
Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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BMS202 hydrochloride (1675203-84-5(free base))
CAS :<p>BMS202 hydrochloride (1675203-84-5) is a potent PD-1/PD-L1 inhibitor (IC50: 18 nM) that promotes PD-L1 dimerization, blocking PD1 binding.</p>Formule :C25H30ClN3O3Degré de pureté :98.29% - 99.47%Couleur et forme :SolidMasse moléculaire :455.97Hexamethylene bisacetamide
CAS :<p>Hexamethylene bisacetamide inhibits BET Bromodomain Proteins.</p>Formule :C10H20N2O2Degré de pureté :99.94%Couleur et forme :White FlakesMasse moléculaire :200.28PDL-1 cpd 10
CAS :<p>PDL-1 cpd 10 is a novel small molecule PD-L1 inhititor.</p>Formule :C21H23N5O2Degré de pureté :97.08%Couleur et forme :SolidMasse moléculaire :377.44Piperacetazine
CAS :<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57(E/Z)-Necrosulfonamide
CAS :<p>(E/Z)-Necrosulfonamide is a novel inhibitor of MLKL.</p>Formule :C18H15N5O6S2Degré de pureté :97.62% - 98%Couleur et forme :SolidMasse moléculaire :461.47Z-VAD-FMK
CAS :<p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>Formule :C21H28FN3O7Degré de pureté :98.24% - 99.79%Couleur et forme :SolidMasse moléculaire :453.46Sinapinic Acid
CAS :<p>Sinapinic Acid (Synapoic acid) is a phenolic isolated from the roots of Hydnophytum formicarumJack. It is an HDAC inhibitor and also inhibits ACE-I activity.</p>Formule :C11H12O5Degré de pureté :99.88% - >99.99%Couleur et forme :SolidMasse moléculaire :224.21Tyrphostin AG1296
CAS :<p>Tyrphostin AG1296 (Tyrphostin AG 1296) is an inhibitor of PDGFR with IC50 of 0.3-0.5 μM, no activity to EGFR.</p>Formule :C16H14N2O2Degré de pureté :99.94% - >99.99%Couleur et forme :SolidMasse moléculaire :266.29Rhapontin
CAS :<p>Rhapontin may reduce liver fat and better blood sugar/lipids, showing potential for treating type 2 diabetes.</p>Formule :C21H24O9Degré de pureté :99% - 99.91%Couleur et forme :Light YellowMasse moléculaire :420.41Perillyl alcohol
CAS :<p>Perillyl Alcohol, a monoterpene with antitumor properties, inhibits protein activation blocking cancer cell growth.</p>Formule :C10H16ODegré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :152.23Licochalcone B
CAS :<p>Licochalcone B inhibits human bladder cancer cells, reduces inflammation by NO, TNFalpha, and MCP-1, and a derivative protects against endotoxin shock.</p>Formule :C16H14O5Degré de pureté :99.33% - 99.93%Couleur et forme :SolidMasse moléculaire :286.28Pitstop 2
CAS :<p>Pitstop2 is an amphipathic protein-bound inhibitor of the clathrin terminal domain. Pitstop2 has antitumor activity. Cost-effective, quality assurance.</p>Formule :C20H13BrN2O3S2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :473.36ZM 336372
CAS :<p>ZM 336372 is a potent and selective c-Raf inhibitor.</p>Formule :C23H23N3O3Degré de pureté :97.24% - 97.51%Couleur et forme :SolidMasse moléculaire :389.45Avelumab
CAS :<p>Avelumab is a fully human IgG1 anti-PD-L1 monoclonal antibody. Avelumab shows potential antibody-dependent cell-mediated cytotoxicity.</p>Degré de pureté :95% - 97.17% (SDS-PAGE)Couleur et forme :LiquidMasse moléculaire :143.8 kDaEvofosfamide
CAS :<p>Evofosfamide (TH-302) is a hypoxia-activated prodrug that releases Br-IPM in tumors to cause DNA damage and potentially induce apoptosis.</p>Formule :C9H16Br2N5O4PDegré de pureté :98.74% - 99.75%Couleur et forme :SolidMasse moléculaire :449.04Buparlisib
