Canal calcique
Les canaux calciques sont des protéines membranaires qui régulent le flux d'ions calcium dans et hors des cellules, ce qui est essentiel pour diverses fonctions cellulaires, y compris la contraction musculaire, la libération de neurotransmetteurs et l'expression génique. La dysrégulation de l'activité des canaux calciques est associée à des conditions telles que l'hypertension, les arythmies cardiaques et les troubles neurologiques. Chez CymitQuimica, nous proposons une large sélection de modulateurs des canaux calciques pour soutenir vos recherches en santé cardiovasculaire, neurobiologie et transduction du signal.
493 produits trouvés pour "Canal calcique"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
O-Desmethylcarvedilol
CAS :<p>O-Desmethylcarvedilol (Desmethylcarvedilol) is an active metabolite of Carvedilol, a non-selective β-adrenergic receptor (β-AR) antagonist. This compound inhibits store overload-induced calcium release in HEK293 cells expressing the RyR2 R4496C mutation (IC50= 7.62 µM). Additionally, O-Desmethylcarvedilol slows the increase in heart rate and prevents diastolic pressure reduction induced by Isoproterenol in conscious rabbits (ED50s = 32 and 5 µg/kg).</p>Formule :C23H24N2O4Couleur et forme :SolidMasse moléculaire :392.45SB-237376
CAS :<p>SB-237376 is a calcium and potassium channel antagonist used to treat cardiac arrhythmias.</p>Formule :C20H25N3O5Degré de pureté :98.88% - 99.81%Couleur et forme :SoildMasse moléculaire :387.43D-myo-Inositol-1,3-diphosphate (sodium salt)
CAS :<p>D-myo-Inositol-1,3-phosphate (Ins(1,3)P) is an inositol phosphate involved in cellular signal transduction.</p>Formule :C6H12Na2O12P2Couleur et forme :SolidMasse moléculaire :384.08TPC2-A1-P
CAS :<p>TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).</p>Formule :C20H21BrF3NO3Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :460.29OPC 8490 free base
CAS :<p>OPC 8490 free base is a positive inotropic vasodilator and a cardiotonic agent that can be used to study cardiovascular diseases.</p>Formule :C24H27N3O3Degré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :405.49D-myo-Inositol-1,4,5-triphosphate trisodium
CAS :<p>D-myo-Inositol-1,4,5-triphosphate trisodium (Inositol 1,4,5-trisphosphate trisodium) is a second messenger produced in cells by phospholipase C-mediated</p>Formule :C6H15Na3O15P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.06Elgodipine
CAS :<p>Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.</p>Formule :C29H33FN2O6Degré de pureté :98.95% - 99.50%Couleur et forme :SolidMasse moléculaire :524.58Cavα2δ-IN-1
CAS :<p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>Formule :C18H27N5OCouleur et forme :SolidMasse moléculaire :329.448Ser-Ala-alloresact acetate
<p>Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.</p>Formule :C44H75N13O16S2Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :1106.281-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS :<p>1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(</p>Formule :C5H10ClNO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :151.59Triphenylethylene
CAS :<p>Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formule :C20H16Couleur et forme :White PowderMasse moléculaire :256.34ω-Conotoxin MVIIC
CAS :<p>Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.</p>Formule :C106H178N40O32S7Degré de pureté :98%Couleur et forme :White Lyophilised SolidMasse moléculaire :2749Myomodulin
CAS :<p>Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A the</p>Formule :C36H67N11O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :846.12PACAP-38 (31-38), human, mouse, rat TFA
<p>PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.</p>Formule :C49H84F3N17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1176.29BTT-266
CAS :<p>BTT-266 is a blocker of voltage-gated calcium channel for pain management.</p>Formule :C34H28N4O4Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :556.61Calcium Channel Compound Library
<p>A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening;</p>Couleur et forme :Odour SolidPD 0299685
