Apoptose
Les inhibiteurs de l'apoptose sont des composés qui empêchent ou retardent le processus de mort cellulaire programmée, connu sous le nom d'apoptose. Ces inhibiteurs sont essentiels pour étudier les mécanismes de survie cellulaire et sont utilisés pour enquêter sur les maladies où l'apoptose est dysrégulée, telles que le cancer, les troubles neurodégénératifs et les maladies auto-immunes. En modulant l'apoptose, ces inhibiteurs peuvent aider au développement de thérapies visant à contrôler la mort cellulaire. Chez CymitQuimica, nous offrons une sélection complète d'inhibiteurs de l'apoptose de haute qualité pour soutenir vos recherches en biologie cellulaire, oncologie et domaines connexes.
Sous-catégories appartenant à la catégorie "Apoptose"
- ASK(6 produits)
- BCL(11 produits)
- Caspase(125 produits)
- FOXO1(3 produits)
- IAP(66 produits)
- Mdm2(12 produits)
- PD-1/PD-L1(125 produits)
- PDK(9 produits)
- PERK(25 produits)
- Sérine/thréonine kinase(15 produits)
- Survivant(13 produits)
- TNF(92 produits)
- c-RET(51 produits)
- p53(62 produits)
Affichez 6 plus de sous-catégories
5592 produits trouvés pour "Apoptose"
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12-HETE
CAS :<p>12-HETE ((±)12-HETE) is a regulator of PGE2, having both antithrombotic and prothrombotic effects.</p>Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.47Daporinad hydrochloride
CAS :<p>Daporinad hydrochloride (FK 866 hydrochloride) is a NAMPT inhibitor with antitumor and antiangiogenic activity that induces apoptosis in tumor cells.</p>Formule :C24H30ClN3O2Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :427.97Bcl-xL antagonist 2
CAS :<p>Bcl-xL antagonist 2 is an effective and selective antagonist of Bcl-xL with an IC50 of 91 nM and a Ki of 65 nM.</p>Formule :C21H16N4O3S2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :436.51MG-277
<p>MG-277 is a molecular glue compound transformed from PROTAC degradation agent, MG-277 potently inhibits tumor cell growth in a p53-independent manner.</p>Formule :C41H42Cl2FN5O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :774.71NDI-Lyso
CAS :<p>NDI-Lyso is an anticancer agent targeting lysosomes, functioning through an enzyme-induced self-assembly (EISA) mechanism catalyzed by Cathepsin B. In cancer cell lysosomes, it forms rigid long fibers, promoting lysosomal swelling, lysosomal membrane permeabilization (LMP), and membrane disruption. This leads to non-classical caspase-independent apoptosis (Apoptosis). NDI-Lyso demonstrates significant selective anticancer activity across various cancer cell lines and drug-resistant cancer cells (IC50 approximately 10 μM), while exhibiting low toxicity to normal cells (IC50 > 60 μM).</p>Formule :C71H100N22O13Couleur et forme :SolidMasse moléculaire :1469.69PROTAC HIF-1α degrader-1
<p>PROTAC HIF-1α degrader-1 (compound V2) is an effective proteolysis-targeting chimeric (PROTAC) degrader of hypoxia-inducible factor-1α (HIF-1α), with an IC50 value of 7.54 µM. This compound exhibits anti-proliferative activity, reduces HIF-1α protein expression, and induces apoptosis.</p>Formule :C51H72N6O7SCouleur et forme :SolidMasse moléculaire :913.22hMcl-1-IN-1
<p>hMcl-1-IN-1 (Compound 9) is an hMcl-1 inhibitor based on a His224 arylsulfonyl fluoride, displaying an IC50 value of 5.8 nM.</p>Formule :C69H113FN20O19SCouleur et forme :SolidMasse moléculaire :1577.82PROTAC TRIB2 degrader-1
<p>PROTAC TRIB2 degrader-1 (Compound 5k) is a potent TRIB2 degrader that selectively induces TRIB2 degradation via the CRBN-dependent ubiquitin-proteasome pathway. It effectively inhibits cell proliferation and induces cell apoptosis (apoptosis), making it useful in cancer research.</p>Formule :C45H45FN8O6Couleur et forme :SolidMasse moléculaire :812.89BIM-46174 HCl
<p>BIM-46174 HCl is a G-protein inhibitor with anticancer activity that induces cysteine 3-dependent apoptosis.</p>Formule :C22H31ClN4OSDegré de pureté :99.77% - 99.77%Couleur et forme :SolidMasse moléculaire :435.03P53R3
CAS :<p>P53R3 is a potent reactivator of p53, effectively restoring sequence-specific DNA binding to several p53 hot spot mutants, namely p53 R175H, p53 R248W, and p53</p>Formule :C32H35Cl2N5O2Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :592.56BM 957
CAS :<p>BM 957 is an effective Bcl-2 and Bcl-xL inhibitor (Kis: 1.2 and <1 nM; IC50s: 5.4 and 6.0 nM).</p>Formule :C52H56ClF3N6O7S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1065.68rac-CCT-250863 HCl
<p>rac-CCT-250863 HCl: NEK 2 inhibitor, halts cell cycle, anti-cancer growth, boosts Pomalidomide-induced apoptosis.</p>Formule :C24H26ClF3N4O2SDegré de pureté :98.21%Couleur et forme :SoildMasse moléculaire :527SPOP-IN-6lc
CAS :<p>SPOP-IN-6lc is a SPOP inhibitor with oncogenic effects in renal cancer cells.SPOP-IN-6lc can be used to study apoptosis.</p>Formule :C26H31N7O2SDegré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :505.64Glutathione arsenoxide hydrochloride
<p>Glutathione arsenoxide hydrochloride: anti-cancer, inhibits tumour metabolism, targets ANT, promotes apoptosis, marks cell proteins.</p>Formule :C18H26AsClN4O9SDegré de pureté :99.74%Couleur et forme :SoildMasse moléculaire :584.866-Bromo-4-methoxypyrazolo[1,5-a]pyridine-3-carbonitrile
CAS :<p>6-Bromo-4-methoxypyrazolo[1,5-a]pyridine-3-carbonitrile is a PDK1 inhibitor with anticancer and antiproliferative activity that can be used to study</p>Formule :C9H6BrN3ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :252.07PROTAC-O4I2
CAS :<p>PROTAC-O4I2, a PROTAC ligand targeting splicing factor 3B1 (SF3B1), induced FLAG-SF3B1 degradation in K562 cells with an IC50 value of 0.244 μM.</p>Formule :C29H29ClN6O5SDegré de pureté :97.45%Couleur et forme :SolidMasse moléculaire :609.1AZD-4877
CAS :<p>AZD-4877: Potent Eg5 inhibitor, IC50 = 2 nM, alters mitosis, induces apoptosis, has antitumor effects.</p>Formule :C28H33N5O2SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :503.66NS3694
CAS :<p>NS3694 is an inhibitor of apoptosis and inhibits apoptosome formation and caspase activation.</p>Formule :C15H10ClF3N2O3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :358.7Lesigercept
