
Canal sodique
Les canaux sodiques sont des protéines membranaires essentielles qui permettent le passage des ions sodium (Na+) à travers la membrane cellulaire, générant et propageant des signaux électriques dans les neurones, les cellules musculaires et d'autres tissus excitables. Ces canaux sont vitaux pour l'initiation et la conduction des potentiels d'action, ce qui les rend cruciaux dans des processus tels que la transmission de l'influx nerveux, la contraction musculaire et la fonction cardiaque. La dysrégulation des canaux sodiques peut entraîner des troubles neurologiques, des arythmies et des conditions de douleur chronique. Chez CymitQuimica, nous proposons une variété de modulateurs de canaux sodiques pour soutenir vos recherches en neurobiologie, cardiologie et gestion de la douleur.
202 produits trouvés pour "Canal sodique"
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Nav1.8-IN-4
CAS :<p>Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.</p>Formule :C20H14F4N2O3Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :406.33Topiramate
CAS :<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formule :C12H21NO8SDegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :339.36Lidocaine Hydrochloride hydrate
CAS :<p>Lidocaine Hydrochloride hydrate is an amide local anesthetic, has anti-inflammatory property.</p>Formule :C14H22N2O·HCl·H2ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :288.82Lamotrigine
CAS :<p>Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.</p>Formule :C9H7Cl2N5Degré de pureté :99.76% - 99.95%Couleur et forme :White To Pale Cream-Colored Powder Crystals From Isopropanol SolidMasse moléculaire :256.09Oxcarbazepine
CAS :<p>Oxcarbazepine (GP 47680), an anti-epileptic, reduces CNS disorganized electrical activity.</p>Formule :C15H12N2O2Degré de pureté :98.46%Couleur et forme :Crystals From Ethanol SolidMasse moléculaire :252.27Diphenidol hydrochloride
CAS :<p>Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.</p>Formule :C21H28ClNODegré de pureté :99.15% - 99.33%Couleur et forme :Crystals Soluble In Methanol WaterMasse moléculaire :345.91Tocainide hydrochloride
CAS :<p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>Formule :C11H17ClN2ODegré de pureté :97%Couleur et forme :SolidMasse moléculaire :228.72Ropivacaine hydrochloride
CAS :<p>Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activity</p>Formule :C17H26N2O·HClDegré de pureté :99.85% - 99.95%Couleur et forme :SolidMasse moléculaire :310.86Tocainide
CAS :<p>Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.</p>Formule :C11H16N2ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :192.26NaV1.7 inhibitor-1
CAS :<p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>Formule :C23H30FNO4SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :435.55Amiloride hydrochloride
CAS :<p>Amiloride hydrochloride (Amiloride HCl) 是上皮钠通道和尿激酶型纤溶酶原激活物受体的抑制剂,也是 polycystin-2通道阻断剂。</p>Formule :C6H9Cl2N7ODegré de pureté :99.72% - 99.95%Couleur et forme :Physical Description Crystalline Solid Or Very Light Yellow Powder (Ntp 1992)Masse moléculaire :266.09Phenytoin
CAS :<p>Phenytoin: a non-sedative hydantoin, antiepileptic with anticonvulsant effects, stabilizes neurons, prevents seizure spread, and relaxes muscles.</p>Formule :C15H12N2O2Degré de pureté :99.95%Couleur et forme :Needles (Alcohol) Tasteless (Ntp 1992)Masse moléculaire :252.27Eleclazine hydrochloride
CAS :<p>Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).</p>Formule :C21H17ClF3N3O3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :451.83Lidocaine
CAS :<p>Lidocaine, an amide local anesthetic, reduces pain and inflammation by dampening ICAM-1, cytokines, and neutrophil influx.</p>Formule :C14H22N2ODegré de pureté :99.95% - >99.99%Couleur et forme :Needles From Benzene Or Alcohol SolidMasse moléculaire :234.34Benzocaine
CAS :<p>Benzocaine is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.</p>Formule :C9H11NO2Degré de pureté :99.16% - 99.88%Couleur et forme :Rhombohedra From Ether DrypowderMasse moléculaire :165.19Primidone
CAS :<p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>Formule :C12H14N2O2Degré de pureté :99.91%Couleur et forme :Crystals (Ntp 1992)Masse moléculaire :218.25Brompheniramine maleate
CAS :<p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>Formule :C16H19BrN2·C4H4O4Degré de pureté :99.80%Couleur et forme :Crystal PowderMasse moléculaire :435.31Oxybuprocaine hydrochloride