CAS :<p>Buparlisib (BKM120) is an orally bioavailable specific oral inhibitor of the pan-class I PI3K (IC50s: 52/166/116/nM for p110α, p110β, and p110δ).</p>Formule :C18H21F3N6O2Degré de pureté :95.32% - 98.45%Couleur et forme :SolidMasse moléculaire :410.39NS-1619
CAS :<p>NS1619 have cardio-protective effects after ischemia-reperfusion injury.</p>Formule :C15H8F6N2O2Degré de pureté :97.66% - 98%Couleur et forme :SolidMasse moléculaire :362.23SSE15206
CAS :<p>SSE15206 is a microtubule polymerization inhibitor that overcomes multidrug resistance.</p>Formule :C19H21N3O3SDegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :371.45Niraparib tosylate
CAS :<p>Niraparib tosylate (MK-4827 (tosylate))(with IC50 of 3.8 nM/2.1 nM) is a selective PARP1/PARP2 inhibitor.</p>Formule :C19H20N4O·C7H8O3SDegré de pureté :99.34% - 99.87%Couleur et forme :SolidMasse moléculaire :492.59Tenovin-1
CAS :<p>Tenovin-1 inhibits protein-deacetylating activities of SirT1 and SirT2 and protects against MDM2-mediated p53 degradation, which involves ubiquitination.</p>Formule :C20H23N3O2SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :369.48SBI-0206965
CAS :<p>SBI-0206965 is a potent, selective and cell-permeable autophagy kinase ULK1 inhibitor with IC50 of 108 nM for ULK1 kinase activity and 711 nM for ULK2.</p>Formule :C21H21BrN4O5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :489.32Iberdomide
CAS :<p>Iberdomide (CC-220) is a modulator of cereblon( IC50 value of 60 nM in a competitive TR-FRET assay).</p>Formule :C25H27N3O5Degré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :449.5AZD1208
CAS :<p>AZD1208 is a novel, orally bioavailable, highly selective PIM kinase inhibitor with single nanomolar potency against all three PIM kinases.</p>Formule :C21H21N3O2SDegré de pureté :97.24% - 99.83%Couleur et forme :SolidMasse moléculaire :379.48Niraparib hydrochloride
CAS :<p>Niraparib hydrochloride (MK-4827) is a PARP inhibitor with potential cancer treatment effects, causing DNA damage and apoptosis.</p>Formule :C19H21ClN4ODegré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :356.85Propylparaben
CAS :<p>Propylparaben (Propyl parahydroxybenzoate) is an antimicrobial agent, preservative, flavouring agent</p>Formule :C10H12O3Degré de pureté :99.84%Couleur et forme :White Solid CrystallineMasse moléculaire :180.20Navitoclax
CAS :<p>View and buy Navitoclax from TargetMol.Navitoclax (ABT-263) is a potent, orally bioavailable Bcl-2 family protein inhibitor that avidly binds Bcl-2.Cited in 4 publications.</p>Formule :C47H55ClF3N5O6S3Degré de pureté :95.82% - >99.99%Couleur et forme :Pale Yellow SolidMasse moléculaire :974.61Dihydrokaempferol
CAS :<p>Dihydrokaempferol (Aromadendrin) is a natural product. It induces apoptosis and inhibits Bcl-2 and Bcl-xL expression, possesses anti-inflammatory activity.</p>Formule :C15H12O6Degré de pureté :97.79% - 99.96%Couleur et forme :SolidMasse moléculaire :288.25Necrostatin-1
CAS :<p>Necrostatin-1 (Nec-1) is a necrotic apoptosis inhibitor and RIP1 inhibitor with specificity.</p>Formule :C13H13N3OSDegré de pureté :99.25% - >99.99%Couleur et forme :SolidMasse moléculaire :259.33SC-236
CAS :<p>SC-236 (Sc 236) is an orally active and selective inhibitor of COX-2 (IC50 of 0.005 μM and 17.8 μM for COX-2 and COX-1, respectively).</p>Formule :C16H11ClF3N3O2SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :401.79Fulvestrant
