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ATPase

ATPase

Les ATPases sont des enzymes qui catalysent la décomposition de l'ATP en ADP et un ion phosphate libre, une réaction qui libère de l'énergie utilisée pour conduire de nombreux processus au sein de la cellule, y compris le transport actif à travers les membranes. Les ATPases jouent un rôle crucial dans le maintien de l'homéostasie cellulaire, de l'équilibre du pH et des gradients ioniques. Les dysfonctionnements de l'activité des ATPases sont associés à des maladies telles que l'insuffisance cardiaque, l'hypertension et la neurodégénérescence. Chez CymitQuimica, nous fournissons des inhibiteurs et des modulateurs d'ATPase de haute qualité pour soutenir vos recherches en énergétique cellulaire, transport membranaire et pathologie des maladies.

98 produits trouvés pour "ATPase"

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  • Permethrin

    CAS :
    Permethrin (NRDC-143) is a pyrethroid insecticide commonly used in the treatment of LICE INFESTATIONS and SCABIES.
    Formule :C21H20Cl2O3
    Degré de pureté :99.37% - 99.54%
    Couleur et forme :Colorless Crystals To A Viscous Liquid; Color White To Pale Yellow Permethrin Is A Pale Brown Liquid Relatively Water Insoluble Used As An Insecticide
    Masse moléculaire :391.29

    Ref: TM-T1332

    100mg
    33,00€
    1mL*10mM (DMSO)
    34,00€
    500mg
    72,00€
  • Fenbufen

    CAS :
    Fenbufen (Lederfen) is a non-steroidal anti-inflammatory drug used primarily to treat inflammation in osteoarthritis, ankylosing spondylitis, and tendinitis.
    Formule :C16H14O3
    Degré de pureté :98.35% - 98.46%
    Couleur et forme :White Solid
    Masse moléculaire :254.28

    Ref: TM-T0859

    200mg
    34,00€
    500mg
    46,00€
    1g
    54,00€
  • Trichlormethiazide

    CAS :
    Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.
    Formule :C8H8Cl3N3O4S2
    Degré de pureté :98.8% - 99.54%
    Couleur et forme :Solid
    Masse moléculaire :380.66

    Ref: TM-T0114

    1g
    37,00€
    2g
    50,00€
    1mL*10mM (DMSO)
    52,00€
  • Prilocaine hydrochloride

    CAS :
    Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.
    Formule :C13H21ClN2O
    Degré de pureté :99.97%
    Couleur et forme :Needles White Or Off White Crystalline Powder
    Masse moléculaire :256.77

    Ref: TM-T0796

    100mg
    34,00€
    1mL*10mM (DMSO)
    34,00€
    500mg
    71,00€
    1g
    92,00€
  • ATP synthase inhibitor 1

    CAS :
    ATP synthase inhibitor 1 is an inhibitor of the c subunit of the F1/FO-ATP synthase complex.
    Formule :C17H18ClN3O3S2
    Degré de pureté :99.83%
    Couleur et forme :Solid
    Masse moléculaire :411.93

    Ref: TM-T10404

    1mg
    56,00€
    5mg
    119,00€
    10mg
    192,00€
    25mg
    383,00€
    50mg
    565,00€
    100mg
    807,00€
  • Suloctidil

    CAS :
    Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.
    Formule :C20H35NOS
    Degré de pureté :99.75% - >99.99%
    Couleur et forme :Solid
    Masse moléculaire :337.56

    Ref: TM-T0712

    5mg
    34,00€
    1mL*10mM (DMSO)
    48,00€
    10mg
    49,00€
    25mg
    73,00€
  • Ciliobrevin D

    CAS :
    Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.
    Formule :C17H8Cl3N3O2
    Degré de pureté :98.09%
    Couleur et forme :Solid
    Masse moléculaire :392.62

    Ref: TM-T14965

    1mg
    60,00€
    2mg
    87,00€
    5mg
    133,00€
    1mL*10mM (DMSO)
    148,00€
    10mg
    203,00€
    25mg
    401,00€
    50mg
    592,00€
    100mg
    827,00€
  • Tolbutamide

    CAS :
    Tolbutamide (HLS 831) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.
    Formule :C12H18N2O3S
    Degré de pureté :99.80% - 99.93%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :270.35

    Ref: TM-T1054

    500mg
    46,00€
    1mL*10mM (DMSO)
    50,00€
    1g
    62,00€
  • Gboxin

    CAS :
    Gboxin is an inhibitor of oxidative phosphorylation that targets glioblastoma,inhibits the activity of F0F1 ATP synthase, with antitumour activity.
    Formule :C22H33ClN2O2
    Degré de pureté :99.96% - >99.99%
    Couleur et forme :Solid
    Masse moléculaire :392.96

    Ref: TM-T15373

    1mg
    42,00€
    2mg
    55,00€
    1mL*10mM (DMSO)
    87,00€
    5mg
    88,00€
    10mg
    126,00€
    25mg
    245,00€
    50mg
    385,00€
    100mg
    612,00€
    200mg
    850,00€
  • Diazoxide

    CAS :
    Diazoxide (Proglycem) is a benzothiadiazine derivative that is a peripheral vasodilator used for hypertensive emergencies.
    Formule :C8H7ClN2O2S
    Degré de pureté :99% - 99.83%
    Couleur et forme :Solid
    Masse moléculaire :230.67

