Canal calcique
Les canaux calciques sont des protéines membranaires qui régulent le flux d'ions calcium dans et hors des cellules, ce qui est essentiel pour diverses fonctions cellulaires, y compris la contraction musculaire, la libération de neurotransmetteurs et l'expression génique. La dysrégulation de l'activité des canaux calciques est associée à des conditions telles que l'hypertension, les arythmies cardiaques et les troubles neurologiques. Chez CymitQuimica, nous proposons une large sélection de modulateurs des canaux calciques pour soutenir vos recherches en santé cardiovasculaire, neurobiologie et transduction du signal.
573 produits trouvés pour "Canal calcique"
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Mast cell degranulating peptide (28-49)
CAS :Mast cell degranulating peptide (28-49) is a bee venom depolarizer that can improve the cGMP content of cerebellum tablets in mice.
Formule :C110H196N40O24S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2591.25NAADP sodium
NAADP sodium is a Ca2+ motor second messenger that targets Ca(2+) channels and can be used to study cancer and immune dysfunction.Formule :C21H27N6O18P3Couleur et forme :SolidMasse moléculaire :744.39D-myo-Inositol-1,3,4,5-tetraphosphate (sodium salt)
CAS :Ins(1,3,4,5)-P4, made via Ins(1,4,5)P3 phosphorylation, boosts calcium by opening ER and plasma membrane channels.Formule :C6H8Na8O18P4Couleur et forme :SolidMasse moléculaire :675.93Mipsagargin
CAS :Mipsagargin (G-202) is a new antibiotic that inhibits DNA biosynthesis.Formule :C66H100N6O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1409.52G-Glu-Ser
CAS :G-Glu-Ser is a calcium receptor activator and Flavor-enriching agent.Formule :C8H14N2O6Couleur et forme :SolidMasse moléculaire :234.21(R)-IDHP
CAS :(R)-IDHP, a salvia derivative, relaxes blood vessels by blocking calcium channels, aiding cardiovascular research.Formule :C12H16O5Couleur et forme :SolidMasse moléculaire :240.25CALP3
CAS :Cell-permeable CaM agonist, binds EF-hand, activates phosphodiesterase without Ca2+, inhibits Ca2+ toxicity, IC50=33μM.Formule :C44H68N10O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :881.08Amlodipine aspartic acid impurity
CAS :Amlodipine aspartic acid: a calcium blocker with antihypertensive effects; contains specific impurities.Formule :C24H29ClN2O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :524.95Ins(1,4,5)-P3 hexapotassium salt
CAS :D-myo-Inositol 1,4,5-trisphosphate hexapotassium salt is promotes endoplasmic The second messenger of net calcium ions.Formule :C6H9K6O15P3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :648.64GTx1-15
GTx1-15, an inhibitor cystine knot (ICK) peptide, antagonizes the voltage-dependent calcium channel Cav3.1, as well as voltage-dependent sodium channels Nav1.3Formule :C176H271N53O45S7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4073.821,4-Dihydropyridine
1,4-Dihydropyridine acts as an antagonist for calcium channels (calcium channel), specifically blocking the L-type calcium channels. This action reduces the influx of calcium ions into cardiac and vascular smooth muscle cells, consequently decreasing cardiac contractility and heart rate, dilating blood vessels, and lowering blood pressure.Formule :C12H17NO4Couleur et forme :SolidMasse moléculaire :239.27CALP3 TFA(261969-05-5 free base)
CALP3 TFA is a potent Ca2+ channel blocker that activates EF-hand motifs of Ca2+-binding proteins.Formule :C46H69F3N10O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :995.1Nesiritide acetate
CAS :Nesiritide, a 32-amino acid natriuretic peptide and recombinant form of human brain natriuretic peptide, enhances vasorelaxation ex vivo in porcine hearts from an acute coronary occlusion model when given as a 2 µg/kg bolus dose followed by a 0.01 µg/kg per minute infusion, facilitated by the calcium ionophore A23187. Formulations containing nesiritide have been utilized in managing congestive heart failure.Formule :C143H244N50O42S4C2H4O2Couleur et forme :SolidMasse moléculaire :3524.1ω-Conotoxin CnVIIA