<p>Lesigercept is a humanized antibody that targets IGHE.</p>Couleur et forme :Odour LiquidTilogotamab
CAS :<p>Tilogotamab (GEN-1029) is an agonistic hexameric complex targeting two independent epitopes on DR5, used for studying multiple myeloma (MM).</p>Degré de pureté :95%Couleur et forme :LiquidHFY-4A
CAS :<p>HFY-4A is a novel HDAC inhibitor.HFY-4A has antitumour activity and has shown antiproliferative activity in breast cancer cells.</p>Formule :C20H19N3O2Degré de pureté :98.66% - 99.22%Couleur et forme :SoildMasse moléculaire :333.38Sandacanol
CAS :<p>Sandacanol (Sandranol) is an olfactory receptor (OR10H1) agonist.Sandacanol induces cell cycle arrest and partial apoptosis in bladder cancer cells.</p>Formule :C14H24ODegré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :208.34Δ8-Tetrahydrocannabinoquinone
CAS :<p>Δ8-Tetrahydrocannabinoquinone (HU-336) is a potent anti-angiogenic agent that inhibits angiogenesis by directly inducing apoptosis in vascular endothelial cells. It achieves this without altering the expression of pro-angiogenic and anti-angiogenic cytokines and receptors. Δ8-Tetrahydrocannabinoquinone also shows significant effectiveness against tumor xenografts in nude mice.</p>Formule :C21H28O3Couleur et forme :SolidMasse moléculaire :328.45FA4-Cu
<p>FA4-Cu is a compound formed from the effective pancreatic cancer inhibitor FA4 and Cu(II), which can induce apoptosis by triggering ER and mitochondrial stress.</p>Formule :C27H33Cl2CuN5O2SCouleur et forme :SolidMasse moléculaire :626.1Anticancer agent 136
<p>Anticancer agent 136 (compound 22), a C17-triazole analogue of Geldanamycin (GDM), exhibits an IC50 value of 3.38 μM against human dermal fibroblasts (HDF) and</p>Formule :C40H50N6O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :742.86Anticancer agent 146
<p>Anticancer Agent 146 (Compound 1.19) acts as a necroptosis inducer and demonstrates anti-tumor efficacy in the MDA-MB-231 mouse xenograft model [1].</p>Formule :C19H16Cl2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :375.25BAY 1892005
CAS :<p>BAY 1892005 is a p53 protein modulator that targets the p53 condenser for the study of diseases associated with misfolded p53 protein</p>Formule :C11H8ClFN2OSDegré de pureté :99.62%Couleur et forme :SoildMasse moléculaire :270.71Anti-inflammatory agent 45
<p>Compound 2v (Anti-inflammatory agent 45) demonstrates anticancer properties with direct inhibitory impacts on the proliferation of various blood malignancies,</p>Formule :C25H22BrNO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :512.35Antitumor agent-96
<p>"Antitumor agent-96 (Compound D34) is a potent MRE11 inhibitor that down-regulates the homologous recombination (HR) pathway by binding to and suppressing the</p>Formule :C27H32N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :416.56Flaccidoside II
CAS :<p>Flaccidoside II, an active triterpenoid saponin from Anemone flaccida rhizome, both inhibits proliferation and induces apoptosis in Malignant Peripheral Nerve</p>Formule :C59H96O25Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1205.38Ara-SH
<p>Ara-SH, a derivative of Cytarabine with a mercaptopropionic acid substitution, serves as the initiator for the self-assembly of a smart, co-loaded Cytarabine</p>Formule :C12H17N3O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.342'-epi-2'-O-Acetylthevetin B
CAS :<p>2'-Epi-2'-O-Acetylthevetin B (GHSC-74), a cardiac glycoside extractable from Cerbera manghas L.</p>Formule :C44H68O19Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :901Apoptosis inducer 11
<p>Apoptosis Inducer 11 (compound 3u) promotes apoptosis via the mitochondrial pathway and elicits a G2/M block alongside a marked reduction in the S phase within</p>Formule :C27H28N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :460.52TAT-BH4 (Bcl-xL)
<p>TAT-BH4 (Bcl-xL), primarily localized at the mitochondria, inhibits apoptotic cell death.</p>Formule :C159H268N58O45Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3712.19TAT-NEP1-40
<p>TAT-NEP1-40, a blood-brain barrier (BBB) permeable peptide, confers protection to PC12 cells against oxygen and glucose deprivation (OGD) while promoting</p>Formule :C268H438N88O77Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :6124.89CPT2
CAS :<p>Carnitine palmitoyltransferase 2 (CPT2), an enzyme involved in fatty acid oxidation, serves as a prognostic biomarker for colorectal cancer (CRC).</p>Degré de pureté :98%Couleur et forme :SolidPyridinium bisretinoid A2E TFA
CAS :<p>Pyridinium bisretinoid A2E (A2E) TFA, a fluorophore derived from retinal pigment epithelium (RPE) lipofuscin, initiates blue-light-induced apoptosis, mediates</p>Formule :C44H58F3NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :705.93Antitumor agent-112
<p>Antitumor agent-112 (compound 3a) is a potent antitumor agent that induces apoptosis and exhibits cytotoxic activity on A549 cells, with an IC50 value of 91.35</p>Formule :C18H17ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :388.87TAT-NEP1-40 TFA
<p>TAT-NEP1-40 TFA, a blood-brain barrier-permeable peptide, safeguards PC12 cells against oxygen and glucose deprivation (OGD) and fosters neurite outgrowth.</p>Formule :C268H438N88O77·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :6124.89 (free base)TP4 (Nile tilapia piscidin)
CAS :<p>TP4 (Nile tilapia piscidin) is an orally active piscidin-like antimicrobial peptide that exhibits inhibition of various gram-positive and negative bacterial</p>Formule :C135H226N50O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2981.56Antitumor agent-113
<p>Antitumor Agent-113 exhibits cytotoxicity in A549 cells, with an IC50 of 46.60 μM, and induces apoptosis, making it applicable for research in non-small cell</p>Formule :C21H22ClN5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :443.95Anticancer agent 106
<p>Compound 106 (compound 10ic) induces apoptosis in B16-F10 melanoma cells and potently inhibits metastatic nodules in mouse models of lung metastatic melanoma,</p>Formule :C26H25N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :475.56FD2157
<p>FD2157, a photosensitive PI3K inhibitor, exhibits inhibitory IC50 values of 43 nM for PI3Kα, 83 nM for PI3Kβ, 84 nM for PI3Kγ, and 14 nM for PI3Kδ.</p>Formule :C27H21ClN6O8SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.01cpm-1285