    Ref: TM-T0126

    25mg
    34,00€
    50mg
    42,00€
    100mg
    52,00€
    1mL*10mM (DMSO)
    52,00€
    500mg
    105,00€
    1g
    152,00€
  • Cyclocreatine

    CAS :
    Cyclocreatine, a creatine analogue and substrate for creatine kinase, inhibits creatine metabolism and prostate cancer cell proliferation.
    Formule :C5H9N3O2
    Degré de pureté :99.864%
    Couleur et forme :Solid
    Masse moléculaire :143.14

    Ref: TM-T40445

    50mg
    37,00€
    100mg
    49,00€
    500mg
    92,00€
    1g
    134,00€
  • 3'-Deoxy-3'-amino-ATP

    CAS :
    3'-Deoxy-3'-amino-ATP is a competitive ATP inhibitor with a 2.3 μM Ki, used to synthesize tRNA.
    Formule :C10H17N6O12P3
    Couleur et forme :Solid
    Masse moléculaire :506.197

    Ref: TM-T40522

    5mg
    873,00€
  • (S)-PF-03716556

    CAS :
    (S)-PF-03716556 can be used as an acid pump inhibitor for the treatment of disease conditions mediated by acid pump inhibitory activity.
    Formule :C22H26N4O3
    Degré de pureté :99.75% - 99.91%
    Couleur et forme :Soild
    Masse moléculaire :394.47

    Ref: TM-T2093L

    1mg
    109,00€
    5mg
    233,00€
    10mg
    344,00€
    25mg
    532,00€
    50mg
    735,00€
    100mg
    982,00€
    200mg
    1.333,00€
  • (±)16-HETE

    CAS :
    Electrolyte and fluid transport in the kidney are regulated in part by arachidonic acid and its metabolites.
    Formule :C20H32O3
    Couleur et forme :Solid
    Masse moléculaire :320.473

    Ref: TM-T35465

    25µg
    329,00€
    50µg
    625,00€
    100µg
    1.179,00€
  • (±)17-HETE

    CAS :
    Electrolyte and fluid transport in the kidney are regulated in part by arachidonic acid and its metabolites.
    Formule :C20H32O3
    Couleur et forme :Solid
    Masse moléculaire :320.473

    Ref: TM-T35523

    25µg
    477,00€
    50µg
    888,00€
    100µg
    1.701,00€
  • SC 4453

    CAS :
    SC 4453 is a digoxin analog and a cardiac glycoside derivative.
    Formule :C41H64N2O12
    Couleur et forme :Solid
    Masse moléculaire :776.965

    Ref: TM-T34554

    25mg
    À demander
    50mg
    À demander
    100mg
    À demander
  • ATP Synthesis-IN-1


    ATP Synthesis-IN-1 (Compound 4), a quinoline derivative, potently inhibits PA ATP synthesis with an IC50 of 11.1μg/mL and exhibits antibacterial properties.
    Couleur et forme :Odour Solid

    Ref: TM-T82945

    5mg
    À demander
    50mg
    À demander
  • Digoxigenin Monodigitoxoside

    CAS :
    Digoxigenin monodigitoxoside is a cardiac glycoside metabolite of digoxin and a Na+/K+ ATPase inhibitor.
    Formule :C29H44O8
    Couleur et forme :Solid
    Masse moléculaire :520.663

    Ref: TM-T36060

    1mg
    767,00€
  • PK095

    CAS :

    PK095 is a proprietary compound in the guanidine - based F1F0-ATPase inhibitor family.

    Formule :C20H18N4O2S
    Degré de pureté :96.84%
    Couleur et forme :Soild
    Masse moléculaire :378.45

    Ref: TM-T67763

    1mg
    67,00€
    5mg
    143,00€
    10mg
    197,00€
    25mg
    314,00€
    50mg
    434,00€
    100mg
    587,00€
    200mg
    785,00€
  • Prilocaine acetate


    Prilocaine acetate, an amino amide compound, functions as a Na/K-ATPase inhibitor, exhibiting neurotoxic effects [1] [2].
    Formule :C15H24N2O3
    Couleur et forme :Solid
    Masse moléculaire :280.36

    Ref: TM-T75280

    5mg
    À demander
    50mg
    À demander
  • 17(S)-HETE

    CAS :
    17(S)-HETE is an arachidonic acid metabolite generated via the CYP450 pathway. 17(S)-HETE acts as an allosteric activator of CYP450 1B1 and an ATPase inhibitor.
    Formule :C20H32O3
    Couleur et forme :Solid
    Masse moléculaire :320.47

    Ref: TM-T35849

    25µg
    477,00€
    50µg
    888,00€
    100µg
    1.701,00€
  • A 80915A

    CAS :
    A80915A: Semi-naphthoquinone antibiotic, blocks gastric (H(+)-K+)-ATPase; potency varies with enzyme conformation; K+ reduces binding rate.
    Formule :C26H31Cl3O5
    Couleur et forme :Solid
    Masse moléculaire :529.88

    Ref: TM-T26450

    25mg
    À demander
    50mg
    À demander
    100mg
    À demander
  • BMS 199264

