Chromatine/Épigénétique
Les inhibiteurs de la chromatine/épigénétique sont des composés qui modulent la structure et la fonction de la chromatine ou interfèrent avec les modifications épigénétiques, telles que la méthylation de l'ADN et la modification des histones. Ces inhibiteurs sont des outils essentiels pour étudier la régulation de l'expression génique et le rôle de l'épigénétique dans des maladies telles que le cancer, les troubles neurologiques et les anomalies du développement. En ciblant les processus épigénétiques, ces inhibiteurs peuvent modifier les schémas d'expression génique et offrir de nouvelles perspectives thérapeutiques. Chez CymitQuimica, nous offrons une large sélection d'inhibiteurs de la chromatine/épigénétique de haute qualité pour soutenir vos recherches en biologie moléculaire, génétique et épigénétique.
Sous-catégories appartenant à la catégorie "Chromatine/Épigénétique"
2612 produits trouvés pour "Chromatine/Épigénétique"
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AMPK activator 1
CAS :AMPK activator 1 is an AMPK activator(compound No.1-75, EC50: <0.1μM).Formule :C32H33F3N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :578.62NV03
CAS :NV03 is a selective antagonist of the UHRF1-H3K9me3 interaction (Kd=2.4 μM) for cancer research. a ligand for E3 ligases in PROTAC synthesis.Formule :C19H27N5O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :389.52M122
CAS :M122 is a selective histone deacetylase HDAC1 and HDAC2 inhibitor and potent antitumor agent.Formule :C24H25N5OS2Couleur et forme :SolidMasse moléculaire :463.62CTK7A
CAS :CTK7A is a water-soluble inhibitor of p300. CTK7A inhibits tumor growth in xenografted mice.Formule :C28H24N2NaO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :507.498HDAC6-IN-6
CAS :HDAC6-IN-6: Potent HDAC6 blocker, BBB-permeable, IC50: 0.025μM; inhibits AChE, Aβ 1-42 aggregation; promotes neurite growth, low neurotoxicity.Formule :C20H15N3O2Couleur et forme :SolidMasse moléculaire :329.35MAT2A inhibitor 1
CAS :MAT2A inhibitor 1 is an inhibitor of methionine adenosyltransferase 2A (MATA2) (IC50 < l00 nM).Formule :C31H22N6OSCouleur et forme :SolidMasse moléculaire :526.61HDAC-IN-5
CAS :HDAC-IN-5 is a histone deacetylase (HDAC) inhibitor.Formule :C26H24F3N5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :527.56CTPB
CAS :CTPB is a potent p300 histone acetyltransferase (HAT) activator that can be used in the preparation of hair growth promoters and/or hair loss treatments.Formule :C31H43ClF3NO2Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :554.13JAK3-IN-12
CAS :JAK3-IN-12 (compound 15k) is a potent inhibitor of JAK3 (IC50: 9.5 nM) and can be used in the study of rheumatoid arthritis.Formule :C19H19N5O4SCouleur et forme :SolidMasse moléculaire :413.45SB-429201
CAS :SB-429201 is an effective, selective inhibitor of HDAC1.Formule :C28H24N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.5JAK3-IN-9
CAS :JAK3-IN-9, potent JAK3 inhibitor, IC50 of 1.7 nM, highly selective, low toxicity, orally bioavailable, shows anti-arthritis activity.Formule :C17H23N5O4SCouleur et forme :SolidMasse moléculaire :393.46CPI-455 HCl
CAS :CPI-455: specific KDM5A inhibitor, IC50=10±1nM, increases H3K4me3, reduces DTPs in cancer cells.Formule :C16H15ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :314.77LB-205
CAS :LB-205 is a Zn 2+ dependent pan-inhibitor of class I and class II HDACs. It also has a long half-life in vivo.Formule :C18H21N3O2SCouleur et forme :SolidMasse moléculaire :343.44INCB16562
CAS :INCB16562: oral JAK1/2 inhibitor, halts IL-6/STAT3 in myeloma cells, boosts drug efficacy, stunts myeloma in mice.Formule :C19H11Cl2N5Couleur et forme :SolidMasse moléculaire :380.23Guadecitabine