CAS :<p>CPM-1285 induces apoptosis by effectively inhibiting the function of intracellular Bcl-2 and associated death antagonists.</p>Formule :C153H240N44O42SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3399.88Anticancer agent 132
<p>Compound Rh1 (Anticancer agent 132) acts as an inducer of apoptosis and autophagy, exhibiting both antitumor and antimetastatic activities.</p>Formule :C24H16Cl3F3N5ORhDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :656.68Antitumor agent-103
<p>Antitumor Agent-103 (compound 24l) induces apoptosis and possesses antiproliferative and anti-colony formation properties.</p>Formule :C36H36N8O9S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :788.85Anticancer agent 153
<p>Anticancer Agent 153 (Compound 3) promotes apoptosis through the generation of Reactive Oxygen Species (ROS) and elevates the loss of Mitochondrial Membrane</p>Formule :C16H11Cl2N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :364.18Pamrevlumab
CAS :<p>FG-3019 (Pamrevlumab), a human antibody, targets CTGF, potentially treating idiopathic pulmonary fibrosis.</p>Degré de pureté :100% (SEC-HPLC) - 95%Couleur et forme :LiquidSACLAC
CAS :<p>SACLAC is a cysteine asparaginase activation inhibitor with antitumor activity used in the study of acute myeloid leukemia and cancer.</p>Formule :C20H40ClNO3Degré de pureté :97.03%Couleur et forme :SoildMasse moléculaire :377.992-aminobenzo[d]thiazol-6-ol
CAS :<p>2-aminobenzo[d]thiazol-6-ol: antimicrobial, antioxidant, anticancer; may trigger cancer cell apoptosis.</p>Formule :C7H6N2OSDegré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :166.2(E/Z)-Squalene
CAS :<p>(E/Z)-Squalene modulates ROS, triggers apoptosis/necrosis, reduces liver cholesterol and triglycerides.</p>Formule :C30H50Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :410.72Bifenthrin
CAS :<p>Bifenthrin is a synthetic pyrethroid insecticide.Bifenthrin induces cell death in bovine mammary epithelial cells through ROS generation, disruption of calcium homeostasis, and alteration of the MAPK signaling cascade.Bifenthrin induces apoptosis by inducing cell-cycle arrest.</p>Formule :C23H22ClF3O2Degré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :422.87Se-Aspirin
CAS :<p>Se-Aspirin (Se-NSAID-8) has anticancer activity and gastroprotective effects, inhibits activation of proinflammatory and pro-survival NF-ĸB pathways, and inhibits the expression of anti-apoptotic targets downstream of NF-ĸB (e.g., Bcl-xL, Mcl-1, and survivin).Se-Aspirin induces Cell cycle arrest and activation of apoptosis accelerates ulcer healing and can be used to study pancreatic and colorectal cancer.</p>Formule :C12H12N2O3SeDegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :311.2Cyclamic acid sodium
CAS :<p>Sodium cyclamate is a carbonic anhydrase inhibitor, artificial sweetener, with anticonvulsant properties, and used in cancer research.</p>Formule :C6H12NNaO3SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :201.22Capsazepine
CAS :Formule :C19H21ClN2O2SDegré de pureté :>98.0%(HPLC)(qNMR)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :376.901-(2-Deoxy-2-fluoro-β-D-arabinofuranosyl)uracil
CAS :<p>1-(2-Deoxy-2-fluoro-beta-D-arabinofuranosyl)uracil is a Nucleoside, fluoro-modified nucleoside; Arabino-nucleosidde.</p>Formule :C9H11FN2O5Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :246.19Belinostat
CAS :Formule :C15H14N2O4SDegré de pureté :>98.0%(HPLC)Couleur et forme :White to Light yellow to Light orange powder to crystalMasse moléculaire :318.35(-)-Gallocatechin Gallate
CAS :Formule :C22H18O11Degré de pureté :>95.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :458.38Parthenolide
CAS :Formule :C15H20O3Degré de pureté :>97.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :248.32Everolimus-d4
CAS :<p>Everolimus-d4 is a deuterated compound of Everolimus.</p>Formule :C53H83NO14Couleur et forme :SolidMasse moléculaire :962.2646-Formylpterin
CAS :<p>6-Formylpterin (Pterin-6-aldehyde) is an inhibitor of Xanthine Oxidase, which induces ROS generation and apoptosis in HL-60 cells.</p>Formule :C7H5N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :191.15Alantolactone
CAS :Formule :C15H20O2Degré de pureté :>95.0%(GC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :232.322'-Deoxy-2'-fluoro-β-D-arabinoguanosine
CAS :<p>2'-Deoxy-2'-fluoro-beta-D-arabinoguanosine is a purine nucleoside analog with a broad spectrum of antitumor activity, targeting malignant tumors of the inert</p>Formule :C10H12FN5O4Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :285.23FMAU
CAS :<p>FMAU (2'-Deoxy-2'-fluoro-5-methyl-beta-D-arabinouridine) is a thymine nucleoside analog with insertional activity on replicating DNA.FMAU can be used to label</p>Formule :C10H13FN2O5Degré de pureté :98.6%Couleur et forme :SolidMasse moléculaire :260.22Octreotide
CAS :<p>Octreotide (SMS 201-995) is a potent inhibitor of growth hormone, glucagon, and insulin.</p>Formule :C49H66N10O10S2Degré de pureté :99.64%Couleur et forme :White PowderMasse moléculaire :1019.24C-DIM 12
CAS :Formule :C23H17ClN2Degré de pureté :>98.0%(HPLC)(qNMR)Couleur et forme :Orange to Amber to Dark red powder to crystalineMasse moléculaire :356.85Olanzapine D3
CAS :<p>Olanzapine D3 is the deuterium labeled Olanzapine.</p>Formule :C17H20N4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.45PBOX 6
CAS :<p>PBOX 6 is a pyrrolo-1,5-benzoxazepine (PBOX) compound with anticancer and antitumor activity that inhibits the growth of breast cancer cells.</p>Formule :C25H20N2O3Degré de pureté :98.18% - 98.71%Couleur et forme :SolidMasse moléculaire :396.4413-Methyltetradecanoic acid
CAS :<p>LeDSF3 controls HSAF production in Lysobacter, has antifungal properties, and acts as an anti-tumor by inhibiting p-AKT and activating caspase-3.</p>Formule :C15H30O2Couleur et forme :SolidMasse moléculaire :242.4VK3-OCH3
CAS :Formule :C14H14O3SDegré de pureté :>98.0%(HPLC)Couleur et forme :Light yellow to Yellow to Orange powder to crystalMasse moléculaire :262.32Hydroxy-PP-Me