    CAS :
    BMS 199264 hydrochlorid a inhibitor of mitochondrial F1F0 ATP hydrolase, thus preventing ATP reduction to ameliorate cardiac necrosis during ischemia.
    Formule :C26H31ClN4O4S
    Degré de pureté :99.83%
    Couleur et forme :Soild
    Masse moléculaire :531.07

    Ref: TM-T26843L

    5mg
    2.288,00€
  • Transdermal Peptide Disulfide

    CAS :
    TD 1 peptide, an 11-amino acid, binds ATP1B1's C-terminus, enhancing transdermal drug delivery.
    Formule :C40H64N14O16S2
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :1061.15

    Ref: TM-TP1033

    1mg
    65,00€
    5mg
    138,00€
    10mg
    207,00€
  • Ouabagenin

    CAS :
    Ouabagenin, a naturally occurring LXR ligand with selective agonist activity, functions as an EC 3.6.3.9 (Na(+)/K(+)-transport ATPase) inhibitor [1] [2].
    Formule :C23H34O8
    Couleur et forme :Solid
    Masse moléculaire :438.51

    Ref: TM-TN7752

    10mg
    À demander
    50mg
    À demander
  • Chlorpropylate

    CAS :
    Chlorpropylate is an insecticide.
    Formule :C17H16Cl2O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :339.21

    Ref: TM-T27010

    25mg
    À demander
    50mg
    À demander
    100mg
    À demander
  • NSC799462


    NSC799462, a triazole inhibitor, specifically targets p97 ATPase, exerting its effect by binding to a designated site on the p97 enzyme. This interaction induces localized structural alterations in p97, effectively inhibiting its ATPase activity with an IC 50 value of 15 nM.
    Formule :C30H32F2N6O3S
    Couleur et forme :Solid
    Masse moléculaire :594.68

    Ref: TM-T200146

    10mg
    À demander
    50mg
    À demander
  • S-WJM992


    S-WJM992 (compound 10ahb) serves as an antiparasitic agent, effectively inhibiting ATPase activity in high [Na+] environments. It also significantly counteracts parasites resistant to PfATP4 inhibitors. Additionally, S-WJM992 acts as a potential transmission blocker by impeding gamete development and halting the transmission of parasites to mosquitoes during blood feeding.
    Formule :C22H18ClFN6O3
    Couleur et forme :Solid
    Masse moléculaire :468.87

    Ref: TM-T200205

    10mg
    À demander
    50mg
    À demander
  • 14-Anhydrodigitoxigenin

    CAS :
    14-Anhydrodigitoxigenin, a digitoxin derivative, inhibits guinea pig heart Na+/K+-ATPase by 15% at 10 μM concentration.
    Formule :C23H32O3
    Couleur et forme :Solid
    Masse moléculaire :356.506

    Ref: TM-T37707

    5mg
    178,00€
    10mg
    349,00€
    25mg
    717,00€
    50mg
    1.288,00€
  • Flavopereirine

    CAS :
    Flavopereirine is a beta-carboline alkaloid.
    Formule :C17H15N2
    Couleur et forme :Solid
    Masse moléculaire :247.31

    Ref: TM-T31799

    25mg
    1.369,00€
  • Lnd 623

    CAS :
    Lnd 623 is an inotropic aminosteroid.
    Formule :C27H47NO6
    Couleur et forme :Solid
    Masse moléculaire :481.674

    Ref: TM-T32829

    25mg
    1.369,00€
  • NSC819701


    NSC819701 is a triazole-based inhibitor of p97ATPase. It inhibits the activity of p97ATPase by binding to specific sites on p97.
    Formule :C30H32F2N8O3S
    Couleur et forme :Solid
    Masse moléculaire :622.69

    Ref: TM-T89915

    10mg
    À demander
    50mg
    À demander
  • Luciferase, firefly

    CAS :
    Luciferase, firefly is a reporter gene in cellular imaging studies to quantify target gene expression levels and measure intracellular ATP content,
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :N/A

    Ref: TM-TP1774

    1mg
    339,00€
    5mg
    854,00€
    10mg
    1.170,00€
  • 5-Hydroxydecanoic acid

    CAS :
    5-Hydroxydecanoic acid is a selective ATP-sensitive K+ (KATP) channel blocker (IC50 of ~30 μM). 5-Hydroxydecanoic acid is a substrate for mitochondrial outer membrane acyl-CoA synthetase and has antioxidant activity.
    Formule :C10H20O3
    Degré de pureté :99.24%
    Couleur et forme :Solid
    Masse moléculaire :188.26

    Ref: TM-T29457

    100mg
    À demander
    200mg
    À demander
    10mg
    91,00€
    1mL*10mM (DMSO)
    100,00€
    25mg
    159,00€
    50mg
    223,00€
  • (+)-SJ733

    CAS :
    (+)-SJ733 (SJ000557733) is a potent Na+-ATPase PfATP4 inhibitor with antimalarial activity for the study of malaria.
    Formule :C24H16F4N4O2
    Degré de pureté :99.21%
    Couleur et forme :Solid
    Masse moléculaire :468.4

