Récepteur GABA
Les récepteurs GABA sont les principaux récepteurs de neurotransmetteurs inhibiteurs du système nerveux central, jouant un rôle crucial dans la régulation de l'excitabilité neuronale et le maintien de l'équilibre entre excitation et inhibition. La dysfonction des récepteurs GABA est impliquée dans divers troubles neurologiques et psychiatriques, notamment l'épilepsie, l'anxiété et la dépression. Chez CymitQuimica, nous proposons une gamme complète de modulateurs des récepteurs GABA pour soutenir vos recherches en neurobiologie, santé mentale et développement thérapeutique.
371 produits trouvés pour "Récepteur GABA"
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Primidone (Standard)
CAS :Primidone (Standard) is the standard substance of Primidone, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential tremor, and psychiatric disorders.Formule :C12H14N2O2Couleur et forme :Crystals (Ntp 1992)Masse moléculaire :218.25Vigabatrin Hydrochloride
CAS :Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Formule :C6H11NO2·HClDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :165.62TACA
CAS :GABAA agonistFormule :C4H7NO2Degré de pureté :98%Couleur et forme :White SolidMasse moléculaire :101.1CGP 36742
CAS :CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Formule :C7H18NO2PCouleur et forme :SolidMasse moléculaire :179.2MRK-016
CAS :MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.Formule :C17H20N8O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :368.39L-655708
CAS :L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.Formule :C18H19N3O4Degré de pureté :99.36%Couleur et forme :PowderMasse moléculaire :341.36Furosemide-d5
CAS :Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.Formule :C12H11ClN2O5SCouleur et forme :SolidMasse moléculaire :335.78(2S)-6-Prenylnaringenin
CAS :(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formule :C20H20O5Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :340.37Acamprosate calcium
CAS :Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Formule :C10H20CaN2O8S2Degré de pureté :98% - 99.93%Couleur et forme :White Odorless Or Nearly Odorless PowderMasse moléculaire :400.48Acetoxyvalerensre
CAS :Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.
Formule :C17H24O4Degré de pureté :98.22%Couleur et forme :SolidMasse moléculaire :292.37Piperazine citrate
CAS :Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Formule :C24H46N6O14Degré de pureté :99.8%Couleur et forme :Crystals IndicationMasse moléculaire :642.65AZD7325
CAS :AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
Formule :C19H19FN4O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :354.38Ginkgolide A
CAS :Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.Formule :C20H24O9Degré de pureté :98.76% - 99.81%Couleur et forme :White PowderMasse moléculaire :408.40Guvacine hydrochloride
CAS :Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)Formule :C6H10ClNO2Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :163.602CL 218872
CAS :CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Formule :C13H9F3N4Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :278.23Pipequaline hydrochloride
CAS :Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.Formule :C22H25ClN2Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :352.9Arecaidine hydrochloride
CAS :Arecaidine hydrochloride may have carcinogenesis.Formule :C7H12ClNO2Degré de pureté :99.69% - ≥95%Couleur et forme :SolidMasse moléculaire :177.63Ref: TM-T5799
2mg34,00€5mg48,00€10mg67,00€25mg100,00€50mg149,00€100mg213,00€200mg316,00€1mL*10mM (DMSO)49,00€(R)-baclofen
CAS :(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Formule :C10H12ClNO2Degré de pureté :97.20% - 98.94%Couleur et forme :SolidMasse moléculaire :213.66Ocinaplon
CAS :Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formule :C17H11N5ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :301.3L-DABA
CAS :L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).Formule :C4H10N2O2Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :118.13Kavain
CAS :Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFormule :C14H14O3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :230.26Songorine
CAS :Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formule :C22H31NO3Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :357.49AZD-6280
CAS :AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formule :C20H22N4O3Degré de pureté :98.99%Couleur et forme :SolidMasse moléculaire :366.41Ref: TM-T7136
1mg215,00€5mg439,00€10mg640,00€25mg1.018,00€50mg1.423,00€100mg1.935,00€1mL*10mM (DMSO)484,00€Cholesterol myristate
CAS :Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.
Formule :C41H72O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :597.01α-Thujone
CAS :α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formule :C10H16ODegré de pureté :97.02% - 98.41%Couleur et forme :Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Masse moléculaire :152.23Temgicoluril
CAS :Temgicoluril (mebikar) acts on GABA Receptor.Formule :C8H14N4O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :198.226-Aminonicotinic acid
CAS :6-Aminonicotinic acid is a natural product.