CAS :<p>Hydroxy-PP-Me is a CBR1 inhibitor that inhibits apoptosis induced by serum withdrawal.Hydroxy-PP-Me is used in the study of leukemia.</p>Formule :C16H18N4ODegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :282.34Sunitinib-d10
CAS :<p>Sunitinib D10, a deuterium-enriched version, inhibits VEGFR2 and PDGFRβ tyrosine kinases (IC50: 80 nM/2 nM).</p>Formule :C22H27FN4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.54Forodesine hydrochloride
CAS :<p>Forodesine hydrochloride blocks lymphocyte growth and induces leukemia cell death by inhibiting PNP, effective across species.</p>Formule :C11H15ClN4O4Couleur et forme :SolidMasse moléculaire :302.714-[Di(1H-indol-3-yl)methyl]phenol
CAS :Formule :C23H18N2ODegré de pureté :>97.0%(T)(HPLC)Couleur et forme :White to Light orange to Yellow powder to crystalMasse moléculaire :338.41Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride
CAS :<p>Thalidomide-O-amido-PEG4-C2-NH2 hydrochloride is a synthesized E3 ligase ligand-linker conjugate incorporating the Thalidomide-based cereblon ligand and a</p>Formule :C25H35ClN4O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :587.02Cis-5-Norbornene-exo-2,3-dicarboxylic Anhydride
CAS :<p>Cis-5-Norbornene-exo-2,3-dicarboxylic Anhydride: sensitizing, induces HepG2/SK-Hep1 apoptosis, inhibits PP2A. IC50: HepG2=62μM, SK-Hep1=151μM.</p>Formule :C9H8O3Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :164.16BAY 11-7082
CAS :Formule :C10H9NO2SDegré de pureté :>98.0%(HPLC)(N)Couleur et forme :White to Almost white powder to crystalMasse moléculaire :207.25Thalidomide-Piperazine 5-fluoride
CAS :<p>Thalidomide-Piperazine 5-fluoride: a cereblon ligand-linked E3 ligase via PROTAC tech.</p>Formule :C17H17FN4O4Couleur et forme :SolidMasse moléculaire :360.34Palmatine hydroxide
CAS :<p>Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.</p>Formule :C21H23NO5Couleur et forme :SolidMasse moléculaire :369.41SB 202190
CAS :Formule :C20H14FN3ODegré de pureté :>95.0%(HPLC)Couleur et forme :White to Light yellow to Light orange powder to crystalMasse moléculaire :331.35Tetrac
CAS :<p>Tetrac (Tetraiodothyroacetic acid) is a derivative of L-thyroxine (T4), a thyroxine integrin receptor antagonist.Tetrac induces antiproliferation by blocking</p>Formule :C14H8I4O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :747.83Necrostatin 2 S enantiomer
CAS :<p>Necrostatin 2 S enantiomer is the S enantiomer of Necrostatin 2</p>Formule :C13H12ClN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :277.71Ezatiostat
CAS :<p>Ezatiostat (TER199(free base)) is a tripeptide analog of glutathione that can selectively inhibit GSTP1-1 catalytic activity.</p>Formule :C27H35N3O6SDegré de pureté :97.95%Couleur et forme :SolidMasse moléculaire :529.65PARG-IN-4
CAS :<p>PARG-IN-4 (compound A) is an orally active and cell-membrane permeable PARG inhibitor (EC50=1.9 nM) that inhibits tumour growth in mice with antitumour .</p>Formule :C20H25F2N7O2S2Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :497.59Tegaserod
CAS :<p>Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).</p>Formule :C16H23N5ODegré de pureté :99.20% - 99.89%Couleur et forme :SolidMasse moléculaire :301.39Thalidomide-O-amido-PEG-C2-NH2
CAS :<p>Thalidomide-based cereblon ligand linked to PEG-C2-NH2 for use in PROTAC E3 ligase conjugates.</p>Formule :C19H22N4O7Couleur et forme :SolidMasse moléculaire :418.42'-Aminoacetophenone
CAS :<p>Compound Fr14273 is a natural product for research related to life sciences. The catalog number is Fr14273 and the CAS number is 551-93-9.</p>Formule :C8H9NODegré de pureté :99.88%Couleur et forme :Pale Yellow Solid Solid CrystallineMasse moléculaire :135.17Rapamycin-d3
CAS :<p>Rapamycin-d3 is the deuterium labeled Rapamycin. Rapamycin is a potent and specific inhibitor of mTOR(IC50 of 0.1 nM in HEK293 cells).</p>Formule :C51H79NO13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :917.19Nutlin-3
CAS :Formule :C30H30Cl2N4O4Degré de pureté :>95.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :581.49p,p'-DDD
CAS :<p>TDE is an organochlorine insecticide with slightly irritating to the skin.</p>Formule :C14H10Cl4Couleur et forme :Colourless To Off-White CrystalsMasse moléculaire :320.03EIF2α activator 2
CAS :<p>EIF2α activator 2 is an activator of eIF2α phosphorylation, anti-proliferative in SRB, K562, and PBMC cells, suitable for cancer research.</p>Formule :C21H20F6N2O2Degré de pureté :98.86%Couleur et forme :SolidMasse moléculaire :446.39Sodium catechol sulfate
CAS :<p>Sodium catechol sulfate is a bioactive chemical.</p>Formule :C6H4Na2O8S2Degré de pureté :98%Couleur et forme :Light Tan PowderMasse moléculaire :314.20Isoalantolactone
CAS :Formule :C15H20O2Degré de pureté :>98.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :232.32(Rac)-Hesperetin
CAS :<p>(Rac)-Hesperetin, a racemic flavanone, inhibits human UGT activity and triggers apoptosis via p38 MAPK activation.</p>Formule :C16H14O6Couleur et forme :SolidMasse moléculaire :302.285-Methoxyuridine
CAS :<p>5-Methoxyuridine (Mo5U) is an antitumor purine analog that inhibits DNA synthesis and induces apoptosis in lymphatic cancers.</p>Formule :C10H14N2O7Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :274.23(S)-Oxiracetam
CAS :<p>(S)-Oxiracetam is a positive allosteric the AMPA receptorsmodulator.</p>Formule :C6H10N2O3Couleur et forme :SolidMasse moléculaire :158.16GO-203
CAS :<p>GO-203 is a useful organic compound for research related to life sciences. The catalog number is T35351 and the CAS number is 1222186-26-6.</p>Formule :C89H171F3N52O21S2Couleur et forme :SolidMasse moléculaire :2426.81Melatonin-d4
CAS :<p>Melatonin D5, a deuterium-labeled version of melatonin, is a hormone produced by the pineal gland, known for its role as a selective ATF-6 inhibitor that promotes apoptosis in human hepatoma cells via COX-2 downregulation. Additionally, it activates melatonin receptors and exhibits antioxidative and anti-inflammatory properties.</p>Formule :C13H16N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :236.32-Thiocytidine
CAS :<p>2-Thiocytidine is a purine nucleoside analog that targets malignant tumors of the inert lymphatic system and has a broad spectrum of antitumor activity.2-</p>Formule :C9H13N3O4SDegré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :259.28Meisoindigo
