Entre las marcas de nuestros más de 25 colaboradores destaca TargetMol
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Termina el 31 dic( quedan 8 días )
GNE-2256
CAS:GNE-2256, also known as molecule 19, is an orally active compound that inhibits Interleukin 1 receptor-associated kinase 4 (IRAK4) with a K i of 1.4 nM and hasFórmula:C24H27FN6O4Forma y color:SolidPeso molecular:482.51TP-030-2
CAS:<p>TP-030-2 is a RIPK1 inhibitor (human K i =0.43 nM ; mouse IC 50 =100 nM) .</p>Fórmula:C23H21BrN4O3Forma y color:SolidPeso molecular:481.34TP-030-1
CAS:TP-030-1, RIPK1 inhibitor: K(i) hRIPK1 at 3.9nM, IC50 mRIPK1 at 4.2μM; targets inflammation, neurodegeneration research.Fórmula:C23H22N4O3Forma y color:SolidPeso molecular:402.45CK2-IN-4
CAS:<p>CK2-IN-4 is a protein kinase (CK2) inhibitor with an IC50 value of 8.6 µM.</p>Fórmula:C18H11N3O4SPureza:99.72%Forma y color:SolidPeso molecular:365.36IGUANA-1
CAS:<p>IGUANA-1 is a highly efficient and selective ALDH1B1 inhibitor that inhibits the growth of colorectal cancer cells and colorectal cancer cell-derived organoids.</p>Fórmula:C27H26ClN3O4Pureza:99.08%Forma y color:SolidPeso molecular:491.97MSC-1186
CAS:<p>MSC-1186 selectively inhibits SRPKs—IC50: 2.7nM (SRPK1), 81nM (SRPK2), 0.6nM (SRPK3)—for cancer research.</p>Fórmula:C19H17ClFN7O2SForma y color:SolidPeso molecular:461.9TMV-IN-1
CAS:TMV-IN-1: a chalcone inhibits TMV with EC50s of 70.7 and 60.8 μg/mL, applicable in infection and tumor studies.Fórmula:C28H26O4Forma y color:SolidPeso molecular:426.5DHBP dibromide
CAS:DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.Fórmula:C24H38Br2N2Pureza:99.73%Forma y color:Yellow To Yellow-Green Powder Or FlakesPeso molecular:514.38CK2-IN-6
CAS:CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.Fórmula:C19H16ClN7O2Forma y color:SolidPeso molecular:409.83BGB-8035
CAS:<p>BGB-8035 is a BTK inhibitor with antitumor activity that inhibits BTK, TEC, and EGFR.BGB-8035 is used in the study of tumors and autoimmune diseases.</p>Fórmula:C24H31N5O4Pureza:96.74%Forma y color:SolidPeso molecular:453.53SZM-1209
CAS:<p>SZM-1209 is a potent and specific RIPK1 inhibitor with oral activity, displaying a dissociation constant (Kd) of 85 nM.</p>Fórmula:C31H29F5N4O5S2Pureza:98%Forma y color:SolidPeso molecular:696.71GLPG3970
CAS:GLPG3970, a pioneering inhibitor of SIK2/SIK3, is utilized in the investigation of inflammation and autoimmune diseases.Fórmula:C25H27F3N4O4Pureza:99.60% - >99.99%Forma y color:SolidPeso molecular:504.5DKFZ-748
CAS:<p>DKFZ-748 is a selective HDAC10 inhibitor and has a dose-dependent growth inhibitory effect on HeLa cells.</p>Fórmula:C18H23N3O3Pureza:98.10%Forma y color:SolidPeso molecular:329.39RGT-068A
CAS:RGT-068A is a potent, selective and oral bioavailable MALT1 inhibitor .Fórmula:C17H16ClN9O2Forma y color:SolidPeso molecular:413.82DHBP
CAS:DHBP (Benzoresorcinol) is an WalKR TCS activator.Fórmula:C13H10O3Pureza:99.95%Forma y color:Light-Yellow Solid CrystallinePeso molecular:214.22Angiotensin (1-7)
CAS:Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) is a synthetic heptapeptide, inhibits canine ACE activity with vasodilator and antiproliferative activities.Fórmula:C41H62N12O11Pureza:>99.99%Forma y color:White Lyophilised SolidPeso molecular:899I-BET432
