ATPase
Les ATPases sont des enzymes qui catalysent la décomposition de l'ATP en ADP et un ion phosphate libre, une réaction qui libère de l'énergie utilisée pour conduire de nombreux processus au sein de la cellule, y compris le transport actif à travers les membranes. Les ATPases jouent un rôle crucial dans le maintien de l'homéostasie cellulaire, de l'équilibre du pH et des gradients ioniques. Les dysfonctionnements de l'activité des ATPases sont associés à des maladies telles que l'insuffisance cardiaque, l'hypertension et la neurodégénérescence. Chez CymitQuimica, nous fournissons des inhibiteurs et des modulateurs d'ATPase de haute qualité pour soutenir vos recherches en énergétique cellulaire, transport membranaire et pathologie des maladies.
93 produits trouvés pour "ATPase"
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Blebbistatin
CAS :<p>Blebbistatin ((±)-Blebbistatin) is a non-muscle myosin II (NMII)-selective and non-muscle myosin heavy chain 9 (MYH9)-specific inhibitor.Cost-effective and quality-assured.</p>Formule :C18H16N2O2Degré de pureté :99.88% - 99.97%Couleur et forme :Bright Yellow SolidMasse moléculaire :292.33Rabeprazole Sulfide
CAS :<p>Rabeprazole Sulfide (Rabeprazole Related Compound E) is an antiulcer drug in the class of proton pump inhibitors.</p>Formule :C18H21N3O2SDegré de pureté :99.34% - 99.78%Couleur et forme :Off-White Crystalline PowderMasse moléculaire :343.44Rbin-1
CAS :<p>Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.</p>Formule :C13H12N4SDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :256.33Omecamtiv mecarbil
CAS :<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Formule :C20H24FN5O3Degré de pureté :98% - 99.23%Couleur et forme :SolidMasse moléculaire :401.43Chloroprocaine hydrochloride
CAS :<p>Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.</p>Formule :C13H20Cl2N2O2Degré de pureté :99.65%Couleur et forme :White Crystalline PowderMasse moléculaire :307.22NPD8733
CAS :<p>NPD8733 is an inhibitor of cancer cell-enhanced fibroblast migration. It specifically binds to valosin-containing protein (VCP)/p97.</p>Formule :C18H15NO4Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :309.32D-α-Hydroxyglutaric acid disodium
CAS :<p>D-α-Hydroxyglutaric acid disodium (Disodium (R)-2-Hydroxyglutarate) is a competitive inhibitor of α-ketoglutarate-dependent dioxygenases with Ki of 0.628 mM.</p>Formule :C5H6Na2O5Degré de pureté :97.16%Couleur et forme :SolidMasse moléculaire :192.08Parimifasor
CAS :<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Formule :C18H11Cl2F4N5ODegré de pureté :96.77% - 98.97%Couleur et forme :SolidMasse moléculaire :460.21Revaprazan hydrochloride
CAS :<p>Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.</p>Formule :C22H24ClFN4Degré de pureté :99.62% - 99.91%Couleur et forme :SolidMasse moléculaire :398.9Transdermal Peptide Disulfide Acetate
<p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>Formule :C42H68N14O18S2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :1121.2(-)-Blebbistatin
CAS :<p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>Formule :C18H16N2O2Degré de pureté :99.38% - 99.61%Couleur et forme :SolidMasse moléculaire :292.33Vonoprazan fumarate
CAS :<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Formule :C17H16FN3O2S·C4H4O4Degré de pureté :99.16% - 99.98%Couleur et forme :SolidMasse moléculaire :461.46BTS
CAS :<p>BTS (N-Tosylbenzylamine) is a potent inhibitor of Ca2+-stimulated myosin S1 ATPase (IC50 : 5 μM) .</p>Formule :C14H15NO2SDegré de pureté :99.45%Couleur et forme :White Crystalline SolidMasse moléculaire :261.34Prilocaine
CAS :<p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>Formule :C13H20N2ODegré de pureté :98.49%Couleur et forme :Needles SolidMasse moléculaire :220.31NSC 617145
CAS :<p>NSC 617145 (NSC617145) is an inhibitor of WRN helicase that inhibits the ATPase, but not exonuclease, activity of WRN helicase in a concentration-dependent</p>Formule :C13H10Cl4N2O4Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :400.04Rostafuroxin
CAS :<p>Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.</p>Formule :C23H34O4Degré de pureté :99.08% - >99.99%Couleur et forme :SolidMasse moléculaire :374.51KM 91104
CAS :<p>KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.</p>Formule :C14H12N2O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :272.26PF 03716556
CAS :<p>PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal reflux</p>Formule :C22H26N4O3Degré de pureté :99.79% - 99.85%Couleur et forme :SolidMasse moléculaire :394.47Tetradifon
CAS :<p>Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.</p>Formule :C12H6Cl4O2SDegré de pureté :99.84%Couleur et forme :Yellowish Odorless OilMasse moléculaire :356.05Ro18-5362