CAS :<p>Fulvestrant (ZM 182780) is an estrogen receptor (ER) antagonist (IC50=9.4 nM) and an agonist of GPR30.</p>Formule :C32H47F5O3SDegré de pureté :99.1% - >99.99%Couleur et forme :White PowderMasse moléculaire :606.77Quercetin
CAS :<p>Quercetin (Sophoretin) is a natural flavonoid and is an agonist of SIRT1.</p>Formule :C15H10O7Degré de pureté :96.29% - 98.05%Couleur et forme :Sensitive To Exposure To Air And Light Insoluble In Water Alcoholic Solutions Taste Very Bitter (Ntp 1992)Masse moléculaire :302.24SecinH3
CAS :<p>SecinH3 is selective cytohesin inhibitor.</p>Formule :C24H20N4O4SDegré de pureté :97.49% - 99.37%Couleur et forme :SolidMasse moléculaire :460.51NVP-CGM097
CAS :<p>NVP-CGM097 (CGM097) is an effective and specific MDM2 inhibitor (IC50: 1.7 nM for hMDM2).</p>Formule :C38H47ClN4O4Degré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :659.26Linifanib
CAS :<p>Linifanib (AL-39324) (ABT-869) is a novel, potent ATP-competitive VEGFR/PDGFR inhibitor for KDR (IC50: 4 nM), CSF-1R (IC50: 3 nM), Flt-1/3 (IC50: 3/4 nM) and</p>Formule :C21H18FN5ODegré de pureté :98% - 98.24%Couleur et forme :SolidMasse moléculaire :375.4Coniferaldehyde
CAS :<p>Coniferaldehyde (Ferulaldehyde) is a member of the class of cinnamaldehydes. Coniferaldehyde has a role as an antifungal agent and a plant metabolite.</p>Formule :C10H10O3Degré de pureté :96.35% - 99.96%Couleur et forme :SolidMasse moléculaire :178.18DC661
CAS :<p>DC661 is a palmitoyl-protein thioesterase 1 (PPT1) inhibitor that acts as an anti-lysosomal agent by inhibiting autophagy, demonstrating anti-cancer activity.</p>Formule :C31H39Cl2N5Degré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :552.58Cobimetinib
CAS :<p>Cobimetinib (GDC-0973) is a MEK1 inhibitor with selective and oral activity. Cobimetinib exhibits antitumor activity. Cost-effective and quality-assured.</p>Formule :C21H21F3IN3O2Degré de pureté :98% - 99.61%Couleur et forme :SolidMasse moléculaire :531.31GW 5074
CAS :<p>GW 5074 (Raf1 Kinase Inhibitor I)(IC50=9 nM) is an effective and specific c-Raf inhibitor.</p>Formule :C15H8Br2INO2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :520.94YH239-EE
CAS :<p>YH239-EE, the ethyl ester of YH239, is a potent p53-MDM2 antagonist and an apoptosis inducer.</p>Formule :C25H27Cl2N3O4Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :504.41Didymin
CAS :<p>Didymin, an antioxidant, may treat neuroblastoma and neurodegeneration by blocking N-Myc and boosting RKIP.</p>Formule :C28H34O14Degré de pureté :99.12% - 99.87%Couleur et forme :Faintly Beige PowderMasse moléculaire :594.56GSK2256098
CAS :<p>GSK2256098 (GTPL7939) is a small molecule FAK kinase inhibitor.</p>Formule :C20H23ClN6O2Degré de pureté :99.46% - 99.74%Couleur et forme :SolidMasse moléculaire :414.893,6-Dihydroxyflavone
CAS :<p>3,6-Dihydroxyflavone suppresses the epithelial-mesenchymal transition in breast cancer cells by inhibiting the Notch signaling pathway.</p>Formule :C15H10O4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :254.24PP1
CAS :<p>PP1 (AGL 1872), a specific and effective Src inhibitor, is with IC50 for Lck/Fyn is 5 nM/ 6 nM, respectively.</p>Formule :C16H19N5Degré de pureté :99% - 99.88%Couleur et forme :Off-White To Grey SolidMasse moléculaire :281.36Oroxin B
CAS :<p>Oroxin B (Hypocretin-2) has antioxidant activity.</p>Formule :C27H30O15Degré de pureté :98.22% - 99.81%Couleur et forme :SolidMasse moléculaire :594.52Nystatin