CAS :Formule :C17H12N2O2Degré de pureté :>98.0%(HPLC)Couleur et forme :Orange to Brown to Dark red powder to crystalMasse moléculaire :276.30(Rac)-Apremilast D5
CAS :<p>(Rac)-Apremilast D5 is a deuterium-labeled version of the enantiomer (R)-Apremilast, also known as (R)-CC-10004, which itself is one specific form of Apremilast</p>Formule :C22H24N2O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.53Barbadin
CAS :<p>Barbadin is an inhibitor of β-arrestin/β2-adaptin interaction.Barbadin enhances the effects of lorcaserin on weight loss and can be used to study obesity.</p>Formule :C19H15N3OSDegré de pureté :98.93% - 99.10%Couleur et forme :SolidMasse moléculaire :333.41MC1742
CAS :<p>MC1742 inhibits class I/IIb HDACs, blocks sarcoma CSC growth, and reactivates latent HIV. IC50: HDAC1-3/8 (0.02-0.61 μM), HDAC6/10 (7-40 nM).</p>Formule :C21H21N3O3SDegré de pureté :99.20%Couleur et forme :SolidMasse moléculaire :395.48Degarelix
CAS :<p>Degarelix is a peptide and selective GnRH (human gonadotropin-releasing hormone) receptor antagonist prostate cancer by lowering testosterone levels.</p>Formule :C82H103ClN18O16Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :1632.26MCL-1/BCL-2-IN-2
CAS :<p>MCL-1/BCL-2-IN-2 is a selective Mcl-1 and Bcl-2 inhibitor with potential antitumor activity for tumor research.</p>Formule :C20H15BrN2O2SDegré de pureté :98.03%Couleur et forme :SolidMasse moléculaire :427.31Bleximenib oxalate
CAS :<p>Bleximenib oxalate (Menin-MLL inhibitor 24 oxalate) is a menin-MLL inhibitor that blocks the binding of the menin-KMT2A complex to chromatin at gene promoters.</p>Formule :C34H52FN7O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :689.824-(Dimethylamino)-N-[7-(hydroxyamino)-7-oxoheptyl]benzamide
CAS :Formule :C16H25N3O3Degré de pureté :>97.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :307.391,4-Dideoxy-1,4-epithio-D-ribitol
CAS :<p>1,4-Dideoxy-1,4-epithio-D-ribitol is a purine nucleoside analog that targets malignant tumors of the inert lymphatic system and possesses a broad spectrum of</p>Formule :C5H10O3SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :150.2Fosfenopril
CAS :<p>Fosfenopril is an ACE inhibitor reducing LPS-induced inflammation via TLR4/NF-κB suppression, used in cardiovascular and anti-inflammatory molecular studies.</p>Formule :C23H34NO5PCouleur et forme :SolidMasse moléculaire :435.49Fluorizoline
CAS :<p>Fluorizoline is a PHB-binding compound with anticancer and antiproliferative activity and induces apoptosis.</p>Formule :C15H8Cl2F3NSDegré de pureté :98.22% - 99.52%Couleur et forme :SolidMasse moléculaire :362.20PRDX1-IN-1
CAS :<p>PRDX1-IN-1 is a and PRDX1 inhibitor with potential anti-inflammatory and anti-cancer activity for the study of breast and esophageal cancer.</p>Formule :C46H55N3O4Degré de pureté :98.04%Couleur et forme :SolidMasse moléculaire :713.95Wedelolactone
CAS :Formule :C16H10O7Degré de pureté :>98.0%(HPLC)Couleur et forme :White to Dark green powder to crystalMasse moléculaire :314.25Metronidazole-d4
CAS :<p>Metronidazole-d4 is a deuterium labeled compound isotopic tracing.Metronidazole is an antibiotic and antiprotozoal oral and BBB penetration anaerobic bacteria.</p>Formule :C6H9N3O3Couleur et forme :SolidMasse moléculaire :175.18Mardepodect hydrochloride
CAS :<p>Mardepodect hydrochloride (Mardepodect HCl) is a PDE10A inhibitor.Mardepodect hydrochloride upregulates genes encoding specific growth factors.</p>Formule :C25H21ClN4ODegré de pureté :95.1%Couleur et forme :SolidMasse moléculaire :428.91J22352
CAS :<p>J22352, a PROTAC (proteolysis-targeting chimeras)-like and highly selective HDAC6 inhibitor with an IC50 value of 4.7 nM, enhances anticancer effects in</p>Formule :C24H21N3O4Couleur et forme :SolidMasse moléculaire :415.44Benzyl selenocyanate
CAS :<p>Benzyl selenocyanate is a chemopreventive agent that effectively inhibits chemically induced tumors at both initiation and postinitiation stages in animal models. It acts as a potent inhibitor of DNA (cytosine-5)-methyltransferase (Mtase) with an IC50 of 8.4 μM.</p>Formule :C8H7NSeDegré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :196.11M47
CAS :<p>M47 is a selective CRY1 (Cryptochrome 1) degradator that enhances nuclear degradation of CRY1, thereby extending the lifespan of p53 knockout mice.</p>Formule :C28H22ClNO4Couleur et forme :SolidMasse moléculaire :471.93Fenitrothion
CAS :<p>Fenitrothion (Arbogal) is a insecticide that exhibits reproductive toxicity, inhibits acetylcholinesterase, and is commonly used in agriculture.</p>Formule :C9H12NO5PSDegré de pureté :95.07%Couleur et forme :Yellow-Brown Liquid Insecticide Against Chewing And Sucking Insects On Rice Orchard Fruits Vegetables Cereals CottonMasse moléculaire :277.23Chiisanoside
CAS :<p>Chiisanoside is a useful organic compound for research related to life sciences. The catalog number is T123983 and the CAS number is 89354-01-8.</p>Formule :C48H74O19Couleur et forme :SolidMasse moléculaire :955.101N-3-oxo-dodecanoyl-L-Homoserine lactone
CAS :<p>N-3-oxo-dodecanoyl-L-Homoserine lactone (3-oxo-C12-HSL), a quorum-sensing signaling molecule synthesized by P. aeruginosa and specific B. cepacia complex strains [1][2], facilitates bacterial gene expression modulation in response to cell density escalation and triggers IL-8 production in 16HBE human bronchial epithelial cells [3].</p>Formule :C16H27NO4Couleur et forme :SolidMasse moléculaire :297.39Dynole 34-2
CAS :<p>Dynole 34-2 is a non-competitive inhibitor of dynamin1 and dynamin2 GTPases that inhibits receptor-mediated endocytosis and synaptic vesicle endocytosis.</p>Formule :C25H36N4ODegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :408.58Thalidomide-piperazine-Boc
CAS :<p>Thalidomide-piperazine-Boc is an intermediate utilized for synthesizing BCL6 PROTAC, which targets B-cell lymphoma 6 protein.</p>Formule :C22H26N4O6Couleur et forme :SolidMasse moléculaire :442.46Methylstat
CAS :<p>Methylstat is a methyl ester prodrug of a Jumonji C domain-containing histone demethylase (JMJD) inhibitor that has favorable cell permeability.</p>Formule :C28H31N3O6Degré de pureté :98.34% - 98.34%Couleur et forme :SolidMasse moléculaire :505.56Busulfan-d8
