Inhibiteur d’enzymes
Les inhibiteurs d'enzymes sont des composés qui diminuent ou arrêtent l'activité des enzymes, en se liant à celles-ci de manière spécifique. Ces inhibiteurs jouent un rôle crucial dans la régulation des processus biologiques et sont largement utilisés dans la recherche médicale et le développement de médicaments. En bloquant l'action des enzymes, ils permettent d'étudier la fonction enzymatique et de développer des traitements contre diverses maladies. Chez CymitQuimica, nous proposons une large gamme d'inhibiteurs enzymatiques de haute qualité pour soutenir vos recherches en biologie et en pharmacologie.
123 produits trouvés pour "Inhibiteur d’enzymes"
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Retorphan
CAS :Produit contrôlé<p>Applications Retorphan is a powerful and selective inhibitors of neprilysin and is being developed as a therapeutic agent. Retorphan behave as the prodrug of the enantiomers of Thiorphan (T369500).<br>References Monteil, T., et al.: Mini. Rev. Med. Chem., 2, 209 (2002); Roques, B.P., et al.: Nature, 288, 286 (1980); Tiraboschi, G., et al.: Protein Engineering, 12, 2, 141 (1999)<br></p>Formule :C21H23NO4SCouleur et forme :NeatMasse moléculaire :385.48(1R,2R)-2-Fluorocyclopentanamine Hydrochloride
CAS :Produit contrôlé<p>Applications A cyclopentanamine used in the preparation of heterocyclic and aromatic ureas and amides as CEPT inhibitors.<br></p>Formule :C5H11ClFNCouleur et forme :NeatMasse moléculaire :139.61-Deoxy-L-altronojirimycin Hydrochloride
CAS :Produit contrôlé<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References Jefferies, I., et al.: Bioorg. Med. Chem. Lett., 7, 1171 (1997), Hassan, A., et al.: Carbohydr. Res., 339, 1565 (2004),<br></p>Formule :C6H13NO4·ClHDegré de pureté :>90%Couleur et forme :NeatMasse moléculaire :199.634-Fluorobenzoic Acid-d4
CAS :Produit contrôlé<p>Applications 4-Fluorobenzoic Acid-d4 is used as a reagent in the synthesis of Flurofamide-d4 (F596687); the isotope labelled analog of Fluorofamide (F596685) which is a compound that acts as a urease inhibitor, useful in the treatment of gastritis and irregular urease activity in the urinary tract.<br>References Loes, A. et al.: Lett. App. Microbiol., 58, 31 (2014); Ohta, T.et al.: Biochem. Biophys, Res. Comm., 285, 728 (2001)<br></p>Formule :C7HD4FO2Couleur et forme :NeatMasse moléculaire :144.14tert-Butyl (3-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)cyclohex-3-en-1-yl)carbamate
CAS :Produit contrôléFormule :C17H30BNO4Couleur et forme :NeatMasse moléculaire :323.24n-Pentyl-d11 chloroformate
CAS :Produit contrôlé<p>Applications n-Pentyl-d11 chloroformate is labelled n-Pentyl chloroformate which can be used to synthesize 1,3-disubstituted ureas as potent inhibitors of the soluble epoxide hydrolase.<br>References Kim, I., et al.: J. Med. Chem., 47, 2110 (2004); Hammock, B., et al.: PCT Int. Appl. (2006), WO 2006045119 A2 20060427.<br></p>Formule :C6D11ClO2Couleur et forme :NeatMasse moléculaire :161.674-Pyridin-2,3,5,6-d4-ol-d
CAS :Produit contrôlé<p>Applications 4-Pyridin-2,3,5,6-d4-ol-d is one of the azepanone derivatives studies as CGRP receptor antagonists.<br>References Liu, J.: PCT Int. Appl. (2010), WO 2010108103 A1 20100923.<br></p>Formule :C5D5NOCouleur et forme :NeatMasse moléculaire :100.13n-Propyl-2,2,3,3,3-d5-amine Hydrochloride
CAS :Produit contrôlé<p>Applications n-Propyl-2,2,3,3,3-d5-amine Hydrochloride is the hydrochloride salt of 1-Propyl-d5-amine (P833702); the isotope labelled analog of 1-Propylamine (P833700) which is used in the synthesis of pyrimidine derivatives as novel and highly potent PDE4 inhibitors. It is also used in the preparation of fluorenone analogs with DNA topisomerase I inhibitors.<br>References Goto, T. et al.: Bioorg. Med. Chem., 21, 7025 (2013); Lee, C. et al.: Bioorg. Med. Chem. 21, 7125, (2013)<br></p>Formule :C3H5D5ClNCouleur et forme :NeatMasse moléculaire :100.6tert-Butyl 4-Bromo-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoate
CAS :Produit contrôléFormule :C18H17BrN2O3Couleur et forme :NeatMasse moléculaire :389.24GW4869 TFA Salt (~90%, ~10% inorganics)