CAS :<p>Nystatin (Fungicidin) is a topical and oral antifungal agent with activity against many species of yeast and candida albicans, which is used largely to treat</p>Formule :C47H75NO17Degré de pureté :69.55% - 99.53%Couleur et forme :Yellow SuspensionMasse moléculaire :926.1Capmatinib
CAS :<p>Capmatinib (INCB28060) is an orally bioavailable inhibitor of the proto-oncogene c-Met (HGFR)with potential antineoplastic activity.</p>Formule :C23H17FN6ODegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :412.42Betulinic acid
CAS :<p>Betulinic acid, a lupane-type triterpene from white birch bark, has antiretroviral, antimalarial, anti-inflammatory, and anticancer properties.</p>Formule :C30H48O3Degré de pureté :99.12% - 99.7%Couleur et forme :White Crystalline PowderMasse moléculaire :456.7MK-4101
CAS :<p>MK-4101 inhibits Hedgehog pathway, causing apoptosis and reduced proliferation in cancer cells.</p>Formule :C24H24F5N5ODegré de pureté :98.2% - 99.13%Couleur et forme :SolidMasse moléculaire :493.47KEA1-97
CAS :<p>Kea1-97 is a selective disruptor of interaction between thioredoxin and caspase-3 (IC50 = 10 μ M).</p>Formule :C15H9Cl2FN4Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :335.16Pralatrexate
CAS :<p>Pralatrexate (10-Propargyl-10-deazaaminopterin) is a folate analogue inhibitor of dihydrofolate reductase (DHFR) exhibiting high affinity for reduced folate</p>Formule :C23H23N7O5Degré de pureté :94.32% - 99.59%Couleur et forme :SolidMasse moléculaire :477.47C188-9
CAS :<p>C188-9 (TTI-101) is a Stat3 inhibitor with an IC50 of 4-7 μM.</p>Formule :C27H21NO5SDegré de pureté :98.07% - >99.99%Couleur et forme :SolidMasse moléculaire :471.52Vatalanib dihydrochloride
CAS :<p>Vatalanib dihydrochloride (PTK787 dihydrochloride)(IC50=37 nM) is an inhibitor of VEGFR2/KDR.</p>Formule :C20H15ClN4·2HClDegré de pureté :99.16%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :419.73NADPH tetrasodium salt
CAS :<p>NADPH tetrasodium salt is the reduced form of the electron acceptor nicotinamide adenine dinucleotide phosphate, which acts as an electron donor in a variety of</p>Formule :C21H26N7Na4O17P3Degré de pureté :97.15% - >99.99%Couleur et forme :SolidMasse moléculaire :833.35ML385
CAS :<p>ML385 is an NRF2 inhibitor (IC50=1.9 μM) with novelty and specificity.</p>Formule :C29H25N3O4SDegré de pureté :98.08% - >99.99%Couleur et forme :SolidMasse moléculaire :511.59Vandetanib
CAS :<p>Vandetanib (ZD6474) is a potent inhibitor of VEGFR2 (IC50: 40 nM). It also inhibits VEGFR3 and EGFR.</p>Formule :C22H24BrFN4O2Degré de pureté :99.7% - >99.99%Couleur et forme :White SolidMasse moléculaire :475.35tubuloside B
CAS :<p>Tubuloside B from Cistanche salsa stems guards SH-SY5Y cells against TNFalpha-induced apoptosis.</p>Formule :C31H38O16Degré de pureté :97.59% - 99.72%Couleur et forme :SolidMasse moléculaire :666.62PF-4989216
CAS :<p>PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.</p>Formule :C18H13FN6OSDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :380.4JX06
CAS :<p>JX06, a potent, selective and covalent PDK inhibitor, inhibits PDK1, PDK2 and PDK3 with IC50 of 49 nM, 101 nM and 313 nM respectively.</p>Formule :C10H16N2O2S4Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :324.51Diosgenin glucoside