CAS :<p>Busulfan-d8 (Sulphabutin-d8) is the 2H-labeled Busulfan. Busulfan is an anticancer agent with immunosuppressive and myeloablative chemotherapy activities.</p>Formule :C6H6D8O6S2Couleur et forme :SolidMasse moléculaire :254.35Pancratistatin
CAS :<p>Pancratistatin, an isoquinoline from Hymenocallis littoralis, triggers apoptosis in melanoma and is studied for neuroblastoma, leukemia, and breast cancer.</p>Formule :C14H15NO8Couleur et forme :SolidMasse moléculaire :325.27Necrostatin 2
CAS :<p>Necrostatin 2 is a RIPK1 inhibitor that can be used to study inner ear disorders such as sudden deafness, dizziness and tinnitus.</p>Formule :C13H12ClN3O2Degré de pureté :99.92% - 99.92%Couleur et forme :SolidMasse moléculaire :277.71Propylparaben sodium
CAS :<p>Propylparaben sodium, a plant-based preservative used in cosmetics, pharma, and food, hinders follicle growth and sperm health.</p>Formule :C10H12NaO3Couleur et forme :SolidMasse moléculaire :203.193L-Cystine, hydrochloride
CAS :<p>L-Cystine, hydrochloride is a useful organic compound for research related to life sciences. The catalog number is T124989 and the CAS number is 34760-60-6.</p>Formule :C6H13ClN2O4S2Couleur et forme :SolidMasse moléculaire :276.75NU 9056
CAS :<p>NU 9056 is an effective and selective inhibitor of KAT5 histone acetyltransferase with an IC50 of 2 µM.</p>Formule :C6H4N2S4Degré de pureté :95.36% - 97.11%Couleur et forme :SolidMasse moléculaire :232.37Tubulin inhibitor 1
CAS :<p>Tubulin inhibitor 1 blocks tubulin polymerization, with strong anti-tumor effects, induces apoptosis and G2/M mitotic arrest.</p>Formule :C21H24N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.43ODN 1826
CAS :<p>ODN 1826 is a TLR9 agonist and immunostimulant, which has antitumor effects and promotes cell apoptosis.</p>Degré de pureté :90% - 90%Couleur et forme :SolidMasse moléculaire :6364.1Lestaurtinib
CAS :<p>Lestaurtinib (CEP 701) is a FLT3 inhibitor that inhibits the phosphorylation of RPTKs and can be used to study leukemia.</p>Formule :C26H21N3O4Degré de pureté :99.17%Couleur et forme :Off-White SolidMasse moléculaire :439.46YZ129
CAS :<p>YZ129, an HSP90-calcineurin-NFAT inhibitor with 820 nM IC50, halts GBM growth, arrests G2/M phase, and induces apoptosis.</p>Formule :C19H12N2O2Couleur et forme :SolidMasse moléculaire :300.31Br-DAPI
CAS :<p>IST5-002 (N6-Benzyladenosine-5'-phosphate) is a Stat5a/b inhibitor with anticancer activity and is used in cancer research.</p>Formule :C16H14BrN5Degré de pureté :100%Couleur et forme :SolidMasse moléculaire :356.22SB 203580
CAS :Formule :C21H16FN3OSDegré de pureté :>98.0%(HPLC)Couleur et forme :White to Orange to Green powder to crystalMasse moléculaire :377.44Cobimetinib hemifumarate
CAS :<p>Cobimetinib hemifumarate is a potent and selective MEK1 inhibitor with an IC50 value of 4.2 nM for MEK1.</p>Formule :C46H46F6I2N6O8Couleur et forme :SolidMasse moléculaire :1178.707PI3Kα-IN-9
CAS :<p>PI3Kα-IN-9 is an inhibitor of PI3Kα and PI3Kα with antiproliferative activity, inhibits PI3Kα, PI3Kγ, PI3Kδ, and PI3Kβ, induces apoptosis.</p>Formule :C18H21N7O3Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :383.4Hydrolyzed Fumonisin B1
CAS :<p>Hydrolyzed Fumonisin B1 is the backbone and the main hydrolysis product of the mycotoxin fumonisin B1 (FB1), can weakly inhibit ceramide synthase.</p>Formule :C22H47NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.62PND-1186 hydrochloride
CAS :<p>PND-1186 hydrochloride (VS-4718 hydrochloride) is a highly specific, reversible and potent inhibitor of FAK (IC50: 1.5 nM), which can selectively induce</p>Formule :C25H27ClF3N5O3Couleur et forme :SolidMasse moléculaire :537.97BIX02188
CAS :<p>BIX02188 is a selective and potent MEK5 inhibitor that inhibits MEK5-induced apoptosis in cells expressing the oncogenic mutant FLT3-ITD.</p>Formule :C25H24N4O2Degré de pureté :97.66%Couleur et forme :SolidMasse moléculaire :412.48Traumatic Acid
CAS :<p>Traumatic Acid aids wound healing in plants by stimulating cell division to create a callus.</p>Formule :C12H20O4Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :228.28Acyclovir-d4
CAS :<p>Acyclovir-d4 is a deuterated compound of Acyclovir. Acyclovir has a CAS number of 59277-89-3. Acyclovir is a synthetic analog of the purine nucleoside, guanosine, with potent antiviral activity against herpes simplex viruses type 1 and 2, varicella-zoster virus and other viruses of the herpesvirus family.</p>Formule :C8H7D4N5O3Couleur et forme :SolidMasse moléculaire :229.23Indirubin-3'-monoxime
CAS :Formule :C16H11N3O2Degré de pureté :>98.0%(HPLC)Couleur et forme :Light yellow to Brown powder to crystalMasse moléculaire :277.28Bz 423
CAS :<p>Bz 423 is a potent immunomodulator that induces apoptosis by activating Bax and Bak to induce mitochondrial outer membrane permeabilization and cytochrome c</p>Formule :C27H21ClN2O2Degré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :440.92Baohuoside I
CAS :Formule :C27H30O10Degré de pureté :>95.0%(T)(HPLC)Couleur et forme :White to Light yellow to Green powder to crystalMasse moléculaire :514.53AZD-5991
CAS :<p>AZD-5991, an antitumor compound, is a highly selective, potent and direct MCL-1 inhibitor, rapid apoptosis by Bak-dependent mitochondrial apoptotic pathway.</p>Formule :C35H34ClN5O3S2Degré de pureté :98.08% - 98.95%Couleur et forme :SolidMasse moléculaire :672.26Z-Ile-Leu-aldehyde
CAS :<p>Z-Ile-Leu-aldehyde is an effective and competitive peptide aldehyde inhibitor of γ-secretase and notch.</p>Formule :C20H30N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :362.46MM-401 TFA
CAS :<p>MM-401 (TFA), an MLL1 H3K4 methylation inhibitor (IC50 = 0.32 µM), blocks MLL1-WDR5, causing cell cycle arrest and apoptosis, for MLL leukemia studies.</p>Formule :C31H47F3N8O7Couleur et forme :SolidMasse moléculaire :700.75Embelin
CAS :Formule :C17H26O4Degré de pureté :>95.0%(T)(HPLC)Couleur et forme :Light yellow to Yellow to Orange powder to crystalMasse moléculaire :294.39Capecitabine-d11