CAS :<p>PD 0299685 is a potent α2δ ligand of the Ca2+ channel for the treatment of interstitial cystitis.</p>Formule :C10H21NO2Degré de pureté :97.20%Couleur et forme :SoildMasse moléculaire :187.28Calcium Channel antagonist 3
CAS :<p>Calcium Channel antagonist 3 is a voltage-gated calcium channel inhibitor (IC50 : 5-20 μM).</p>Formule :C23H26N2O4SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :426.53Fasudil
CAS :<p>Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.</p>Formule :C14H17N3O2SDegré de pureté :99.79% - 99.84%Couleur et forme :SolidMasse moléculaire :291.37Linoleic Acid Amide
CAS :<p>Linoleic Acid Amide (Linoleamide) is derived from linoleic acid and regulates Ca2+ flux by inhibiting the sarco/endoplasmic reticulum Ca2+-ATPase.</p>Formule :C18H33NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :279.46Flosatidil
CAS :<p>Flosatidil is a small molecule voltage-gated calcium channel complex (VDCCs) blocker for the treatment of neurological disorders and cardiovascular diseases,</p>Formule :C26H34F3N3O3SDegré de pureté :98.29% - 99.60%Couleur et forme :SolidMasse moléculaire :525.63Ziconotide
CAS :<p>Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.</p>Formule :C102H172N36O32S7Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :2639.13Atagabalin HCl
CAS :<p>Atagabalin HCl is a novel voltage-dependent calcium channel (VDCC) α2δ subunit (1 and 2) ligand that affects slow-wave sleep and can be used to treat insomnia.</p>Formule :C10H20ClNO2Degré de pureté :99.96% - ≥98%Couleur et forme :SoildMasse moléculaire :221.72Huwentoxin I
CAS :<p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>Formule :C161H246N48O44S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3750.36KT-362 free base
CAS :<p>KT-362 is a calcium channel blocker with antihypertensive properties that can be used in the study of cardiovascular disease.</p>Formule :C22H28N2O3SDegré de pureté :99.76%Couleur et forme :SoildMasse moléculaire :400.5317R(18S)-EpETE
CAS :<p>17R(18S)-EpETE: Oxylipin, eicosapentaenoic acid metabolite, activates BKCa channels, has negative chronotropic effects.</p>Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.4571,4-Dihydropyridine
<p>1,4-Dihydropyridine acts as an antagonist for calcium channels (calcium channel), specifically blocking the L-type calcium channels. This action reduces the influx of calcium ions into cardiac and vascular smooth muscle cells, consequently decreasing cardiac contractility and heart rate, dilating blood vessels, and lowering blood pressure.</p>Formule :C12H17NO4Couleur et forme :SolidMasse moléculaire :239.27Chlorocresol
CAS :<p>Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.</p>Formule :C7H7ClOCouleur et forme :SolidMasse moléculaire :142.58Levamlodipine besylate Hemipentahydrate
CAS :<p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>Formule :C20H25ClN2O5·C6H6O3SH2OCouleur et forme :SolidMasse moléculaire :1224.18NAADP sodium
<p>NAADP sodium is a Ca2+ motor second messenger that targets Ca(2+) channels and can be used to study cancer and immune dysfunction.</p>Formule :C21H27N6O18P3Couleur et forme :SolidMasse moléculaire :744.39D-myo-Inositol-1,4,5-triphosphate tripotassium
CAS :<p>D-myo-Inositol-1,4,5-triphosphate tripotassium is a second messenger in the intracellular signaling system that induces Ca2+ mobilization.</p>Formule :C6H12K3O15P3Couleur et forme :SolidMasse moléculaire :534.37Ethacrynic acid D5
CAS :<p>Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.</p>Formule :C13H12Cl2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.17Cyclic ADP-ribose ammonium
<p>cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.</p>Couleur et forme :LiquidsFTX-3.3
CAS :<p>sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.</p>Formule :C12H29N7OCouleur et forme :SolidMasse moléculaire :287.412Candidalysin
CAS :<p>Candidalysin is a cytolytic peptide toxin initially isolated from *Candida albicans*, exhibiting both toxic and non-toxic properties. It activates epithelial cell signaling pathways by interacting with the epithelial growth factor receptor (EGFR) on host cells, leading to the activation of matrix metalloproteinases (MMP) and calcium ion influx, which results in inflammatory responses and immune cell recruitment. Additionally, Candidalysin exhibits cytotoxicity by causing membrane damage to host cells.</p>Formule :C153H266N38O38S2Couleur et forme :SolidMasse moléculaire :3310.11Ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate
