
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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Teneligliptin hydrobromide
CAS :<p>Teneligliptin hydrobromide: potent, novel DPP-4 inhibitor; inhibits human/rat plasma DPP-4 with ~1 nM IC50.</p>Formule :C22H30N6OSBrHDegré de pureté :97.83% - 99.92%Couleur et forme :SolidMasse moléculaire :628.86Aniline mustard
CAS :<p>Aniline mustard (Mesylerythrol) is alkylating mustard with anti-neoplastic activity.</p>Formule :C10H13Cl2NDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :218.129-Methoxycamptothecin
CAS :<p>9-Methoxycamptothecin (MCPT) has antitumour activities through topoisomerase inhibition.</p>Formule :C21H18N2O5Degré de pureté :98.49% - 99.56%Couleur et forme :SolidMasse moléculaire :378.38Radotinib
CAS :<p>Radotinib (IY-5511), and sometimes referred to by its investigational name IY5511, is a drug for the treatment of different types of Y, most notably</p>Formule :C27H21F3N8ODegré de pureté :99.13% - 99.97%Couleur et forme :SolidMasse moléculaire :530.5NSC 73150
CAS :<p>6-Methyl-1H-pyrimidin-4-one (NSC 73150) shows antitumor effects, impeding growth in breast, lung, liver cancer, and inducing apoptosis.</p>Formule :C12H12N4O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :244.25Ispinesib
CAS :<p>Ispinesib (SB-715992), a selective, effectvie and reversible inhibitor of kinesin spindle protein (KSP), is derived from quinazolinone, with antineoplastic</p>Formule :C30H33ClN4O2Degré de pureté :98% - 99.09%Couleur et forme :SolidMasse moléculaire :517.064E1rcat
CAS :<p>4E1RCat is a dual inhibitor of eIF4E:eIF4 g and eIF4E:4E-BP1 interaction. And it inhibits the binding of eIF4 g to eIF4E with IC50 of 3.2 μM.</p>Formule :C28H18N2O6Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :478.45pimpinellin
CAS :<p>Pimpinellin is a natural product that acts as antagonist of proteins with GABA receptor activity.</p>Formule :C13H10O5Degré de pureté :99.85% - ≥95%Couleur et forme :SolidMasse moléculaire :246.22β-Lapachone
CAS :<p>β-Lapachone (ARQ-501) is a specific DNA topoisomerase I inhibitor, and no inhibitory activities against DNA topoisomerase II or ligase.</p>Formule :C15H14O3Degré de pureté :99.76% - 99.88%Couleur et forme :SolidMasse moléculaire :242.27MX69
CAS :<p>MX69 is the MDM2/XIAP inhibitor, blocking the MDM2 protein-XIAP RNA interaction, leading to MDM2 degradation.</p>Formule :C27H26N2O4SDegré de pureté :97.27% - 99.57%Couleur et forme :SolidMasse moléculaire :474.57Isatin
CAS :<p>Isatin (2,3-Indolinedione) is an endogenous MAO inhibitor.</p>Formule :C8H5NO2Degré de pureté :98.92%Couleur et forme :Yellow To Reddish Crystalline SolidMasse moléculaire :147.13BDA-366
CAS :<p>BDA-366, a potent Bcl2 antagonist, selectively binds the Bcl2-BH4 domain with high affinity (Ki = 3.3 nM), inducing a conformational change that nullifies its</p>Formule :C24H29N3O4Degré de pureté :98.61%Couleur et forme :SoildMasse moléculaire :423.53BDO
CAS :<p>3BDO is a new mTOR activator. 3BDO inhibits autophagy.</p>Formule :C18H17NO5Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :327.33Sodium dichloroacetate
CAS :<p>Sodium dichloroacetate (BCA) inhibits PDK (IC50: 183 μM PDK2, 80 μM PDK4), triggers cancer cell apoptosis, and impedes tumor growth.</p>Formule :C2HCl2NaO2Degré de pureté :99.32% - 99.87%Couleur et forme :White PowderMasse moléculaire :150.92AES-350
