuclei, triggers apoptosis, and targets A549R cancer cells.
    Fórmula:C30H36Cl2N5O3Zn
    Pureza:98%
    Forma y color:Solid
    Peso molecular:650.92
  • UniPR505

    CAS:
    <p>UniPR505 is a potent EphA2 antagonist (IC50: 0.95 µM), a novel 3α-carbamoyloxy derivative with antiangiogenic properties.</p>
    Fórmula:C39H57N3O5
    Pureza:98.23%
    Forma y color:Solid
    Peso molecular:647.89
  • UR-MB108

    CAS:
    UR-MB108 is a potent and selective inhibitor of ABCG2 (BCRP), displaying an IC50 value of 79 nM, and exhibits stability in blood plasma.
    Fórmula:C40H38N6O4
    Forma y color:Solid
    Peso molecular:666.77
  • Kinetin riboside

    CAS:
    Kinetin riboside (N6-Furfuryladenosine) can induce apoptosis in cancer cells. It inhibits the proliferation of HCT-15 cells(IC50 of 2.5 μM)
    Fórmula:C15H17N5O5
    Pureza:98.17%
    Forma y color:White Solid
    Peso molecular:347.33
  • RSV-IN-7

    CAS:
    <p>RSV-IN-7 (example 253) is a RSV inhibitor ( EC 50 : &lt; 0.4 μΜ) .</p>
    Fórmula:C27H22F3N7O3
    Forma y color:Solid
    Peso molecular:549.50
  • BAY-3153

    CAS:
    BAY-3153 is a selective CCR1 ( C-C motif chemokine receptor 1 ) antagonist (human IC 50 =3 nM ; rat IC 50 =11 nM ; mice IC 50 =81 nM) .
    Fórmula:C25H29Cl2N3O4
    Forma y color:Solid
    Peso molecular:506.42
  • GNE-2256

    CAS:
    GNE-2256, also known as molecule 19, is an orally active compound that inhibits Interleukin 1 receptor-associated kinase 4 (IRAK4) with a K i of 1.4 nM and has
    Fórmula:C24H27FN6O4
    Forma y color:Solid
    Peso molecular:482.51