    Ref: TM-T17313

    1mg
    180,00€
  • 1-N-Methyl-4-mercaptohistidine disulfide

    CAS :
    1-N-Methyl-4-mercaptohistidine disulfide is a Duchenne chloroplast coupling factor 1 redox modulator that inhibits light-triggered CF1 ATPase activity.
    Formule :C14H20N6O4S2
    Degré de pureté :97.67% - ≥98%
    Couleur et forme :Soild
    Masse moléculaire :400.48

    Ref: TM-T83633

    50mg
    À demander
    1mg
    989,00€
    5mg
    1.324,00€
  • Anti-ATP7B Antibody (7M703)


    Anti-ATP7B Antibody (7M703) is an antibody targeting ATP7B. Anti-ATP7B Antibody (7M703) can be used in ELISA, IF, FCM.
    Couleur et forme :Odour Liquid

    Ref: TM-TMAH-00095

    50µl
    202,00€
    100µl
    339,00€
  • L-Palmitoylcarnitine

    CAS :
    L-Palmitoylcarnitine (L-PC) inhibits Na/K ATPase activity and potentiates fibrinolytic enzymes and tPA to inhibit thrombosis.
    Formule :C23H45NO4
    Degré de pureté :97% - 99.81%
    Couleur et forme :Solid
    Masse moléculaire :399.61

    Ref: TM-T15698

    1mg
    99,00€
    5mg
    289,00€
    10mg
    432,00€
    25mg
    692,00€
    50mg
    945,00€
  • Anti-ATP7B Antibody (4W208)


    Anti-ATP7B Antibody (4W208) is an antibody targeting ATP7B. Anti-ATP7B Antibody (4W208) can be used in ELISA, IHC, IF, FCM.
    Couleur et forme :Odour Liquid

    Ref: TM-TMAH-00094

    50µl
    203,00€
    100µl
    341,00€
  • Blebbistatin

    CAS :
    Blebbistatin ((±)-Blebbistatin) is a non-muscle myosin II (NMII)-selective and non-muscle myosin heavy chain 9 (MYH9)-specific inhibitor.Cost-effective and quality-assured.
    Formule :C18H16N2O2
    Degré de pureté :99.88% - 99.97%
    Couleur et forme :Bright Yellow Solid
    Masse moléculaire :292.33

    Ref: TM-T21550

    1mg
    34,00€
    2mg
    49,00€
    5mg
    73,00€
    1mL*10mM (DMSO)
    81,00€
    10mg
    124,00€
    25mg
    203,00€
    50mg
    358,00€
    100mg
    538,00€
  • Apoptozole

    CAS :
    Apoptozole (Apoptosis Activator VII) is an inhibitor of the ATPase domain of Hsc70 and Hsp70, and can induce apoptosis.
    Formule :C33H25F6N3O3
    Degré de pureté :99.75%
    Couleur et forme :Solid
    Masse moléculaire :625.56

    Ref: TM-T3293

    2mg
    34,00€
    5mg
    48,00€
    1mL*10mM (DMSO)
    63,00€
    10mg
    79,00€
    25mg
    130,00€
    50mg
    222,00€
    100mg
    331,00€
    200mg
    489,00€
  • Rabeprazole Sulfide

    CAS :
    Rabeprazole Sulfide (Rabeprazole Related Compound E) is an antiulcer drug in the class of proton pump inhibitors.
    Formule :C18H21N3O2S
    Degré de pureté :99.34% - 99.78%
    Couleur et forme :Off-White Crystalline Powder
    Masse moléculaire :343.44

    Ref: TM-T1734

    1mL*10mM (DMSO)
    33,00€
    200mg
    34,00€
    500mg
    49,00€
    1g
    63,00€
  • Esomeprazole Magnesium

    CAS :
    Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.
    Formule :C34H36MgN6O6S2
    Degré de pureté :98.76% - 99.73%
    Couleur et forme :Solid
    Masse moléculaire :713.12

    Ref: TM-T2686

    1mL*10mM (DMSO)
    34,00€
    100mg
    42,00€
    500mg
    92,00€
    1g
    120,00€
  • Rbin-1

    CAS :
    Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.
    Formule :C13H12N4S
    Degré de pureté :99.83%
    Couleur et forme :Solid
    Masse moléculaire :256.33

    Ref: TM-T7411

    5mg
    66,00€
    1mL*10mM (DMSO)
    73,00€
    10mg
    90,00€
    25mg
    205,00€
    50mg
    356,00€
    100mg
    530,00€
  • Omecamtiv mecarbil

    CAS :
    Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic
    Formule :C20H24FN5O3
    Degré de pureté :98% - 99.23%
    Couleur et forme :Solid
    Masse moléculaire :401.43

    Ref: TM-T2006

    1mg
    38,00€
    2mg
    50,00€
    1mL*10mM (DMSO)
    71,00€
    5mg
    80,00€
    10mg
    117,00€
    25mg
    187,00€
    50mg
    333,00€
    100mg
    495,00€
  • Chloroprocaine hydrochloride

    CAS :
    Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.
    Formule :C13H20Cl2N2O2
    Degré de pureté :99.65%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :307.22

    Ref: TM-T6443

    1mL*10mM (DMSO)
    33,00€
    10mg
    39,00€
    25mg
    64,00€
    50mg
    88,00€
    100mg
    133,00€
  • NPD8733

    CAS :

    NPD8733 is an inhibitor of cancer cell-enhanced fibroblast migration. It specifically binds to valosin-containing protein (VCP)/p97.

