CAS 2974489-09-1

BMS-818251

CAS : 2974489-09-1

BMS-818251 is a potent small-molecule inhibitor that targets HIV-1 entry, with an EC50 value of 0.019 nM. It exhibits over 10 times greater efficacy on the cross-subtype panels of the 208-HIV-1 strain compared to BMS-626529. BMS-818251 enhances potency through interactions with gp120 residues in the conserved β20-β21 hairpin.

Formule : C₂₉H₂₆N₆O₅S

Couleur et forme : Solid

Masse moléculaire : 570.619

Ref: TM-T204307