ATPase
Les ATPases sont des enzymes qui catalysent la décomposition de l'ATP en ADP et un ion phosphate libre, une réaction qui libère de l'énergie utilisée pour conduire de nombreux processus au sein de la cellule, y compris le transport actif à travers les membranes. Les ATPases jouent un rôle crucial dans le maintien de l'homéostasie cellulaire, de l'équilibre du pH et des gradients ioniques. Les dysfonctionnements de l'activité des ATPases sont associés à des maladies telles que l'insuffisance cardiaque, l'hypertension et la neurodégénérescence. Chez CymitQuimica, nous fournissons des inhibiteurs et des modulateurs d'ATPase de haute qualité pour soutenir vos recherches en énergétique cellulaire, transport membranaire et pathologie des maladies.
100 produits trouvés pour "ATPase"
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NPD8733
CAS :<p>NPD8733 is an inhibitor of cancer cell-enhanced fibroblast migration. It specifically binds to valosin-containing protein (VCP)/p97.</p>Formule :C18H15NO4Degré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :309.32D-α-Hydroxyglutaric acid disodium
CAS :D-α-Hydroxyglutaric acid disodium (Disodium (R)-2-Hydroxyglutarate) is a competitive inhibitor of α-ketoglutarate-dependent dioxygenases with Ki of 0.628 mM.Formule :C5H6Na2O5Degré de pureté :97.16%Couleur et forme :SolidMasse moléculaire :192.08Eniporide
CAS :Eniporide is a Na(+)/H(+) exchange inhibitor.Formule :C14H16N4O3SDegré de pureté :96.78% - 99.26%Couleur et forme :SolidMasse moléculaire :320.37Rostafuroxin
CAS :Rostafuroxin (PST 2238) has been used in trials studying the treatment of Essential Hypertension.Formule :C23H34O4Degré de pureté :98.24% - >99.99%Couleur et forme :SolidMasse moléculaire :374.51Tegoprazan
CAS :Tegoprazan is an orally active, highly selective gastric H+/K+-ATPase inhibitor.Cost-effective and quality-assured.Formule :C20H19F2N3O3Degré de pureté :98.22%Couleur et forme :SolidMasse moléculaire :387.38BRITE-338733
CAS :<p>BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.</p>Formule :C27H35N3O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :433.59Parimifasor
CAS :Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.Formule :C18H11Cl2F4N5ODegré de pureté :96.77% - 98.97%Couleur et forme :SolidMasse moléculaire :460.21Mitiglinide Calcium
CAS :Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-Formule :(C19H24NO3)2·CaDegré de pureté :99.83%Couleur et forme :White Crystal PosderMasse moléculaire :668.88Tirofiban hydrochloride monohydrate
CAS :<p>Tirofiban（MK383） hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>Formule :C22H39ClN2O6SDegré de pureté :98.81% - >99.99%Couleur et forme :White SolidMasse moléculaire :495.07BTS
CAS :BTS (N-Tosylbenzylamine) is a potent inhibitor of Ca2+-stimulated myosin S1 ATPase (IC50 : 5 μM) .Formule :C14H15NO2SDegré de pureté :99.45%Couleur et forme :White Crystalline SolidMasse moléculaire :261.34Transdermal Peptide Disulfide Acetate
<p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>Formule :C42H68N14O18S2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :1121.2Prilocaine
CAS :Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread ofFormule :C13H20N2ODegré de pureté :98.49%Couleur et forme :Needles SolidMasse moléculaire :220.31(-)-Blebbistatin
CAS :(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.Formule :C18H16N2O2Degré de pureté :99.38% - 99.61%Couleur et forme :SolidMasse moléculaire :292.33CB-5083
CAS :CB-5083 is a potent, selective, and orally bioavailable p97 AAA ATPase inhibitor ( IC50=11 nM).Formule :C24H23N5O2Degré de pureté :95.95% - 99.92%Couleur et forme :SolidMasse moléculaire :413.47Tenatoprazole
CAS :Tenatoprazole (TU-199), a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM).Formule :C16H18N4O3SDegré de pureté :99.57%Couleur et forme :White Crystalline PowderMasse moléculaire :346.4Rabeprazole sodium
CAS :Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.Formule :C18H20N3NaO3SDegré de pureté :98% - 99.912%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :381.42Esomeprazole Magnesium
CAS :Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.Formule :C34H36MgN6O6S2Degré de pureté :98.76% - 99.73%Couleur et forme :SolidMasse moléculaire :713.12Revaprazan hydrochloride
CAS :Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.Formule :C22H24ClFN4Degré de pureté :99.62% - 99.91%Couleur et forme :SolidMasse moléculaire :398.9FCCP
CAS :FCCP (Trifluoromethoxy carbonylcyanide phenylhydrazone) is an oxidative phosphorylation (OXPHOS) inhibitor and mitochondrial proton carrier uncoupler.Formule :C10H5F3N4ODegré de pureté :98% - 99.65%Couleur et forme :White SolidMasse moléculaire :254.17Chloroprocaine
CAS :Chloroprocaine: Na,K-ATPase inhibitor, IC50=13 mM, local anesthetic.Formule :C13H19ClN2O2Couleur et forme :SolidMasse moléculaire :270.76KM 91104
CAS :KM 91104 is a cell permeable inhibitor of V-ATPase. KM91104 specifically targets the interaction between V-ATPase subunit A3 and subunit B2.Formule :C14H12N2O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :272.26PF 03716556
CAS :PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal refluxFormule :C22H26N4O3Degré de pureté :99.79% - 99.95%Couleur et forme :SolidMasse moléculaire :394.47Tetradifon
CAS :Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.Formule :C12H6Cl4O2SDegré de pureté :99.84%Couleur et forme :Yellowish Odorless OilMasse moléculaire :356.05Istaroxime oxalate
