Entre las marcas de nuestros más de 25 colaboradores destaca TargetMol
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Termina el 31 dic( quedan 8 días )
4-Biphenylboronic acid
CAS:<p>4-Biphenylboronic acid is a boric acid substance widely used in medicine and other fields.</p>Fórmula:C12H11BO2Pureza:99.53%Forma y color:SolidPeso molecular:198.034-Biphenylcarboxylic acid
CAS:<p>4-Biphenylcarboxylic acid is a polarographic reagent used in pharmaceutical synthesis, with potent antifungal and antibacterial properties.</p>Fórmula:C13H10O2Pureza:99.58%Forma y color:SolidPeso molecular:198.221Topoisomerase IIα-IN-9
CAS:Compound EN300-20599, with CAS No. 16346-97-7, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound EN300-20599 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Fórmula:C14H14O4SForma y color:SolidPeso molecular:278.321,4-Cineole
CAS:1,4-Cineole (Isocineole) is a natural, oxygenated monoterpene. 1,4-Cineole can activate both human TRPM8 and human TRPA1.Fórmula:C10H18OPureza:97.15%Forma y color:Colorless Liq LiquidPeso molecular:154.25A-317491
CAS:A-317491 (ABT 202) is a non-nucleotide P2X3 ( Ki: 22 nM) and P2X2/3 receptor (Ki: 9 nM) antagonist, which inhibits calcium flux mediated by the receptors.Fórmula:C33H27NO8Pureza:98.08%Forma y color:SolidPeso molecular:565.57A-317491 sodium
A-317491 blocks P2X3 and P2X2/3 receptors, easing inflammatory pain and neuropathy in rats.Fórmula:C33H24NNa3O8Forma y color:SolidPeso molecular:631.12740 Y-P
CAS:740 Y-P (740YPDGFR) is a PI3K activator with cell permeability,binds GST fusion proteins containing the N-and C-terminal SH2 domains of p85. Low-Cost!Fórmula:C141H222N43O39PS3Pureza:98.3% - 99.87%Forma y color:SolidPeso molecular:3270.7740 Y-P(TFA)
<p>740 Y-P(TFA)(1236188-16-1 free base) (740YPDGFR(TFA)) is a potent and cell-permeable activator of PI3K.</p>Fórmula:C143H223F3N43O41PS3Pureza:98%Forma y color:SolidPeso molecular:3384.73740 Y-P acetate
740 Y-P acetate (740YPDGFR acetate) is a potent and cell-permeable PI3K activator.740 Y-P acetate tends to bind to GST fusion proteins containing the N- and C-Fórmula:C143H226N43O41PS3Pureza:99.92%Forma y color:SoildPeso molecular:3330.79Albiglutide Fragment
CAS:<p>Albiglutide fragment is a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36).</p>Fórmula:C148H224N40O45Pureza:98%Forma y color:SolidPeso molecular:3283.6KO-947
CAS:<p>KO-947 is a potent and specific inhibitor of ERK1/2 kinases.</p>Fórmula:C21H17N5OPureza:97.84%Forma y color:SolidPeso molecular:355.39Cintirorgon
CAS:Cintirorgon (LYC-55716) is a selective, oral agonist of RORγ. Cintirorgon modulates gene expression of RORγ expressing T lymphocyte immune cells.Fórmula:C27H23F6NO6SPureza:99.92%Forma y color:SolidPeso molecular:603.53Cintirorgon sodium
CAS:Cintirorgon (LYC-55716) is an oral RORgamma agonist with immunomodulatory and anticancer effects.Fórmula:C27H23F6NNaO6SPureza:98%Forma y color:SolidPeso molecular:626.52MT-DADMe-ImmA
CAS:<p>MT-DADMe-ImmA (MTDIA) is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP, Ki: 90 pM).</p>Fórmula:C13H19N5OSPureza:99.56%Forma y color:SolidPeso molecular:293.39UCB9608
CAS:UCB9608 is a selective and orally active PI4KIIIβ inhibitor (IC50: 11 nM), selective over PI3KC2 α, β, and γ lipid kinases.Fórmula:C20H26N8O2Pureza:97.53% - 99.59%Forma y color:SolidPeso molecular:410.47Brepocitinib