    Formule :C18H15NO4
    Degré de pureté :98.48%
    Couleur et forme :Solid
    Masse moléculaire :309.32

    Ref: TM-T9008

    1mg
    42,00€
    5mg
    87,00€
    10mg
    125,00€
    25mg
    245,00€
    50mg
    399,00€
    100mg
    645,00€
    200mg
    898,00€
  • DHQ

    CAS :
    DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.
    Formule :C8H6N2O2
    Degré de pureté :99.89%
    Couleur et forme :Solid
    Masse moléculaire :162.15

    Ref: TM-T20436

    1mL*10mM (DMSO)
    33,00€
    100mg
    46,00€
    500mg
    103,00€
    1g
    148,00€
  • Rabeprazole sodium

    CAS :
    Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.
    Formule :C18H20N3NaO3S
    Degré de pureté :98% - 99.91%
    Couleur et forme :White Or Off White Crystalline Powder
    Masse moléculaire :381.42

    Ref: TM-T1651

    1mL*10mM (DMSO)
    33,00€
    10mg
    39,00€
    25mg
    63,00€
    50mg
    90,00€
    100mg
    114,00€
    200mg
    167,00€
  • Transdermal Peptide Disulfide Acetate


    Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly
    Formule :C42H68N14O18S2
    Degré de pureté :99.97%
    Couleur et forme :Solid
    Masse moléculaire :1121.2

    Ref: TM-TP1033L

    1mg
    81,00€
    5mg
    159,00€
    10mg
    236,00€
    25mg
    427,00€
    50mg
    625,00€
    100mg
    889,00€
    500mg
    1.783,00€
  • Rostafuroxin

    CAS :
    Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.
    Formule :C23H34O4
    Degré de pureté :98.24% - >99.99%
    Couleur et forme :Solid
    Masse moléculaire :374.51

    Ref: TM-T2621

    2mg
    46,00€
    5mg
    66,00€
    1mL*10mM (DMSO)
    73,00€
    10mg
    106,00€
    25mg
    208,00€
    50mg
    354,00€
    100mg
    588,00€
  • Prilocaine

    CAS :
    Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of
    Formule :C13H20N2O
    Degré de pureté :98.49%
    Couleur et forme :Needles Solid
    Masse moléculaire :220.31

    Ref: TM-T6953

    25mg
    34,00€
    50mg
    46,00€
    1mL*10mM (DMSO)
    49,00€
    100mg
    66,00€
    200mg
    96,00€
    500mg
    144,00€
  • Tenatoprazole

    CAS :
    Tenatoprazole (TU-199), a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM).
    Formule :C16H18N4O3S
    Degré de pureté :99.57%
    Couleur et forme :White Crystalline Powder
    Masse moléculaire :346.4

    Ref: TM-T6700

    5mg
    34,00€
    1mL*10mM (DMSO)
    35,00€
    10mg
    50,00€
    25mg
    65,00€
    50mg
    80,00€
    100mg
    92,00€
    500mg
    221,00€
  • CB-5083

    CAS :
    CB-5083 is a potent, selective, and orally bioavailable p97 AAA ATPase inhibitor ( IC50=11 nM).
    Formule :C24H23N5O2
    Degré de pureté :95.95% - 99.92%
    Couleur et forme :Solid
    Masse moléculaire :413.47

    Ref: TM-T6796

    1mg
    43,00€
    2mg
    56,00€
    1mL*10mM (DMSO)
    92,00€
    5mg
    93,00€
    10mg
    130,00€
    25mg
    281,00€
    50mg
    444,00€
    100mg
    650,00€
    500mg
    1.369,00€
  • D-α-Hydroxyglutaric acid disodium

    CAS :
    D-α-Hydroxyglutaric acid disodium (Disodium (R)-2-Hydroxyglutarate) is a competitive inhibitor of α-ketoglutarate-dependent dioxygenases with Ki of 0.628 mM.
    Formule :C5H6Na2O5
    Degré de pureté :97.16%
    Couleur et forme :Solid
    Masse moléculaire :192.08

    Ref: TM-T6820

    5mg
    34,00€
    10mg
    49,00€
    25mg
    70,00€
    50mg
    104,00€
    100mg
    177,00€
    200mg
    264,00€
    500mg
    442,00€
  • FCCP

    CAS :
    FCCP (Trifluoromethoxy carbonylcyanide phenylhydrazone) is an oxidative phosphorylation (OXPHOS) inhibitor and mitochondrial proton carrier uncoupler.
    Formule :C10H5F3N4O
    Degré de pureté :98% - 99.65%
    Couleur et forme :White Solid
    Masse moléculaire :254.17

    Ref: TM-T6834

    5mg
    35,00€
    10mg
    52,00€
    1mL*10mM (DMSO)
    52,00€
    25mg
    86,00€
    50mg
    140,00€
    100mg
    253,00€
  • Tegoprazan

    CAS :
    Tegoprazan is an orally active, highly selective gastric H+/K+-ATPase inhibitor.Cost-effective and quality-assured.
    Formule :C20H19F2N3O3
    Degré de pureté :98.22%
    Couleur et forme :Solid
    Masse moléculaire :387.38