CAS :ω-Conotoxin CnVIIA, a 27-amino-acid neuropeptide toxin, serves as an N-type calcium current blocker [1].Formule :C110H179N39O36S7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2848.29ω-Conotoxin GVIA
CAS :Peptide neurotoxin; selectively and reversibly blocks N-type calcium channels (IC50 = 0.15 nM). Reduces (RS)-3,5-DHPG -induced long term depression in vivo.Formule :C120H182N38O43S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3037OPC 8490 free base
CAS :OPC 8490 free base is a positive inotropic vasodilator and a cardiotonic agent that can be used to study cardiovascular diseases.Formule :C24H27N3O3Degré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :405.49RyRs activator 5
Compound A-1 (RyRs activator 5) is an efficacious agonist of ryanodine receptors, exhibiting activity against Spodoptera frugiperda [1].Couleur et forme :Odour SolidCalcium Channel antagonist 5
CAS :Calcium Channel antagonist5 (compound 32) is a calcium channel antagonist with a pIC50 of 5.50.Formule :C17H18N2O6Couleur et forme :SolidMasse moléculaire :346.34Lyso-Globotriaosylceramide (d18:1)
CAS :Lyso-Gb3, lacking fatty acyl, binds Stx1 with cholesterol and phosphatidylcholine, not Stx2; lowers neutrophil viability; accumulates in Fabry disease.Formule :C36H67NO17Couleur et forme :SolidMasse moléculaire :785.922ω-conotoxin MoVIA
ω-Conotoxin MVIIA is a potent, selective inhibitor of Ca_v2.2, exhibiting an IC_50 of 0.33 μM in the SH-SY5Y fluorimetric hCa_v2.2 assay [1].Formule :C147H233N45O47S7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3607.15Ion Channel Targeted Library
A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;
Couleur et forme :Odour SolidNSC156529
CAS :NSC156529 suppresses AKT1, reduces cancer cell growth in vitro, and inhibits prostate tumors in vivo.Formule :C28H21ClS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.05ω-Conotoxin SO3
CAS :ω-Conotoxin SO3 is an analgesic peptide that functions as an antagonist to N-type voltage-sensitive calcium channels, and can be isolated from the venom ofFormule :C100H166N36O31S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2561PDDHV
CAS :PDDHV: a capsaicin-like vanilloid selective for rat TRPV1; induces Ca2+ uptake in neurons, EC50 of 70 nM.Formule :C49H72O11Couleur et forme :SolidMasse moléculaire :837.0917R(18S)-EpETE
CAS :17R(18S)-EpETE: Oxylipin, eicosapentaenoic acid metabolite, activates BKCa channels, has negative chronotropic effects.Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.457ProTx-I
CAS :Selective blocker for CaV3.1 (IC50 = 0.2 μM), CaV3.2 (31.8 μM), also inhibits NaV1.8 and blocks KV2.1 channels.
Formule :C171H245N53O47S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3987.51FS-2
FS-2 is a potent, specific inhibitor of L-type CaV channels, effectively impeding high K+ or glucose-induced L-type Ca2+ influx in RIN beta cells [1].Formule :C297H462N92O86S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7018.061-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS :1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(
Formule :C5H10ClNO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :151.59Glutarimide
CAS :Compound PDK0025, with CAS No. 1121-89-7, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0025 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C5H7NO2Couleur et forme :White SolidMasse moléculaire :113.11Elgodipine
CAS :Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.Formule :C29H33FN2O6Degré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :524.58Cavα2δ-IN-1
CAS :Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a KiFormule :C18H27N5OCouleur et forme :SolidMasse moléculaire :329.448Calciseptin
CAS :Calciseptine, a neurotoxin isolated from the Black Mamba (Dendroaspis p.Formule :C299H468N90O87S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7036.12BTT-266
CAS :BTT-266 is a blocker of voltage-gated calcium channel for pain management.
