CAS 1093412-18-0

Roflupram

CAS : 1093412-18-0

Roflupram is a selective inhibitor of the enzyme response element binding protein (RBP), which is responsible for the activation of gene expression in the nucleus. It has been shown to inhibit the production of inflammatory mediators such as TNF-α, IL-1β, and IL-6. Roflupram also inhibits the production of amyloid protein by microglia cells, which may be related to its clinical relevance in treating Alzheimer's disease. Roflupram binds to RBP with high affinity and specificity, blocking its interaction with DNA and preventing gene expression. This drug may be used to treat autoimmune diseases or even cancer due to its ability to inhibit tumor growth.

Formule : C₁₆H₂₀F₂O₄

Degré de pureté : Min. 95%

Masse moléculaire : 314.32 g/mol

Ref: 3D-TTB41218

FFPM

CAS : 1093412-18-0

FFPM is a novel PDE4 inhibitor (IC50: 6 nM) and good selectivity over other PDEs. The drug also penetrates the blood brain barrier well.

Formule : C₁₆H₂₀F₂O₄

Couleur et forme : Solid

Masse moléculaire : 314.32

Ref: TM-T24061