CAS :<p>ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate inhibits NAD(P)H: quinone oxidoreductase 1.</p>Formule :C12H10ClNO3Degré de pureté :99.19%Couleur et forme :SolidMasse moléculaire :251.67ProTx-I
CAS :<p>Selective blocker for CaV3.1 (IC50 = 0.2 μM), CaV3.2 (31.8 μM), also inhibits NaV1.8 and blocks KV2.1 channels.</p>Formule :C171H245N53O47S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3987.51(±)5(6)-DiHETE
CAS :<p>Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.</p>Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.472MMK 1
CAS :<p>Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.</p>Formule :C75H123N19O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1610.97ω-Agatoxin TK
CAS :<p>Selective blocker of CaV2.1 P/Q-type calcium channels.</p>Formule :C215H337N65O70S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5273.02Catharanthine
CAS :<p>Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).</p>Formule :C21H24N2O2Degré de pureté :99.11%Couleur et forme :White PowderMasse moléculaire :336.43CCT129957
CAS :<p>CCT129957 is a novel and potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of about 3 μM and a GC50 of 15 μM.CCT129957 exhibits anticancer activity and</p>Formule :C17H15N3O3Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :309.32(R)-(+)-Bay-K-8644
CAS :<p>(R)-(+)-Bay-K-8644, a Ca2+ channel agonist, is a dihydropyridine agonist that induces central respiratory depression and inhibits platelet activation in cats.</p>Formule :C16H15F3N2O4Degré de pureté :96.51% - 96.51%Couleur et forme :SolidMasse moléculaire :356.3N-Palmitoyl Glycine
CAS :<p>Acyl amides like AEA modulate pain/inflammation. PalGly, similar to N-acyl ethanolamines, inhibits nociception and induces calcium influx in cells.</p>Formule :C18H35NO3Couleur et forme :SolidMasse moléculaire :313.48TPC2-A1-N
CAS :<p>TPC2-A1-N is a TPC2 small molecule agonist that can be used to detect different functions of TPC2 channels in intact cells.</p>Formule :C17H9Cl2F3N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :401.17(S)-Lercanidipine D3 hydrochloride
CAS :<p>(S)-Lercanidipine D3 hydrochloride is a deuterium labeled Lercanidipine D3 hydrochloride. (S)-Lercanidipine hydrochloride is an agent of antihypertensive.</p>Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.21(R)-Nicardipine
CAS :<p>(R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Formule :C26H29N3O6Couleur et forme :SolidMasse moléculaire :479.53β-Cyfluthrin
CAS :<p>β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.</p>Formule :C22H18Cl2FNO3Couleur et forme :SolidMasse moléculaire :434.29(R)-Lercanidipine-d3 hydrochloride
CAS :<p>(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.</p>Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.21YM-244769
CAS :<p>YM-244769 (3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-) is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3)</p>Formule :C26H22FN3O3Degré de pureté :95.62%Couleur et forme :SolidMasse moléculaire :443.47Nicardipine-d3 hydrochloride
CAS :<p>Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.</p>Formule :C26H30ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :519YM-244769 dihydrochloride
CAS :<p>YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.</p>Formule :C26H24Cl2FN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :516.39HSK16149
CAS :<p>HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.</p>Formule :C12H19NO2Couleur et forme :SolidMasse moléculaire :209.28MRS1845
CAS :<p>MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).</p>Formule :C21H22N2O6Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :398.41(S)-Nicardipine
CAS :<p>(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Formule :C26H29N3O6Couleur et forme :SolidMasse moléculaire :479.53Almorexant hydrochloride
CAS :<p>Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.</p>Formule :C29H32ClF3N2O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :549.02Norverapamil-d7
