CAS 1262769-98-1

CP-346086 dihydrate

CAS : 1262769-98-1

CP-346086 dihydrate is a strong oral MTP inhibitor with 2.0 nM IC50, reducing cholesterol and triglycerides in vivo.

Formule : C₂₆H₂₆F₃N₅O₃

Couleur et forme : Solid

Masse moléculaire : 513.521

Ref: TM-T38666

CP 346086 dihydrate

CAS : 1262769-98-1

CP 346086 is a statin that inhibits the production of cholesterol by blocking the enzyme HMG-CoA reductase. It has been shown to reduce LDL cholesterol and increase HDL cholesterol levels, as well as having an effect on VLDL and triglycerides. CP 346086 also shows efficacy in reducing cardiovascular disease risk factors such as hyperlipidemias, hypertension, and diabetic nephropathy. This drug is absorbed from the intestine and is excreted unchanged in the feces. The plasma concentration of this drug increases when taken with food or other lipid-rich substances. CP 346086 may cause liver steatosis, which can lead to hepatic steatosis.

Formule : C₂₆H₂₂F₃N₅O•(H₂O)₂

Degré de pureté : Min. 97 Area-%

Couleur et forme : Powder

Masse moléculaire : 513.51 g/mol

Ref: 3D-LHA39048