I-BET432, a BET inhibitor, blocks BRD4 BD1/BD2 (pIC50: 7.5/7.2), is oral, and targets cancer/inflammation.Fórmula:C18H21N3O3Forma y color:SolidPeso molecular:327.38BLM-IN-2
BLM-IN-2: BLM inhibitor, IC50=0.8 μM; hinders CRC cell growth, invasion, cycle arrest, and death.Fórmula:C33H38BrFN4OForma y color:SolidPeso molecular:605.58TUL01101
CAS:<p>TUL01101, a selective oral JAK1 inhibitor (IC50: 3 nM), also targets JAK2, JAK3, TYK2; for rheumatoid arthritis research.</p>Fórmula:C22H25F2N5O2Forma y color:SolidPeso molecular:429.46BAY-7081
BAY-7081 is a cyanopyridone-based compound that functions as a potent, selective, and orally active PDE9A inhibitor, demonstrating an inhibition concentration (Fórmula:C19H27ClN4OForma y color:SolidPeso molecular:362.9ASPER-29
CAS:ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.Fórmula:C31H29BrN2O5SForma y color:SolidPeso molecular:621.54ARS-2102
CAS:ARS-2102 is a potent covalent KRAS G12C inhibitor for use in cancer research .Fórmula:C28H31ClF2N6O2Forma y color:SolidPeso molecular:557.03ENT-C225
CAS:ENT-C225 is a potent TrkB neurotrophin receptor (TrkBR) activator with neuroprotective activity for the study of Alzheimer's disease and Parkinson's disease.Fórmula:C26H40N4O5Pureza:99.36% - 99.36%Forma y color:SolidPeso molecular:488.62FTX-6746
CAS:FTX-6746 is an orally active and selective PPARG reverse inhibitor with anticancer activity. It can be used in research on urothelial carcinoma.Fórmula:C16H7ClF2N2OPureza:98.68%Forma y color:SolidPeso molecular:316.695'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Fórmula:C12H16N6O4Pureza:98.95% - ≥95%Forma y color:PowderPeso molecular:308.29PG-11047
CAS:PG-11047 (CGC-11047) is a polyamine analogue utilized in breast cancer research.Fórmula:C14H32N4Forma y color:SolidPeso molecular:256.43PG-11047 2HCl
PG-11047 2HCl treats genitourinary, immune, genetic, ocular, blood/lymphatic disorders, and aids lymphoma/prostate cancer research.Fórmula:C14H34Cl2N4Pureza:97.47%Forma y color:SolidPeso molecular:329.35Debneyol
CAS:Debneyol exhibits more potent fungicidal activity than validamycin.Fórmula:C15H26O2Forma y color:SolidPeso molecular:238.37Flavipin
CAS:Flavipin: Ahr agonist, alters Ahr genes in T cells/macrophages, disrupts Arid5a, scavenges DPPH (IC50=7.2μM), inhibits α-glucosidase (IC50=33.8μM).Fórmula:C9H8O5Forma y color:SolidPeso molecular:196.16Aviculin
CAS:Aviculin, a lignan glycoside, exhibits anticancer properties by inducing apoptosis in breast cancer cells with an IC50 of 75.47 μM.Fórmula:C26H34O10Forma y color:SolidPeso molecular:506.54JNJ-9350
CAS:<p>JNJ-9350: SMOX inhibitor (IC50 0.01 μM), PAO inhibitor (IC50 0.79 μM), for cancer research.</p>Fórmula:C25H22N6OForma y color:SolidPeso molecular:422.48Immepip
CAS:Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.Fórmula:C9H15N3Forma y color:SolidPeso molecular:165.24SBI-993
CAS:SBI-993 is a potent SBI-477 analog with good pharmacokinetics and enhances insulin signaling by inhibiting MondoA.Fórmula:C23H24N4O4SForma y color:SolidPeso molecular:452.53Diclofensine
CAS:<p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>Fórmula:C17H17Cl2NOPureza:97.01% - 98.13%Forma y color:SolidPeso molecular:322.23MK-4541
