Entre las marcas de nuestros más de 25 colaboradores destaca TargetMol
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Termina el 31 dic( quedan 8 días )
2-Hydroxy atorvastatin calcium salt
CAS:2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).Fórmula:C33H34FN2O60·5CaPureza:97.06%Forma y color:SolidPeso molecular:593.68Bavisant
CAS:<p>Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.</p>Fórmula:C19H27N3O2Pureza:99.21% - 99.65%Forma y color:SolidPeso molecular:329.44DG051
CAS:DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM).Fórmula:C21H25Cl2NO4Pureza:98.26%Forma y color:SolidPeso molecular:426.33BI-882370
CAS:BI-882370 is a specific RAF kinase inhibitor.Fórmula:C28H33F2N7O2SPureza:97.33% - 99.07%Forma y color:SolidPeso molecular:569.67MC-DOXHZN hydrochloride
CAS:<p>MC-DOXHZN hydrochloride is an albumin-binding prodrug of Doxorubicin. Doxorubicin is a DNA topoisomerase II inhibitor.</p>Fórmula:C37H43ClN4O13Pureza:98%Forma y color:SolidPeso molecular:787.22NCGC00244536
CAS:NCGC00244536 (KDM4B Inhibitor B3) is a potent KDM4B inhibitor (IC50: 10 nM).Fórmula:C25H22N2O2Pureza:97.2% - 99.72%Forma y color:SolidPeso molecular:382.45MK-7246
CAS:MK-7246 is a potent and specific CRTH2 antagonist (Ki: 2.5 nM).Fórmula:C21H21FN2O4SForma y color:SolidPeso molecular:416.47SH5-07
CAS:<p>SH5-07 is a hydroxamic acid-based Stat3 inhibitor (IC50: 3.9 μM).</p>Fórmula:C29H28F5N3O5SPureza:95.54%Forma y color:SolidPeso molecular:625.61Fadraciclib
CAS:<p>Fadraciclib (CYC065) is an orally available, second-generation ATP-competitive inhibitor of CDK2/CDK9 kinases (IC50s: 5/26 nM).</p>Fórmula:C21H31N7OPureza:99.75%Forma y color:SolidPeso molecular:397.52Purpureaside C
CAS:Purpureaside C is a phenolic glycoside with significant proinflammatory, immunomodulating and antimicrobial effects.Fórmula:C35H46O20Pureza:97.42%Forma y color:SolidPeso molecular:786.73AMG-3969
CAS:AMG-3969 is an effective glucokinase-glucokinase regulatory protein interaction (GK-GKRP) disruptor (IC50: 4 nM).Fórmula:C21H20F6N4O3SPureza:99.65%Forma y color:SolidPeso molecular:522.46Cefuracetime
CAS:<p>Cefuracetime (SKF81367) (SKF81367) is a cephalosporin antibiotic.</p>Fórmula:C17H17N3O8SPureza:98.33%Forma y color:SolidPeso molecular:423.4AVE 0991
CAS:<p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>Fórmula:C29H32N4O5S2Pureza:98.69%Forma y color:SolidPeso molecular:580.72MI-463
CAS:MI-463 is a potent and orally bioavailable inhibitor of the menin-mLL interaction (IC50: 15.3 nM).Fórmula:C24H23F3N6SPureza:99.18% - >99.99%Forma y color:SolidPeso molecular:484.54Ilorasertib
CAS:Ilorasertib (ABT-348) inhibits Aurora kinases A/B/C & RET, PDGFRβ, Flt1 (IC50: 1-120 nM).Fórmula:C25H21FN6O2SPureza:96.17% - 97.49%Forma y color:SolidPeso molecular:488.54LY2857785
CAS:LY2857785 is a type I competitive and reversible ATP kinase inhibitor against CDK7/CDK8/CDK9 (IC50s: 246 nM/16 nM/11 nM).Fórmula:C26H36N6OPureza:99.68%Forma y color:Solid PowderPeso molecular:448.6CHZ868
CAS:<p>CHZ868 is a type II JAK inhibitor with potential antitumor activity that reverses the persistence of type I JAK inhibitors and can be used to study leukemia.</p>Fórmula:C22H19F2N5O2Pureza:99.38%Forma y color:SolidPeso molecular:423.42Nastorazepide
