Inhibiteur d’enzymes
Les inhibiteurs d'enzymes sont des composés qui diminuent ou arrêtent l'activité des enzymes, en se liant à celles-ci de manière spécifique. Ces inhibiteurs jouent un rôle crucial dans la régulation des processus biologiques et sont largement utilisés dans la recherche médicale et le développement de médicaments. En bloquant l'action des enzymes, ils permettent d'étudier la fonction enzymatique et de développer des traitements contre diverses maladies. Chez CymitQuimica, nous proposons une large gamme d'inhibiteurs enzymatiques de haute qualité pour soutenir vos recherches en biologie et en pharmacologie.
123 produits trouvés pour "Inhibiteur d’enzymes"
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Benzyl Methyl Carbonate
CAS :Produit contrôlé<p>Applications Benzyl Methyl Carbonate is used in designing of inhibitors for serine and thiol proteases.<br></p>Formule :C9H10O3Couleur et forme :NeatMasse moléculaire :166.17(R)-Pinocembrin
CAS :Produit contrôlé<p>Applications (2R)-Pinocembrin is the (R)-enantiomer of Pinocembrin, a flavanoid with antioxidant activity found in damiana, honey, and propolis. (2R)-Pinocembrin is a potential inhibitor of PIM1 kinase, an oncogene that has been implicated in the development of leukemias, lymphomas, and prostate cancer.<br>References Zhao, J. et al.: J. Ethnopharmacol., 120, 387 (2008); Holder, S. et al.: Mol. Cancer Ther., 6, 163 (2007); Holder, S. et al.: Bioorg. Med. Chem., 15, 6463 (2007);<br></p>Formule :C15H12O4Couleur et forme :WhiteMasse moléculaire :256.25Teneligliptin Hydrobromide (2:5)
CAS :Produit contrôlé<p>Applications Teneligliptin Hydrobromide (2:5) is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. It is eliminated via excretion, and has a half-life of 24.2 hours in the human body.<br>References Goda, M. & Kadowaki, T.: Drugs Today, 49, 615 (2013); Kishimoto, M.: Diabetes Metab. Syndr. Obes., 6, 187 (2012)<br></p>Formule :C22H32·5Br2·5N6OSCouleur et forme :NeatMasse moléculaire :628.86Bis(2-butoxyethyl) 2-(3-Hydroxybutoxy)ethyl Phosphate Triester
CAS :Produit contrôlé<p>Applications Bis(2-butoxyethyl) 2-(3-Hydroxybutoxy)ethyl Phosphate Triester is derived from 2-Butoxyethanol (B692895), which is a reagent in the synthesis of 4-butoxyethoxy-N-octadecyl-1,8-naphthalimide as a new fluorescent probe for the determination of proteins. Also used as a reagent in the synthesis of 4-hydroxybenzaldehyde derivatives as tyrosinase inhibitors.<br>References Sun, Y., et al.: Bioorg. Med. Chem. Lett., 21, 3798 (2011); Yi, W., et al.: Eur. J. Med. Chem., 45, 639 (2010)<br></p>Formule :C18H39O8PCouleur et forme :Colourless To Light YellowMasse moléculaire :414.47Daidzein Diglucuronide
CAS :Produit contrôléFormule :C27H26O16Couleur et forme :White To Off-WhiteMasse moléculaire :606.49Nicotelline
CAS :Produit contrôlé<p>Applications Nicotelline is a Nicotine (N412420) related metabolite with potential as an inhibitor of human cytochrome P-450 2A6.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Denton, T. et al.: Biochem. Pharm., 67, 751 (2004); Gorrod, J. et al.: Anal. Det. Nic. Rel. Comp. Metab., 69, (1999);<br></p>Formule :C15H11N3Couleur et forme :NeatMasse moléculaire :233.27(3S,5S)-Atorvastatin Calcium Salt
CAS :Produit contrôlé<p>Impurity Atorvastatin Related Compound E<br>Applications Impuritiy of Atorvaststin (A791750), a selective, competitive HMG-CoA reductase inhibitor. Atorvastatin is the only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and triglycerides in patients with hypercholesterolemia. Atorvastatin Related Compound E<br>References Kearney, A.S., et al.: Pharm. Res., 10, 1461 (1993), Heinonen, T.M., et al.: Clin. Ther., 18, 853 (1996), Whitfield, L.R., et al.: Eur. J. Drug Metab. Pharmacokinet., 25, 97 (2000),<br></p>Formule :C33H34FN2O5·CaCouleur et forme :NeatMasse moléculaire :1155.34N-(2-Hydroxyethyl)-1-deoxy-L-idonojirimycin Hydrochloride
CAS :Produit contrôlé<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References van de Water, F., et al.: Drug Metab. Rev., 37, 443 (2005), Koepsell, H., et al.: Pharm. Res., 24, 1227 (2007), Jappar, D., et al.: Pharm. Res., 26, 172 (2009),<br></p>Formule :C8H18ClNO5Couleur et forme :NeatMasse moléculaire :243.69N-(2-Hydroxyethyl)-1-deoxy-L-altronojirimycin Hydrochloride Salt