CAS:MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.Fórmula:C22H31F3N2O3Forma y color:SolidPeso molecular:428.49PV-1019
CAS:PV-1019 (NSC 744039), a potent Chk2 inhibitor, has an IC50 of 24 nM and blocks Chk2 autophosphorylation and IR-induced apoptosis.Fórmula:C18H17N7O3Forma y color:SolidPeso molecular:379.37Cadein1
Cadein1, an isoquinolinium derivative, induces G2/M phase delay and caspase-dependent apoptosis in cancer cells lacking functional p53.Fórmula:C33H48F2INO2Forma y color:SolidPeso molecular:655.64EDP-305
CAS:<p>EDP-305, an oral FXR agonist, has EC50s of 34 nM/8 nM in CHO/HEK cells, aids in PBC and NASH research with antifibrotic properties.</p>Fórmula:C36H58N2O5SForma y color:SolidPeso molecular:630.92Miclxin
CAS:Miclxin (DS37262926) is a novel MIC60 inhibitor that induces apoptosis through mitochondrial stress in mutant tumor cells via β-catenin.Miclxin is a potentFórmula:C26H27N5O2Pureza:99.17% - 99.99%Forma y color:SolidPeso molecular:441.52BiCAPPA
CAS:BiCAPPA, a bivalent antiprion, reduces scrapie-infected prion proteins with 0.32 μM efficiency.Fórmula:C38H40Cl2N6O2Forma y color:SolidPeso molecular:683.67Con B-1
CAS:ConB-1 is a potent and selective ALK inhibitor with low toxicity to normal cells .Fórmula:C38H52ClN7O6SForma y color:SolidPeso molecular:770.38JMX0293
<p>JMX0293, a salicylamide derivative, inhibits STAT3, inducing MDA-MB-231 cell apoptosis with IC50=3.38μM, while sparing MCF-10A (IC50>60μM).</p>Fórmula:C25H30Cl2N4O7Forma y color:SolidPeso molecular:569.43BM212
CAS:BM212 is an antimycobacterial compound.It inhibits the growth of laboratory and clinical isolate M. tuberculosis strains.Fórmula:C23H25Cl2N3Pureza:99.13%Forma y color:SolidPeso molecular:414.37SP-471P
CAS:SP-471P inhibits DENV protease; EC50: DENV1-5.9 μM, DENV2-1.4 μM, DENV3-5.1 μM, DENV4-1.7 μM; CC50 >100 μM; lowers viral RNA synthesis.Fórmula:C33H26BrN5O2Forma y color:SolidPeso molecular:604.5CPT-Se3
CAS:CPT-Se3, a camptothecin derivative, boosts anticancer activity, triggers apoptosis in Hep G2, and is cytotoxic to various cells with IC50 of 2.19-4.7 μM.Fórmula:C24H20N2O6Se2Pureza:98%Forma y color:SolidPeso molecular:590.35CPT-Se4
CAS:CPT-Se4, a seleno-derivative of CPT, effectively kills cancer cells, triggers apoptosis, and is cytotoxic against various cell lines.Fórmula:C25H24N2O7Se2Pureza:98%Forma y color:SolidPeso molecular:622.39GA-O-02
GA-O-02, an 18β-Glycyrrhetinic acid derivative, inhibits NO/cytokines and fights Gram-positive bacteria; potent anti-inflammatory/antimicrobial.Fórmula:C37H46ClNO6Forma y color:SolidPeso molecular:636.22GA-O-06
GA-O-06: 18β-Glycyrrhetinic acid derivative with powerful antimicrobial effects on Gram-positive bacteria and anti-inflammatory properties.Fórmula:C37H46FNO6Forma y color:SolidPeso molecular:619.76CFT8634
CAS:CFT8634 degrades BRD9, for synovial sarcoma and SMARCB1 tumor research, from patent WO2021178920A1.Fórmula:C37H45F3N6O5Forma y color:SolidPeso molecular:710.79VT02956
CAS:<p>VT02956 inhibits LATS1 (IC50: 0.76 nM) & LATS2 (0.52 nM), targets Hippo pathway, and hampers ER+ breast cancer growth.</p>Fórmula:C22H23N5OForma y color:SolidPeso molecular:373.45
