Somatostatine
La somatostatine est une hormone peptidique qui inhibe la libération de plusieurs autres hormones, y compris l'hormone de croissance, l'insuline et le glucagon. Elle agit en se liant aux récepteurs de la somatostatine, qui sont des récepteurs couplés aux protéines G exprimés dans divers tissus. Les analogues de la somatostatine sont utilisés dans le traitement de l'acromégalie, des tumeurs neuroendocrines et des troubles gastro-intestinaux. Ces analogues sont également des outils précieux pour étudier la sécrétion hormonale et la signalisation. Chez CymitQuimica, nous offrons une gamme complète d'analogues de la somatostatine de haute qualité pour soutenir vos recherches en endocrinologie, régulation hormonale et développement thérapeutique.
49 produits trouvés pour "Somatostatine"
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(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS :<p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>Formule :C20H29N3O8Degré de pureté :99.72%Couleur et forme :SoildMasse moléculaire :439.46Somatostatin acetate
<p>Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.</p>Degré de pureté :99.11%Couleur et forme :Odour SolidCortistatin 14, human, rat acetate
<p>Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects and</p>Formule :C80H112N18O19S2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :1693.98Cortistatin-14 acetate
<p>Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).</p>Formule :C83H118N20O20S2Degré de pureté :98.24% - 99.63%Couleur et forme :SoildMasse moléculaire :1780.08Seglitide acetate
CAS :<p>Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.</p>Formule :C46H60N8O9Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :869.02Cyclosomatostatin Acetate
<p>Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell</p>Formule :C46H61N7O8Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :840.02Seglitide
CAS :<p>Peptide agonist targets sst2/sst5 receptors. IC50/Kd: sst1 >1000, sst2 = 0.2-1.5, sst3 = 27-36, sst4 >127, sst5 = 0.06-23 nM.</p>Formule :C44H56N8O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :808.98Ilatreotide
CAS :<p>Ilatreotide is a Amadori compound of octreotide.</p>Formule :C61H86N10O20S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1343.53CYN 154806
CAS :<p>CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).</p>Formule :C56H68N12O14S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1197.34Cortistatin 14, human, rat
CAS :<p>Cortistatin 14: a neuropeptide similar to somatostatin; induces sleep, depresses neuronal activity; found in cortex, hippocampus.</p>Formule :C81H113N19O19S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1721.01Veldoreotide
CAS :Veldoreotide (Somatoprim): a somatostatin analogue targeting receptors 2, 4, 5, reduces GH in pituitary adenomas.Formule :C60H74N12O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1123.3Somatostatin(3-6)
CAS :<p>Somatostatin(3-6) is a somatostatin fragment.</p>Formule :C22H34N6O6SCouleur et forme :SolidMasse moléculaire :510.61MMC(TMZ)-TOC TFA
<p>MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.</p>Formule :C74H99F3N20O21S2Couleur et forme :SolidMasse moléculaire :1725.82Cortistatin 29
<p>Cortistatin 29: neuropeptide, relieves neuropathic pain, binds SS receptors (IC50: 2.8-13.7 nM), anti-fibrotic.</p>Formule :C161H242N46O41S2Couleur et forme :SolidMasse moléculaire :3539.77Satoreotide
CAS :<p>Satoreotide (JR11) is an SSTR2 antagonist, typically conjugated with radiolabeled chelators for use in neuroendocrine tumor imaging [1].</p>Formule :C58H72ClN15O14S2Couleur et forme :SolidMasse moléculaire :1302.87L-796,778
CAS :<p>L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.</p>Formule :C29H40N6O7Degré de pureté :96.20%Couleur et forme :SolidMasse moléculaire :584.66BIM-23190 hydrochloride
<p>BIM-23190 hydrochloride, somatostatin analog, SSRT2/5 agonist, Ki: 0.34 nM (SSTR2), 11.1 nM (SSTR5). Used in cancer, acromegaly research.</p>Couleur et forme :LiquidDOTA-JR11
CAS :<p>DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.</p>Formule :C74H98ClN19O21S2Couleur et forme :SolidMasse moléculaire :1689.27Dotanoc
CAS :<p>Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.</p>Formule :C69H94N14O17S2Couleur et forme :SolidMasse moléculaire :1455.71Cyclic SSTR agonist octreotide
<p>Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .</p>Formule :C53H71N11O14S2Couleur et forme :SolidMasse moléculaire :1150.33Cyclosomatostatin TFA
<p>Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.</p>Formule :C46H58F3N7O8Couleur et forme :SolidMasse moléculaire :893.99L-796,778 acetate
<p>L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.</p>Formule :C31H44N6O9Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :644.72Tau conotoxin CnVA