CAS :Produit contrôlé<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References Jefferies, I., et al.: Bioorg. Med. Chem. Lett., 7, 1171 (1997), Hassan, A., et al.: Carbohydr. Res., 339, 1565 (2004),<br></p>Formule :C8H18ClNO5Couleur et forme :NeatMasse moléculaire :243.68523'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt (>90%)
CAS :<p>Stability Hygroscopic<br>Applications 3'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt, is a nucleotide and was proposed to be a possible inhibitor of DNA synthesis.<br>References Frederiksen, Sune.: Biochimica et Biophysica Acta, 76(3), 366-71 (1963)<br></p>Formule :C10H15N5O9P2•xC6H15NDegré de pureté :>90%Couleur et forme :NeatMasse moléculaire :411.20 + x(101.19)Naringenin chalcone
CAS :Produit contrôléFormule :C15H12O5Couleur et forme :NeatMasse moléculaire :272.25Nitromifene Citrate (E/Z mixture)
CAS :Produit contrôlé<p>Applications Nitromifene citrate is a non-steroidal estrogen antagonist. It is structurally similar to Tamoxifen (T006000) which is a selective estrogen response modifier (SERM).<br>References Rudick, C., et al.: Endorcrinol., 144, 179 (2003); Sutherland, R., et al.: Nature, 267, 434 (1977)<br></p>Formule :C33H36N2O11Couleur et forme :Yellow To OrangeMasse moléculaire :636.65LCZ696
CAS :<p>Applications LCZ696 is a novel dual-acting inhibitor of angiotensin II receptor and neprilysin, which can be used for blood pressure reduction.<br>References Ruilope, L.M.; et al.: Lancet, 375, 1255 (2010)<br></p>Formule :C24H28NO5·C24H27N5O3·3Na·x(H2O)Couleur et forme :MixtureMasse moléculaire :479.48 + (433.47) + x(18.02)2,5-Dideoxy-2,5-imino-D-mannitol
CAS :Produit contrôlé<p>Stability Hygroscopic<br>Applications A glucosidase inhibitor.<br>References Fellows, L.E.: Pestic. Sci., 17, 602 (1986)<br></p>Formule :C6H13NO4Couleur et forme :Off White SolidMasse moléculaire :163.17Vitamin B12 e-Monocarboxylic Acid
CAS :<p>Stability Hygroscopic<br>Applications Vitamin B12 Monocarboxylic Acid is an impurity of Vitamin B12 (V676005) which is a water-soluble vitamin with a key role in the normal functioning of the brain and nervous system, and for the formation of blood.<br>References Rickes, et al.: Science, 107, 396 (1948); Kirschbaum, J., et al.: Anal. Profiles Drug Subs., 10, 183 (1981); Grasbeck, R., et al.: Clin. Biochem., 17, 99 (1984)<br></p>Formule :C63H87CoN13O15PCouleur et forme :Dark Red SolidMasse moléculaire :1356.35Abamine
CAS :Produit contrôlé<p>Applications Abamine is an inhibitor of 9-Cis-Epoxycarotenoid dioxygenase (NCED), the key regulatory enzyme in the plant hormone abscisic acid (ABA) biosynthesis pathway.<br>References Kitahata, N., et al.: Bioorg. Med. Chem., 14, 5555 (2006); Han, S., et al.: Bioorg. Med. Chem. Lett., 14, 3033 (2004)<br></p>Formule :C21H24FNO4Couleur et forme :NeatMasse moléculaire :373.42tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate
CAS :Produit contrôlé<p>Applications tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate is an orally anti-diabetic agent as a inhibitors of dipeptidylpeptidase IV (DPP-4).<br>References Yoshida, T., et al.: Bioorg. Med. Chem., 20, 5705-5719 (2012);<br></p>Formule :C27H38N6O3SCouleur et forme :NeatMasse moléculaire :526.69CP-10447
CAS :<p>Applications CP-10447 is an inhibitor apolipoprotein B (apoB) and triglyceride secretion in human hepatoma cells (HepG2) by inhibiting MTP activity and stimulating the early ER degradation of apoB. It is useful tool for further study of the mechanisms of apoB secretion and triglyceride-rich lipoprotein assembly.<br>References Haghpassand, M. et al.: J. Lipid. Res., 37, 1468 (1996); Pan, M. et al.: J. Biol. chem., 275, 27399 (2000);<br></p>Formule :C16H13BrN2OCouleur et forme :NeatMasse moléculaire :329.19N-(10-Aminodecyl)-5-chloro-1-naphthalenesulfonamide Hydrochloride
CAS :Produit contrôlé<p>Applications Naphthalenesulfonamides derivatives are neoplasm inhibitors.<br>References Hidaka, H., et al.: Proc. Nat. Acad. Sci. USA, 78, 4354 (1981)<br></p>Formule :C20H29ClN2O2S·ClHCouleur et forme :NeatMasse moléculaire :433.44
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