Formule :C34H28N4O4Degré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :556.61ω-Conotoxin CVIE
ω-Conotoxin CVIE selectively inhibits voltage-gated Ca^2+ channels (Ca_v 2.2) [1].Formule :C98H164N40O34S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2638.99ω-Hexatoxin-Hv1a
CAS :ω-Hexatoxin-Hv1a, a neurotoxin extracted from the venom of the spider Hadronyche versuta, inhibits voltage-gated calcium channels [1] [2].Formule :C162H247N49O61S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4049.38ω-Conotoxin Bu8
ω-Conotoxin Bu8 is a 25-amino-acid-residue ω-conotoxin that features three disulfide bridges.Formule :C103H174N42O35S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2753.13PACAP-38 (31-38), human, mouse, rat TFA
PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.Formule :C49H84F3N17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1176.29wt hMLN
Wild-type human myoregulin (wt hMLN) is a microprotein that inhibits the sarcoplasmic reticulum Ca²⁺ pump (SERCA), playing a crucial role in the regulation ofFormule :C245H404N54O66SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :5194.22Calcium Ionophore I
CAS :Calcium Ionophore I has a wide range of applications in life science related research.Formule :C38H72N2O8Couleur et forme :SolidMasse moléculaire :685.0ω-Tbo-IT1
ω-Tbo-IT1, a peptide toxin extracted from the venom of Tibellus oblongus, functions as an inhibitor of insect calcium channels [1].Formule :C171H285N61O53S9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4332.05IP3RPEP6
CAS :IP3RPEP6 serves as a competitive inhibitor of IP3R. Its IC50 values for IP3R1, IP3R2, and IP3R3 are 9.0 μM, 3.9 μM, and 4.3 μM, respectively. This compound does not affect ryanodine receptors and Cx43 hemichannels, and it is capable of modulating intracellular calcium signaling.Formule :C49H79N15O24Couleur et forme :SolidMasse moléculaire :1262.24Myr-TAT-CBD3
Myr-TAT-CBD3, a CRMP2-CaV2.2 interaction inhibitor, has been shown to significantly attenuate carrageenan-induced thermal hypersensitivity and reverse thermalFormule :C148H269N59O33Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3403.09ω-Conotoxin MVIIC
CAS :Peptide neurotoxin; wide spectrum blocker of N, P and Q type calcium channels.Formule :C106H178N40O32S7Degré de pureté :98%Couleur et forme :White Lyophilised SolidMasse moléculaire :2749D-myo-Inositol-1,2-diphosphate (sodium salt)
CAS :Ins(1,2)P2, a less potent InsP isomer than Ins(1,4,5)P3, acts as a secondary messenger in cellular signal transmission.Formule :C6H12Na2O12P2Couleur et forme :SolidMasse moléculaire :384.08Ethacrynic acid D5
CAS :Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.Formule :C13H12Cl2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.17Flosatidil
CAS :Flosatidil is a small molecule voltage-gated calcium channel complex (VDCCs) blocker for the treatment of neurological disorders and cardiovascular diseases,Formule :C26H34F3N3O3SDegré de pureté :99.87% - 99.99%Couleur et forme :SolidMasse moléculaire :525.63Imperatoxin A TFA
Imperatoxin A TFA, a peptide toxin derived from the venom of the African scorpion Pandinus imperator, acts as an activator of Ca2+-release channels/ryanodine receptors (RyRs). It facilitates the influx of Ca2+ from the sarcoplasmic reticulum into the cell.Formule :C148H254N58O45S6·xC2HF3O2Couleur et forme :SolidMasse moléculaire :3758.35 (free base)Myoregulin
Myoregulin (MLN peptide), a regulin family member, modulates muscle performance through intracellular calcium handling.Formule :C239H391N53O67S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5175.17Triphenylethylene
CAS :Compound PDK0283, with CAS No. 58-72-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0283 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C20H16Couleur et forme :White PowderMasse moléculaire :256.34Calcicludine
CAS :Calcicludine, a protein toxin derived from the green mamba (Dendroaspis angusticeps) venom, selectively inhibits high-voltage-activated, particularly L-type,Formule :C321H476N86O78S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :6980.13Sulcardine 2HCl
CAS :Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 channels and can be used to study atrial fibrillation.Formule :C24H35Cl2N3O4SDegré de pureté :99.33% - 99.76%Couleur et forme :SoildMasse moléculaire :532.523Ziconotide
CAS :Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.Formule :C102H172N36O32S7Degré de pureté :98%Couleur et forme :White PowderMasse moléculaire :2639.13Budiodarone tartrate
CAS :Budiodarone tartrate (ATI-2042 tartrate) is an antiarrhythmic agent that inhibits calcium channels, and can be used in atrial fibrillation research.Formule :C31H37I2NO11Degré de pureté :97.44%Couleur et forme :SolidMasse moléculaire :853.44Ref: TM-T74678
1mg166,00€5mg402,00€10mg652,00€25mg1.238,00€50mg1.932,00€100mg2.721,00€1mL*10mM (DMSO)626,00€ω-Conotoxin FVIA
ω-Conotoxin FVIA is an inhibitor of N-type Ca²⁺ channels (Caᵥ2.2), shown to alleviate mechanical and thermal pain abnormalities in a rat model of caudal nerveFormule :C98H164N36O33S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2566.96Calcium Channel Compound Library
A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening;Couleur et forme :Odour SolidRef: TM-L7200
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demanderω-Agatoxin TK
CAS :Selective blocker of CaV2.1 P/Q-type calcium channels.Formule :C215H337N65O70S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5273.02Huwentoxin I
CAS :Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.Formule :C161H246N48O44S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3750.36Ser-Ala-alloresact acetate
Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.Formule :C44H75N13O16S2Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :1106.28Vesnarinone HCl
Vesnarinone HCl is an oral PDE3 inhibitor improving heart contractility, affecting calcium and potassium flux. Used in heart failure research.Formule :C22H26ClN3O4Degré de pureté :99.17%Couleur et forme :SoildMasse moléculaire :431.91Myoregulin TFA
Myoregulin (MLN peptide) TFA, belonging to the regulin family, is a regulator of muscle performance through modulation of intracellular calcium dynamics.Formule :C239H391N53O67S3·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5175.17 (free base)(±)5(6)-DiHETE
CAS :Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.Formule :C20H32O4Couleur et forme :SolidMasse moléculaire :336.472Chlorocresol
CAS :Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.Formule :C7H7ClOCouleur et forme :SolidMasse moléculaire :142.58Ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate
CAS :ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate inhibits NAD(P)H: quinone oxidoreductase 1.Formule :C12H10ClNO3Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :251.67Caloxin 3A1
Caloxin 3A1, a biologically active peptide, is a member of the caloxins, which are inhibitors of the extracellular plasma membrane (PM) Ca2+ pumps.Formule :C83H126N22O30Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1912.02Cyclic ADP-ribose ammonium
cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.Couleur et forme :Liquidω-Conotoxin CVIF
ω-Conotoxin CVIF is a selective inhibitor of Ca v 2.2 channels, demonstrating an IC50 value of 34.3 nM in isolated rat DRG neurons.Formule :C101H170N40O33S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2665.07Levamlodipine besylate Hemipentahydrate
CAS :Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.Formule :C20H25ClN2O5·C6H6O3SH2OCouleur et forme :SolidMasse moléculaire :1224.18MCU-i11
CAS :MCU-i11 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.Formule :C28H28N4O5SDegré de pureté :98.3%Couleur et forme :SolidMasse moléculaire :532.61Ref: TM-T9960
1mg152,00€5mg340,00€10mg485,00€25mg802,00€50mg1.099,00€100mg1.485,00€1mL*10mM (DMSO)400,00€KT-362 free base
CAS :KT-362 is a calcium channel blocker with antihypertensive properties that can be used in the study of cardiovascular disease.Formule :C22H28N2O3SDegré de pureté :99.91%Couleur et forme :SoildMasse moléculaire :400.53MMK 1
CAS :Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.Formule :C75H123N19O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1610.97Candidalysin
CAS :Candidalysin is a cytolytic peptide toxin initially isolated from *Candida albicans*, exhibiting both toxic and non-toxic properties. It activates epithelial cell signaling pathways by interacting with the epithelial growth factor receptor (EGFR) on host cells, leading to the activation of matrix metalloproteinases (MMP) and calcium ion influx, which results in inflammatory responses and immune cell recruitment. Additionally, Candidalysin exhibits cytotoxicity by causing membrane damage to host cells.Formule :C153H266N38O38S2Couleur et forme :SolidMasse moléculaire :3310.11Flunarizine
CAS :Flunarizine is an orally administered peripheral vasodilator, a dual blocker of voltage-gated Na+/Ca2+ channels and a D2 dopamine receptor antagonist.Formule :C26H26F2N2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :404.50Fasudil
CAS :Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.Formule :C14H17N3O2SDegré de pureté :99.79% - 99.84%Couleur et forme :SolidMasse moléculaire :291.37Lnd 796
CAS :Lnd 796 is an aminosteroid related to LND 623.Formule :C27H45NO7Couleur et forme :SolidMasse moléculaire :495.65Maurocalcine TFA
Maurocalcine TFA acts as an agonist for ryanodine receptor (RyR) channels 1, 2, and 3, demonstrating cell-penetrating capabilities. It induces binding of [3H]ryanodine to RyR1 with an EC50 of 2558 nM and exhibits an apparent affinity of 14 nM for RyR2. This compound is applicable for in vivo cell tracking or other cellular imaging techniques.Formule :C156H270N56O46S6·xC2HF3O2Couleur et forme :SolidMasse moléculaire :3858.55 (free base)PD 0299685
CAS :PD 0299685 is a potent α2δ ligand of the Ca2+ channel for the treatment of interstitial cystitis.Formule :C10H21NO2Degré de pureté :97.20%Couleur et forme :SoildMasse moléculaire :187.28WU-07047
CAS :WU-07047 is a simplified analog of the selective Gαq/11 inhibitor YM-25489.Formule :C39H58N4O11Couleur et forme :SolidMasse moléculaire :758.90N-Palmitoyl Glycine
CAS :Acyl amides like AEA modulate pain/inflammation. PalGly, similar to N-acyl ethanolamines, inhibits nociception and induces calcium influx in cells.Formule :C18H35NO3Couleur et forme :SolidMasse moléculaire :313.48YM-244769 dihydrochloride
CAS :YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.Formule :C26H24Cl2FN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :516.39YM-244769
CAS :YM-244769 (3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-) is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3)Formule :C26H22FN3O3Degré de pureté :95.62%Couleur et forme :SolidMasse moléculaire :443.47MRS1845
CAS :MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).Formule :C21H22N2O6Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :398.41Almorexant hydrochloride
CAS :Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.Formule :C29H32ClF3N2O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :549.02(R)-(+)-Bay-K-8644
CAS :(R)-(+)-Bay-K-8644, a Ca2+ channel agonist, is a dihydropyridine agonist that induces central respiratory depression and inhibits platelet activation in cats.
