CymitQuimica logo

CAS 3068489-78-8

:

Trier par
Le filtre de pureté n’est pas visible car les produits actuels ne disposent pas de données de pureté associées pour le filtrage.
1 produits concernés.
  • AR antagonist 10
    Targetmol
    + Info

    AR antagonist 10

    CAS :
    <p>AR antagonist 10 (Compound Y5) is a potent, orally active androgen receptor (AR) antagonist with an IC50 value of 0.04 μM. It demonstrates a dual mechanism of action: antagonizing AR by disrupting AR dimerization and inducing AR degradation through the ubiquitin-proteasome pathway. This compound shows excellent activity against various resistant AR mutants and effectively inhibits the growth of LNCaP xenograft tumors. AR antagonist 10 is applicable for research in resistant prostate cancer.</p>
    Formule :C18H17ClN4O3S
    Couleur et forme :Solid
    Masse moléculaire :404.871

    Ref: TM-T205420