CAS 554403-08-6

SAX-187 hydrochloride

CAS : 554403-08-6

WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.

Formule : C₁₅H₁₄Cl₂N₄O₂S₂

Couleur et forme : Solid

Masse moléculaire : 417.33

Ref: TM-T69104

2-[1-[(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]-1H-indol-3-yl]ethylamine Hydrochloride

Produit contrôlé

CAS : 554403-08-6

Applications 2-[1-[(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]-1H-indol-3-yl]ethylamine Hydrochloride is the HCl salt of 2-[1-[(6-Chloroimidazo[2,1-b][1,3]thiazol-5-yl)sulfonyl]-1H-indol-3-yl]ethylamine which is a selective 5-HT6 receptor agonist. It has been proven to have antidepressant and anxiolytic effects on rats suggesting its usefulness as a potential antidepressant.
References Carr, G., et al.: Psychopharmacology, 213, 499 (2011);

Formule : C₁₅H₁₃ClN₄O₂S₂·ClH

Couleur et forme : Neat

Masse moléculaire : 417.333

Ref: TR-C368405