CAS :<p>AES-350, an HDAC6 inhibitor (IC50: 0.0244 μM), also targets HDAC-3, -8, -11, induces AML cell apoptosis, and aids AML research.</p>Formule :C18H20N2O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :312.36N-Formyl-Met-Leu-Phe
CAS :<p>N-Formyl-Met-Leu-Phe (N-Formyl-MLF) (fMLF) is a synthetic peptide that acts as an agonist at formyl peptide receptors (FPR; Ki = 0.8 pM).</p>Formule :C21H31N3O5SDegré de pureté :98.69% - ≥95%Couleur et forme :SolidMasse moléculaire :437.55Rotundic acid
CAS :<p>Rotundic acid fights various cancers: HepG2, A375, NCI-H446, MCF-7, and HT-29.</p>Formule :C30H48O5Degré de pureté :96.91% - 99.97%Couleur et forme :SolidMasse moléculaire :488.7Isobavachalcone
CAS :<p>Isobavachalcone (Corylifolinin) is a chalcone constituent of Angelica keiskei, has potent anti-inflammatory activity, possible can ameliorate neuronal injury in</p>Formule :C20H20O4Degré de pureté :98% - 99.76%Couleur et forme :SolidMasse moléculaire :324.37Palmatine chloride
CAS :<p>Palmatine chloride an isoquinoline alkaloid, is an important medicinal herbal extract with diverse pharmacological and biological properties.</p>Formule :C21H22ClNO4Degré de pureté :97.9% - 99.47%Couleur et forme :SolidMasse moléculaire :387.857Bortezomib
CAS :<p>Bortezomib (LDP 341) is a 20S proteasome inhibitor (Ki=0.6 nM) that is reversible and selective.</p>Formule :C19H25BN4O4Degré de pureté :97.79% - >99.99%Couleur et forme :Yellow SolidMasse moléculaire :384.24IACS-010759
CAS :<p>IACS-010759 is an orally bioavailable inhibitor of complex I of oxidative phosphorylation of the mitochondrial electron transport chain.</p>Formule :C25H25F3N6O4SDegré de pureté :99.54% - 99.73%Couleur et forme :SolidMasse moléculaire :562.56Ketorolac
CAS :<p>Ketorolac (Acuvail) is an NSAID that blocks prostaglandin synthesis, related to heterocyclic acetic acids.</p>Formule :C15H13NO3Degré de pureté :99.68%Couleur et forme :White Crystalline Or White PowderMasse moléculaire :255.27TPCA-1
CAS :<p>TPCA-1 (TPCA1) is an effective and specific IKK-2 inhibitor (IC50: 17.9 nM); shows >22-fold selectivity over IKK-1 and >550-fold selectivity over others kinases</p>Formule :C12H10FN3O2SDegré de pureté :95.03% - 97.86%Couleur et forme :SolidMasse moléculaire :279.29ML162
CAS :<p>ML162 is a covalent glutathione peroxidase 4 (GPX4) inhibitor that induces ferroptosis. ML162 has antitumor activity. Cost-effective and quality-assured.</p>Formule :C23H22Cl2N2O3SDegré de pureté :98.42% - 99.55%Couleur et forme :SolidMasse moléculaire :477.4Poziotinib
CAS :<p>Poziotinib (NOV120101)(NOV120101; HM781-36B) is an irreversible HER1/2/4 inhibitor (IC50s: 3/5/23 nM).</p>Formule :C23H21Cl2FN4O3Degré de pureté :98.69% - 99.78%Couleur et forme :SolidMasse moléculaire :491.34BG45
CAS :<p>BG45 is an HDAC I type inhibitor with IC50 of 289 nM, 2.0 μM, 2.2 μM and >20 μM for HDAC3/1/2/6 in cell-free assays, respectively.</p>Formule :C11H10N4ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :214.22INCB-057643
CAS :<p>INCB057643 is a potent, selective and orally bioavailable BET inhibitor.</p>Formule :C20H21N3O5SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :415.46Thapsigargin
CAS :<p>Thapsigargin is a natural product, an inhibitor of sarcoplasmic/endoplasmic reticulum Ca2+ ATPase (SERCA) and an endoplasmic reticulum stress inducer.</p>Formule :C34H50O12Degré de pureté :99.07% - 99.3%Couleur et forme :Colourless FilmMasse moléculaire :650.75PS-1145