    Ref: TM-T17030

    1mg
    50,00€
    5mg
    114,00€
    1mL*10mM (DMSO)
    126,00€
    10mg
    170,00€
    25mg
    281,00€
    50mg
    371,00€
    100mg
    485,00€
    200mg
    690,00€
  • Eniporide

    CAS :
    Eniporide is a Na(+)/H(+) exchange inhibitor.
    Formule :C14H16N4O3S
    Degré de pureté :96.78% - 99.26%
    Couleur et forme :Solid
    Masse moléculaire :320.37

    Ref: TM-T2089

    1mg
    34,00€
    5mg
    73,00€
    1mL*10mM (DMSO)
    84,00€
    10mg
    113,00€
    25mg
    187,00€
    50mg
    279,00€
    100mg
    404,00€
    200mg
    570,00€
  • (-)-Blebbistatin

    CAS :
    (-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.
    Formule :C18H16N2O2
    Degré de pureté :99.38% - 99.61%
    Couleur et forme :Solid
    Masse moléculaire :292.33

    Ref: TM-T6038

    2mg
    39,00€
    5mg
    59,00€
    10mg
    90,00€
    25mg
    170,00€
    50mg
    268,00€
    100mg
    430,00€
  • BTS

    CAS :
    BTS (N-Tosylbenzylamine) is a potent inhibitor of Ca2+-stimulated myosin S1 ATPase (IC50 : 5 μM) .
    Formule :C14H15NO2S
    Degré de pureté :99.45%
    Couleur et forme :White Crystalline Solid
    Masse moléculaire :261.34

    Ref: TM-T7144

    1g
    33,00€
    1mL*10mM (DMSO)
    33,00€
  • Parimifasor

    CAS :
    Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.
    Formule :C18H11Cl2F4N5O
    Degré de pureté :96.77% - 98.97%
    Couleur et forme :Solid
    Masse moléculaire :460.21

    Ref: TM-T4640

    1mg
    46,00€
    2mg
    59,00€
    5mg
    90,00€
    1mL*10mM (DMSO)
    90,00€
    10mg
    137,00€
    25mg
    268,00€
    50mg
    394,00€
    100mg
    582,00€
  • Chloroprocaine

    CAS :
    Chloroprocaine: Na,K-ATPase inhibitor, IC50=13 mM, local anesthetic.
    Formule :C13H19ClN2O2
    Couleur et forme :Solid
    Masse moléculaire :270.76

    Ref: TM-T60469

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Mitiglinide Calcium

    CAS :
    Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-
    Formule :(C19H24NO3)2·Ca
    Degré de pureté :99.83%
    Couleur et forme :White Crystal Posder
    Masse moléculaire :668.88

    Ref: TM-T6587

    200mg
    46,00€
  • BTB06584

    CAS :
    BTB06584: IF1-dependent F1 Fo-ATPase inhibitor; novel AHAS inhibitor targeting MTB.
    Formule :C19H12ClNO6S
    Degré de pureté :97.63% - ≥95%
    Couleur et forme :Solid
    Masse moléculaire :417.82

    Ref: TM-T1940

    2mg
    34,00€
    5mg
    50,00€
    1mL*10mM (DMSO)
    56,00€
    10mg
    70,00€
    25mg
    92,00€
    50mg
    116,00€
    100mg
    202,00€
    200mg
    314,00€
  • NSC 617145

    CAS :
    NSC 617145 (NSC617145) is an inhibitor of WRN helicase that inhibits the ATPase, but not exonuclease, activity of WRN helicase in a concentration-dependent
    Formule :C13H10Cl4N2O4
    Degré de pureté :99.78%
    Couleur et forme :Solid
    Masse moléculaire :400.04

    Ref: TM-T9168

    1mg
    34,00€
    2mg
    49,00€
    5mg
    73,00€
    1mL*10mM (DMSO)
    80,00€
    10mg
    90,00€
    25mg
    164,00€
    50mg
    227,00€
    100mg
    358,00€
    500mg
    842,00€
  • KM 91104

    CAS :
    KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.
    Formule :C14H12N2O4
    Degré de pureté :99.04%
    Couleur et forme :Solid
    Masse moléculaire :272.26

    Ref: TM-T9230

    1mg
    84,00€
    5mg
    160,00€
    1mL*10mM (DMSO)
    221,00€
    10mg
    245,00€
    25mg
    494,00€
    50mg
    713,00€
    100mg
    982,00€
    500mg
    1.998,00€
  • Tirofiban hydrochloride monohydrate

    CAS :
    Tirofiban(MK383) hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.
    Formule :C22H39ClN2O6S
    Degré de pureté :98.81% - >99.99%
    Couleur et forme :White Solid
    Masse moléculaire :495.07

    Ref: TM-T2537

    5mg
    46,00€
    10mg
    66,00€
    25mg
    112,00€
    50mg
    177,00€
    100mg
    294,00€
    500mg
    702,00€
  • PF 03716556

    CAS :
    PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal reflux
    Formule :C22H26N4O3
    Degré de pureté :99.79% - 99.95%
    Couleur et forme :Solid
    Masse moléculaire :394.47

    Ref: TM-T2093

    2mg
    39,00€
    5mg
    57,00€
    10mg
    92,00€
    25mg
    165,00€
    50mg
    304,00€
    100mg
    479,00€
  • trans-Permethrin-d6 (dimethyl-d6)