CAS :<p>Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.</p>Formule :C17H29ClN2O3Degré de pureté :>99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :344.88Butamben
CAS :<p>Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.</p>Formule :C11H15NO2Degré de pureté :99.43%Couleur et forme :Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Masse moléculaire :193.24Mexiletine hydrochloride
CAS :<p>Mexiletine hydrochloride is a lidocaine-like antiarrhythmic (Class IB) and anesthetic, stabilizing heartbeats by inhibiting sodium in cardiac cells.</p>Formule :C11H18ClNODegré de pureté :99.88%Couleur et forme :White To Off-White SolidMasse moléculaire :215.72Ropivacaine
CAS :<p>Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.</p>Formule :C17H26N2ODegré de pureté :97.75% - >99.99%Couleur et forme :SolidMasse moléculaire :274.40Dibucaine
CAS :<p>Dibucaine (Cinchocaine), a local anesthetic of the amide type, is now usually used for surface anesthesia.</p>Formule :C20H29N3O2Degré de pureté :99.698% - 99.88%Couleur et forme :Colorless Or Almost Colorless Powder SolidMasse moléculaire :343.46Articaine hydrochloride
CAS :<p>Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.</p>Formule :C13H21ClN2O3SDegré de pureté :99.76%Couleur et forme :White Crystalline PowderMasse moléculaire :320.84Bupivacaine hydrochloride
CAS :<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Formule :C18H28N2O·HClDegré de pureté :99.9% - >99.99%Couleur et forme :SolidMasse moléculaire :324.89Disopyramide
CAS :<p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>Formule :C21H29N3ODegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :339.47E 0747 FA
<p>E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax in Purkinje fibers of porcine heart.E 0747 FA inhibits Na channels in cardiac cells.</p>Formule :C22H30ClN3O6Degré de pureté :98.54%Couleur et forme :SolidMasse moléculaire :467.94Phenazopyridine hydrochloride
CAS :<p>Phenazopyridine HCl, an oral urinary analgesic, may cause nausea, anemia, and liver/kidney toxicity. Possibly carcinogenic.</p>Formule :C11H12ClN5Degré de pureté :99.27%Couleur et forme :Brownish-Yellow Crystals Aqueous Solutions Are Yellow To Brick-Red And Slightly Acidic; They May Be Stabilized By The AdditionMasse moléculaire :249.7Vinpocetine
CAS :<p>Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).</p>Formule :C22H26N2O2Degré de pureté :99.85% - 99.98%Couleur et forme :White Crystalline SolidMasse moléculaire :350.45DSP-2230
CAS :<p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>Formule :C20H20F3N5O2Degré de pureté :97.14%Couleur et forme :SolidMasse moléculaire :419.4Methocarbamol
CAS :<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Formule :C11H15NO5Degré de pureté :99.96%Couleur et forme :Crystals From Benzene SolidMasse moléculaire :241.24Ranolazine dihydrochloride
CAS :<p>Ranolazine 2HCl, an antianginal, treats arrhythmia by inhibiting sodium current without changing blood pressure or heart rate.</p>Formule :C24H35Cl2N3O4Degré de pureté :99.30% - >99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :500.46Lidocaine hydrochloride
CAS :<p>Lidocaine HCl: local anesthetic, antiarrhythmic, stronger & longer-lasting than procaine but shorter than bupivacaine/prilocaine.</p>Formule :C14H23ClN2ODegré de pureté :99.81% - 99.92%Couleur et forme :White Crystal PowderMasse moléculaire :270.798Propafenone
CAS :<p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>Formule :C21H27NO3Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :341.44QX-314 chloride
CAS :<p>QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.</p>Formule :C16H27ClN2ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :298.85Phenytoin sodium
CAS :<p>Phenytoin sodium (Diphantoine) is an inactive stabilizer for voltage-gated sodium channel .</p>Formule :C15H11N2NaO2Degré de pureté :99.88% - 99.92%Couleur et forme :SolidMasse moléculaire :274.25Amitriptyline hydrochloride
CAS :<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Formule :C20H24ClNDegré de pureté :97% - 99.94%Couleur et forme :Crystals White To Off-White PowderMasse moléculaire :313.86Meticrane
CAS :<p>Meticrane (Arresten) is a sulphonamide-derivative with thiazide-like diuretic activity.</p>Formule :C10H13NO4S2Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :275.34PF-04885614
CAS :<p>PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.</p>Formule :C13H14F3N3ODegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :285.27Mebeverine hydrochloride