CAS :<p>PS-1145 (IKK Inhibitor X) is a specific IKK inhibitor with IC50 of 88 nM.</p>Formule :C17H11ClN4ODegré de pureté :98.81% - >99.99%Couleur et forme :SolidMasse moléculaire :322.75RAF265
CAS :<p>RAF265 (CHIR-265) inhibits C-Raf/B-Raf/V600E (IC50: 3-60 nM), blocks VEGFR2 (EC50: 30 nM), in Phase 2 trials.</p>Formule :C24H16F6N6ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :518.41LASSBio-1135
CAS :<p>LASSBio-1135 is an orally effective antagonist of TRPV1 and inhibitor of TNF-α production.</p>Formule :C18H14N4Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :286.33Epieriocalyxin A
CAS :<p>Epieriocalyxin A can suppress Caco-2 colon cancer cell growth. It could be a potential drug for colon cancer therapy in the future.</p>Formule :C20H24O5Degré de pureté :97.00%Couleur et forme :SolidMasse moléculaire :344.4Eprenetapopt
CAS :<p>Eprenetapopt (PRIMA-1Met) restores wild-type conformation and function to mutant p53, and triggers apoptosis in tumor cells.</p>Formule :C10H17NO3Degré de pureté :98.75% - 99.57%Couleur et forme :SolidMasse moléculaire :199.25Tandutinib
CAS :<p>Tandutinib (CT53518) (MLN518, CT53518), an effective FLT3 antagonist (IC50: 0.22 μM), can also inhibit c-Kit and PDGFR, 15-20 fold higher potency for FLT3</p>Formule :C31H42N6O4Degré de pureté :99.45% - ≥98%Couleur et forme :White SolidMasse moléculaire :562.7Quinidine sulfate dihydrate
CAS :<p>Quinidine sulfate dihydrate (Pitayine Sodium) is a potent and selective cytochrome P450db inhibitor</p>Formule :C40H54N4O10SDegré de pureté :99.85%Couleur et forme :White To Light Yellow Crystal PowdeMasse moléculaire :782.9Paederosidic acid
CAS :<p>Paederosidic acid shows anti-tumor, anticonvulsant, and sedative properties, may treat epilepsy by modulating brain GABA and glutamate levels.</p>Formule :C18H24O12SDegré de pureté :98% - 99.56%Couleur et forme :SolidMasse moléculaire :464.44DMU-212
CAS :<p>DMU-212, a Resveratrol derivative, has antimitotic, antiproliferative, antioxidant properties; induces apoptosis via ERK1/2.</p>Formule :C18H20O4Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :300.35(Rac)-Idroxioleic acid
CAS :<p>(Rac)-Idroxioleic acid (2-Hydroxyoleic acid) is a fatty acid amide hydrolase inhibitor with anti-tumor effect.</p>Formule :C18H34O3Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :298.46K-Ras(G12C) inhibitor 12
CAS :<p>K-Ras(G12C) inhibitor 12 is an allosteric inhibitor of oncogenic K-Ras(G12C).</p>Formule :C15H17ClIN3O3Degré de pureté :97.16%Couleur et forme :SolidMasse moléculaire :449.67LY-411575
CAS :<p>LY-411575, a potent γ-secretase inhibitor, is with IC50 of 0.078 nM in the membrane and 0.082 nM in cell-based. It also suppresses Notch clevage.</p>Formule :C26H23F2N3O4Degré de pureté :97.03% - 99.38%Couleur et forme :SolidMasse moléculaire :479.48Mycophenolate Mofetil
CAS :<p>Mycophenolate Mofetil (TM-MMF), is an immunosuppressive agent, 2-morpholinoethyl ester of MPA, and an inhibitor of inosine monophosphate dehydrogenase (IMPDH).</p>Formule :C23H31NO7Degré de pureté :98.27% - 99.85%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :433.49Carfilzomib
CAS :<p>Carfilzomib (PR-171) is a proteasome inhibitor that irreversibly binds to the chymotrypsin of the 20S proteasome.</p>Formule :C40H57N5O7Degré de pureté :99.6% - 99.84%Couleur et forme :SolidMasse moléculaire :719.91TW-37
