Canal calcique
Les canaux calciques sont des protéines membranaires qui régulent le flux d'ions calcium dans et hors des cellules, ce qui est essentiel pour diverses fonctions cellulaires, y compris la contraction musculaire, la libération de neurotransmetteurs et l'expression génique. La dysrégulation de l'activité des canaux calciques est associée à des conditions telles que l'hypertension, les arythmies cardiaques et les troubles neurologiques. Chez CymitQuimica, nous proposons une large sélection de modulateurs des canaux calciques pour soutenir vos recherches en santé cardiovasculaire, neurobiologie et transduction du signal.
578 produits trouvés pour "Canal calcique".
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Gallopamil hydrochloride
CAS :Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.Formule :C28H41ClN2O5Degré de pureté :99.86%Couleur et forme :Yellow SolidMasse moléculaire :521.09Ref: TM-T11353L
1mg35,00€5mg70,00€1mL*10mM (DMSO)86,00€10mg95,00€25mg133,00€50mg173,00€100mg268,00€500mg655,00€Norverapamil
CAS :Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .Formule :C26H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.58CaV1.3 antagonist-1
CAS :CaV1.3 antagonist-1 is a selective CaV1.3L-type calcium channel antagonist useful for researching neurological disorders and cardiovascular diseases.Formule :C17H19ClN2O3Couleur et forme :SolidMasse moléculaire :334.8Dopropidil
CAS :Dopropidil: anti-angina calcium regulator with anti-ischemic properties in animal models.Formule :C20H35NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.5NC 1100
CAS :NC 1100 is a calcium channel antagonist.Formule :C27H34Cl2N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :505.48RS 30026
CAS :RS 30026 is a potent calcium channel agonist.Formule :C23H21NO4SCouleur et forme :SolidMasse moléculaire :407.48ITH-12575
CAS :ITH-12575 is an inhibitor of Mitochondrial Na+/Ca2+ exchange (mNCX). ITH12575 reduces Ca(2+) influx through CALHM1 at low micromolar concentrations.Formule :C18H18ClNOSDegré de pureté :99.53%Couleur et forme :White SolidMasse moléculaire :331.86ML218 hydrochloride
CAS :ML218 hydrochloride inhibits T-type Ca2+ channels Cav3.1-3.3; most effective on Cav3.2 and Cav3.3 (IC50s: 310 nM, 270 nM).Formule :C19H27Cl3N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.79Diltiazem malate
CAS :Diltiazem malate is an ACE inhibitor and non-dihydropyridine calcium channel blocker used in the treatment of hypertension.Formule :C26H32N2O9SCouleur et forme :SolidMasse moléculaire :548.60(R)-Amlodipine
CAS :(R)-Amlodipine is the R-enantiomer of Amlodipine and functions as an orally active dihydropyridine calcium channel blocker with antianginal properties.Formule :C20H25ClN2O5Degré de pureté :99.97%Couleur et forme :White SolidMasse moléculaire :408.88Palonidipine
CAS :Palonidipine is an antagonist of calcium, is potential for the therapy of angina-pectoris and hypertension.Formule :C29H34FN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :539.6BK 129
CAS :BK 129 is a local anesthetic with relaxant properties. BK 129 inhibits Ca2+ entry into the smooth muscle cell and Ca2+ release from sarcoplasmic reticulum.Formule :C22H36N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :392.53PD 122860
CAS :PD 122860 is a dihydropyridine enhancing heart contractility, altering ECG, and relaxing aortic rings.Formule :C23H20F3N3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :491.48Topiramate lithium
CAS :Topiramate lithium: antiepileptic, GluR5 antagonist, enhances GABA, inhibits kainate/AMPA, Na+/Ca2+ channels; ↑ K+ conductance; ↓ carbonic anhydrase.Formule :C12H20LiNO8SCouleur et forme :SolidMasse moléculaire :345.29YS-201
CAS :YS-201 is an antagonist of dihydropyridine-type calcium channel.Formule :C24H31N3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.52UK51656
CAS :UK51656 is an antagonist of calcium (IC50: 4 nM).Formule :C22H28ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :465.93Flordipine
CAS :Flordipine is used as a calcium channel blocker.Formule :C26H33F3N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.55JTV-519 free base
CAS :JTV-519 free base (K201 free base), recognized for its antiarrhythmic and cardioprotective properties, functions as a Ca2+-dependent blocker of sarcoplasmicFormule :C25H32N2O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :424.6TTA-Q6(isomer)
CAS :TTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective antagonist of the T-type Ca2+ channel.Formule :C20H15ClF3N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.8Hyperforin dicyclohexylammonium salt
CAS :Hyperforin dicyclohexylammonium is a TRPC6 activator and antidepressant that modulates Ca2+ levels.Formule :C47H75NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :718.10SQ-31765
CAS :SQ-31765 is a blocker of benzazepine calcium channel.Formule :C24H27F3N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :464.48BMS-192364
CAS :BMS-192364 is a bio-active chemical.Formule :C15H9ClF3N3O2Couleur et forme :SolidMasse moléculaire :355.70Diproteverine
CAS :Diproteverine is a calcium antagonist, it has antianginal property.Formule :C26H35NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.56GSK-5503A
CAS :GSK-5503A is a novel channel blocker of CRAC.Formule :C23H17F2N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :405.4Lemildipine
CAS :Lemildipine is a new blocker of dihydropyridine calcium entry.Formule :C20H22Cl2N2O6Couleur et forme :SolidMasse moléculaire :457.3GSK-5498A