    CAS :
    trans-Permethrin-d6 (dimethyl-d6) is a deuterated compound of trans-Permethrin. trans-Permethrin has a CAS number of 551877-74-8.
    Formule :C21H14D6Cl2O3
    Couleur et forme :Solid
    Masse moléculaire :397.33

    Ref: TM-TMIJ-0462

    1mg
    À demander
    5mg
    À demander
  • Tetradifon

    CAS :
    Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.
    Formule :C12H6Cl4O2S
    Degré de pureté :99.84%
    Couleur et forme :Yellowish Odorless Oil
    Masse moléculaire :356.05

    Ref: TM-T20559

    25mg
    36,00€
  • SKF-97574 HCl

    CAS :
    SKF-97574 is proton pump inhibitor.
    Formule :C22H25ClN2O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :400.9

    Ref: TM-T28794

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • FSBA hydrochloride

    CAS :
    FSBA hydrochloride(5'-p-Fluorosulfonylbenzoyladenosine) is an ATP analogue serving as an affinity probe for the ATP site of Na/K-ATPase.
    Formule :C17H17ClFN5O7S
    Degré de pureté :97.96%
    Couleur et forme :Solid
    Masse moléculaire :489.86

    Ref: TM-T27391

    1mg
    92,00€
    5mg
    226,00€
    10mg
    356,00€
    25mg
    597,00€
  • Istaroxime

    CAS :
    Istaroxime is an effective inhibitor of Na+, K+-ATPase (IC50: 0.11 μM).
    Formule :C21H32N2O3
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :360.49

    Ref: TM-T15600

    25mg
    2.178,00€
    50mg
    2.862,00€
    100mg
    3.870,00€
  • Istaroxime oxalate

    CAS :
    Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.
    Formule :C23H34N2O7
    Couleur et forme :Solid
    Masse moléculaire :450.53

    Ref: TM-T69975

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FCPT

    CAS :
    FCPT is an ATP competitive kinesin-5 inhibitor.
    Formule :C17H13FN2S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :296.36

    Ref: TM-T25409

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • RS 029

    CAS :
    RS 029 is a nitroimidazole that has been exhibited to significantly inhibit (Na+K+) ATP-ase activity.
    Formule :C13H16N6O6
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :352.3

    Ref: TM-T26130

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Azeloprazole

    CAS :
    Azeloprazole, a proton pump inhibitor, is used potentially for the treatment of gastroesophageal reflux disease (GERD).
    Formule :C22H27N3O4S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :429.53

    Ref: TM-T26727

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Ro18-5362

    CAS :
    Ro18-5362 is the less active prodrug of Ro 18-5364.
    Formule :C22H25N3O2S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :395.52

    Ref: TM-T19549

    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • Laurinterol

    CAS :
    Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.
    Formule :C15H19BrO
    Couleur et forme :Solid
    Masse moléculaire :295.21

    Ref: TM-T25638

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Bifenazate

    CAS :
    Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.
    Formule :C17H20N2O3
    Degré de pureté :99.62%
    Couleur et forme :Solid Crystalline
    Masse moléculaire :300.35

    Ref: TM-T14571

    25mg
    33,00€
    1mL*10mM (DMSO)
    49,00€
  • Dicirenone

    CAS :
    Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal
    Formule :C26H36O5
    Degré de pureté :99.1%
    Couleur et forme :Solid
    Masse moléculaire :428.56

    Ref: TM-T13881

    1mg
    630,00€
    5mg
    1.620,00€
  • ATPase-IN-2

    CAS :
    ATPase-IN-2: ATPase inhibitor (IC50 = 0.9μM), also blocks C. difficile toxin B (AC50 = 30.91μM). Used in ATP research.
    Formule :C22H20N2O4
    Couleur et forme :Solid
    Masse moléculaire :376.41

    Ref: TM-T61553

    500mg
    1.791,00€
  • Istaroxime hydrochloride

    CAS :
    Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a novel positive inotropic compound.
    Formule :C21H33ClN2O3
    Couleur et forme :Solid
    Masse moléculaire :396.95

    Ref: TM-T15599

    2mg
    125,00€
    5mg
    207,00€
    1mL*10mM (DMSO)
    226,00€
    10mg
    339,00€
    50mg
    710,00€
    100mg
    1.063,00€
  • Leminoprazole

    CAS :
    Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.
    Formule :C19H23N3OS
    Degré de pureté :99.08% - 99.79%
    Couleur et forme :Solid
    Masse moléculaire :341.47

    Ref: TM-T27812

    1mg
    81,00€
    5mg
    172,00€
    10mg
    259,00€
    25mg
    424,00€
    50mg
    583,00€
    100mg
    800,00€
  • SKF96067

    CAS :
    SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.
    Formule :C21H22N2O2
    Degré de pureté :99.89%
    Couleur et forme :Solid
    Masse moléculaire :334.41

    Ref: TM-T16894

    1mg
    264,00€
    5mg
    650,00€
    10mg
    888,00€
    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • AGN-201904

    CAS :
    AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.
    Formule :C25H25N3O8S2
    Degré de pureté :97.32%
    Couleur et forme :Solid
    Masse moléculaire :559.61