CAS :<p>TW-37 is an nonpeptide inhibitor to recombinant Bcl-2, Bcl-xL and Mcl-1 (Ki: 0.29/1.11/0.26 μM).</p>Formule :C33H35NO6SDegré de pureté :97.06% - ≥95%Couleur et forme :SolidMasse moléculaire :573.7Eltrombopag
CAS :<p>Eltrombopag (SB-497115-GR), an orally active thrombopoietin receptor agonist with megakaryopoiesis stimulating activity, binds to and stimulates the platelet</p>Formule :C25H22N4O4Degré de pureté :99.27%Couleur et forme :Orange To Red SolidMasse moléculaire :442.47Valproic Acid
CAS :<p>Valproic Acid (2-Propylpentanoic Acid) is a branched chain fatty acid which potentially enhances central GABAergic neurotransmission and inhibits Na+ channels.</p>Formule :C8H16O2Degré de pureté :97.78% - 99%Couleur et forme :Colourless To Pale Yellow Liquid ViscousMasse moléculaire :144.21Brassinolide
CAS :<p>Brassinolide (Brassin lactone) is a plant hormone isolated from rapeseed (Brassica napus) promoting stem elongation and cell division.</p>Formule :C28H48O6Degré de pureté :98% - 99.189%Couleur et forme :Off-White SolidMasse moléculaire :480.68TCS7010
CAS :<p>TCS7010 (Aurora A Inhibitor I) is a novel, potent, and selective inhibitor of Aurora A with IC50 of 3.4 nM in a cell-free assay.</p>Formule :C31H31ClFN7O2Degré de pureté :98.49% - 99.62%Couleur et forme :SolidMasse moléculaire :588.07SB 202190
CAS :<p>SB 202190 (FHPI) is a p38 MAPK inhibitor that inhibits p38α and p38β2 (IC50=50/100 nM) selectively and cell-permeably.</p>Formule :C20H14FN3ODegré de pureté :98% - 99.84%Couleur et forme :Pale YellowMasse moléculaire :331.34Rosmarinic acid
CAS :<p>Rosmarinic acid (Labiatenic acid) is widely found in plants and has antioxidant, anti-inflammatory, and antibacterial activities.</p>Formule :C18H16O8Degré de pureté :98.88% - 99.73%Couleur et forme :Brown Fine PowderMasse moléculaire :360.31SRS11-92
CAS :<p>SRS11-92 (AA9) is a ferroptosis inhibitor and a derivative of ferrostatin-1</p>Formule :C22H28N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :352.47Millepachine
CAS :<p>Millepachine is a natural product found in the Chinese herbal medicine with strong antitumor effects against numerous human cancer cells.</p>Formule :C22H22O4Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :350.41Vanillyl Alcohol
CAS :<p>Vanillyl Alcohol (3-Methoxy-4-hydroxybenzyl alcohol) possesses anti-angiogenic, anticonvulsive, anti-inflammatory, anti-oxidant and anti-nociceptive activities.</p>Formule :C8H10O3Degré de pureté :97.02% - 98.42%Couleur et forme :Crystalline White To Off-White PowderMasse moléculaire :154.16Pyrogallol
CAS :<p>Pyrogallol (Piral) is a white crystalline powder and a powerful reducing agent prepared by heating gallic acid.</p>Formule :C6H6O3Degré de pureté :99.88%Couleur et forme :SoildMasse moléculaire :126.11Ixabepilone
CAS :<p>Ixabepilone (Azaepothilone B) is an orally bioavailable microtubule inhibitor.</p>Formule :C27H42N2O5SDegré de pureté :98% - 99.50%Couleur et forme :SolidMasse moléculaire :506.7Taurolidine
CAS :<p>Taurolidine is a synthetic taurine analog with antimicrobial and anti-neoplastic actions. It displays broad bactericidal and fungicidal activity.</p>Formule :C7H16N4O4S2Degré de pureté :99.79% - 99.81%Couleur et forme :SolidMasse moléculaire :284.36Rimiducid
CAS :<p>Rimiducid, a tacrolimus analogue, dimerizes FKBP domains to activate Caspase 9 and induce apoptosis; binds FKBP12 weakly.</p>Formule :C78H98N4O20Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :1411.63CCCP