CAS :<p>Diosgenin glucoside (Trillin) and other synthetic glycosides with similar activities may be of use in the management of hypercholesterolemia and atherosclerosis</p>Formule :C33H52O8Degré de pureté :97.17% - 99.44%Couleur et forme :SolidMasse moléculaire :576.76MK-2206 dihydrochloride
CAS :<p>MK-2206 dihydrochloride (MK-2206 2HCl) is a variant Akt inhibitor that inhibits Akt1, Akt2, and Akt3 (IC50=8/12/65 nM) with orally active, highly potent and</p>Formule :C25H23Cl2N5ODegré de pureté :99.228% - 99.94%Couleur et forme :SolidMasse moléculaire :480.39Tauroursodeoxycholate dihydrate
CAS :<p>Tauroursodeoxycholate (TUDCA ,Taurolite) dihydrate is a bile acid that reduces Caspase-3, Caspase-12, ERK, reducing endoplasmic reticulum stress mediated death.</p>Formule :C26H49NO8SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :535.73Geranyl acetate
CAS :<p>Geranyl acetate is a monoterpene that has been found in C. sativa with diverse biological activities.</p>Formule :C12H20O2Degré de pureté :98% - 99.36%Couleur et forme :Physical Description Clear Colorless Liquid With An Odor Of Lavender (Ntp 1992)Masse moléculaire :196.29Tubastatin A
CAS :<p>Tubastatin A: Selective HDAC6 inhibitor, IC50 of 15 nM, 1000x less effective on other isozymes except HDAC8.</p>Formule :C20H21N3O2Degré de pureté :97.22% - 99.51%Couleur et forme :SolidMasse moléculaire :335.4Alisertib
CAS :<p>Alisertib (MLN 8237) is a specific Aurora A inhibitor (IC50: 1.2 nM). The selectivity of Alisertib(MLN 8237) is >200-fold higher for Aurora A than Aurora B.</p>Formule :C27H20ClFN4O4Degré de pureté :98.31% - >99.99%Couleur et forme :SolidMasse moléculaire :518.92Linalool
CAS :<p>Linalool, in essential oils, offers antinociceptive, antimicrobial, and anti-inflammatory effects, protects the liver, and boosts plant defense.</p>Formule :C10H18ODegré de pureté :98.22%Couleur et forme :Colorless Liquid Drypowder Liquid Othersolid LiquidMasse moléculaire :154.25SRS16-86
CAS :<p>SRS16-86 is a novel third-generation ferrostatin, is an inhibitor of ferroptosis.</p>Formule :C26H32N4O2Degré de pureté :97.73%Couleur et forme :SolidMasse moléculaire :432.56dl-Maackiain
CAS :<p>1. dl-Maackiain (Demethylpterocarpin) induces apoptosis and growth suppression 2. MAK1 is the second functional gene cloned from Maackiain detoxification.</p>Formule :C16H12O5Degré de pureté :97.36% - 99.89%Couleur et forme :SolidMasse moléculaire :284.26AT7519 Hydrochloride
CAS :<p>AT7519 Hydrochloride (AT7519 HCl) is a multi-CDK inhibitor for CDK1, 2, 4, 6 and 9.</p>Formule :C16H18Cl3N5O2Degré de pureté :99.66% - 99.9%Couleur et forme :SolidMasse moléculaire :418.71Juglanin
CAS :<p>Juglanin is a JNK activator. Juglanin with inflammation and anti-tumor activities. It can induce apoptosis and autophagy on human breast cancer cells.</p>Formule :C20H18O10Degré de pureté :98.8% - 99.33%Couleur et forme :SolidMasse moléculaire :418.35Obacunone
CAS :<p>Obacunone: cytotoxic to prostate cells, anti-S. Typhimurium, may inhibit breast cancer and aromatase, trigger apoptosis.</p>Formule :C26H30O7Degré de pureté :98% - ≥95%Couleur et forme :White PowderMasse moléculaire :454.51PhiKan 083
CAS :<p>PhiKan 083 is a carbazole derivative</p>Formule :C16H18N2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :238.33Hirsutine
CAS :<p>Hirsutine induces apoptosis and is a potent Dengue virus inhibitor exhibiting low cytotoxicity.Hirsutine has anticancer, cardioprotective, anti-hypertensive and</p>Formule :C22H28N2O3Degré de pureté :99.36% - 99.98%Couleur et forme :SolidMasse moléculaire :368.47(Rac)-Antineoplaston A10
