CAS 113158-34-2

Norbinaltorphimine dihydrochloride

CAS : 113158-34-2

Norbinaltorphimine dihydrochloride

Degré de pureté : ≥98%

Masse moléculaire : 734.71g/mol

Ref: 54-BUP21440

Norbinaltorphimine Dihydrochloride Salt-d6

Produit contrôlé

CAS : 113158-34-2

Formule : C₄₀H₃₉D₆Cl₂N₃O₆

Couleur et forme : Neat

Masse moléculaire : 667.823

Ref: TR-N661127

Norbinaltorphimine Dihydrochloride Salt

Produit contrôlé

CAS : 113158-34-2

Applications Norbinaltorphimine Dihydrochloride Salt is a synthetic derivative of Naltrexone (N285750, HCl) and is useful as a κ-opioid antagonist.
References Agmo, A., et al.: Neuropharmacology, 37, 223 (1998); Nagase, H., et al.: Jpn. Kokai Tokkyo Koho. JP 03193782 A 19910823. Aug 23, 1991; Portoghese, P.S., et al.: J. Med. Chem., 31, 836 (1988)

Formule : C₄₀H₄₃N₃O₆·2ClH

Couleur et forme : Neat

Masse moléculaire : 734.708

Ref: TR-N661125

Norbinaltorphimine dihydrochloride

Produit contrôlé

CAS : 113158-34-2

Norbinaltorphimine dihydrochloride is a potent, selective κ-opioid receptor agonist. It binds to the κ-opioid receptor on the cell surface and blocks the signal pathway that leads to the production of endothelin-a in cells. Norbinaltorphimine dihydrochloride has been shown to be effective for the treatment of oral pathogens such as Streptococcus pyogenes, Streptococcus pneumoniae, and Neisseria sp., as well as for prevention of myocardial infarction. Norbinaltorphimine dihydrochloride also has anti-inflammatory effects, which are mediated by its ability to inhibit prostaglandin synthesis through inhibition of cyclooxygenase activity.

Formule : C₄₀H₄₅Cl₂N₃O₆

Degré de pureté : Min. 95%

Masse moléculaire : 734.71 g/mol

Ref: 3D-NEA15834

Norbinaltorphimine dihydrochloride

CAS : 113158-34-2

Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.

Formule : C₄₀H₄₅Cl₂N₃O₆

Degré de pureté : 98.17% - 99.88%

Couleur et forme : Solid

Masse moléculaire : 734.71

Ref: TM-T12241