CAS :Guadecitabine is a second-generation DNA methyltransferases inhibitor. It is used for research on acute myeloid leukemia and myelodysplastic syndromes.Formule :C18H24N9O10PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :557.41PB131
CAS :PB131, a selective and brain-permeable HDAC6 inhibitor, exhibits high binding affinity (IC50: 1.8 nM) and potent anti-inflammatory activity, making it suitableFormule :C16H16FN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :301.32ZL0454
CAS :ZL0454 is an effective and selective Bromodomain-containing protein 4 inhibitors (IC50: 49 and 32 nM for BD1 and BD2).Formule :C18H22N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.46MPT0G211
CAS :MPT0G211: oral HDAC6 inhibitor with IC50=0.291 nM, 1000x selectivity, neuroprotective, anti-metastatic, crosses blood-brain barrier for Alzheimer's.Formule :C17H15N3O2Degré de pureté :99.93% - 99.98%Couleur et forme :SolidMasse moléculaire :293.32Ref: TM-T60616
1mg92,00€5mg222,00€10mg356,00€25mg560,00€50mg782,00€100mg1.063,00€200mg1.459,00€1mL*10mM (DMSO)245,00€Bromodomain inhibitor-8
CAS :Bromodomain inhibitor-8 is an inhibitor of BET bromodomain used to treat autoimmune and inflammatory diseases.Formule :C26H25ClN2O3Couleur et forme :SolidMasse moléculaire :448.94Exifone
CAS :Exifone (NSC-680919) is a mixed, nonessential activator of HDAC1 that is capable of binding to both free and substrate-bound enzyme, resulting in an increasedFormule :C13H10O7Degré de pureté :99.77% - 99.95%Couleur et forme :Yellow SolidMasse moléculaire :278.21Bromodomain inhibitor-9
CAS :Bromodomain inhibitor-9 selectively targets BRD4-1 (Kd 12 nM), used in metabolic, inflammatory, fibrotic, and autoimmune disease studies.Formule :C24H28N4O5SCouleur et forme :SolidMasse moléculaire :484.571,2,3,4,5,6-Hexabromocyclohexane
CAS :Inhibits JAK2 autophosphorylation; non-cytotoxic at 100μM; 1μM reduces activity by 50%, 50μM nearly abolishes it.Formule :C6H6Br6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :557.54Tankyrase-IN-2
CAS :Tankyrase-IN-2 is a selective, potent and orally active inhibitor of tankyrase with IC50s of 10, 7, and 710 nM for TNKS1, TNKS2 as well as PARP1, respectivelyFormule :C17H14F2N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :316.36(5H)-Phenanthridinone
CAS :6(5H)-Phenanthridinone suppresses PARP1/2, reduces RDM4 cell growth, downregulates pro-inflammatory genes, and alleviates EAE symptoms in rats.Formule :C13H9NOCouleur et forme :SolidMasse moléculaire :195.22NCC-149
CAS :NCC-149 is a HDAC8 inhibitor.Formule :C16H14N4O2SCouleur et forme :SolidMasse moléculaire :326.37MS-1020
CAS :MS-1020 inhibits JAK3/STAT3, blocks active JAK3, suppresses JAK3/STAT5 signaling, and targets STAT3 in certain cells.Formule :C21H18N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :346.38AC-93253 iodide
CAS :AC-93253 iodide is a selective inhibitor of SIRT2. It significantly enhances the acetylation of tubulin p53 and histone H4.Formule :C23H25IN2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :488.43GNE-272
CAS :GNE-272 is a selective inhibitor of CBP/EP300 (IC50: 0.02, 0.03, and 13 μM for CBP, EP300, and BRD4, respectively) and a selective in vivo probe for CBP/EP300.Formule :C22H25FN6O2Couleur et forme :SolidMasse moléculaire :424.47Ac-Lys-AMC
CAS :Ac-Lys-AMC (Hexanamide) is a fluorescent substrate for histone deacetylase HDACs.Formule :C18H23N3O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :345.39PS315