CAS :<p>Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .</p>Formule :C26H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :447.62Hexadecylphosphoserine TFA
<p>Hexadecylphosphoserine is a type of phospholipid molecule that incorporates a long-chain alkyl group (hexadecyl) and a phosphatidylserine group, granting it high affinity for cell membranes. This compound exhibits antitumor activity by modulating [Ca++]i and related signaling pathways, making it useful for breast cancer research.</p>Formule :C21H41F3NO8PCouleur et forme :SolidMasse moléculaire :523.52Dronedarone
CAS :<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Formule :C31H44N2O5SDegré de pureté :98.85% - 99.58%Couleur et forme :SolidMasse moléculaire :556.76Azumolene
CAS :<p>Azumolene (EU4093 free base)</p>Formule :C13H9BrN4O3Degré de pureté :98.1% - 98.35%Couleur et forme :SolidMasse moléculaire :349.14Ginsenoside Rd
CAS :<p>Ginsenoside Rd (Gypenoside VIII) may have properties that inhibit or prevent the growth of tumors.</p>Formule :C48H82O18Degré de pureté :99.13% - 99.92%Couleur et forme :SolidMasse moléculaire :947.15JNJ-26990990
CAS :<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Formule :C9H10N2O2S2Degré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :242.32Efonidipine
CAS :<p>Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.</p>Formule :C34H38N3O7PDegré de pureté :98.35% - 99.47%Couleur et forme :SolidMasse moléculaire :631.66Bepridil hydrochloride
CAS :<p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>Formule :C24H35ClN2ODegré de pureté :99.45% - 99.68%Couleur et forme :SolidMasse moléculaire :4032,5-Di-tert-butylhydroquinone
CAS :<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Formule :C14H22O2Degré de pureté :97.11%Couleur et forme :PelletslargecrystalsMasse moléculaire :222.32DHBP dibromide
CAS :<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Formule :C24H38Br2N2Degré de pureté :99.73%Couleur et forme :Yellow To Yellow-Green Powder Or FlakesMasse moléculaire :514.38L-Phenylalanine
CAS :<p>L-Phenylalanine (3-Phenyl-L-alanine) is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.</p>Formule :C9H11NO2Degré de pureté :99.37% - 99.87%Couleur et forme :Solid CrystallineMasse moléculaire :165.19GSK1016790A
CAS :<p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>Formule :C28H32Cl2N4O6S2Degré de pureté :97.37% - 99.38%Couleur et forme :SolidMasse moléculaire :655.61Propiverine hydrochloride
CAS :<p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>Formule :C23H30ClNO3Degré de pureté :99.93%Couleur et forme :White Crystalling PowerMasse moléculaire :403.94Dantrolene sodium hemiheptahydrate
CAS :<p>Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium</p>Formule :C14H9N4NaO5·5H2ODegré de pureté :99.72%Couleur et forme :Orange PowderMasse moléculaire :399.29Pranidipine
CAS :<p>Pranidipine (OPC-13340) is a novel, long-acting 1,4-dihydropyridine calcium channel blocker.</p>Formule :C25H24N2O6Degré de pureté :99.95%Couleur et forme :Yellow SolidMasse moléculaire :448.47Aranidipine
CAS :<p>Aranidipine (MPC1304) (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.</p>Formule :C19H20N2O7Degré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :388.37(±)-Praeruptorin A
CAS :<p>(±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation.</p>Formule :C21H22O7Degré de pureté :98.9% - 99.73%Couleur et forme :SolidMasse moléculaire :386.4(+)-Kavain
CAS :<p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>Formule :C14H14O3Degré de pureté :97% - ≥95%Couleur et forme :White Fine PowderMasse moléculaire :230.26Suvecaltamide
CAS :<p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>Formule :C20H23F3N2O2Degré de pureté :99.29% - 99.70%Couleur et forme :SolidMasse moléculaire :380.4NS-638
CAS :<p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>Formule :C15H11ClF3N3Degré de pureté :98.44%Couleur et forme :SolidMasse moléculaire :325.72NFAT Inhibitor-2
CAS :<p>NFAT Inhibitor-2 is a compound used as a molecular building block.</p>Formule :C22H20F2N2O4SDegré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :446.47Efonidipine hydrochloride monoethanolate