Formule :C16H15F3N2O4Degré de pureté :96.51% - 96.51%Couleur et forme :SolidMasse moléculaire :356.3Catharanthine
CAS :Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).Formule :C21H24N2O2Degré de pureté :99.11%Couleur et forme :White PowderMasse moléculaire :336.43CCT129957
CAS :CCT129957 is a novel and potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of about 3 μM and a GC50 of 15 μM.CCT129957 exhibits anticancer activity andFormule :C17H15N3O3Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :309.32Ref: TM-T14903
1mg44,00€5mg93,00€10mg126,00€25mg220,00€50mg330,00€100mg497,00€500mg1.054,00€1mL*10mM (DMSO)92,00€TPC2-A1-N
CAS :TPC2-A1-N is a TPC2 small molecule agonist that can be used to detect different functions of TPC2 channels in intact cells.Formule :C17H9Cl2F3N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :401.17(S)-Lercanidipine D3 hydrochloride
CAS :(S)-Lercanidipine D3 hydrochloride is a deuterium labeled Lercanidipine D3 hydrochloride. (S)-Lercanidipine hydrochloride is an agent of antihypertensive.Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.21Norverapamil-d7 HCl
CAS :Norverapamil-d7 HCl (D591-d7 HCl) is a 2H-labeled Norverapamil HCl, a calcium channel blocker and P-gp inhibitor, also a coronary vasodilator.Formule :C26H37ClN2O4Couleur et forme :SolidMasse moléculaire :484.08(R)-Nicardipine
CAS :(R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).Formule :C26H29N3O6Couleur et forme :SolidMasse moléculaire :479.53β-Cyfluthrin
CAS :β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.Formule :C22H18Cl2FNO3Couleur et forme :SolidMasse moléculaire :434.29(R)-Lercanidipine-d3 hydrochloride
CAS :(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :651.21Nicardipine-d3 hydrochloride
CAS :Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.Formule :C26H30ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :519HSK16149
CAS :HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.Formule :C12H19NO2Couleur et forme :SolidMasse moléculaire :209.28A 839977
CAS :A 839977 is a P2X7 receptor antagonist with analgesic activity that inhibits BzATP-induced calcium efflux from the P2X7 receptor for the study of renal fibrosisFormule :C19H14Cl2N6ODegré de pureté :98.01%Couleur et forme :SolidMasse moléculaire :413.26(S)-Nicardipine
CAS :(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).Formule :C26H29N3O6Couleur et forme :SolidMasse moléculaire :479.53Norverapamil-d7
CAS :Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .Formule :C26H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :447.62Hexadecylphosphoserine TFA
Hexadecylphosphoserine is a type of phospholipid molecule that incorporates a long-chain alkyl group (hexadecyl) and a phosphatidylserine group, granting it high affinity for cell membranes. This compound exhibits antitumor activity by modulating [Ca++]i and related signaling pathways, making it useful for breast cancer research.Formule :C21H41F3NO8PCouleur et forme :SolidMasse moléculaire :523.52Magnesium sulfate
CAS :Magnesium sulfate: anticonvulsant for eclampsia, tocolytic agent.Formule :MgSO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :120.37Etripamil
CAS :Etripamil is a fast-acting intranasal L-type calcium-channel blocker for Paroxysmal Supraventricular Tachycardia.Formule :C27H36N2O4Degré de pureté :99.47% - 99.83%Couleur et forme :SolidMasse moléculaire :452.59Ref: TM-T15257
1mg52,00€2mg74,00€5mg110,00€10mg169,00€25mg295,00€50mg447,00€100mg670,00€200mg1.054,00€Dronedarone
CAS :Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Formule :C31H44N2O5SDegré de pureté :98.85% - 99.99%Couleur et forme :SolidMasse moléculaire :556.76