CAS :PS315, a PS48 derivative, allosterically inhibits PKCζ/η (IC50: 10/30 μM), targeting aPKC's PIF-pocket, with anti-cancer properties.Formule :C23H19ClO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :362.85ZYJ-34v
CAS :ZYJ-34v is an oral histone deacetylase inhibitor (HDACi) with potent antitumor activities.Formule :C27H35N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :497.58SD-1029
CAS :SD-1029 is a JAK2 inhibitor and a novel Stat3 activation inhibitor that inhibits Stat3 phosphorylation and JAK-STAT signaling.Formule :C25H32Br2Cl2N2O3Couleur et forme :SolidMasse moléculaire :639.25Jaspamycin
CAS :Jaspamycin (7-CN-7-C-Ino) does not bind with purified human PKARIα.Formule :C12H12N4O5Couleur et forme :SolidMasse moléculaire :292.25(R)-UT-155
CAS :(R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.Formule :C20H15F4N3O2Couleur et forme :SolidMasse moléculaire :405.35ARTD10/PARP10-IN-1
CAS :ARTD10/PARP10-IN-1 is a PARP inhibitor that inhibits ARTD8/PARP14 and has anticancer and antitumour activity for the study of prostate cancer.Formule :C12H12N2O4Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :248.233-Deazaneplanocin A
CAS :3-Deazaneplanocin A (DZNep) is an EZH2 and AHCY inhibitor with antipoxigenic activity that inhibits fibrosis in the liver, kidneys, peritoneum, and airways.Formule :C12H14N4O3Degré de pureté :99.03% - 99.68%Couleur et forme :SolidMasse moléculaire :262.27GS-626510
CAS :GS-626510 is an orally bioavailable inhibitor of BET family bromodomains (Kd: 0.59-3.2 nM for BRD2/3/4; IC50: 83 nM and 78 nM for BD1 and BD2).Formule :C25H22N4OCouleur et forme :SolidMasse moléculaire :394.47AMPK activator
CAS :AMPK activatorFormule :C22H21FO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.4LW479
CAS :LW479 is a novel inhibitor of HDAC and is a promising candidate for the prevention of breast cancer.Formule :C21H23BrN2O4SCouleur et forme :SolidMasse moléculaire :479.39KDM5A-IN-1
CAS :KDM5A-IN-1 is a pan-histidine lysine demethylase 5 KDM5 inhibitor that inhibits KDM5A, KDM5B, and KDM5C.Can be used in the study of cancer.Formule :C15H22N4O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :290.36DC_517
CAS :DC_517 is an inhibitor of DNA methyltransferase 1 (DNMT1) ( IC50: 1.7 μM; Kd: 0.91 μM).Formule :C33H35N3O2Couleur et forme :SolidMasse moléculaire :505.65Sirt2-IN-1
CAS :Sirt2-IN-1 is an inhibitor of sirtuin 2 (IC50 = 163 nM).Formule :C28H27N7O2S2Degré de pureté :99.57% - 99.84%Couleur et forme :SolidMasse moléculaire :557.69Ref: TM-T12920
1mg100,00€5mg203,00€10mg323,00€25mg513,00€50mg697,00€100mg888,00€500mg1.783,00€1mL*10mM (DMSO)253,00€L 888607 Racemate
CAS :L 888607 Racemate blocks DP1 and TP receptors with 132 nM and 17 nM affinity.Formule :C19H15ClFNO2SCouleur et forme :SolidMasse moléculaire :375.84Ilorasertib hydrochloride
CAS :Ilorasertib hydrochloride (ABT-348 hydrochloride) is an ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A (IC50s:Formule :C25H22ClFN6O2SDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :525Tetrahydrouridine
CAS :Tetrahydrouridine (NSC-112907; THU) is a multidrug resistance modulator.Formule :C9H16N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :248.23ITF3756
CAS :ITF3756 is a selective HDAC6 inhibitor.Formule :C13H11N5O2SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :301.32Tyk2-IN-7
CAS :Tyk2-IN-7 is an inhibitor of TYK2 JH2, binds to the TYK2 JH2 domain (IC50: 0.00053 μM; Ki.app: 0.00007 μM).Formule :C18H15D3N6O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :401.46Givinostat hydrochloride monohydrate
CAS :Givinostat hydrochloride monohydrate (ITF2357) is an HDAC inhibitor.Formule :C24H27N3O4·HCl·H2ODegré de pureté :97.97% - 99.51%Couleur et forme :SolidMasse moléculaire :475.97Pulrodemstat Methylbenzenesulfonate