CAS :<p>Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gut</p>Formule :C25H35NO5Degré de pureté :99.81% - 99.81%Couleur et forme :SolidMasse moléculaire :429.55Flunarizine dihydrochloride
CAS :<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Formule :C26H28Cl2F2N2Degré de pureté :99.53% - 99.89%Couleur et forme :White Crystalline Powder Odorless And TastelessMasse moléculaire :477.42BIIB 722 Mesylate
CAS :<p>BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.</p>Formule :C19H23F3N6O5SDegré de pureté :99.57%Couleur et forme :SoildMasse moléculaire :504.483Zoniporide
CAS :<p>Zoniporide (CP-597396) is an NHE-1 inhibitor that inhibits platelet swelling and can be used in the study of cardiovascular diseases.</p>Formule :C17H16N6ODegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :320.35LTGO-33
CAS :<p>LTGO-33 is a voltage-gated sodium channel NaV1.8 inhibitor that inhibits NaV1.8, NaV1.1-NaV1.7, and NaV1.9.</p>Formule :C21H17F4N3O3SDegré de pureté :97.6%Couleur et forme :SoildMasse moléculaire :467.44Veratridine
CAS :<p>Veratridine is a benzoate-cevane found in Veratrum and Schoenocaulon. It activates sodium channels to stay open longer than normal.</p>Formule :C36H51NO11Degré de pureté :98.07% - 99.27%Couleur et forme :Yellowish-White Amorphous Powder PowderMasse moléculaire :673.79GpTx-1 TFA
<p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with >20-fold and >950-fold selectivity, respectively.</p>Couleur et forme :Odour SolidTrapencaine
CAS :<p>Trapencaine is a newly synthesized carbamate type local anesthetic that induces conformational changes in sodium channels on hypertrophic cell membranes.</p>Formule :C22H34N2O3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :374.52SLC26A3-IN-2
CAS :<p>Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.</p>Formule :C19H13ClN2O2SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :368.84Nav1.3 channel inhibitor 1
<p>Nav1.3 Channel Inhibitor 1 (Compound 15b) is a state-dependent inhibitor of the voltage-gated sodium channel Na v 1.3, with an IC50 value of 20 nM.</p>Formule :C19H15F2N3O3S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :435.47Halazone
CAS :<p>Halazone (Pantocid) is fine white powder with an odor of chlorine. It has been widely used to disinfect drinking water.</p>Formule :C7H5Cl2NO4SDegré de pureté :98.64%Couleur et forme :Physical Description Fine White Powder With An Odor Of Chlorine (Ntp 1992)Masse moléculaire :270.09ProTx II TFA
<p>ProTx-II TFA is a potent and highly selective Nav1.7 sodium channel blocker, exhibiting an IC50 of 0.3 nM and demonstrating at least 100-fold selectivity over</p>Formule :C168H250N46O41S8·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3826.59 (free base)Ancistrotecine B
<p>Ancistrotecine B (Compound 2), a Nav1.7 channel inhibitor (IC50: 0.73 μM), has been shown to alleviate inflammatory pain in mice [1].</p>Formule :C26H31NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :421.53PF-06456384 trihydrochloride
CAS :<p>PF-06456384 trihydrochloride is a selective NaV1.7 inhibitor acting through protein-ligand binding. intravenous infusion and pain research.</p>Formule :C35H35Cl3F3N7O3S2Degré de pureté :99.16%Couleur et forme :SolidMasse moléculaire :829.18Solpecainol
CAS :<p>solpecainol is a sodium channel blocker used in the study of neurological and cardiovascular diseases.</p>Formule :C18H23NO3Degré de pureté :99.71%Couleur et forme :SoildMasse moléculaire :301.38Analgesic agent-2
<p>Analgesic Agent-2, a selective orally active inhibitor of the NaV1.8 channel, demonstrates an IC50 of 50.18 nM in HEK293 cells that stably express the human</p>Formule :C21H21ClF2N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.871-(1-Methyl-1h-pyrazol-4-yl)-ethanone
CAS :<p>1-(1-Methyl-1h-pyrazol-4-yl)-ethanone is a high purity biochemical reagent that can be used in research related to life sciences.</p>Formule :C6H8N2ODegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :124.14Nav1.7-IN-18
<p>Nav1.7-IN-18 (Compound 31) is a Nav1.7 inhibitor with a Ki value of 4.9 nM and an IC50 of 13 nM, demonstrating analgesic effects in transgenic mice with inherited erythromelalgia (IEM).</p>Formule :C30H33Cl2F2NO4Couleur et forme :SolidMasse moléculaire :580.49Myomodulin
CAS :<p>Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A the</p>Formule :C36H67N11O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :846.12ASG-5ME