CAS :<p>Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.</p>Formule :C72H116N24O17S4Couleur et forme :SolidMasse moléculaire :1718.1SSTR4 agonist-1
CAS :<p>SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.</p>Formule :C16H23N3O2Couleur et forme :SolidMasse moléculaire :289.37L-797,591 hydrochloride
<p>L-797,591 HCl activates SSTR1, boosts p-ERK5 with AG1478, and enhances p38 phosphorylation, reversible by AG1478.</p>Formule :C38H50ClN5O2Degré de pureté :98.65% - >99.99%Couleur et forme :SoildMasse moléculaire :644.30Somatostatin-28 (1-14)
CAS :<p>Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.</p>Formule :C61H105N23O21SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1528.71CH 275
CAS :<p>Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.</p>Formule :C74H96N14O15S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1485.8Somatostatin 1-28 acetate
<p>Somatostatin 1-28 acetate circulates in human plasma.</p>Degré de pureté :99.22%Couleur et forme :SoildSomatostatin
CAS :<p>Somatostatin: a peptide hormone inhibiting growth hormone, insulin, and glucagon; secreted by hypothalamus and pancreatic D cells.</p>Degré de pureté :98%Couleur et forme :PowderMasse moléculaire :1637.88Neuronostatin-13 (human)
CAS :<p>Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.</p>Formule :C64H110N20O16Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1415.68[D-Trp8,Tyr11] Somatostatin
CAS :[D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,Formule :C76H104N18O20S2Masse moléculaire :1653.88[Tyr11]-Somatostatin
CAS :[Tyr11]-Somatostatin, a neuroactive peptide, aids proteomics research and modulates retinal function.Formule :C76H104N18O20S2Masse moléculaire :1653.89DOTA-EB-TATE
DOTA-EB-TATE is formed by combining the SST peptide derivative DOTA-octreotate with an Evans blue analog (EB). This peptide drug conjugate (PDC) enhances the pharmacokinetics of SSTR2 analogs and reduces PRRT toxicity. Additionally, DOTA-EB-TATE serves in the synthesis/research of radiopharmaceutical conjugates (RDC).Formule :C105H133N21O30S5Masse moléculaire :2329.63Cortistatin-14
CAS :<p>Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.</p>Formule :C81H114N20O18S2Degré de pureté :98.06% - 98.23%Couleur et forme :SolidMasse moléculaire :1720.03Lanreotide
CAS :Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formule :C54H69N11O10S2Couleur et forme :SolidMasse moléculaire :1096.32Anti-Somatostatin Antibody (9L93)
<p>Anti-Somatostatin Antibody (9L93) is a Rabbit antibody targeting Somatostatin. Anti-Somatostatin Antibody (9L93) can be used in ELISA.</p>Couleur et forme :Odour LiquidBIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Formule :C59H83N13O14S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :1262.5Paltusotine
CAS :<p>Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.</p>Formule :C27H22F2N4ODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :456.49Pasireotide Acetate
CAS :<p>The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.</p>Formule :C60H70N10O11Degré de pureté :98.64% - 99.92%Couleur et forme :SolidMasse moléculaire :1107.26Octreotide Acetate
CAS :<p>Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.</p>Formule :C51H70N10O12S2Degré de pureté :99.03% - 99.87%Couleur et forme :Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidMasse moléculaire :1079.3FK962
CAS :<p>FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.</p>Formule :C14H17FN2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :264.3Somatostatin Impurity 2 (13-Dha) Trifluoroacetate
Formule :C76H102N18O18S2·C2HF3O2Masse moléculaire :1619.88 114.02CYN 154806 TFA
CAS :<p>CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.</p>Formule :C58H69F3N12O16S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :1311.36Edotreotide
CAS :<p>Edotreotide (SMT-487) is an Indicator and Reagent. It also is used in the Diagnosis and Staging of Tumors Expressing Somatostatin Receptors.</p>Formule :C65H92N14O18S2Degré de pureté :96.95%Couleur et forme :SolidMasse moléculaire :1421.64L-803087
CAS :<p>L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.</p>Formule :C25H29F2N5O3Degré de pureté :97.58%Couleur et forme :SolidMasse moléculaire :485.53L-796778 acetate
CAS :<p>L-796778 acetate is a selective sst3 receptor agonist. In CHO-K1 cells expressing hsst3 receptors, it acts as a partial agonist that inhibits Forskolin-induced cAMP production, with an IC50 value of 18 nM. Additionally, L-796778 acetate exhibits anticonvulsant properties.</p>Formule :C31H44N6O9Couleur et forme :SolidMasse moléculaire :644.716SSTR5 antagonist 6
CAS :<p>SSTR5 antagonist 6, an orally active antagonist specific to the somatostatin receptor subtype 5 (SSTR5), exhibits an IC50 value of 24 nM. This compound is utilized in researching type 2 diabetes [1].</p>Formule :C22H28ClN3O4Couleur et forme :SolidMasse moléculaire :433.93
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