CAS :LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.Formule :C31H31F2N5O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :623.67HDAC3-IN-T247
CAS :HDAC3-IN-T247 (HDAC3 inhibitor T247) is a histone deacetylase 3 (HDAC3) inhibitor with antiviral activity that inhibits the proliferation of cancer cells.Formule :C21H19N5OSDegré de pureté :98.11% - 98.94%Couleur et forme :SolidMasse moléculaire :389.47Ref: TM-T24131
1mg87,00€5mg178,00€10mg295,00€25mg610,00€50mg867,00€100mg1.153,00€1mL*10mM (DMSO)203,00€YM-53601 free base
CAS :YM-53601 free base is an inhibitor of squalene synthetase which suppresses lipogenic biosynthesis and lipid secretion in rodents.Formule :C21H21FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.4EP009
CAS :EP009, a novel, selective, and orally active inhibitor of JAK3, induces therapeutic response in T-cell malignancies.Formule :C14H24O2Couleur et forme :SolidMasse moléculaire :224.34MDK8228
CAS :MDK8228 is an inhibitor of CBP/p300 and BRD4 bromodomain. MDK8228 downregulates IL-6, IL-ß and IFN-ß in macrophages.Formule :C31H41N5O3Couleur et forme :SolidMasse moléculaire :531.69AJH-836
CAS :AJH-836 is a compound that activates Munc13-1 and PKC ε/α, demonstrating a dissociation constant (Kd) of 4.5 nM for PKCα, and facilitates the translocation ofFormule :C22H38O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :382.53SIRT2-IN-9
CAS :SIRT2-IN-9: selective SIRT2 inhibitor; IC50=1.3μM; halts MCF-7 cell growth; for cancer study.Formule :C21H22N6OS2Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :438.57RM65
CAS :RM65 is an arginine methyltransferase inhibitor.Formule :C34H32N2O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :596.76HDAC-IN-58
CAS :HDAC-IN-58, a selective HDAC6 inhibitor, exhibits potent inhibitory activity with an IC50 of 2.06 nM, rendering it suitable for research into chronicFormule :C16H13ClF2N4O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :414.81JAK-IN-21
CAS :JAK-IN-21 is a selective and potent JAK inhibitor that inhibits JAK1, JAK2, J2V617F and TYK2 with IC50 values of 1.73, 2.04, 109 and 62.9 nM, respectively.Formule :C19H16N8ODegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :372.38JAK-IN-14
CAS :JAK-IN-14 (compound 16) is a specific JAK1 inhibitor. It prevents JAK1 phosphorylation by binding to the active site of JAK in immune, inflammation and cancer.Formule :C19H15FN4ODegré de pureté :98.27%Couleur et forme :SolidMasse moléculaire :334.35Ref: TM-T9764
1mg81,00€5mg170,00€10mg268,00€25mg555,00€50mg888,00€100mg1.414,00€200mg1.882,00€1mL*10mM (DMSO)178,00€LSD1-IN-6
CAS :LSD1-IN-6, a potent LSD1 inhibitor (IC50: 123 nM), enhances H3K4me2 without altering LSD1 expression. Reversible.Formule :C15H13BrN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.18IDO1 and HDAC1 Inhibitor
CAS :IDO1 and HDAC1 Inhibitor is a dual IDO1 and HDAC1 inhibitor (IC50s: 69.0 nM and 66.5 nM).Formule :C25H22BrFN8O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :597.4HDAC-IN-49
HDAC-IN-49: potent, broad HDAC inhibitor; IC50s: 10-1880 nM for HDAC1-6; strong anti-leukemic, low toxicity to healthy cells.Formule :C26H27FN4O4Couleur et forme :SolidMasse moléculaire :478.52Sirt1/2-IN-1
CAS :Sirt1/2-IN-1 inhibits SIRT1 (IC50: 1.81 μg/mL) and SIRT2 (2.10 μg/mL), less on SIRT3 (20.5 μg/mL), with anticancer properties.Formule :C22H13ClN2OS2Couleur et forme :SolidMasse moléculaire :420.93PIM-1 Inhibitor 2
CAS :PIM-1 Inhibitor 2 (PIM1-IN-2) is a potent Pim-1 inhibitor with potential anti-cancer activity, used in cancer research.Formule :C17H11ClN4ODegré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :322.752′-Deoxy-5-nitrocytidine