    Ref: TM-T23667

    1mg
    164,00€
    2mg
    234,00€
    5mg
    389,00€
    10mg
    532,00€
    25mg
    820,00€
  • NC-1300-B

    CAS :
    NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.
    Formule :C17H19N3OS
    Degré de pureté :99.50%
    Couleur et forme :Solid
    Masse moléculaire :313.42

    Ref: TM-T28136

    1mg
    164,00€
    5mg
    389,00€
    10mg
    532,00€
    25mg
    820,00€
  • FR-167356

    CAS :
    FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone metastasis.
    Formule :C19H17Cl2NO3
    Degré de pureté :98.44% - 99.74%
    Couleur et forme :Solid
    Masse moléculaire :378.25

    Ref: TM-T27371

    1mg
    110,00€
    5mg
    259,00€
    10mg
    353,00€
    25mg
    533,00€
    50mg
    718,00€
    100mg
    945,00€
    200mg
    1.251,00€
  • SCH28080

    CAS :
    SCH28080 is a reversible and K+-competitive inhibitor of gastric H+/K+-ATPase with an IC50 value of 20 nM (rabbit microsomal membrane).SCH28080 is a potent
    Formule :C17H15N3O
    Degré de pureté :99.24%
    Couleur et forme :Solid
    Masse moléculaire :277.32

    Ref: TM-T16865

    1mg
    34,00€
    1mL*10mM (DMSO)
    82,00€
    5mg
    84,00€
    10mg
    130,00€
    25mg
    251,00€
    50mg
    374,00€
    100mg
    533,00€
  • Tiludronate disodium

    CAS :
    Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.
    Formule :C7H7ClNa2O6P2S
    Degré de pureté :>99.99% - >99.99%
    Couleur et forme :Fine White To Off-White Crystalline Powder
    Masse moléculaire :362.57

    Ref: TM-T13159

    5mg
    75,00€
    10mg
    109,00€
    25mg
    178,00€
    50mg
    268,00€
    100mg
    396,00€
    500mg
    800,00€
  • Ro 18-5364

    CAS :
    Ro 18-5364 is a potent inhibitor of the gastric (H+ + K+)-ATPase with an apparent Ki of 0.1 μM at pH 6.
    Formule :C22H25N3O3S
    Degré de pureté :98%
    Couleur et forme :Solid
    Masse moléculaire :411.52

    Ref: TM-T28563

    25mg
    1.639,00€
    50mg
    2.142,00€
    100mg
    2.790,00€
  • BMS-199264 hydrochloride

    CAS :
    BMS-199264 hydrochloride is selective inhibitor of mitochondrial F1F0 ATP hydrolase,inhibit decline of ATP and myocardial necrosis during myocardial ischemia.
    Formule :C26H32Cl2N4O4S
    Degré de pureté :99.86%
    Couleur et forme :Solid
    Masse moléculaire :567.53

    Ref: TM-T26843

    1mg
    105,00€
    5mg
    250,00€
    10mg
    401,00€
    25mg
    803,00€
    50mg
    1.305,00€
    100mg
    2.088,00€
  • 3′-Acetate-ATP

    CAS :
    3’-Acetate-ATP, an analogue of ATP and its acetylation product, exhibits maximum ultraviolet absorption at 259 nm in neutral aqueous solutions.
    Formule :C12H18N5O14P3
    Couleur et forme :Solid
    Masse moléculaire :549.22

    Ref: TM-T79586

    5mg
    À demander
    50mg
    À demander
  • Suloctidil HCl

    CAS :
    Suloctidil HCl is a peripheral vascular dilator.
    Formule :C20H36ClNOS
    Couleur et forme :Solid
    Masse moléculaire :374.02

    Ref: TM-T0712L

    25mg
    1.998,00€
    50mg
    2.412,00€
    100mg
    2.880,00€
  • ATP synthase inhibitor 2

    CAS :
    ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.
    Formule :C21H22N2O3S
    Couleur et forme :Solid
    Masse moléculaire :382.48

    Ref: TM-T61649

    25mg
    690,00€
    50mg
    897,00€
    100mg
    1.341,00€
  • Antimalarial agent 7


    Antimalarial agent 7 is a potent and effective inhibitor of PfATP4. Antimalarial agent 7 has potential for the study of the human plasmodium falciparum.
    Formule :C23H22F2N4O3
    Couleur et forme :Solid
    Masse moléculaire :440.44

    Ref: TM-T62537

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Hsp90-IN-38

    CAS :
    Hsp90-IN-38 (compound 20m) is an inhibitor of HSP90 (heat shock protein). It demonstrates a strong binding affinity to HSP90 with a Kd of 87 nM. The compound inhibits ATPase activity with an IC50 of 0.13 μM. Hsp90-IN-38 also shows inhibitory effects on HCT116, MCF-7, SKBr3, K562, and A549 cells with IC50 values of 0.187, 0.072, 0.105, 0.403, and 0.031 μM, respectively.
    Formule :C28H35N3O5
    Couleur et forme :Solid
    Masse moléculaire :493.595

    Ref: TM-T205493

    10mg
    À demander
    50mg
    À demander
  • Vonoprazan fumarate

    CAS :

    Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.

    Formule :C17H16FN3O2S·C4H4O4
    Degré de pureté :99.16% - 99.98%
    Couleur et forme :Solid
    Masse moléculaire :461.46