CAS :<p>CCCP blocks STING activation, TBK1, IRF3 signaling, and IFN-β production by disrupting MMP.</p>Formule :C9H5ClN4Degré de pureté :97.15% - 99.64%Couleur et forme :Yellow To Orange PowderMasse moléculaire :204.62Eriocitrin
CAS :<p>Eriocitrin: an antioxidative flavonoid; reduces exercise-induced oxidative damage and lipids; fights fatty liver and inhibits carbonic anhydrase VA.</p>Formule :C27H32O15Degré de pureté :98.41% - 99.11%Couleur et forme :SolidMasse moléculaire :596.53Mirodenafil dihydrochloride
CAS :<p>Mirodenafil dihydrochloride is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>Formule :C26H39Cl2N5O5SDegré de pureté :99.64% - 99.78%Couleur et forme :SolidMasse moléculaire :604.59Sinomenine
CAS :<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Formule :C19H23NO4Degré de pureté :99.02% - 99.73%Couleur et forme :White PowderMasse moléculaire :329.39Tacedinaline
CAS :<p>Tacedinaline (CI994) is a selective class I HDAC inhibitor with potential antineoplastic activity.</p>Formule :C15H15N3O2Degré de pureté :96.83% - 99.15%Couleur et forme :WhiteMasse moléculaire :269.3W-7 hydrochloride
CAS :<p>W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochloride</p>Formule :C16H22Cl2N2O2SDegré de pureté :99.63%Couleur et forme :White Crystalline SolidMasse moléculaire :377.32ISOGINKGETIN
CAS :<p>ISOGINKGETIN (4',4'''-Dimethylamentoflavone), a compound derived from the leaves of Ginkgo biloba, to up-regulate adiponectin secretion.</p>Formule :C32H22O10Degré de pureté :98% - 99.72%Couleur et forme :SolidMasse moléculaire :566.51Cysteamine hydrochloride
CAS :<p>Cysteamine hydrochloride (Thioethanolamine Hydrochloride) is an agent for the treatment of nephropathic cystinosis and an antioxidant.</p>Formule :C2H7NS·HClDegré de pureté :99.34% - 99.87%Couleur et forme :White Crystalline Powder With A Strong And Disagreeable SmellMasse moléculaire :113.61SCR130
CAS :<p>SCR130 (1,7,9-Triazaspiro[4.5]dec-1-ene-6,10-dione, 2,4-bis(4-chlorophenyl)-8-thioxo-) 是基于 SCR7 的 DNA 非同源末端连接抑制剂,可诱导细胞凋亡并,具有抗癌活性。 它特异性依赖连接酶 IV,抑制 DNA 的末端连接。</p>Formule :C19H13Cl2N3O2SDegré de pureté :98.9%Couleur et forme :SolidMasse moléculaire :418.3Otenaproxesul
CAS :<p>Otenaproxesul (ATB 346) is a novel hydrogen sulphide-releasing derivative of naproxen with markedly reduced toxicity.</p>Formule :C21H19NO3SDegré de pureté :98.76% - 99.13%Couleur et forme :SolidMasse moléculaire :365.45Flavokawain A
CAS :<p>NSC-37445 shows anti-tumor properties; Flavokawain A may reduce inflammation by hindering specific signaling in macrophages.</p>Formule :C18H18O5Degré de pureté :97.1% - 99.72%Couleur et forme :SolidMasse moléculaire :314.332Nivolumab
CAS :<p>Nivolumab is a monoclonal antibody, a humanized IgG4 antibody to PD-1. Nivolumab has antitumor activity. Cost-effective and quality-assured.</p>Degré de pureté :98% - 98%Couleur et forme :LiquidMasse moléculaire :146 kDaGanoderic acid D
CAS :<p>Ganoderic acid D, a Ganoderma component, inhibits HeLa cell growth with an IC50 of 17.3µM after 48h.</p>Formule :C30H42O7Degré de pureté :98.06% - 99.98%Couleur et forme :SolidMasse moléculaire :514.65EGFR-IN-12
CAS :<p>EGFR-IN-12 (EGFR Inhibitor) is a cell permeable and selective inhibitor of EGFR kinase (IC50: 21 nM) and blocks receptor autophosphorylation in cells.</p>Formule :C21H18F3N5ODegré de pureté :98.3% - 99.76%Couleur et forme :SolidMasse moléculaire :413.4IITZ-01
