CAS 1104599-69-0

MK-4256

CAS : 1104599-69-0

MK-4256 is a synthetic β-carboline alkaloid that binds to the dopamine D2 receptor. It has an imidazole ring and a carboxylic acid. The binding of MK-4256 to the D2 receptor induces an increase in intracellular calcium levels, which leads to an inhibition of various enzymes and protein kinases, such as diastereomer and glipizide. In vitro assays have shown that MK-4256 inhibits the release of insulin from pancreatic cells without affecting other types of cells. This drug has also been shown to be effective in reducing food intake in animals; however, further studies are needed for its clinical use in humans. MK-4256 has been observed to have neuroprotective effects on dopaminergic neurons, as well as anti-inflammatory and analgesic effects in animal models.

Formule : C₂₇H₂₃FN₈O

Degré de pureté : Min. 95%

Masse moléculaire : 494.5 g/mol

Ref: 3D-EUB59969

MK-4256

CAS : 1104599-69-0

MK-4256 is an effective and selective SSTR3 antagonist (IC50s: 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively).

Formule : C₂₇H₂₃FN₈O

Couleur et forme : Solid

Masse moléculaire : 494.52

Ref: TM-T16095