CAS :<p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>Formule :C36H45ClN3O8PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :714.18Praeruptorin E
CAS :<p>Praeruptorin C/E relaxes arteries, reduces heart contractility, acting like calcium blockers. D/E protect mice from acid lung injury by halting PMNs and IL-6.</p>Formule :C24H28O7Degré de pureté :98.04% - 99.95%Couleur et forme :SolidMasse moléculaire :428.47SR33805
CAS :<p>SR33805 is a potent antagonist of Ca2+ channel(EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively)</p>Formule :C32H40N2O5SDegré de pureté :99.15%Couleur et forme :SolidMasse moléculaire :564.74Ibutilide Fumarate
CAS :<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Formule :(C20H36N2O3S)2·C4H4O4Degré de pureté :99.68% - 99.74%Couleur et forme :SolidMasse moléculaire :885.23Azumolene sodium anhydrous
CAS :<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Formule :C13H8BrN4NaO3Couleur et forme :SolidMasse moléculaire :371.13Argireline
CAS :<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formule :C34H60N14O12SDegré de pureté :96.79% - 99.65%Couleur et forme :White PowderMasse moléculaire :888.99TGR5 Receptor Agonist
CAS :<p>TGR5 is a potent TGR5(GPCR19) agonist.</p>Formule :C18H14Cl2N2O2Degré de pureté :99.77% - ≥95%Couleur et forme :SolidMasse moléculaire :361.22Ethacrynic acid
CAS :<p>Ethacrynic acid (Edecrin) 是谷胱甘肽 S-转移酶抑制剂，也是NF-κB 信号传导途径的有效抑制剂，并且还调节白三烯的形成。它还可抑制 L 型电压依赖性和储存操作的钙通道，从而导致气道平滑肌细胞松弛。它是利尿剂，具有抗炎特性，可减轻类维生素 A 诱导的小鼠耳部水肿。</p>Formule :C13H12Cl2O4Degré de pureté :98.61% - 99.85%Couleur et forme :Crystals Physical Description White Solid (Ntp 1992)Masse moléculaire :303.14Glaucine
CAS :<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Formule :C21H25NO4Degré de pureté :99.42% - 99.56%Couleur et forme :SolidMasse moléculaire :355.43HC-056456
CAS :<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Formule :C12H6N2O4S2Degré de pureté :99.62% - 99.65%Couleur et forme :SolidMasse moléculaire :306.32Psoralenoside
CAS :<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Formule :C17H18O9Degré de pureté :99.03% - 99.49%Couleur et forme :SolidMasse moléculaire :366.32Quadrol
CAS :<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formule :C14H32N2O4Degré de pureté :99.91% - 99.92%Couleur et forme :Viscous Liquid Liquid ViscousMasse moléculaire :292.41Mirogabalin
CAS :<p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>Formule :C12H19NO2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :209.28Efonidipine hydrochloride
CAS :<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Formule :C34H39ClN3O7PCouleur et forme :SolidMasse moléculaire :668.12NP118809
CAS :<p>NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).</p>Formule :C32H32N2ODegré de pureté :97.74% - 98.68%Couleur et forme :SolidMasse moléculaire :460.61Praeruptorin C
CAS :<p>Praeruptorin C: an antioxidant, calcium antagonist, protects neurons, reduces vascular hypertrophy, affects cellular signals.</p>Formule :C24H28O7Degré de pureté :99.6% - 99.92%Couleur et forme :SolidMasse moléculaire :428.47CDN1163
CAS :<p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>Formule :C20H20N2O2Degré de pureté :99.83% - ≥95%Couleur et forme :SolidMasse moléculaire :320.39ABT-639 hydrochloride
CAS :<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Formule :C20H21Cl2F2N3O3SCouleur et forme :SolidMasse moléculaire :492.36Pyr6
CAS :<p>Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx</p>Formule :C17H9F7N4ODegré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :418.27Gabapentin hydrochloride
CAS :<p>Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.</p>Formule :C9H17NO2·HClDegré de pureté :99.71%Couleur et forme :Off-White SolidMasse moléculaire :207.7Pinaverium bromide
CAS :<p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>Formule :C26H41Br2NO4Degré de pureté :99.52%Couleur et forme :White Crystalline PowderMasse moléculaire :591.42Taurolithocholic acid sodium salt
CAS :<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Formule :C26H44NNaO5SDegré de pureté :99.79% - 99.93%Couleur et forme :SolidMasse moléculaire :505.69FPL64176
CAS :<p>FPL64176 is a L-type calcium channels activator.</p>Formule :C22H21NO3Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :347.41