CAS:Brepocitinib (PF-06700841) is a potent dual JAK1/TYK2 inhibitor (IC50s: 17 nM/23 nM). Brepocitinib also inhibits JAK2/3 (IC50s: 77 nM/6.49 μM).Fórmula:C18H21F2N7OPureza:99.82%Forma y color:SolidPeso molecular:389.4PF-06869206
CAS:PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).Fórmula:C15H14ClF3N4O2Pureza:99.79% - 99.88%Forma y color:SolidPeso molecular:374.75AZ3451
CAS:<p>AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).</p>Fórmula:C30H27BrN4O3Pureza:98.12%Forma y color:SolidPeso molecular:571.46BTTAA
CAS:<p>BTTAA, a Cu(I)-stabilizing ligand, performs potently with ubiquitin Glu18AzF.</p>Fórmula:C19H30N10O2Pureza:99.01%Forma y color:White SolidPeso molecular:430.51GNE-131
CAS:<p>GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).</p>Fórmula:C23H30N4O3SPureza:98.54% - 99.59%Forma y color:SolidPeso molecular:442.57PRN1371
CAS:<p>PRN1371 is a specific and potent FGFR1-4 and CSF1R inhibitor (IC50s: 0.6/1.3/4.1/19.3/8.1 nM for FGFR1/2/3/4 and CSF1R).</p>Fórmula:C26H30Cl2N6O4Pureza:98.65%Forma y color:SolidPeso molecular:561.46NKP-1339
CAS:NKP-1339 (IT-139) induces G2/M cell cycle arrest, blockage of DNA synthesis, and induction of apoptosis via the mitochondrial pathway.Fórmula:C14H12Cl4N4NaRuPureza:98%Forma y color:SolidPeso molecular:502.14AB-423
CAS:<p>AB-423 is an inhibitor of HBV capsid assembly, and potently inhibits HBV replication (EC50/EC90: 0.08-0.27 μM/0.33-1.32 μM in cells).</p>Fórmula:C17H17F3N2O3SPureza:99.72% - 99.89%Forma y color:SolidPeso molecular:386.396-Amino-5-azacytidine
CAS:<p>6-Amino-5-azacytidine has an inhibitory of the growth of E. coli.</p>Fórmula:C8H13N5O5Pureza:99.6%Forma y color:SolidPeso molecular:259.22RR6
CAS:RR6 acts as a selective, reversible, and competitive vanin inhibitor at nanomolar concentration.Fórmula:C16H23NO4Pureza:98.98%Forma y color:SolidPeso molecular:293.36AMG 837 calcium hydrate
CAS:<p>AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.</p>Fórmula:C52H44CaF6O8Pureza:98.07%Forma y color:SolidPeso molecular:950.97Ningetinib
CAS:<p>Ningetinib (CT-053) (CT053PTSA) is an orally bioavailable tyrosine kinase inhibitor with IC50s of <1.0, 1.9 and 6.7 nM for Axl, VEGFR2, and c-Met, respectively.</p>Fórmula:C31H29FN4O5Pureza:99.95% - 99.98%Forma y color:SolidPeso molecular:556.58Capromorelin Tartrate
CAS:<p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>Fórmula:C32H41N5O10Pureza:97.69%Forma y color:SolidPeso molecular:655.7Lorediplon
CAS:<p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>Fórmula:C20H15FN4O2SPureza:99.12% - 99.19%Forma y color:SolidPeso molecular:394.423-Hydroxyglutaric acid
CAS:3-Hydroxyglutaric acid is one of several metabolites produced when insufficient levels of GCDH are available. It is used as a biomarker of GCDH deficiency.Fórmula:C5H8O5Pureza:99.93%Forma y color:SolidPeso molecular:148.11E7046
CAS:E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.Fórmula:C22H18F5N3O4Pureza:99.86%Forma y color:SolidPeso molecular:483.4MDR-1339
CAS:MDR-1339 is a blood-brain-barrier-permeable inhibitor of amyloid-β (Aβ) aggregation.Fórmula:C20H22O4Pureza:98.57%Forma y color:SolidPeso molecular:326.39Transcrocetinate disodium
CAS:Transcrocetinate disodium (Disodium trans-crocetinate), extracted from saffron (Crocus sativus L.), is a high-affinity antagonist of NMDA receptor.Fórmula:C20H22Na2O4Pureza:98.27% - 99.22%Forma y color:SolidPeso molecular:372.37EX229