CAS :2′-Deoxy-5-nitrocytidine is a DNA Methyltransferase inhibitor that can be used for cancer research[1].Formule :C9H12N4O6Couleur et forme :SolidMasse moléculaire :272.21SB-284851-BT
CAS :SB-284851-BT: BRD4/p38α/BRDT inhibitor; IC50: BRD4-BD1 1.7µM, BRDT 18µM, BRD4 3.7µM; Kd p38α 0.47nM; reduces IL-8, affects c-Myc/NF-κB.Formule :C26H26FN5OCouleur et forme :SolidMasse moléculaire :443.52PKC-IN-4
CAS :PKC-IN-4 (compound 7l) is a highly potent and orally active inhibitor of atypical protein kinase C (aPKC), exhibiting an IC 50 value of 0.52 μM.Formule :C21H25N5SCouleur et forme :SolidMasse moléculaire :379.52CD161
CAS :CD161: powerful, selective oral BET inhibitor; IC50: 28.2 nM (BRD4 BD1), 7.2 nM (BRD4 BD2); strong anticancer properties.Formule :C26H21N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :435.48YF479
CAS :YF479 is an inhibitor of histone deacetylase that acts by inhibiting breast tumor growth, metastasis, and recurrence.Formule :C22H27BrN2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.36DC-CPin7
CAS :DC-CPin7, a powerful inhibitor of the bromodomain of CREB-binding protein (CBP), exhibits an IC50 value of 2.5 μM [1].Formule :C19H22N2O5Couleur et forme :SolidMasse moléculaire :358.39OICR-0547
CAS :OICR-0547 is an inactive derivative of OICR-9429 and is commonly used as a negative control for OICR-9429.Formule :C28H29F3N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :542.55HIF-1α inhibitor-1
CAS :HIF-1α inhibitor-1 is a HIF-1 alpha inhibitor.Formule :C15H11N3O4Couleur et forme :SolidMasse moléculaire :297.27SMYD2-IN-1
CAS :SMYD2-IN-1 is an inhibitor of SMYD2 (IC50 of 4.45 nM).Formule :C25H25Cl2F2N7O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :564.41Bisindolylmaleimide II
CAS :protein kinase C (PKC) inhibitorFormule :C27H26N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.52LSD1-IN-12
CAS :LSD1-IN-12 (compound 2) is an effective inhibitor of LSD1, demonstrating inhibitory Ki values of 1.1 μM (LSD1), 61 μM (LSD2), 2.3 μM (MAO-A), and 3.5 μM (MAO-BFormule :C16H16N2OCouleur et forme :SolidMasse moléculaire :252.31SRTCX1002
CAS :SRTCX1002 is a SIRT1 Activator Suppressing Inflammatory Responses through Promotion of p65 Deacetylation and NF-κB Activity inhibitor.Formule :C21H19N5O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.47PU141
CAS :PU141 is a novel inhibitor of histone acetyltransferase (HAT).Formule :C14H9F3N2OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.29CHIC35
CAS :CHIC-35 is a selective deacetylase SIRT1 inhibitor.Formule :C14H15ClN2OCouleur et forme :SolidMasse moléculaire :262.73OTS186935 trihydrochloride
CAS :OTS186935 trihydrochloride is a protein methyltransferase inhibitor of SUV39H2(IC50 of 6.49 nM).Formule :C25H29Cl4N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :573.34HDAC-IN-45
CAS :HDAC-IN-45, a small HDAC blocker, forms H-bonds with Y303 and shows anticancer properties; IC50 for HDAC1/2/3: 0.108/0.585/0.563 μM.Formule :C25H20ClFN8OCouleur et forme :SolidMasse moléculaire :502.93dBRD9-A
CAS :Potent BRD9 degrader that binds selectively, fully degrades BRD9 at low doses, and hinders synovial sarcoma growth in vitro and in mice.Formule :C42H49N7O8Couleur et forme :SolidMasse moléculaire :779.88ET-JQ1-OH
CAS :ET-JQ1-OH is an allele-specific BET inhibitor.Formule :C21H21ClN4O2SCouleur et forme :SolidMasse moléculaire :428.93Y02224
CAS :Y02224 is a BET inhibitor. It shows the reasonable antiproliferative effect on leukemia cells.Formule :C20H17BrN2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :461.33PB118
