CAS 183658-72-2

CYN 154806

CAS : 183658-72-2

CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).

Formule : C₅₆H₆₈N₁₂O₁₄S₂

Degré de pureté : 98%

Couleur et forme : Solid

Masse moléculaire : 1197.34

Ref: TM-TP1877

CYN 154806 trifluoroacetate

CAS : 183658-72-2

CYN 154806 is a novel anti-inflammatory drug that inhibits the vasoactive intestinal peptide receptor and has a neuroprotective effect. It also prevents the activation of microglia, which are cells of the central nervous system responsible for immune defense. CYN 154806 is membrane permeable and can inhibit the transcription-polymerase chain reaction (PCR) in mouse hippocampal tissue and human macrophages. CYN 154806 has been shown to have a low bioavailability and a short half-life, making it difficult to measure its pharmacokinetic properties in vivo. However, CYN 154806 does not appear to be toxic at high doses.

Formule : C₅₆H₆₈N₁₂O₁₄S₂•(C₂HF₃O₂)x

Degré de pureté : Min. 95%

Couleur et forme : Powder

Masse moléculaire : 1,197.34 g/mol

Ref: 3D-IHA65872