CAS :<p>Ro18-5362 is the less active prodrug of Ro 18-5364.</p>Formule :C22H25N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :395.52FSBA hydrochloride
CAS :<p>FSBA hydrochloride(5'-p-Fluorosulfonylbenzoyladenosine) is an ATP analogue serving as an affinity probe for the ATP site of Na/K-ATPase.</p>Formule :C17H17ClFN5O7SDegré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :489.86Dicirenone
CAS :<p>Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal</p>Formule :C26H36O5Degré de pureté :99.1%Couleur et forme :SolidMasse moléculaire :428.56Bifenazate
CAS :<p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>Formule :C17H20N2O3Degré de pureté :99.62%Couleur et forme :Solid CrystallineMasse moléculaire :300.35Istaroxime hydrochloride
CAS :<p>Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a novel positive inotropic compound.</p>Formule :C21H33ClN2O3Couleur et forme :SolidMasse moléculaire :396.95Azeloprazole
CAS :<p>Azeloprazole, a proton pump inhibitor, is used potentially for the treatment of gastroesophageal reflux disease (GERD).</p>Formule :C22H27N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :429.53RS 029
CAS :<p>RS 029 is a nitroimidazole that has been exhibited to significantly inhibit (Na+K+) ATP-ase activity.</p>Formule :C13H16N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.3FCPT
CAS :<p>FCPT is an ATP competitive kinesin-5 inhibitor.</p>Formule :C17H13FN2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.36Laurinterol
CAS :<p>Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.</p>Formule :C15H19BrOCouleur et forme :SolidMasse moléculaire :295.21Istaroxime oxalate
CAS :<p>Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.</p>Formule :C23H34N2O7Couleur et forme :SolidMasse moléculaire :450.53Istaroxime
CAS :<p>Istaroxime is an effective inhibitor of Na+, K+-ATPase (IC50: 0.11 μM).</p>Formule :C21H32N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.49Tiludronate disodium
CAS :<p>Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.</p>Formule :C7H7ClNa2O6P2SDegré de pureté :>99.99% - >99.99%Couleur et forme :Fine White To Off-White Crystalline PowderMasse moléculaire :362.57SCH28080
CAS :<p>SCH28080 is a reversible and K+-competitive inhibitor of gastric H+/K+-ATPase with an IC50 value of 20 nM (rabbit microsomal membrane).SCH28080 is a potent</p>Formule :C17H15N3ODegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :277.32Leminoprazole
CAS :<p>Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.</p>Formule :C19H23N3OSDegré de pureté :99.08% - 99.56%Couleur et forme :SolidMasse moléculaire :341.47NC-1300-B
CAS :<p>NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.</p>Formule :C17H19N3OSDegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :313.42SKF96067
CAS :<p>SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.</p>Formule :C21H22N2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :334.41AGN-201904
CAS :<p>AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.</p>Formule :C25H25N3O8S2Degré de pureté :97.32%Couleur et forme :SolidMasse moléculaire :559.61FR-167356
CAS :<p>FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone metastasis.</p>Formule :C19H17Cl2NO3Degré de pureté :98.44% - 99.74%Couleur et forme :SolidMasse moléculaire :378.253′-Acetate-ATP
CAS :<p>3’-Acetate-ATP, an analogue of ATP and its acetylation product, exhibits maximum ultraviolet absorption at 259 nm in neutral aqueous solutions.</p>Formule :C12H18N5O14P3Couleur et forme :SolidMasse moléculaire :549.22BMS-199264 hydrochloride
CAS :<p>BMS-199264 hydrochloride is selective inhibitor of mitochondrial F1F0 ATP hydrolase,inhibit decline of ATP and myocardial necrosis during myocardial ischemia.</p>Formule :C26H32Cl2N4O4SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :567.53ATP synthase inhibitor 2
CAS :<p>ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.</p>Formule :C21H22N2O3SCouleur et forme :SolidMasse moléculaire :382.48Suloctidil HCl
CAS :<p>Suloctidil HCl is a peripheral vascular dilator.</p>Formule :C20H36ClNOSCouleur et forme :SolidMasse moléculaire :374.02Hsp90-IN-38
CAS :<p>Hsp90-IN-38 (compound 20m) is an inhibitor of HSP90 (heat shock protein). It demonstrates a strong binding affinity to HSP90 with a Kd of 87 nM. The compound inhibits ATPase activity with an IC50 of 0.13 μM. Hsp90-IN-38 also shows inhibitory effects on HCT116, MCF-7, SKBr3, K562, and A549 cells with IC50 values of 0.187, 0.072, 0.105, 0.403, and 0.031 μM, respectively.</p>Formule :C28H35N3O5Couleur et forme :SolidMasse moléculaire :493.595Antimalarial agent 7
<p>Antimalarial agent 7 is a potent and effective inhibitor of PfATP4. Antimalarial agent 7 has potential for the study of the human plasmodium falciparum.</p>Formule :C23H22F2N4O3Couleur et forme :SolidMasse moléculaire :440.44