CAS :<p>IITZ-01 is potent autophagy inhibitor with single-agent anticancer activity ( IC50 of 2.62 μM for PI3Kγ.)</p>Formule :C26H23FN8ODegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :482.513-Nitropropanoic acid
CAS :<p>3-Nitropropanoic acid (Bovinocidin) is an irreversible inhibitor of succinate dehydrogenase.</p>Formule :C3H5NO4Degré de pureté :98.35% - 99.94%Couleur et forme :Crystals From Chloroform Physical Description Golden Crystals (From Chloroform) (Ntp 1992)Masse moléculaire :119.08CCG-1423
CAS :<p>CCG-1423, a selective RhoA pathway inhibitor, suppresses SRF-mediated transcription.</p>Formule :C18H13ClF6N2O3Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :454.75TM5441
CAS :<p>TM5441 is an orally bioavailable fibrinogen activator inhibitor-1 inhibitor that inhibits several cancer cell lines with IC50 values ranging from 13.9 to 51.1 μM.Cost-effective and quality-assured.Cost-effective and quality-assured.</p>Formule :C21H17ClN2O6Degré de pureté :97.62% - 99.09%Couleur et forme :SolidMasse moléculaire :428.82BTdCPU
CAS :<p>BTdCPU is a potent activator of heme-regulated eIF2α kinase (HRI) . BTdCPU promotes eIF2α phosphorylation and induced apoptosis in resistant cell.</p>Formule :C13H8Cl2N4OSDegré de pureté :98.94% - 99.59%Couleur et forme :SolidMasse moléculaire :339.2Demethylzeylasteral
CAS :<p>Demethylzeylasteral (T-96), isolated from Tripterygium wilfordii, has anti-inflammatory, immunosuppressive and anti-tumor activities.</p>Formule :C29H36O6Degré de pureté :98.74% - 99.82%Couleur et forme :SolidMasse moléculaire :480.59Mancozeb
CAS :<p>Mancozeb is a fungicide of ethylene-bis-dithiocarbamate.</p>Formule :C8H12MnN4S8ZnDegré de pureté :98%Couleur et forme :Grayish-Yellow PowderMasse moléculaire :541.08EF24
CAS :<p>EF24 treatment boosts caspase 3/9 activity, hinders MEK1/ERK phosphorylation, and exhibits strong anti-tumor effects in OSCC by deactivating MAPK/ERK.</p>Formule :C19H15F2NODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :311.33Deferitrin
CAS :<p>Deferitrin (GT-56-252) is an iron chelator. It potentially for the treatment of thalassemia and iron overload.</p>Formule :C11H11NO4SDegré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :253.27Simazine
CAS :<p>Simazine (Tafazine), a chlorotriazine herbicide/pesticide, may cause reproductive harm, endocrine disruption, and cancer.</p>Formule :C7H12ClN5Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :201.66TASIN-1
CAS :<p>TASIN-1 is a small molecule inhibitor of mutant adenomatous polyposis coli (APC).</p>Formule :C18H28N2O3SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :352.49NUN82647
CAS :<p>NUN82647 (CU-242) is an Inhibitor of cell cycle at G2 phase, and apoptosis inducer.</p>Formule :C15H13N3O2SDegré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :299.35Z-VAD(OMe)-FMK
CAS :<p>View and buy Z-VAD(OMe)-FMK from TargetMol.Z-VAD(OMe)-FMK is a cell-permeable and irreversible pan-caspase inhibitor.Cited in 10 publications.</p>Formule :C22H30FN3O7Degré de pureté :95.92% - 99.71%Couleur et forme :SolidMasse moléculaire :467.49Glafenine Hydrochloride
CAS :<p>Glafenine Hydrochloride is an anti-inflammatory agent.</p>Formule :C19H17ClN2O4·HClDegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :409.26Pevonedistat
CAS :<p>Pevonedistat (MLN4924) is a potent and selective NEDD8 activating enzyme (NAE) inhibitor (IC50=4.7 nM).</p>Formule :C21H25N5O4SDegré de pureté :95% - 99.92%Couleur et forme :SolidMasse moléculaire :443.52TASIN-1 Hydrochloride
