CAS 1610954-97-6

N-(1-((2-(Dimethylamino)ethyl)amino)-2-methyl-1-oxopropan-2-yl)-4-(4-(2-methyl-5-(3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran -2-yl)benzyl)phenyl)butanamide

CAS : 1610954-97-6

N-(1-((2-(dimethylamino)ethyl)amino)-2-methyl-1-oxopropan-2-yl)-4-(4-(2-methyl-5-(3,4,5-trihydroxytetrahydrofuran -2-yl)benzyl)phenyl)butanamide is a peptide activator of the human ion channel TRPM8. This peptide has been shown to inhibit the binding of a ligand (AITC) to the human receptor hM3Dq and to activate TRPM8 channels in rat dorsal root ganglion neurons. It has also been shown that this peptide can modulate the activity of voltage gated sodium channels.

Formule : C₃₂H₄₇N₃O₆S

Degré de pureté : Min. 95%

Masse moléculaire : 601.8 g/mol

Ref: 3D-KPC95497

LX2761

CAS : 1610954-97-6

LX2761 is a stable inhibitor for SGLT1/2 with IC50s of 2.2/2.7 nM; it targets SGLT1 in the GI tract.

Formule : C₃₂H₄₇N₃O₆S

Degré de pureté : 98%

Couleur et forme : Solid

Masse moléculaire : 601.80

Ref: TM-T15797