CAS 2535970-65-9

EST73502 HCl

CAS : 2535970-65-9

EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.

Formule : C₁₉H₂₇ClF₂N₂O₂

Degré de pureté : 99.96%

Couleur et forme : Solid

Masse moléculaire : 388.88

Ref: TM-T39284

EST73502 hydrochloride

CAS : 2535970-65-9

EST73502 hydrochloride is a potent and selective activator of TRPA1 ion channels. It binds to the extracellular domain of TRPA1, which is located on the cytoplasmic side of the cell membrane. EST73502 hydrochloride has been shown to modulate neuronal activity in cultured cells. This compound may be used as a research tool for studying protein interactions and for developing new drug targets. TRPA1 activation by EST73502 hydrochloride leads to an increase in intracellular calcium levels, which can lead to neuronal excitation, pain perception, and other effects.

Formule : C₁₉H₂₇ClF₂N₂O₂

Degré de pureté : Min. 95%

Masse moléculaire : 388.9 g/mol

Ref: 3D-KBE97065