CAS :GSK-5498A: Selective CARC blocker, inhibits release of mediators from mast cells and cytokines from T-cells (IC50, 1 μM).Formule :C18H11F6N3OCouleur et forme :SolidMasse moléculaire :399.29SOCE inhibitor 1
CAS :SOCE inhibitor 1 is a inhibitor of store-operated calcium entry (SOCE)(IC50 of 4.4 μM).Formule :C25H22F3N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :513.47(S)-Lercanidipine hydrochloride
CAS :(S)-Lercanidipine hydrochloride is the S-enantiomer of Lercanidipine hydrochloride. (S)-lercanidipine hydrochloride is a potent blocker of calcium channel.Formule :C36H42ClN3O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :648.19Anipamil
CAS :Anipamil is a long-acting blocker of calcium channel,and for the treatment of cardiovascular disease.Formule :C34H52N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.79Norbormide
CAS :Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker.Formule :C33H25N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :511.57YS-035 hydrochloride
CAS :inhibitor of outward K+ currentsFormule :C21H30ClNO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :395.92Clopimozide
CAS :Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.Formule :C28H28ClF2N3ODegré de pureté :98.99% - 99.66%Couleur et forme :White SolidMasse moléculaire :495.99Sulcardine sulfate
CAS :Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.Formule :C24H35N3O8S2Degré de pureté :98.74%Couleur et forme :SolidMasse moléculaire :557.68Gallopamil
CAS :Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.Formule :C28H40N2O5Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :484.63Ref: TM-T11353
1mg35,00€5mg74,00€1mL*10mM (DMSO)80,00€10mg113,00€25mg178,00€50mg268,00€100mg408,00€500mg888,00€Upacicalcet
CAS :Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.Formule :C11H14ClN3O6SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :351.76NecroX-5
CAS :NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.Formule :C27H39N3O9S3Degré de pureté :99.94%Couleur et forme :White SolidMasse moléculaire :645.81Ref: TM-T12204
100mgÀ demander1mg52,00€2mg70,00€5mg105,00€1mL*10mM (DMSO)149,00€10mg152,00€25mg235,00€50mg334,00€Fenoverine
CAS :Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.Formule :C26H25N3O3SDegré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :459.56Ref: TM-T62889
1mg66,00€5mg142,00€1mL*10mM (DMSO)145,00€10mg222,00€25mg447,00€50mg715,00€100mg1.063,00€200mg1.459,00€O-1602
CAS :O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatmentFormule :C17H22O2Degré de pureté :99.85%Couleur et forme :Yellow OilMasse moléculaire :258.36Ref: TM-T23097
1mg44,00€5mg95,00€1mL*10mM (DMSO)95,00€10mg137,00€25mg254,00€50mg358,00€100mg537,00€200mg762,00€AZD-1305
CAS :AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.Formule :C22H31FN4O4Degré de pureté :97.32% - 99.31%Couleur et forme :SolidMasse moléculaire :434.5Ref: TM-T30251
1mg92,00€5mg200,00€1mL*10mM (DMSO)225,00€10mg289,00€25mg447,00€50mg622,00€100mg850,00€200mg1.153,00€Ticolubant
CAS :Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.Formule :C23H19Cl2NO3SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :460.37Crobenetine
CAS :Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.Formule :C25H33NO2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :379.54DS16570511
CAS :DS16570511 is a novel, cell-permeable inhibitor targeting the mitochondrial calcium uniporter.Formule :C30H25Cl2N3O4Degré de pureté :98.34% - 98.45%Couleur et forme :White SolidMasse moléculaire :562.44Enecadin
CAS :Enecadin is a neuroprotective agent.Formule :C21H28FN3ODegré de pureté :98.53%Couleur et forme :White SolidMasse moléculaire :357.46JNJ-26489112
CAS :JNJ-26489112 is a CNS-active agent and an inhibitor of voltage-gated Na+ channels and N-type Ca2+ channels.Formule :C9H11ClN2O4SDegré de pureté :99.31%Couleur et forme :White SolidMasse moléculaire :278.71Opc 8490
CAS :Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.Formule :C30H35N3O10Degré de pureté :98.88%Couleur et forme :Yellow SolidMasse moléculaire :597.61Cerebrocrast
CAS :Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.Formule :C26H35F2NO7Degré de pureté :99.71%Couleur et forme :Yellow SolidMasse moléculaire :511.56Terflavoxate
CAS :Terflavoxate is a novel, orally active, semisynthetic statin microtubule inhibitor commonly used in combination with capecitabine.Formule :C26H29NO4Degré de pureté :99.76%Couleur et forme :Yellow SolidMasse moléculaire :419.51Ref: TM-T67964
1mg85,00€5mg170,00€1mL*10mM (DMSO)188,00€10mg245,00€25mg371,00€50mg532,00€100mg737,00€200mg982,00€Vatanidipine
CAS :Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lastingFormule :C41H42N4O6Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :686.8Ref: TM-T24932
1mg177,00€5mg430,00€10mg588,00€1mL*10mM (DMSO)692,00€25mg892,00€50mg1.198,00€100mg1.575,00€SERCA2a activator 1
CAS :SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.Formule :C32H29N3O4SDegré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :551.66Ref: TM-T16873
1mg177,00€5mg447,00€1mL*10mM (DMSO)533,00€10mg625,00€25mg982,00€50mg1.404,00€100mg1.963,00€CP-060
CAS :CP-060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.Formule :C30H42N2O5SDegré de pureté :99.54%Couleur et forme :Yellow OilMasse moléculaire :542.73Ref: TM-T10874
1mg225,00€5mg449,00€10mg605,00€1mL*10mM (DMSO)608,00€25mg900,00€50mg1.215,00€100mg1.639,00€200mg2.215,00€