<p>ASG-5ME is a drug-antibody coupling targeting SLC44A4 that shows anti-tumor activity in xenograft models and may be used to study pancreatic and gastric cancer.</p>Degré de pureté :98.1% (SDS-PAGE); 98.5% (SEC-HPLC) - 98.1% (SDS-PAGE); 98.5% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145.5 kDaZandatrigine
CAS :<p>Zandatrigine (NBI-921352) is a blocker of sodium channel protein type 8 subunit alpha and can be used in studies about nervous system pathologies of epilepsy</p>Formule :C22H25FN4O2S2Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :460.59Zoniporide hydrochloride
CAS :<p>Zoniporide hydrochloride: selective NHE-1 inhibitor, IC50 14 nM, >150x selectivity over other NHEs, inhibits platelet swelling (IC50 59 nM).</p>Formule :C17H17ClN6ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :356.81ETD001
CAS :<p>ETD001 is a long-acting ENaC inhibitor with an IC50 value of 57.5 nM in HBE cells. It is applicable for research in cystic fibrosis.</p>Formule :C41H57F6N9O16Couleur et forme :SolidMasse moléculaire :1045.935-Tridecanol
CAS :<p>5-Tridecanol blocks ion flux in sodium channels.</p>Formule :C13H28ODegré de pureté :97.87%Couleur et forme :SolidMasse moléculaire :200.36NHE-1-IN-2
NHE-1-IN-2 (compound 7g) is a potent NHE-1 inhibitor with an IC50 of 0.78 μM. It mitigates left ventricular systolic dysfunction in mouse models of heart failure.Formule :C23H20ClN3O3Couleur et forme :SolidMasse moléculaire :421.11932APETx2
CAS :<p>ASIC3 inhibitor; IC50: 63 nM (rat), 175 nM (human). Blocks NaV1.8, NaV1.2; analgesic for acid/inflammatory pain.</p>Formule :C196H280N54O61S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4561.06Mambalgin 1
CAS :<p>ASIC1a inhibitor; IC50: 192 nM (human), 72 nM (dimer); inactive channel binding; selective; pain response delay.</p>Formule :C272H429N85O84S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :6554.51CL-424032
CAS :<p>CL-424032 is an inhibitor of sodium channels (sodium channel).</p>Formule :C12H7F3N4O2Couleur et forme :SolidMasse moléculaire :296.21ProTx II
CAS :<p>Selective NaV1.7 inhibitor, alters activation, reduces current, 100x more selective for 1.7 over other Na+ channels.</p>Formule :C168H250N46O41S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3826.59Indenebart
<p>Indenebart is a humanized IgG1λ2 monoclonal antibody targeting SNCA, with HumanIgG1lambda2, Isotype Control serving as the corresponding isotype control.</p>Couleur et forme :Odour LiquidIon Channel Targeted Library
<p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>Couleur et forme :Odour SolidHuwentoxin-IV
CAS :<p>Selective NaV1.7 blocker; also inhibits NaV1.2, 1.3; less effect on NaV1.4, 1.5. Binds to neurotoxin site, traps voltage sensor. IC50: 26-338 nM.</p>Formule :C174H278N52O51S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4106.79OD1
<p>Activates rat Nav1.7, human Nav1.4, rat Nav1.6 (EC50: 7, 10, 47 nM); minimal on Nav1.2, 1.3, 1.5 (EC50 >3 μM); blocks fast inactivation; triggers pain.</p>Formule :C308H466N90O95S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7206.1Phrixotoxin 3
CAS :<p>Potent NaV blocker: IC50 - 0.6 nM (NaV1.2), 42 nM (NaV1.3), 72 nM (NaV1.5); voltage-dependent inhibition.</p>Formule :C176H269N51O48S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4059.74Sodium Channel Targeted Library
<p>A unique collection of xnum sodium channel blockers and agonists for high throughput and high content screening;</p>Couleur et forme :Odour SolidLifarizine FA
<p>Lifarizine FA is a sodium channel blocker used in the treatment of neurological disorders and cardiovascular diseases, study of stroke.</p>Formule :C30H34N4O2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :482.62Benzonatate (PEGn)
CAS :<p>Benzonatate (PEGn) is a unique non-narcotic cough suppressant featuring sodium channel blocking properties and anesthetic effects on respiratory tract stretch receptors.</p>Formule :(C2H4O)nC12H17NO2Couleur et forme :SolidGX 201
CAS :<p>GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.</p>Formule :C25H27ClF4N2O4SDegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :563Mepivacaine hydrochloride
CAS :<p>Mepivacaine hydrochloride (Mepivacaine HCl) is the hydrochloride salt form of mepivacaine, an amide derivative with local anesthetic properties.</p>Formule :C15H22N2O·HClDegré de pureté :98.76% - 99.94%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :282.81Amlenetug