CAS :<p>Antineoplaston A10 is the first identified human antineoplaston, naturally occurring with anti-proliferative properties.</p>Formule :C13H14N2O3Degré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :246.26A-1210477
CAS :<p>A-1210477 is an effective and specific MCL-1 and Bcl-2 inhibitor (Ki/IC50: 0.454/26.2 nM).</p>Formule :C46H55N7O7SDegré de pureté :99.17% - 99.37%Couleur et forme :SolidMasse moléculaire :850.04Echinocystic acid
CAS :<p>EA, a natural triterpene, is found in herbs; it has anti-inflammatory and antioxidant properties.</p>Formule :C30H48O4Degré de pureté :98% - 99.57%Couleur et forme :SolidMasse moléculaire :472.7Pseudolaric Acid B
CAS :<p>Pseudolaric acid B, a natural diterpenoid compound, is isolated from Pseudolarix kaempferi.</p>Formule :C23H28O8Degré de pureté :98.91% - 99.84%Couleur et forme :SolidMasse moléculaire :432.46NVP-HSP990
CAS :<p>NVP-HSP990 (HSP990) is an effective and specific HSP90α/β inhibitor (IC50: 0.6 /0.8 nM).</p>Formule :C20H18FN5O2Degré de pureté :98.03% - 99.32%Couleur et forme :SolidMasse moléculaire :379.39PF-3758309 hydrochloride
CAS :<p>PF-3758309 hydrochloride (PF-03758309 hydrochloride) , is a PAK4 inhibitor, is also a n orally bioavailable small-molecule inhibitor of p21-activated kinase 4 (</p>Formule :C25H31ClN8OSDegré de pureté :98.83% - >99.99%Couleur et forme :SolidMasse moléculaire :527.08Cabozantinib S-malate
CAS :<p>Cabozantinib S-malate (XL184) is the salt form of cabozantinib, an orally bioavailable, small molecule RTK inhibitor with potential antineoplastic activity.</p>Formule :C32H30FN3O10Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :635.59Liproxstatin-1
CAS :<p>Liproxstatin-1 is a potent and selective inhibitor of iron death (IC50=22 nM).</p>Formule :C19H21ClN4Degré de pureté :97.11% - 99.44%Couleur et forme :SolidMasse moléculaire :340.85SZL P1-41
CAS :<p>SZL P1-41 inhibits Skp2, blocks complex formation, and halts ubiquitination, promoting cell senescence, reducing glycolysis, and exhibiting antitumor effects.</p>Formule :C24H24N2O3SDegré de pureté :99.60% - 99.87%Couleur et forme :SolidMasse moléculaire :420.52Panobinostat
CAS :<p>Panobinostat (NVP-LBH589) is a broad-spectrum HDAC inhibitor (IC50=5 nM) with oral activity and non-selectivity.</p>Formule :C21H23N3O2Degré de pureté :97.2% - 99.81%Couleur et forme :Yellow SolidMasse moléculaire :349.43HS-1793
CAS :<p>HS-1793, resveratrol-like, reduces HIF-1, VEGF in hypoxia, and curbs human breast cancer growth in mouse model.</p>Formule :C16H12O3Degré de pureté :98.16% - 99.82%Couleur et forme :SolidMasse moléculaire :252.26Cucurbitacin B
CAS :<p>Cucurbitacin B (Cuc B) has profound in vitro and in vivo antiproliferative effects against human pancreatic Y cells.</p>Formule :C32H46O8Degré de pureté :97.1% - 99.33%Couleur et forme :SolidMasse moléculaire :558.7Rosiglitazone hydrochloride
CAS :<p>Rosiglitazone hydrochloride (BRL-49653 HCl) is a blood glucose-lowering drugs, stimulating insulin secretion by binding to the PPAR receptors in fat cells.</p>Formule :C18H19N3O3S·HClDegré de pureté :99.63% - 99.79%Couleur et forme :SolidMasse moléculaire :393.89ZM-447439
CAS :<p>ZM 447439 selectively inhibits Aurora A/B (IC50: 110/130 nM); 8x less effective on MEK1, Src, Lck; minimal impact on CDK1/2/4, Plk1, Chk1.</p>Formule :C29H31N5O4Degré de pureté :99.11% - 99.59%Couleur et forme :Pale Yellow SolidMasse moléculaire :513.59SP600125
