CAS 106266-06-2
:Rispéridone
Description :
Rispéridone est un médicament antipsychotique atypique principalement utilisé pour traiter la schizophrénie, le trouble bipolaire et l'irritabilité associée à l'autisme. Il fonctionne comme un antagoniste de la sérotonine et de la dopamine, influençant l'activité des neurotransmetteurs dans le cerveau, en particulier les récepteurs de la sérotonine et de la dopamine. Rispéridone se caractérise par sa formule chimique C23H27N3O2 et un poids moléculaire d'environ 410,48 g/mol. La substance apparaît sous forme de poudre cristalline blanche à blanc cassé et est généralement administrée par voie orale, bien que des formulations injectables soient également disponibles. Sa pharmacocinétique indique une demi-vie relativement longue, permettant une posologie une fois par jour dans de nombreux cas. Les effets secondaires courants peuvent inclure la sédation, la prise de poids et des changements métaboliques, nécessitant une surveillance pendant le traitement. Le profil d'efficacité et de sécurité de Rispéridone en fait une option largement prescrite en soins psychiatriques, bien qu'il soit essentiel d'adapter le traitement aux besoins individuels du patient et de surveiller les effets indésirables potentiels.
Formule :C23H27FN4O2
InChI :InChI=1/C23H27FN4O2/c1-15-18(23(29)28-10-3-2-4-21(28)25-15)9-13-27-11-7-16(8-12-27)22-19-6-5-17(24)14-20(19)30-26-22/h5-6,14,16H,2-4,7-13H2,1H3
Code InChI :InChIKey=RAPZEAPATHNIPO-UHFFFAOYSA-N
SMILES :FC=1C=C2C(C(=NO2)C3CCN(CCC=4C(=O)N5C(=NC4C)CCCC5)CC3)=CC1
Synonymes :- 1,2-Benzisoxazole, 4H-pyrido[1,2-a]pyrimidin-4-one deriv.
- 3-(2-(4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one
- 3-[2-[4-(6-Fluor-1,2-benzisoxazol-3-yl)piperidino]ethyl]-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-on
- 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one
- 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-
- Apexidone
- Psychodal
- R 64766
- Rbp 7000
- Resperidone
- Ripedon
- Risbiodal
- Rispa
- Rispadal
- Risperdal
- Risperdal Consta
- Risperdine
- Risperid
- Risperid fort
- Risperidal
- Risperidone ACIS
- Risperidone intermediates
- Spiron
- Zophrenal
- Risperidone
- 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-(9CI)
- 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one, R-64766, Belivon, Risperdal
- Risoeridone
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-
- Kesperidone
- 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydropyrido[2,1-b]pyrimidin-4-one
- 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one, R-64766, Belivon, Risperdal
- 4h-pyrido(1,2-a)pyrimidin-4-one,6,7,8,9-tetrahydro-3-(2-(4-(6-fluoro-1,2-benzi
- 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-
- soxazol-3-yl)-1-piperidinyl)ethyl)-2-methyl-
- 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2,a]pyrimidin-4-one
- Voir plus de synonymes
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23 produits concernés.
Risperidone
CAS :RisperidoneFormule :C23H27FN4O2Degré de pureté :100.0%Couleur et forme :WhiteMasse moléculaire :410.2118RISPERIDONE FOR SYSTEM SUITABILITY CRS
CAS :<p>RISPERIDONE FOR SYSTEM SUITABILITY CRS</p>Formule :C23H27FN4O2Masse moléculaire :410.4845RISPERIDONE CRS
CAS :<p>RISPERIDONE CRS</p>Formule :C23H27FN4O2Couleur et forme :White. Powder.Masse moléculaire :410.4845Risperidone
CAS :Nucleic acids and their salts, whether or not chemically defined; other heterocyclic compounds, nesoiFormule :C23H27FN4O2Couleur et forme :White Off-White PowderMasse moléculaire :410.2118Risperidone
CAS :Formule :C23H27FN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.4845Risperidone
CAS :<p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>Formule :C23H27FN4O2Degré de pureté :99.73%Couleur et forme :Crystalline SolidMasse moléculaire :410.48Risperidone
CAS :Formule :C23H27FN4O2Couleur et forme :White To Off-White SolidMasse moléculaire :410.49Risperidone
CAS :Formule :C23H27FN4O2Degré de pureté :98.0 - 102.0 % (dried basis)Couleur et forme :White to almost white powderMasse moléculaire :410.48Risperidone
CAS :Formule :C23H27FN4O2Degré de pureté :>98.0%(T)(HPLC)Couleur et forme :White to Almost white powder to crystalMasse moléculaire :410.49Risperidone
CAS :<p>Applications Risperidone is a combined serotonin (5-HT2) and dopamine (D2) receptor antagonist.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Jannssen, P.A.J., et al.: J. Pharmacol. Exp. Ther., 244, 685 (1988); Gelders, Y.G., et al.: Pharmacopsychiatry, 23, 206 (1990); Green, B.: Curr. Med. Res. Opin., 16, 57 (2000);<br></p>Formule :C23H27FN4O2Couleur et forme :NeatMasse moléculaire :410.48Risperidone - Bio-X ™
CAS :Produit contrôlé<p>Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs.<br> Risperidone is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.</p>Formule :C23H27FN4O2Degré de pureté :Min. 99.0 Area-%Couleur et forme :White PowderMasse moléculaire :410.48 g/molRisperidone
CAS :Produit contrôlé<p>Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs. Consequently leading to hyperprolactinemia, a negative adverse effect when Risperidone is used as a drug. Risperidone has been shown to have cardiac effects, including increasing heart rate and QT interval. It is also metabolized by cytochrome P450 enzymes and can be detected in wastewater after oral administration of a single dose (0.5 mg/kg).</p>Formule :C23H27FN4O2Degré de pureté :Min. 98.5 Area-%Couleur et forme :White Off-White PowderMasse moléculaire :410.48 g/molRisperidone
CAS :Formule :C23H27FN4O2Degré de pureté :98%Couleur et forme :Solid, White to off-white powderMasse moléculaire :410.212