PB118 clears Aβ, boosts phagocytosis, enhances tubulin networks, reduces p-tau & inflammation in AD; HDAC6 IC50: 5.6 nM.Formule :C18H19FN2O2Couleur et forme :SoildMasse moléculaire :314.35HDAC3-IN-T326
CAS :HDAC3-IN-T326: potent, selective HDAC3 inhibitor, boosts NF-κB acetylation, activates latent HIV gene expression.Formule :C21H18N6O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.47Dot1L-IN-5
CAS :Dot1L-IN-5 is a potent inhibitor of the disruptor of telomeric silencing 1-like protein ( DOT1L ) with an IC 50 SPA DOT1L of 0.17 nM [1].Formule :C23H19ClF2N8O5SCouleur et forme :SolidMasse moléculaire :592.96Helenalin Acetate
CAS :Helenalin Acetate: anti-inflammatory, anti-cancer, hinders C/EBPß and p300 cooperation.Formule :C17H20O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.34PS432
CAS :PS432 inhibits atypical PKCs, targets PIF-pocket, reduces tumors in mice sans side effects.Formule :C25H19ClN2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :494.95DM-01
CAS :DM-01 is a potent and selective inhibitor of EZH2.Formule :C23H24F3N3O2Couleur et forme :SolidMasse moléculaire :431.45Kgp-IN-1
CAS :Kgp-IN-1 is an arginine-specific gingipain (Rgp) inhibitor.Formule :C19H24F4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.41(1S,2R)-Tranylcypromine hydrochloride
CAS :(1S,2R)-Tranylcypromine hydrochloride ((1S,2R)-SKF 385), a potent antidepressant, functions by inhibiting both MAO and LSD1.Formule :C9H12ClNCouleur et forme :SolidMasse moléculaire :169.651Gue1654
CAS :Gue1654 is an OXE-R inhibitor and cardiomyocyte apoptosis.Gue1654 can be used for the study of cardiovascular diseases.Formule :C23H17N3OS3Degré de pureté :98.02% - 98.04%Couleur et forme :SolidMasse moléculaire :447.6CID-4785700
CAS :CID-4785700 is a potent pan-GTPase inhibitor that inhibits Rab7 and inhibits the fungal histone acetyltransferase Rtt109 that binds to Asf1 and Vps75Formule :C22H23ClFN3O3Degré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :431.89Ref: TM-T71740
1mg315,00€5mg873,00€10mg1.080,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.419,00€PARP-1/2-IN-1
CAS :PARP-1-/2-IN-1 is a potent inhibitor of PARP-1 (IC50: 0.51 nM) and PARP-2 (IC50: 23.11 nM).Formule :C24H27FN4O3Couleur et forme :SolidMasse moléculaire :438.49Akt Inhibitor X
CAS :Akt Inhibitor X is a cell-permeable and reversible inhibitor of Akt phosphorylation.Formule :C20H25ClN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :344.88Resminostat
CAS :Resminostat (4SC-201) is an orally bioavailable inhibitor of histone deacetylases (HDACs) with potential antineoplastic activity.Formule :C16H19N3O4SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :349.4NSC-636819
CAS :NSC-636819 is a novel inhibitor of KDM4A/KDM4B.Formule :C22H12Cl4N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.15PNZ5
CAS :PNZ5, an isoxazole-based pan-BET inhibitor, demonstrates potent activity and high selectivity comparable to the established (+)-JQ1, exhibiting a dissociationFormule :C20H18N2O2Degré de pureté :99.51% - 99.61%Couleur et forme :SolidMasse moléculaire :318.37Ref: TM-T12513
1mg109,00€5mg243,00€10mg355,00€25mg532,00€50mg750,00€100mg1.009,00€200mg1.369,00€1mL*10mM (DMSO)240,00€JAK-IN-10
CAS :JAK-IN-10 is a JAK inhibitor. JAK-IN-10 can be used for the research of dry eye disorders.Formule :C20H18FN5O3SDegré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :427.45Ref: TM-T13571
1mg82,00€5mg167,00€10mg246,00€25mg405,00€50mg572,00€100mg772,00€500mg1.539,00€1mL*10mM (DMSO)178,00€SW155246
CAS :SW155246 is a potent and selective inhibitor of DNMT1 (DNA methyltransferase 1; IC50 of 1.2 μM).Formule :C16H11ClN2O5SDegré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :378.79