CAS:Nastorazepide is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity.Fórmula:C29H36N4O5Pureza:99.83%Forma y color:SolidPeso molecular:520.62Zoliflodacin
CAS:Zoliflodacin (ETX0914) (ETX0914, AZD0914) is a new bacterial DNA gyrase/topoisomerase inhibitor.Fórmula:C22H22FN5O7Pureza:99.82% - 99.93%Forma y color:SolidPeso molecular:487.44Peretinoin
CAS:Peretinoin (NIK333) is an oral acyclic retinoid with a vitamin A-like structure that targets retinoid nuclear receptors such as RXR and RAR.Fórmula:C20H30O2Pureza:97.23%Forma y color:SolidPeso molecular:302.45Pseudobufarenogin
CAS:Pseudobufarenogin (ψ-Bufarenogin), a novel anti-tumor compound, suppresses liver cancer growth by inhibiting receptor tyrosine kinase-mediated signaling.Fórmula:C24H32O6Pureza:99.34%Forma y color:SolidPeso molecular:416.51GSK189254A
CAS:<p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>Fórmula:C21H25N3O2Pureza:98.71% - 99.858%Forma y color:SolidPeso molecular:351.44GSK484 hydrochloride
CAS:GSK484 hydrochloride (GTPL8577) is a reversible peptidyl-arginine deiminase 4 (PAD4) inhibitor.Cost-effective and quality-assured.Fórmula:C27H32ClN5O3Pureza:98.32% - 99.62%Forma y color:SolidPeso molecular:510.03NVP-LCQ195
CAS:NVP-LCQ195 (LCQ-195) (AT9311) is a potent inhibitor of CDK1, CDK2, CDK3 and CDK5 (IC50: 1-42 nM).Fórmula:C17H19Cl2N5O4SPureza:99.56% - 99.85%Forma y color:SolidPeso molecular:460.33MI-503
CAS:<p>MI-503 is an efficient and selective Menin-MLL inhibitor. MI-503 has a significant inhibitory effect on human MLL leukemia cell line. Cost-effective and quality-assured.</p>Fórmula:C28H27F3N8SPureza:99.87% - 99.99%Forma y color:SolidPeso molecular:564.63Luteolin-3-O-β-D-glucuronide
CAS:<p>Luteolin-3-O-beta-D-glucuronide is active in the inhibition of nitrite production in macrophages.</p>Fórmula:C21H18O12Pureza:98.56% - 99.51%Forma y color:SolidPeso molecular:462.36Navoximod
CAS:Navoximod (GDC-0919) (NLG- 919, GDC-0919) is a potent indoleamine-(2,3)-dioxygenase (IDO) pathway inhibitor (Ki/EC50: 7 nM/75 nM).Fórmula:C18H21FN2O2Pureza:99.37%Forma y color:SolidPeso molecular:316.37Warangalone
CAS:Warangalone inhibits malaria parasites 3D7 and K1 with IC50s: 4.8 and 3.7 μg/mL, respectively.Fórmula:C25H24O5Pureza:98%Forma y color:SolidPeso molecular:404.46Andropanolide
CAS:Andropanolide is a dipterocarp from Andrographis paniculata with antimalarial and anticancer activity and inhibits the overproduction of nitric oxide.Fórmula:C20H30O5Pureza:98.82% - 98.90%Forma y color:SolidPeso molecular:350.45ACY-775
CAS:<p>ACY-775 is an effective and specific inhibitor of HDAC6 (IC50: 7.5 nM).</p>Fórmula:C17H19FN4O2Pureza:97.67% - 98.83%Forma y color:SolidPeso molecular:330.36KIRA6
CAS:<p>KIRA6 is an effective inhibitor of IRE1α RNase kinase (IC50: 0.6 μM). It can trigger an apoptotic response.</p>Fórmula:C28H25F3N6OPureza:97.91%Forma y color:SolidPeso molecular:518.53Ceftobiprole
CAS:<p>Ceftobiprole (Ro 63-9141) is a β-lactam antibacterial agent that exhibits potent bactericidal activity by binding to PBPs.Cost-effective and quality-assured.</p>Fórmula:C20H22N8O6S2Pureza:95%Forma y color:SolidPeso molecular:534.57CDK-IN-2
