CAS 376641-65-5

BVT-2733 hydrochloride

CAS : 376641-65-5

BVT-2733 hydrochloride is a potent, selective, and orally active non-steroidal 11β-HSD1 inhibitor. It exhibits stronger inhibition on mouse 11β-HSD1 enzyme (IC50=96 nM) compared to the human 11β-HSD1 enzyme (IC50=3341 nM). BVT-2733 hydrochloride shows potential for research in arthritis and obesity-related diseases.

Formule : C₁₇H₂₂Cl₂N₄O₃S₂

Couleur et forme : Solid

Masse moléculaire : 465.42

Ref: TM-T203621

Bvt 2733 hydrochloride

CAS : 376641-65-5

BVT 2733 hydrochloride is a research tool that is used to inhibit ion channels. It binds to ligand-gated ion channels, such as nicotinic acetylcholine receptors and serotonin receptors, and blocks the flow of ions across cell membranes. BVT 2733 hydrochloride has been shown to be a good inhibitor of chloride channels in rat cortical neurons. This compound binds to the receptor site and prevents the binding of natural ligands, such as acetylcholine or serotonin. It also inhibits the activity of peptides that are involved in protein interactions. BVT 2733 hydrochloride may have some therapeutic potential for treating neurological disorders like Alzheimer's disease or Parkinson's disease.

Formule : C₁₇H₂₂Cl₂N₄O₃S₂

Degré de pureté : Min. 95%

Masse moléculaire : 465.4 g/mol

Ref: 3D-BQA64165