CAS :<p>Capecitabine-d11 is a deuterated compound of Capecitabine. Capecitabine has a CAS number of 154361-50-9. Capecitabine is a fluoropyrimidine carbamate belonging to the class of antineoplastic agents called antimetabolites. As a prodrug, capecitabine is selectively activated by tumor cells to its cytotoxic moiety, 5-fluorouracil (5-FU); subsequently, 5-FU is metabolized to two active metabolites, 5-fluoro-2-deoxyuridine monophosphate (FdUMP) and 5-fluorouridine triphosphate (FUTP) by both tumor cells and normal cells. FdUMP inhibits DNA synthesis and cell division by reducing normal thymidine production, while FUTP inhibits RNA and protein synthesis by competing with uridine triphosphate for incorporation into the RNA strand.</p>Formule :C15H11D11FN3O6Couleur et forme :SolidMasse moléculaire :370.42Condurango glycoside A
CAS :<p>Condurango glycoside A activates p53, induces ROS generation, up-regulates p53 expression, and triggers apoptosis as well as premature senescence associated</p>Formule :C53H78O17Couleur et forme :SolidMasse moléculaire :987.18Methopterin
CAS :<p>Methopterin shows the activation and bone resorption function of murine osteoclasts.</p>Formule :C20H21N7O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.43AZT triphosphate
CAS :<p>AZT triphosphate is a Nucleoside Triphosphate.</p>Formule :C10H16N5O13P3Couleur et forme :SolidMasse moléculaire :507.18PT-262
CAS :<p>PT-262: ROCK inhibitor, causes cytoskeleton change, halts lung cancer cell migration.</p>Formule :C14H13ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :276.72Pitavastatin D4
CAS :<p>Pitavastatin D4 is deuterium labeled Pitavastatin. Pitavastatin is a potent inhibitor of HMG-CoA reductase.</p>Formule :C25H24FNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.49Isoginkgetin
CAS :Formule :C32H22O10Degré de pureté :>95.0%(HPLC)Couleur et forme :White to Light yellow powder to crystalMasse moléculaire :566.52PB28 dihydrochloride
CAS :<p>ZD-6888 Hydrochloride (ZD-6888 HCl) is an angiotensin II antagonist that mediates AII receptor blockade and induces AII-mediated inhibition of renin release.</p>Formule :C24H40Cl2N2ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :443.49Iodoacetyl-LC-Biotin
CAS :<p>Iodoacetyl-LC-Biotin (Iaa-Biotin) is a sulfhydryl-responsive probe that forms irreversible thioether bonds at alkaline pH, label protein cysteines.</p>Formule :C18H31IN4O3SDegré de pureté :97.47%Couleur et forme :SolidMasse moléculaire :510.43Amoscanate
CAS :<p>Amoscanate is an antiparasitic agent. It is highly effective in animals against the four major species of schistosomes which infect humans.</p>Formule :C13H9N3O2SCouleur et forme :SolidMasse moléculaire :271.294-PQBH
CAS :<p>4-PQBH is a potent Nur77-binding agent with antitumour activity.4-PQBH is used in the study of hepatocellular carcinoma.</p>Formule :C22H17N5ODegré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :367.4KS100
CAS :<p>KS100 inhibits ALDH1A1, ALDH2, ALDH3A1, boosts ROS, triggers apoptosis, and has anti-cancer properties.</p>Formule :C17H14Br3N3O2SDegré de pureté :97.05%Couleur et forme :SolidMasse moléculaire :564.09Mepazine hydrochloride
CAS :<p>Mepazine hydrochloride (Pecazine hydrochloride) is a MALT1 inhibitor with anticancer and antitumor activity, inhibiting RANK-induced osteoclastogenesis.</p>Formule :C19H23ClN2SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :346.92PR-924
CAS :<p>PR-924 is a selective inhibitor of tripeptide epoxyketone immunoproteasome subunit LMP-7 (IC50: 22 nM).</p>Formule :C37H38N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :618.72Tamoxifen-d5
CAS :<p>Tamoxifen-d5 is a deuterium labeled Tamoxifen.</p>Formule :C26H29NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.55RKI-1447 dihydrochloride
CAS :<p>RKI 1447 dihydrochloride: selective ROCK inhibitor, inhibits colorectal cancer growth, promotes apoptosis (ROCK1 IC50=14.5 nM, ROCK2 IC50=6.2 nM).</p>Formule :C16H16Cl2N4O2SCouleur et forme :SolidMasse moléculaire :399.29Edaravone-d5
CAS :<p>Edaravone, a potent free radical scavenger, prevents MMP-9-induced brain bleeds in rats and has a deuterium variant, Edaravone D5.</p>Formule :C10H10N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :179.23Demethoxycurcumin
CAS :Formule :C20H18O5Degré de pureté :>98.0%(HPLC)Couleur et forme :Light red to Yellow to Red powder to crystalMasse moléculaire :338.36Pyridoclax
CAS :<p>Pyridoclax is an inhibitor of potential Mcl-1.</p>Formule :C29H22N4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.51AZD5582
CAS :<p>AZD5582 is an inhibitor of IAPs, which binds to the BIR3 domains cIAP1, cIAP2, and XIAP with IC50s of 15, 21, and 15 nM, respectively. It induces apoptosis.</p>Formule :C58H78N8O8Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :1015.29Cerivastatin sodium
CAS :<p>Cerivastatin sodium (BAY W 6228 sodium) is an HMG-CoA reductase inhibitor with lipid-lowering activity that reduces LDL cholesterol levels.</p>Formule :C26H33FNNaO5Degré de pureté :98.50% - 99.67%Couleur et forme :SolidMasse moléculaire :481.53Vitamin E succinate
CAS :<p>Vitamin E succinate (D-alpha-Tocopherol Succinate) is an antioxidant tocopherol with antitumor activity that induces apoptosis.</p>Formule :C33H54O5Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :530.78Thalidomide-O-C6-NH2 TFA
CAS :<p>Thalidomide-O-C6-NH2 TFA is a synthesized E3 ligase ligand-linker conjugate used in the PROTAC dTAG-13, a degrader of FKBP12F36V and BET[1].</p>Formule :C21H24F3N3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :487.43Lacto-N-neotetraose
CAS :<p>LNnT is a metabolite that reduces IL-8, has anti-inflammatory effects, and aids in wound healing.</p>Formule :C26H45NO21Couleur et forme :SolidMasse moléculaire :707.63Macitentan-d4
CAS :<p>Macitentan-d4 (ACT-064992 D4) is a C13-labeled inhibitor of the peptides ETA and ETB used to study diseases mediated by endothelin receptor mediation.</p>Formule :C19H20Br2N6O4SDegré de pureté :96.51%Couleur et forme :SolidMasse moléculaire :592.3Etoposide Phosphate
CAS :<p>Etoposide Phosphate is a selective and orally active topoisomerase II inhibitor and anticancer chemotherapy drug that apoptosise, the p53, and G2/M</p>Formule :C29H33O16PCouleur et forme :SolidMasse moléculaire :668.54CuATSP
