Canal calcique
Les canaux calciques sont des protéines membranaires qui régulent le flux d'ions calcium dans et hors des cellules, ce qui est essentiel pour diverses fonctions cellulaires, y compris la contraction musculaire, la libération de neurotransmetteurs et l'expression génique. La dysrégulation de l'activité des canaux calciques est associée à des conditions telles que l'hypertension, les arythmies cardiaques et les troubles neurologiques. Chez CymitQuimica, nous proposons une large sélection de modulateurs des canaux calciques pour soutenir vos recherches en santé cardiovasculaire, neurobiologie et transduction du signal.
573 produits trouvés pour "Canal calcique"
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Levamlodipine besylate Hemipentahydrate
CAS :Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.Formule :C20H25ClN2O5·C6H6O3SH2OCouleur et forme :SolidMasse moléculaire :1224.181-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS :1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(
Formule :C5H10ClNO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :151.59sFTX-3.3
CAS :sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.Formule :C12H29N7OCouleur et forme :SolidMasse moléculaire :287.412WU-07047
CAS :WU-07047 is a simplified analog of the selective Gαq/11 inhibitor YM-25489.Formule :C39H58N4O11Couleur et forme :SolidMasse moléculaire :758.90SNX-482
CAS :Potent CaV2.3 calcium channel blocker, selective, voltage-dependent, with 30 nM IC50. Offers antinociceptive effects on C and Aδ fibres.Formule :C192H274N52O60S7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4495.01ω-Conotoxin FVIA
ω-Conotoxin FVIA is an inhibitor of N-type Ca²⁺ channels (Caᵥ2.2), shown to alleviate mechanical and thermal pain abnormalities in a rat model of caudal nerveFormule :C98H164N36O33S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2566.96Ethacrynic acid D5
CAS :Ethacrynic acid: a diuretic, anti-inflammatory, inhibits calcium channels, GSTs, NF-kB pathway, and modulates leukotriene; has deuterium-labeled form.Formule :C13H12Cl2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.17Fasudil
CAS :Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.Formule :C14H17N3O2SDegré de pureté :99.79% - 99.84%Couleur et forme :SolidMasse moléculaire :291.37IP3RPEP6
CAS :IP3RPEP6 serves as a competitive inhibitor of IP3R. Its IC50 values for IP3R1, IP3R2, and IP3R3 are 9.0 μM, 3.9 μM, and 4.3 μM, respectively. This compound does not affect ryanodine receptors and Cx43 hemichannels, and it is capable of modulating intracellular calcium signaling.Formule :C49H79N15O24Couleur et forme :SolidMasse moléculaire :1262.24Lyso-Globotriaosylceramide (d18:1)
CAS :Lyso-Gb3, lacking fatty acyl, binds Stx1 with cholesterol and phosphatidylcholine, not Stx2; lowers neutrophil viability; accumulates in Fabry disease.Formule :C36H67NO17Couleur et forme :SolidMasse moléculaire :785.922Myoregulin
Myoregulin (MLN peptide), a regulin family member, modulates muscle performance through intracellular calcium handling.Formule :C239H391N53O67S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5175.17Flunarizine
CAS :Flunarizine is an orally administered peripheral vasodilator, a dual blocker of voltage-gated Na+/Ca2+ channels and a D2 dopamine receptor antagonist.Formule :C26H26F2N2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :404.50MCU-i11
CAS :MCU-i11 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.Formule :C28H28N4O5SDegré de pureté :98.3%Couleur et forme :SolidMasse moléculaire :532.61Ref: TM-T9960
1mg152,00€5mg340,00€10mg485,00€25mg802,00€50mg1.099,00€100mg1.485,00€1mL*10mM (DMSO)400,00€D-myo-Inositol-1,4,5,6-tetraphosphate (sodium salt)
CAS :Ins(1,4,5,6)-P4, a signal-transducing inositol oligophosphate, increases 2-14x in cells post-Salmonella infection and modulates EGF signaling.Formule :C6H12Na4O18P4Couleur et forme :SolidMasse moléculaire :588Calciseptin
CAS :Calciseptine, a neurotoxin isolated from the Black Mamba (Dendroaspis p.Formule :C299H468N90O87S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7036.12Myomodulin
CAS :Myomodulin is a neuropeptide present in molluscs, insects, and gastropods.Myomodulin is present in two identified aplysia neurons that contain myomodulin A theFormule :C36H67N11O8S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :846.12Calcium Channel antagonist 5
CAS :Calcium Channel antagonist5 (compound 32) is a calcium channel antagonist with a pIC50 of 5.50.Formule :C17H18N2O6Couleur et forme :SolidMasse moléculaire :346.34TPC2-A1-N
CAS :TPC2-A1-N is a TPC2 small molecule agonist that can be used to detect different functions of TPC2 channels in intact cells.Formule :C17H9Cl2F3N2O2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :401.17(R)-(+)-Bay-K-8644
CAS :(R)-(+)-Bay-K-8644, a Ca2+ channel agonist, is a dihydropyridine agonist that induces central respiratory depression and inhibits platelet activation in cats.
Formule :C16H15F3N2O4Degré de pureté :96.51% - 96.51%Couleur et forme :SolidMasse moléculaire :356.3Catharanthine
CAS :Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).Formule :C21H24N2O2Degré de pureté :99.11%Couleur et forme :White PowderMasse moléculaire :336.43