CAS :<p>TASIN-1 Hydrochloride (TASIN-1 HCl) is a selective inhibitor of truncated APC that acts by selectively killing colorectal cancer cells that express truncated</p>Formule :C18H29ClN2O3SDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :388.95Paroxetine
CAS :<p>Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression.</p>Formule :C19H20FNO3Degré de pureté :98.89% - 99.45%Couleur et forme :White To Off-White PowderMasse moléculaire :329.37Romidepsin
CAS :<p>Romidepsin (NSC-630176), an IV histone deacetylase inhibitor, treats refractory cutaneous/peripheral T-cell lymphomas.</p>Formule :C24H36N4O6S2Degré de pureté :99.4% - 99.94%Couleur et forme :SolidMasse moléculaire :540.7TPCK
CAS :<p>TPCK is an irreversible inhibitor of chymotrypsin-like proteases that affect cell proliferation, apoptosis, and tumorigenesis</p>Formule :C17H18ClNO3SDegré de pureté :97.33%Couleur et forme :PowderMasse moléculaire :351.85PX-12
CAS :<p>PX-12, a Trx-1 inhibitor, promotes apoptosis, reduces HIF-1α/VEGF, and inhibits tumor growth, suggesting use in advanced cancer therapy.</p>Formule :C7H12N2S2Degré de pureté :98% - 99.21%Couleur et forme :SolidMasse moléculaire :188.31L524-0366
CAS :<p>L524-0366 ([1-(3-chlorophenyl)triazol-4-yl]-thiomorpholino-methanone) is a TWEAK-Fn14 signaling cascade inhibitor.</p>Formule :C13H13ClN4OSDegré de pureté :98.6% - 99.13%Couleur et forme :SolidMasse moléculaire :308.79Saquinavir
CAS :<p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>Formule :C38H50N6O5Degré de pureté :99.50% - >99.99%Couleur et forme :SolidMasse moléculaire :670.84Tenilsetam
CAS :<p>Tenilsetam: an endonuclease, nootropic, AGE inhibitor potential for Alzheimer's.</p>Formule :C8H10N2OSDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :182.244-IBP
CAS :<p>4-IBP is a selective σ1 agonist with a high level of affinity for the σ1 receptor (Ki = 1.7 nM) and a moderate affinity for the σ2 receptor (Ki = 25.2 nM) .</p>Formule :C19H21IN2ODegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :420.29Lubiprostone
CAS :<p>Lubiprostone (RU-0211), an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.</p>Formule :C20H32F2O5Degré de pureté :97.31% - 98.54%Couleur et forme :White Odorless Crystals Or Crystalline PowderMasse moléculaire :390.46RH01687
CAS :<p>RH01687 is a potent β-cell protector , exhibits β-cell-protective activities against endoplasmic reticulum (ER) stress.</p>Formule :C12H9ClN6O2SDegré de pureté :97.93%Couleur et forme :SolidMasse moléculaire :336.76Clodronic acid disodium salt
CAS :<p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>Formule :CH4Cl2O6P0·2NaDegré de pureté :>99.99% - ≥98%Couleur et forme :White SolidMasse moléculaire :288.86Sodium benzoate
CAS :<p>Sodium benzoate (Benzoic acid sodium salt) is a D-Amino Acid Oxidase Inhibitor.Sodium Benzoate is a Food Preservative.</p>Formule :C7H5NaO2Degré de pureté :99.72%Couleur et forme :White Solid CrystallineMasse moléculaire :144.10HX 531
CAS :<p>HX 531 is a RXR antagonist (IC50 of 18 nM).Cost-effective and quality-assured.</p>Formule :C29H29N3O4Degré de pureté :98.59% - 99.86%Couleur et forme :SolidMasse moléculaire :483.56Dantrolene sodium hemiheptahydrate
CAS :<p>Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium</p>Formule :C14H9N4NaO5·5H2ODegré de pureté :99.72%Couleur et forme :Orange PowderMasse moléculaire :399.29