CAS :<p>CuATSP is a potent free radical trapping antioxidant (RTA) and ferroptosis inhibitor inhibit lipid peroxidation, for (ALS) and Parkinson's disease.</p>Formule :C18H18CuN6S2Degré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :446.05Fenvalerate
CAS :<p>Fenvalerate (Evercide 2362) is a protein phosphatase 2B (calcineurin) inhibitor, a synthetic pyrethroid insecticide, that inhibits PP2B-Aα.</p>Formule :C25H22ClNO3Degré de pureté :99.62%Masse moléculaire :419.90MRT00033659
CAS :<p>MRT00033659 inhibits CK1 (IC50=0.9 μM), CHK1 (IC50=0.23 μM), activates p53, and destabilizes E2F-1; it's a pyrazolo-pyridine.</p>Formule :C15H14N4OCouleur et forme :SolidMasse moléculaire :266.3CLZ-8
CAS :<p>CLZ-8 (Mcl1-IN-8) is a Mcl-1-PUMA inhibitor with radioprotective activity and inhibits radiation-induced overexpression of PUMA.</p>Formule :C22H23N3O2SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :393.5KT-474
CAS :<p>KT-474 (KYM-001) is a PROTAC degrader targeting IRAK4 with antitumor activity for the study of autoimmune diseases.</p>Formule :C44H49F2N11O6Degré de pureté :98.50% - 99.57%Couleur et forme :SolidMasse moléculaire :865.93NCX 4040
CAS :<p>COX-2 expression inhibitor</p>Formule :C16H13NO7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.28Apremilast-d5
CAS :<p>Apremilast D5 (CC-10004 D5) is a deuterium-labeled Apremilast.</p>Formule :C22H24N2O7SCouleur et forme :SolidMasse moléculaire :465.53Thalidomide-O-amido-PEG3-C2-NH2 hydrochloride
CAS :<p>Thalidomide-based E3 ligase linker for PROTACs with a PEG3 chain and hydrochloride salt.</p>Formule :C23H31ClN4O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :542.97Ulipristal Acetate
CAS :Formule :C30H37NO4Degré de pureté :>98.0%(T)(HPLC)Couleur et forme :White to Yellow to Green powder to crystalMasse moléculaire :475.63Rutin trihydrate
CAS :<p>Rutin trihydrate is a natural flavonoid with antioxidant, anti-inflammatory, anti-diabetic, and anti-cancer benefits, plus heart and brain protection.</p>Formule :C27H36O19Couleur et forme :SolidMasse moléculaire :664.56PI-103 Hydrochloride
CAS :<p>PI-103 Hydrochloride is a dual PI3K/Akt and mTOR inhibitor exhibiting nM-level inhibition of p110α, p110β, p110δ, p110γ, DNA-PK, mTORC1, and mTORC2.</p>Formule :C19H17ClN4O3Degré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :384.82Mycophenolic acid-d3
CAS :<p>Mycophenolic acid-d3 is a derivative that lowers GTP, affects RNA polymerase II transcription, changes polyadenylation, and counters cordyceps.</p>Formule :C17H20O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.36Prexasertib dimesylate
CAS :<p>Prexasertib dimesylate is a selective CHK1 inhibitor with K i 0.9 nM, blocks CHK2 & RSK1, induces DNA breakage, and has potent anti-tumor effects.</p>Formule :C20H27N7O8S2Couleur et forme :SolidMasse moléculaire :557.6Thalidomide-O-amido-C4-NH2
CAS :<p>Thalidomide-O-amido-C4-NH2 is a thalidomide cereblon ligand-linker used for PROTAC synthesis as an E3 ligase.</p>Formule :C19H22N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :402.45-(N,N-Hexamethylene)-amiloride
CAS :<p>5-(N,N-Hexamethylene)-amiloride (5-HMA) is an amiloride derivative that inhibits TRPA1-mediated calcium signaling (IC50: 35 μM). It functions as an inhibitor of the Na+/H+ exchanger (NHE) with Ki values ranging from 0.013 to 2.4 μM for various NHE isoforms. Additionally, 5-HMA blocks ASIC3 channels by 51% at 20 μM.</p>Formule :C12H18ClN7ODegré de pureté :85.48%Couleur et forme :SolidMasse moléculaire :311.77Methoxyacetic acid
CAS :<p>Methoxyacetic acid is an endogenous metabolite.</p>Formule :C3H6O3Couleur et forme :Less Liquid (Ntp 1992) Physical Description Colorless Liquid (Ntp 1992)Masse moléculaire :90.08Prinaberel
CAS :<p>Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.</p>Formule :C15H10FNO3Degré de pureté :97.1%Couleur et forme :SolidMasse moléculaire :271.24(E/Z)-E64FC26
CAS :<p>(E/Z)-E64FC26 is a protein disulfide isomerase (PDI) family inhibitor with affinity for PDIA1, PDIA3, PDIA4, TXNDC5, and PDIA6.</p>Formule :C19H23F3O2Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :340.38Curcumin-d6
CAS :<p>Curcumin D6 (difluoroformylmethane D6) is deuterium-labeled curcumin (Turmeric yellow). Curcumin (Turmeric yellow) is a natural phenolic compound with various pharmacological effects, including anti-inflammatory, antioxidant, anti-proliferative and anti-a</p>Formule :C21H20O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.422Buparlisib Hydrochloride
CAS :<p>Buparlisib Hydrochloride is an inhibitor of pan-class I PI3K (IC50: 52 nM/166 nM/116 nM/262 nM for p110α/p110β/p110δ/p110γ, respectively).</p>Formule :C18H22ClF3N6O2Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :446.85Givinostat
CAS :<p>Givinostat (ITF-2357) is a non-selective, orally active HDAC inhibitor capable of inhibiting STAT5 phosphorylation which is antitumour and anti-inflammatory .</p>Formule :C24H27N3O4Degré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :421.5GSK-843
CAS :<p>GSK-843 (GSK'843) is a RIP3 inhibitor with analgesic activity, inhibits RIP3 expression, and can be used as an adjunctive treatment for inflammation.</p>Formule :C19H15N5S2Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :377.49Acyclovir hydrochloride
CAS :<p>Acyclovir (Aciclovir) hydrochloride is an effective oral antiviral agent with potent anti-herpetic activity. It exhibits IC50 values of 0.85 μM for HSV-1 and 0.86 μM for HSV-2, indicating strong inhibitory effects against these strains. Additionally, Acyclovir hydrochloride induces cell cycle disturbances and apoptosis. This compound also prevents bacterial infections during induction therapy for acute leukemia.</p>Formule :C8H12ClN5O3Couleur et forme :SolidMasse moléculaire :261.67Thalidomide-5,6-F
CAS :<p>Thalidomide-5,6-F, a cereblon ligand for CRBN protein recruitment, forms PROTACs for targeted protein degradation.</p>Formule :C13H8F2N2O4Couleur et forme :SolidMasse moléculaire :294.21Ancitabine
CAS :<p>Ancitabine is an antitumour drug that improves Hailey-Hailey disease-related phenotypes in yeast models. inhibits DNA synthesis, acute leukaemia.</p>Formule :C9H11N3O4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :225.2
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