CAS 1221186-52-2

6-[(3-Methoxyphenyl)methyl]-4-methyl-2-methylsulfinylthieno[3,4]pyrrolo[1,3-d]pyridazin-5-one

CAS : 1221186-52-2

6-[(3-Methoxyphenyl)methyl]-4-methyl-2-methylsulfinylthieno[3,4]pyrrolo[1,3-d]pyridazin-5-one is a potent inhibitor of the voltage gated sodium channels. It blocks the function of ion channels and inhibits the action of the neurotransmitter acetylcholine on postsynaptic neuromuscular junctions. The IC50 value for this compound is 1 µM, making it one of the most potent inhibitors of voltage gated sodium channels currently known. 6-[(3-Methoxyphenyl)methyl]-4-methyl-2-methylsulfinylthieno[3,4]pyrrolo[1,3-d]pyridazin-5-one has been used as a research tool in cell biology and pharmacology to study protein interactions and peptides.

Formule : C₁₈H₁₇N₃O₃S₂

Degré de pureté : Min. 95%

Masse moléculaire : 387.5 g/mol

Ref: 3D-WYB18652

ML202

CAS : 1221186-52-2

ML202 activates human pyruvate kinase M2, affecting PEP cooperativity with minimal impact on ADP binding.

Formule : C₁₈H₁₇N₃O₃S₂

Couleur et forme : Solid

Masse moléculaire : 387.48

Ref: TM-T73525