CAS :Produit contrôlé<p>Applications GW4869 is a selective inhibitor of N-SMase.<br>References Lallemand, T., et al.: Arterioscler. Thromb. Vasc. Biol., 38, 1479 (2018); Figuera-Losada, M., et al.: PLoS One, 10, 0124481 (2015)<br></p>Formule :C30H28N6O2·xC2HF3O2Couleur et forme :NeatMasse moléculaire :504.58 + x(114.02)N-Fmoc-glycine-d2
CAS :Produit contrôlé<p>Applications Isotope labelled N-Fmoc-glycine is an N-Fmoc-protected form of Glycine (G615990). Glycine is a nonessential amino acid that acts as an inhibitory neyrotransmitter in the vertebrate central nervous system. Glycine also posesses cytoprotective against oxidant damage in the kidney.<br>References Eulenberg, V., et al.: Trend. Biochem. Sci., 30, 325 (2005); Gundersen, R., et al.: Acta Anaesth. Scand., 49, 1108 (2005); Lockart, R. & Eagle, H.: Science, 129, 252 (1959); Sogabe, K., et al.: Kidn. Int., 50, 845 (1996)<br></p>Formule :C17H13D2NO4Couleur et forme :NeatMasse moléculaire :299.32Ethyl Palmitate-d31
CAS :Produit contrôlé<p>Applications A labelled fatty acid found in Amaranth oil; it shows inhibitory activity.<br>References Fidler, N., et al.: J. Lipid Res., 41, 1376 (2000), Yang, T., et al.: Food Chem., 80, 473 (2003), Gamel, T., et al.: J. Food Lipids, 14, 323 (2007),<br></p>Formule :C18H5D31O2Couleur et forme :NeatMasse moléculaire :315.671-Propyl-d5-amine
CAS :Produit contrôlé<p>Applications 1-Propyl-d5-amine is labelled 1-Propylamine (P833700) which is used in the synthesis of pyrimidine derivatives as novel and highly potent PDE4 inhibitors. It is also used in the preparation of fluorenone analogs with DNA topisomerase I inhibitors.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Formule :C3H4D5NCouleur et forme :NeatMasse moléculaire :64.14(3R,5S,6E)-7-(2-Cyclopropyl-4-phenyl-3-quinolinyl)-3,5-dihydroxy-6-heptenoic Acid Sodium Salt
CAS :Produit contrôlé<p>Stability Hygroscopic<br>Applications (3R,5S,6E)-7-(2-cyclopropyl-4-phenyl-3-quinolinyl)-3,5-dihydroxy-6-heptenoic Acid Sodium Salt is an impurity of Pitavastatin (P531000), a HMG CoA reductase inhibitor and an antilipemic agent.<br>References Suzukim M., et al.: Bioorg. Med. Chem., 9, 2977 (1999); Yen, H., et al.: J. Clin. Invest., 98, 1253 (1996); Zou, Y., et al.: J. Biol. Chem., 274, 9760 (1999); Sun, X., et al.: Cancer Res., et al.: 61, 3382 (2001); Ladas, E.J., et al.: Clin. Oncol., 22, 517 (2004);<br></p>Formule :C25H24NNaO4Couleur et forme :NeatMasse moléculaire :425.45rac-1,2-Dioctanoyl-3-Chloropropanediol
CAS :Produit contrôlé<p>Stability Moisture Sensitive<br>Applications rac-1,2-Dioctanoyl-3-Chloropropanediol was studied for its ability to act as an inhibitor of protein kinase C.<br>References Briggs, Josie C., et al.: Carbohydrate Res., 234, 23-35 (1992)<br></p>Formule :C19H35ClO4Couleur et forme :NeatMasse moléculaire :362.93N-(n-Butyl)phosphoric Triamide
CAS :<p>Applications N-Alkyl phosphoric triamide useful as urease inhibitors.<br></p>Formule :C4H14N3OPCouleur et forme :White SolidMasse moléculaire :151.153-Amino-N-(Tertbutylbenzenesulfonamide
CAS :Produit contrôlé<p>Applications 3-Amino-N-(Tert-Butyl)Benzenesulfonamide (cas# 608523-94-0) is a useful research chemical.<br></p>Formule :C10H16N2O2SCouleur et forme :NeatMasse moléculaire :228.31(E)-a-Hydroxy Tamoxifen
CAS :Produit contrôlé<p>Applications A metabolite of the chemotherapeutic drug Tamoxifen (T006000). Exhibits a more potent estrogen agonist/antagonist activity than the parent drug. Also active as an intramembranous inhibitor of lipid peroxidation.<br>References Kupfer, D., et al.: Cancer Res., 54, 3140 (1994), Custodio, J.B.A., et al.: Biochem. Pharmacol., 47, 1989 (1994),<br></p>Formule :C26H29NO2Couleur et forme :NeatMasse moléculaire :387.51Valtrate
CAS :Produit contrôlé<p>Applications Valtrate is a Rev-transport inhibitor with anti-HIV activity from Valerianae Radix.<br>References Murakami, N., et al.: Bioorg. Med. Chem. Lett., 12, 2807 (2002); Watanabe, K., et al.: Drug Discoveries Ther., 5, 26 92011)<br></p>Formule :C22H30O8Couleur et forme :Light Brown To Dark YellowMasse moléculaire :422.47A 83-01
CAS :Produit contrôlé<p>Stability Moisture Sensitive<br>Applications A 83-01 is a selective inhibitor of TGF-β type I receptor. A 83-01 treatment increases tumor permeability.<br>References Minowa, T. et al.: British. J. Canc., 101, 1884 (2009)<br></p>Formule :C25H19N5SCouleur et forme :Off-WhiteMasse moléculaire :421.52
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