CAS:EX229 (C991) is an allosteric activator of AMPK, with Kds of 0.06 μM, 0.06 μM and 0.51 μM for α1β1γ1, α2β1γ1, and α1β2γ1, respectively.Fórmula:C24H18ClN3O3Pureza:99.20% - 99.36%Forma y color:SolidPeso molecular:431.87ASTX660
CAS:Tolinapant (ASTX660) is an orally bioavailable cIAP1/2 and XIAP antagonist.Cost-effective and quality-assured.Fórmula:C30H42FN5O3Pureza:98.33% - 99.85%Forma y color:SolidPeso molecular:539.68Tomeglovir
CAS:Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).Fórmula:C23H27N3O4SPureza:98%Forma y color:SolidPeso molecular:441.54Rosiptor
CAS:<p>Rosiptor (AQX-1125) (AQX-1125) is an orally-active and specific phosphatase SHIP1 activator with anti-inflammatory effects.</p>Fórmula:C20H35NO2Pureza:99.53% - 99.73%Forma y color:SolidPeso molecular:321.5Rosiptor acetate
CAS:Rosiptor (AQX-1125) activates SHIP1, inhibits Akt, and reduces inflammation and allergy in rodents.Fórmula:C22H39NO4Pureza:98%Forma y color:Solid PowderPeso molecular:381.55Zegocractin
CAS:<p>Zegocractin (CM-4620) is a calcium-release activated calcium-channel (CRAC channel) inhibitor.</p>Fórmula:C19H11ClF3N3O3Pureza:98.82%Forma y color:SolidPeso molecular:421.76Lumicitabine
CAS:Lumicitabine (ALS-008176) is an inhibitor of RSV polymerase.Fórmula:C18H25ClFN3O6Forma y color:SolidPeso molecular:433.86Fulacimstat
CAS:Fulacimstat (BAY1142524) (BAY1142524) is a chymase inhibitor, with IC50s of 3, 4 nM for hamster and human chymase enzyme, respectively.Fórmula:C23H16F3N3O6Pureza:99.77%Forma y color:SolidPeso molecular:487.38Anemarrhenasaponin I
CAS:Anemarrhenasaponin I shows the remarkable inhibiting effect on platelet aggregation.Fórmula:C39H66O14Pureza:98.29% - 99.85%Forma y color:SolidPeso molecular:758.93Abrocitinib
CAS:<p>Abrocitinib (PF-04965842) (PF-04965842) is a potent, specific and orally-active JAK1 inhibitor (IC50s: 29/803 nM for JAK1/2).</p>Fórmula:C14H21N5O2SPureza:99.09% - 99.91%Forma y color:SolidPeso molecular:323.41Brensocatib
CAS:<p>Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).</p>Fórmula:C23H24N4O4Pureza:97.55%Forma y color:SolidPeso molecular:420.46(±)-Zanubrutinib
CAS:(±)-Zanubrutinib ((±)-BGB-3111) is a potent and orally available Bruton's tyrosine kinase (Btk) inhibitor that demonstrates superior oral bioavailability,Fórmula:C27H29N5O3Pureza:99.09%Forma y color:SolidPeso molecular:471.55ONO-8590580
CAS:ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Fórmula:C21H21FN6Pureza:99.43%Forma y color:SolidPeso molecular:376.43Ningetinib Tosylate
CAS:Ningetinib Tosylate is an orally bioavailable tyrosine kinase inhibitor with IC50s of <1.0, 1.9 and 6.7 nM for Axl, VEGFR2, and c-Met, respectively.Fórmula:C38H37FN4O8SPureza:99.93%Forma y color:SolidPeso molecular:728.79BAY-1436032
CAS:<p>BAY-1436032 is a novel, selective and orally available inhibitor of pan-mutant isocitrate dehydrogenase 1 (IDH1).</p>Fórmula:C26H30F3N3O3Pureza:99.65% - 99.71%Forma y color:SolidPeso molecular:489.53Dofequidar
CAS:<p>Dofequidar (MS-209 free base) is a quinoline derivative that inhibits the efflux of chemotherapeutic agents.</p>Fórmula:C30H31N3O3Pureza:98%Forma y color:SolidPeso molecular:481.59Seletalisib
CAS:Seletalisib (UCB5857) (UCB5857) is a potent and specific PI3Kδ inhibitor (IC50: 12 nM).Fórmula:C23H14ClF3N6OPureza:99.81%Forma y color:SolidPeso molecular:482.85
