Somatostatine
La somatostatine est une hormone peptidique qui inhibe la libération de plusieurs autres hormones, y compris l'hormone de croissance, l'insuline et le glucagon. Elle agit en se liant aux récepteurs de la somatostatine, qui sont des récepteurs couplés aux protéines G exprimés dans divers tissus. Les analogues de la somatostatine sont utilisés dans le traitement de l'acromégalie, des tumeurs neuroendocrines et des troubles gastro-intestinaux. Ces analogues sont également des outils précieux pour étudier la sécrétion hormonale et la signalisation. Chez CymitQuimica, nous offrons une gamme complète d'analogues de la somatostatine de haute qualité pour soutenir vos recherches en endocrinologie, régulation hormonale et développement thérapeutique.
61 produits trouvés pour "Somatostatine".
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L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Formule :C31H44N6O9Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :644.72Tau conotoxin CnVA
CAS :Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Formule :C72H116N24O17S4Couleur et forme :SolidMasse moléculaire :1718.1L-797,591 hydrochloride
L-797,591 HCl activates SSTR1, boosts p-ERK5 with AG1478, and enhances p38 phosphorylation, reversible by AG1478.Formule :C38H50ClN5O2Degré de pureté :98.65% - >99.99%Couleur et forme :White SolidMasse moléculaire :644.30Anti-Somatostatin Antibody (9L93)
Anti-Somatostatin Antibody (9L93) is a Rabbit antibody targeting Somatostatin. Anti-Somatostatin Antibody (9L93) can be used in ELISA.Couleur et forme :Odour LiquidLanreotide
CAS :Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formule :C54H69N11O10S2Couleur et forme :SolidMasse moléculaire :1096.32CYN 154806 TFA
CAS :CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.Formule :C58H69F3N12O16S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :1311.36Edotreotide
CAS :Edotreotide (SMT-487) is an Indicator and Reagent. It also is used in the Diagnosis and Staging of Tumors Expressing Somatostatin Receptors.Formule :C65H92N14O18S2Degré de pureté :96.95%Couleur et forme :White SolidMasse moléculaire :1421.64Octreotide Acetate
CAS :Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formule :C51H70N10O12S2Degré de pureté :99.03% - 99.87%Couleur et forme :White SolidMasse moléculaire :1079.30Paltusotine
CAS :Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Formule :C27H22F2N4ODegré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :456.49Pasireotide Acetate
CAS :The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.Formule :C60H70N10O11Degré de pureté :98.64% - 99.92%Couleur et forme :SolidMasse moléculaire :1107.26Ref: TM-TP2207
1mg90,00€2mg138,00€5mg236,00€10mg409,00€25mg745,00€50mg1.189,00€100mg1.684,00€200mg2.268,00€Somatostatin Impurity 2 (13-Dha) Trifluoroacetate
Formule :C76H102N18O18S2·C2HF3O2Masse moléculaire :1619.88 114.02BIM-23190 aceate
BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.Formule :C59H83N13O14S2Degré de pureté :99.31%Couleur et forme :White SolidMasse moléculaire :1262.5FK962
CAS :FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Formule :C14H17FN2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :264.3Ref: TM-T7829
2mg34,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg82,00€25mg144,00€50mg200,00€100mg278,00€200mg389,00€L-803087
CAS :L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.Formule :C25H29F2N5O3Degré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :485.53Ref: TM-T11800
1mg50,00€5mg112,00€1mL*10mM (DMSO)126,00€10mg175,00€25mg366,00€50mg585,00€100mg928,00€200mg1.234,00€SSTR4 agonist 5
CAS :SSTR4 agonist5 (Compound 5) is an orally active agonist of the somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. It demonstrates good stability in human/rat liver microsomes and can inhibit mechanical hyperalgesia in rat models.Formule :C20H26N4OMasse moléculaire :338.447SST1 receptor antagonist-1
CAS :SST1 receptor antagonist-1 (Compound 23) is a selective antagonist of the somatostatin receptor 1 (SST1), showing a pKd of 9.11 for rSST1 and 8.79 for hSST1. This compound is applicable in research related to retinal and endocrine dysfunction, cancer, and neuropsychiatric disorders.Formule :C29H31F2N3O2Couleur et forme :SolidMasse moléculaire :491.57L-796778 acetate
CAS :L-796778 acetate is a selective sst3 receptor agonist. In CHO-K1 cells expressing hsst3 receptors, it acts as a partial agonist that inhibits Forskolin-induced cAMP production, with an IC50 value of 18 nM. Additionally, L-796778 acetate exhibits anticonvulsant properties.Formule :C31H44N6O9Couleur et forme :SolidMasse moléculaire :644.716SSTR5 antagonist 6
CAS :SSTR5 antagonist 6, an orally active antagonist specific to the somatostatin receptor subtype 5 (SSTR5), exhibits an IC50 value of 24 nM. This compound is utilized in researching type 2 diabetes [1].Formule :C22H28ClN3O4Couleur et forme :SolidMasse moléculaire :433.93