CAS:<p>CDK-IN-2 (CDK inhibitor II) is a potent and specific CDK9 inhibitor (IC50: <8 nM).</p>Fórmula:C18H19ClFN3O2Pureza:99.67%Forma y color:SolidPeso molecular:363.81GNE-495
CAS:GNE-495 is a potent and specific MAP4K4 inhibitor (IC50: 3.7 nM).Fórmula:C22H20FN5O2Pureza:99.22% - 99.57%Forma y color:SolidPeso molecular:405.42SU14813 maleate
CAS:SU14813 maleate is an inhibitor of multi-targeted receptor tyrosine kinases (IC50s: 2, 50, 4, 15 nM for VEGFR1, VEGFR2, PDGFRβ, and KIT).Fórmula:C27H31FN4O8Pureza:98%Forma y color:SolidPeso molecular:558.56JPH203
CAS:<p>JPH203 (KYT-0353) is a potent and specific inhibitor of L-type amino acid transporter protein 1 (LAT-1).</p>Fórmula:C23H19Cl2N3O4Pureza:97.32% - 99.43%Forma y color:SolidPeso molecular:472.32Aticaprant
CAS:<p>Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.</p>Fórmula:C26H27FN2O2Pureza:99.53% - 99.93%Forma y color:SolidPeso molecular:418.5NI-57
CAS:<p>NI-57 inhibits BRPF family proteins: BRPF1 (IC50=3.1nM), BRPF2 (IC50=46nM), BRPF3 (IC50=140nM).</p>Fórmula:C19H17N3O4SPureza:99.88% - >99.99%Forma y color:SolidPeso molecular:383.42lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Forma y color:SolidPeso molecular:565.7Presatovir
CAS:Presatovir (GS-5806) (GS-5806) is a novel, orally bioavailable RSV fusion inhibitor (mean EC50: 0.43 nM).Fórmula:C24H30ClN7O3SPureza:99.14% - 99.92%Forma y color:SolidPeso molecular:532.06AF38469
CAS:AF38469 is a new, specific and orally bioavailable Sortilin inhibitor (IC50: 330 nM).Fórmula:C15H11F3N2O3Pureza:99.18%Forma y color:SolidPeso molecular:324.25NKP608
CAS:NKP608 is a NK-1 receptor antagonist with anticancer and anxiolytic activities.Fórmula:C31H24ClF6N3O2Pureza:99.88% - 99.88%Forma y color:SolidPeso molecular:619.99Exatecan Mesylate
CAS:<p>Exatecan Mesylate (DX8951f) is a DNA topoisomerase I inhibitor (IC50: 2.2 μM, 0.975 μg/mL).</p>Fórmula:C25H26FN3O7SPureza:97.32% - 99.9%Forma y color:SolidPeso molecular:531.55Juglanin
CAS:Juglanin is a JNK activator. Juglanin with inflammation and anti-tumor activities. It can induce apoptosis and autophagy on human breast cancer cells.Fórmula:C20H18O10Pureza:98.8% - 99.33%Forma y color:SolidPeso molecular:418.35Nesbuvir
CAS:Nesbuvir: HCV NS5B polymerase inhibitor, IC50 9 nM against HCV 1b replicon in liver cancer cells.Fórmula:C22H23FN2O5SPureza:99.99%Forma y color:SolidPeso molecular:446.49LY2795050
CAS:<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Fórmula:C23H22ClN3O2Pureza:97.77%Forma y color:SolidPeso molecular:407.89Naquotinib
CAS:Naquotinib (ASP8273) (ASP8273) is an orally available, mutant-selective and irreversible EGFR inhibitor; (IC50s: 8-33 nM and 230 nM toward EGFR mutants and EGFRFórmula:C30H42N8O3Pureza:97.49%Forma y color:SolidPeso molecular:562.71JNJ-40411813
CAS:<p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>Fórmula:C20H25ClN2OPureza:99.74%Forma y color:SolidPeso molecular:344.88Brincidofovir
CAS:Brincidofovir (HDP-CDV) is an orally active, lipophilic form of cidofovir.Fórmula:C27H52N3O7PPureza:98% - 99.62%Forma y color:SolidPeso molecular:561.69Scabertopin
CAS:Scabertopin is a sesquiterpene lactone isolated from Gentiana scabra with anticancer and bacteriostatic activities.Fórmula:C20H22O6Pureza:98.13% - 99.13%Forma y color:SolidPeso molecular:358.39