CAS :Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.Formule :C23H34N2O7Couleur et forme :SolidMasse moléculaire :450.53FCPT
CAS :FCPT is an ATP competitive kinesin-5 inhibitor.Formule :C17H13FN2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :296.36RS 029
CAS :RS 029 is a nitroimidazole that has been exhibited to significantly inhibit (Na+K+) ATP-ase activity.Formule :C13H16N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.3Azeloprazole
CAS :Azeloprazole, a proton pump inhibitor, is used potentially for the treatment of gastroesophageal reflux disease (GERD).Formule :C22H27N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :429.53Ro18-5362
CAS :Ro18-5362 is the less active prodrug of Ro 18-5364.Formule :C22H25N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :395.52Laurinterol
CAS :Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.Formule :C15H19BrOCouleur et forme :SolidMasse moléculaire :295.21Bifenazate
CAS :Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Formule :C17H20N2O3Degré de pureté :99.62%Couleur et forme :Solid CrystallineMasse moléculaire :300.35Dicirenone
CAS :Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renalFormule :C26H36O5Degré de pureté :99.1%Couleur et forme :SolidMasse moléculaire :428.56ATPase-IN-2
CAS :ATPase-IN-2: ATPase inhibitor (IC50 = 0.9μM), also blocks C. difficile toxin B (AC50 = 30.91μM). Used in ATP research.Formule :C22H20N2O4Couleur et forme :SolidMasse moléculaire :376.41Istaroxime hydrochloride
CAS :Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a novel positive inotropic compound.Formule :C21H33ClN2O3Couleur et forme :SolidMasse moléculaire :396.95FSBA hydrochloride
CAS :FSBA hydrochloride(5'-p-Fluorosulfonylbenzoyladenosine) is an ATP analogue serving as an affinity probe for the ATP site of Na/K-ATPase.Formule :C17H17ClFN5O7SDegré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :489.86Istaroxime
CAS :Istaroxime is an effective inhibitor of Na+, K+-ATPase (IC50: 0.11 μM).Formule :C21H32N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :360.49Leminoprazole
CAS :Leminoprazole is an orally available H+,K(+)-ATPase inhibitor that protects gastric mucosal cells from various cellular damages.Formule :C19H23N3OSDegré de pureté :99.08% - 99.56%Couleur et forme :SolidMasse moléculaire :341.47Tiludronate disodium
CAS :Tiludronate disodium: osteoclast inhibitor for metabolic bone disorder research.Formule :C7H7ClNa2O6P2SDegré de pureté :>99.99% - >99.99%Couleur et forme :Fine White To Off-White Crystalline PowderMasse moléculaire :362.57SCH28080
CAS :SCH28080 is a reversible and K+-competitive inhibitor of gastric H+/K+-ATPase with an IC50 value of 20 nM (rabbit microsomal membrane).SCH28080 is a potentFormule :C17H15N3ODegré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :277.32FR-167356
CAS :<p>FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone metastasis.</p>Formule :C19H17Cl2NO3Degré de pureté :98.44% - 99.74%Couleur et forme :SolidMasse moléculaire :378.25AGN-201904
CAS :AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.Formule :C25H25N3O8S2Degré de pureté :97.32%Couleur et forme :SolidMasse moléculaire :559.61SKF96067
CAS :SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.Formule :C21H22N2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :334.41NC-1300-B
CAS :NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.Formule :C17H19N3OSDegré de pureté :99.50%Couleur et forme :SolidMasse moléculaire :313.42BMS-199264 hydrochloride
CAS :<p>BMS-199264 hydrochloride is selective inhibitor of mitochondrial F1F0 ATP hydrolase,inhibit decline of ATP and myocardial necrosis during myocardial ischemia.</p>Formule :C26H32Cl2N4O4SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :567.53Ro 18-5364
CAS :Ro 18-5364 is a potent inhibitor of the gastric (H+ + K+)-ATPase with an apparent Ki of 0.1 μM at pH 6.Formule :C22H25N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.523′-Acetate-ATP
CAS :3’-Acetate-ATP, an analogue of ATP and its acetylation product, exhibits maximum ultraviolet absorption at 259 nm in neutral aqueous solutions.Formule :C12H18N5O14P3Couleur et forme :SolidMasse moléculaire :549.22ATP synthase inhibitor 2
CAS :ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.Formule :C21H22N2O3SCouleur et forme :SolidMasse moléculaire :382.48Hsp90-IN-38
CAS :<p>Hsp90-IN-38 (compound 20m) is an inhibitor of HSP90 (heat shock protein). It demonstrates a strong binding affinity to HSP90 with a Kd of 87 nM. The compound inhibits ATPase activity with an IC50 of 0.13 μM. Hsp90-IN-38 also shows inhibitory effects on HCT116, MCF-7, SKBr3, K562, and A549 cells with IC50 values of 0.187, 0.072, 0.105, 0.403, and 0.031 μM, respectively.</p>Formule :C28H35N3O5Couleur et forme :SolidMasse moléculaire :493.595Suloctidil HCl
CAS :Suloctidil HCl is a peripheral vascular dilator.Formule :C20H36ClNOSCouleur et forme :SolidMasse moléculaire :374.02Antimalarial agent 7
Antimalarial agent 7 is a potent and effective inhibitor of PfATP4. Antimalarial agent 7 has potential for the study of the human plasmodium falciparum.Formule :C23H22F2N4O3Couleur et forme :SolidMasse moléculaire :440.44Vonoprazan fumarate
CAS :<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Formule :C17H16FN3O2S·C4H4O4Degré de pureté :99.16% - 99.98%Couleur et forme :SolidMasse moléculaire :461.46