CAS :<p>SP600125 (JNK Inhibitor II) is a JNK inhibitor that inhibits JNK1, JNK2, and JNK3 (IC50=40/40/90 nM) with oral potency, reversibility, and ATP-competitive</p>Formule :C14H8N2ODegré de pureté :97.63% - 99.82%Couleur et forme :SolidMasse moléculaire :220.23Mimosine
CAS :<p>L-Mimosine (Leucenol) is an antineoplastic alanine-substituted pyridine derivative isolated from Leucena glauca and acts as an iron chelator.</p>Formule :C8H10N2O4Degré de pureté :99.2% - 99.84%Couleur et forme :Crystals From Water SolidMasse moléculaire :198.18PHA-767491 hydrochloride
CAS :<p>PHA-767491 (CAY-10572) is a potent Cdc7/CDK9 inhibitor (IC50: 10/34 nM), selective against GSK3-β, CDK1/2, CDK5, MK2, CHK2, PLK1.</p>Formule :C12H12ClN3ODegré de pureté :99.56% - 99.92%Couleur et forme :SolidMasse moléculaire :249.69KY-05009
CAS :<p>KY-05009 blocks TGF-β1 EMT in lung cancer cells, inhibits TNIK, Wnt genes, induces apoptosis, and is an ATP-competitive TNIK inhibitor (Ki = 100 nM).</p>Formule :C18H16N4O2SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :352.411A-116
CAS :<p>1A-116 is a specific Rac1 inhibitor.</p>Formule :C16H16F3N3Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :307.31CCT 137690
CAS :<p>CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).</p>Formule :C26H31BrN8ODegré de pureté :98.51% - 99.89%Couleur et forme :SolidMasse moléculaire :551.48BTZO-1
CAS :<p>BTZO-1 is an antioxidant response element (ARE) activator with cardioprotective activity.</p>Formule :C13H8N2OSDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :240.28Salidroside
CAS :<p>Salidroside is a bioactive phenolic glycoside compound isolated from Rhodiola rosea and is a prolyl endopeptidase inhibitor.Cost-effective and quality-assured.</p>Formule :C14H20O7Degré de pureté :97.81%Couleur et forme :Red-Brown Fine PowderMasse moléculaire :300.3C-DIM12
CAS :<p>C-DIM12 boosts Nurr1 gene expression, heightens Nurr1 protein in neurons, and improves survival against 6-OHDA.</p>Formule :C23H17ClN2Degré de pureté :97.72% - ≥95%Couleur et forme :SolidMasse moléculaire :356.85SJ-172550
CAS :<p>SJ-172550 is a small molecule inhibitor of MDMX (EC50: 5 μM).</p>Formule :C22H21ClN2O5Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :428.87L-685458
CAS :<p>L-685458 (L-685,458) is a specific and potent inhibitor of A beta PP gamma-secretase activity with Ki of 17 nM.</p>Formule :C39H52N4O6Degré de pureté :99.62% - 99.80%Couleur et forme :SolidMasse moléculaire :672.85Momelotinib
CAS :<p>Momelotinib (LM-1149), an oral JAK1/2 inhibitor with IC50s 11/18 nM, blocks ATP binding, disrupting JAK-STAT pathway and reducing tumor growth.</p>Formule :C23H22N6O2Degré de pureté :97.47% - 99.56%Couleur et forme :SolidMasse moléculaire :414.46TC11
CAS :<p>TC11 (1H-Isoindole-1,3(2H)-dione, 5-amino-2-[2,6-bis(1-methylethyl)phenyl]-TC11) is a potent inhibitor of tumor cell proliferation and an inducer of apoptosis</p>Formule :C20H22N2O2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :322.4Oleic acid
CAS :<p>Oleic acid, a common unsaturated fat, is used in oleates, lotions, and as a pharma solvent.</p>Formule :C18H34O2Degré de pureté :97.14% - 99.91%Couleur et forme :Colorless Or Nearly Colorless Liq (Above 5-7 Deg C) Oleic Acid Is A Colorless To Pale Yellow Liquid With A Mild Odor Floats On Water (Uscg 1999)Masse moléculaire :282.46