<p>Amlenetug is a humanized IgG1κ antibody targeting SNCA, with its corresponding isotype control being HumanIgG1kappa, Isotype Control.</p>Couleur et forme :Odour LiquidMexiletine-d6 hydrochloride
CAS :<p>Mexiletine D6 hydrochloride is a non-selective voltage-gated sodium channel blocker,is a Class IB antianhythmic.</p>Formule :C11H18ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :221.76Triamterene D5
CAS :<p>Triamterene D5 is a deuterium-labeled Triamterene and can block epithelial Na+ channel (ENaC) in a voltage-dependent manner, used as a mild diuretic.</p>Formule :C12H11N7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :258.29BI-9627
CAS :<p>BI-9627 is an inhibitor of sodium-hydrogen exchanger isoform 1 (NHE1) (EC50: 31 nM).</p>Formule :C16H19F3N4O2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :356.34Poneratoxin acetate
<p>Poneratoxin acetate is a neurotoxic peptide and modulator of NaV1.6/NaV1.7, lowering the activation threshold of voltage-gated sodium channels and causing pain.</p>Formule :C129H215N33O31S·xC2H4O2Couleur et forme :SolidMasse moléculaire :2756.35 (free base)Ethacizine hydrochloride
CAS :<p>Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.</p>Formule :C22H28ClN3O3SDegré de pureté :98.08% - 98.08%Couleur et forme :SolidMasse moléculaire :449.99Dibucaine hydrochloride
CAS :<p>Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.</p>Formule :C20H30ClN3O2Degré de pureté :99.66%Couleur et forme :White PowderMasse moléculaire :379.92Bulleyaconitine A
CAS :<p>Bulleyaconitine A, an analgesic and antiinflammatory drug isolated from Aconitum plants, has several potential targets, such as voltage-gated Na+ channels.</p>Formule :C35H49NO9Degré de pureté :99.56% - 99.76%Couleur et forme :SolidMasse moléculaire :627.76AM-2099
CAS :<p>AM-2099 is a selective voltage-gated sodium channel Nav1.7 inhibitor used in pain research.</p>Formule :C19H13F3N4O3S2Couleur et forme :SolidMasse moléculaire :466.46PF-04856264
CAS :<p>PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.</p>Formule :C20H15N5O3S2Degré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :437.5Mepivacaine
CAS :<p>Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.</p>Formule :C15H22N2ODegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :246.35Raxatrigine
CAS :<p>Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.</p>Formule :C18H19FN2O2Degré de pureté :98% - 99.43%Couleur et forme :SolidMasse moléculaire :314.35DS-1971a
CAS :<p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>Formule :C20H21ClFN5O3SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :465.93A-803467
CAS :<p>A-803467 is a selective NaV1.8 channel blocker.</p>Formule :C19H16ClNO4Degré de pureté :96.94% - 98%Couleur et forme :SolidMasse moléculaire :357.79Flecainide hydrochloride
CAS :<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Formule :C17H21ClF6N2O3Degré de pureté :97.79%Couleur et forme :SolidMasse moléculaire :450.81Ropivacaine hydrochloride monohydrate
CAS :<p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>Formule :C17H29ClN2O2Degré de pureté :99.94% - 99.95%Couleur et forme :White SolidMasse moléculaire :328.88Fosphenytoin disodium
CAS :<p>Fosphenytoin disodium (ACC-9653) is a prodrug of phenytoin that is rapidly converted to phenytoin, a voltage-gated sodium channel blocker</p>Formule :C16H13N2Na2O6PDegré de pureté :99.97%Couleur et forme :White Crystalline PowderMasse moléculaire :406.24Metergoline
CAS :<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Formule :C25H29N3O2Degré de pureté :99.83% - 99.97%Couleur et forme :SolidMasse moléculaire :403.52Rimeporide
CAS :<p>Rimeporide (EMD-87580) (EMD-87580) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>Formule :C11H15N3O5S2Degré de pureté :97.66%Couleur et forme :SolidMasse moléculaire :333.38λ-Cyhalothrin
CAS :<p>λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.</p>Formule :C23H19ClF3NO3Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :449.85Flecainide acetate
CAS :<p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>Formule :C19H24F6N2O5Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :474.39Nicainoprol
CAS :<p>Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.</p>Formule :C21H27N3O3Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :369.46Pilsicainide HCl
CAS :<p>Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker</p>Formule :C17H25ClN2ODegré de pureté :99.01% - 99.80%Couleur et forme :SolidMasse moléculaire :308.85

