Entre las marcas de nuestros más de 25 colaboradores destaca TargetMol
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Termina el 31 dic( quedan 8 días )
STAT3-IN-42
<p>STAT3-IN-42 is a ligand for target proteins in PROTACs (Proteolysis Targeting Chimeras). It is utilized in the synthesis of SD-2301.</p>Fórmula:C34H42N7O11PSForma y color:SolidPeso molecular:787.24006Carumonam
CAS:<p>Carumonam, an antibiotic, could enhance the reactivity of Escherichia coli with mono- and polyclonal antisera to rough Escherichia coli J5.</p>Fórmula:C12H14N6O10S2Pureza:98%Forma y color:SolidPeso molecular:466.40EGFR-IN-162
<p>EGFR-IN-162 (compound 20) is an effective EGFR inhibitor that enhances both early and late apoptosis (EGFR) as well as necrosis (necrosis). It shows potential for use in breast cancer research.</p>Fórmula:C27H31N3O2Forma y color:SolidPeso molecular:429.241635-Hydroxypentanoic acid
CAS:5-Hydroxypentanoic acid is a PROTAC linker utilized in the synthesis of PROTAC AR-V7 degrader-1.Fórmula:C5H10O3Forma y color:SolidPeso molecular:118.13CS-VIP 8
CS-VIP 8 is a selective allosteric inhibitor of the WDR5 protein (Ki= 0.008 μM). It induces conformational changes in the MLL1 complex, causing the dissociation of MLL1 from the complex and inhibiting MLL1 histone methyltransferase activity, thereby regulating HOX gene expression. CS-VIP 8 shows potential for research in hematological diseases such as leukemia.Fórmula:C43H52F4N12O7Forma y color:SolidPeso molecular:924.4018DM-4111
CAS:<p>DM-4111, one of the primary monohydroxy metabolites of Tolvaptan, is an effective vasopressin V2 receptor (vasopressin V2 receptor) inhibitor. By inhibiting water reabsorption in renal tubules, it facilitates the excretion of electrolyte-free water. DM-4111 holds potential for research in cardiovascular diseases.</p>Fórmula:C26H25ClN2O4Forma y color:SolidPeso molecular:464.94Aminopeptidase N inhibitor 2
<p>AminopeptidaseN inhibitor 2 is an APN inhibitor (IC50: 4.3 μM) with antitumor properties.</p>Fórmula:C12H16F2N2O4SForma y color:SolidPeso molecular:322.07988Biebrich scarlet
CAS:<p>Biebrich scarlet, a scarlet dye, stains collagen in Masson's trichrome and eosinophils.</p>Fórmula:C22H16N4Na2O7S2Forma y color:Dark Red PowderPeso molecular:558.5Alvespimycin TFA
<p>Alvespimycin (17-DMAG) TFA is a potent inhibitor of Hsp90, binding with an EC50 of 62 ± 29 nM.</p>Fórmula:C34H49F3N4O10Forma y color:SolidPeso molecular:730.34008CDK9/EZH2-IN-1
CAS:CDK9/EZH2-IN-1 is a dual-target inhibitor of CDK9 and EZH2 with IC50 values of 83.9 nM and 108.6 nM, respectively. It induces apoptosis and causes DNA double-strand breaks (DSB). Additionally, CDK9/EZH2-IN-1 inhibits the proliferation of MKN45, MDA-MB-453, and SW620 cancer cells, with respective IC50 values of 136.3 nM, 171.3 nM, and 315.7 nM.Fórmula:C47H59N11O4S2Forma y color:SolidPeso molecular:906.17RNAP-σ interaction inhibitor-1
CAS:<p>RNAP-σ interaction inhibitor-1 (compound 5d) acts as an inhibitor of the interaction between RNA polymerase and the sigma factor. It exhibits activity against Streptococci with a minimum inhibitory concentration (MIC) ranging from 1-2 µg/mL.</p>Fórmula:C19H11Cl3N2O6S2Forma y color:SolidPeso molecular:533.79Omadacycline tosylate
CAS:<p>Omadacycline tosylate (PTK 0796 tosylate) is an orally available antibacterial agent and tetracycline antibiotic, broad-spectrum antimicrobial activity.</p>Fórmula:C36H48N4O10SPureza:98%Forma y color:SolidPeso molecular:728.85ADP-β-S trisodium
ADP-β-S (trisodium) is an analog of ADP and acts as a partial agonist. It can induce human platelet aggregation and inhibit PGE1-stimulated adenylate cyclase.Fórmula:C10H12N5Na3O9P2SForma y color:SolidPeso molecular:508.95241CAXII-IN-2
CAXII-IN-2 (compound 3j) is a highly effective inhibitor of CAXII. It demonstrates inhibitory activity against CA IX and CAXII, with Ki values of 27.4 nM and 4.0 nM, respectively.Fórmula:C16H13FNO4PForma y color:SolidPeso molecular:333.05662PD-1/PD-L1-IN-55
CAS:PD-1/PD-L1-IN-55 (compound D6) is a potent PD-1/PD-L1 inhibitor with an IC50 of 4.8 nM. It enhances IFN-γ secretion and decreases the proportion of late apoptosis due to PD-L1.Fórmula:C25H23ClN2O3Forma y color:SolidPeso molecular:434.92Androgen receptor antagonist 13
CAS:Androgen receptor antagonist 13 (compound 8a) is an orally active androgen receptor antagonist with an IC50 of 0.20 μM. It is used in prostate cancer research.Fórmula:C16H15N3O3SForma y color:SolidPeso molecular:329.37Mitochondrial-IN-1
CAS:Mitochondrial-IN (C458) is a potent inhibitor of mitochondrial complex I. It offers significant protection against Aβ toxicity, exhibits favorable pharmacokinetic properties, and has minimal off-target effects.Fórmula:C22H30N2OForma y color:SolidPeso molecular:338.49Deltamethrin
CAS:<p>Deltamethrin, a pyrethroid insecticide, causes reversible hind limb rigidity in rats and is used for crop protection and disease control.</p>Fórmula:C22H19Br2NO3Pureza:99.25% - 99.85%Forma y color:White To Off-White Crystals Or PowderPeso molecular:505.20CDA-IN-4
CAS:<p>CDA-IN-4 (compound VS-24) is an inhibitor of chitin deacetylase (CDA). At a concentration of 100 μg/mL, CDA-IN-4 provides a protective effect of 61.2% against rice blast disease.</p>Fórmula:C10H9BrN4O2SForma y color:SolidPeso molecular:329.17Trimegestone
CAS:Trimegestone, a highly effective oral progestogen, is used for endometrial protection, all doses inducing secretory endometrial transformation.Fórmula:C22H30O3Pureza:98%Forma y color:SolidPeso molecular:342.47