Formule :C6H6N2O2Degré de pureté :99.94%Couleur et forme :SoildMasse moléculaire :138.1238rac-BHFF
CAS :rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Formule :C17H21F3O3Degré de pureté :99.69% - >99.99%Couleur et forme :SolidMasse moléculaire :330.34Ref: TM-T4176
2mg43,00€5mg60,00€10mg96,00€25mg187,00€50mg311,00€100mg472,00€200mg657,00€1mL*10mM (DMSO)71,00€α-Asarone
CAS :alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formule :C12H16O3Degré de pureté :99.64% - 99.64%Couleur et forme :Monoclinic Needles From Water Monoclinic Needles From WaterMasse moléculaire :208.25Fipronil
CAS :Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formule :C12H4Cl2F6N4OSDegré de pureté :97.21%Couleur et forme :Solid PowderMasse moléculaire :437.15Thiocolchicoside
CAS :Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.Formule :C27H33NO10SDegré de pureté :99.11% - 99.39%Couleur et forme :SolidMasse moléculaire :563.62γ-Acetylenic GABA
CAS :γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Formule :C6H9NO2Couleur et forme :SolidMasse moléculaire :127.143Tiagabine hydrochloride
CAS :Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formule :C20H25NO2S2·HClDegré de pureté :99.09% - 99.77%Couleur et forme :White To Off-White SolidMasse moléculaire :412.01Gabazine free base
CAS :Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Formule :C15H17N3O3Couleur et forme :SolidMasse moléculaire :287.31Lorediplon
CAS :Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Formule :C20H15FN4O2SDegré de pureté :99.12% - 99.19%Couleur et forme :SolidMasse moléculaire :394.42Loreclezole hydrochloride
CAS :Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.Formule :C10H7Cl4N3Couleur et forme :SolidMasse moléculaire :310.99Tiagabine hydrochloride hydrate
CAS :Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formule :C20H28ClNO3S2Couleur et forme :SolidMasse moléculaire :430.022'MeO6MF
CAS :2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormule :C17H14O3Degré de pureté :99.28% - 99.63%Couleur et forme :SolidMasse moléculaire :266.29Ref: TM-T8887
1mg49,00€5mg102,00€10mg152,00€25mg243,00€50mg340,00€100mg460,00€200mg627,00€1mL*10mM (DMSO)96,00€Piperazine
CAS :Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formule :C4H10N2Couleur et forme :SolidMasse moléculaire :86.14Pikamilone
CAS :Pikamilone (Picamilon) is an intelligent medicine.Formule :C10H12N2O3Degré de pureté :99.38%Couleur et forme :White Crystalline PowderMasse moléculaire :208.21(+)-Kavain
CAS :(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formule :C14H14O3Degré de pureté :97% - ≥95%Couleur et forme :White Fine PowderMasse moléculaire :230.26(-)-Securinine
CAS :(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formule :C13H15NO2Degré de pureté :99.58% - 99.87%Couleur et forme :SolidMasse moléculaire :217.26Isonipecotic acid
CAS :Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.Formule :C6H11NO2Degré de pureté :99.82%Couleur et forme :White To Faint Pink-Beige PowderMasse moléculaire :129.16SKF89976A hydrochloride
CAS :SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormule :C22H26ClNO2Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :371.9Ref: TM-T12930
1mg34,00€5mg65,00€10mg89,00€25mg167,00€50mg264,00€100mg409,00€200mg590,00€1mL*10mM (DMSO)71,00€Miltirone
CAS :Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formule :C19H22O2Degré de pureté :99.22% - 99.66%Couleur et forme :SolidMasse moléculaire :282.38Phenibut (hydrochloride)
CAS :Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formule :C10H14ClNO2Degré de pureté :99.93%Couleur et forme :White Crystalline PowderMasse moléculaire :215.684-Acetamidobutanoic acid
CAS :4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formule :C6H11NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :145.16CGP52432
CAS :CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formule :C15H24Cl2NO4PDegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :384.24(E)-3,4,5-Trimethoxycinnamic acid
CAS :(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formule :C12H14O5Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :238.24Imidazenil
CAS :Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.Formule :C18H12BrFN4ODegré de pureté :98.4%Couleur et forme :SolidMasse moléculaire :399.22Isoflurane
CAS :Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.Formule :C3H2ClF5ODegré de pureté :98%Couleur et forme :Clear Colorless Liquid LiquidMasse moléculaire :184.49Cyclothiazide
CAS :Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).Formule :C14H16ClN3O4S2Degré de pureté :98.23% - 99.49%Couleur et forme :Crystals From Dilute Alcohol SolidMasse moléculaire :389.88SSD114 HCl
CAS :SSD114 is a novel GABAB receptor positive allosteric modulator.Formule :C18H21ClF3N3ODegré de pureté :99.03% - 99.95%Couleur et forme :SolidMasse moléculaire :387.83Ref: TM-T4522
2mg34,00€5mg50,00€10mg75,00€25mg111,00€50mg172,00€100mg290,00€200mg419,00€1mL*10mM (DMSO)46,00€p-Hydroxybenzaldehyde
CAS :1.Formule :C7H6O2Degré de pureté :99.05% - 99.86%Couleur et forme :SolidMasse moléculaire :122.12Aminooxyacetic acid hemihydrochloride
CAS :Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABAFormule :C2H5NO3·5HClDegré de pureté :98.03%Couleur et forme :Light Beige Crystalline PowderMasse moléculaire :109.3Amentoflavone
CAS :Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formule :C30H18O10Degré de pureté :98.21% - 99.22%Couleur et forme :Odourless Whitish SolidMasse moléculaire :538.46Ref: TM-T3417
2mg34,00€5mg50,00€10mg80,00€25mg126,00€50mg215,00€100mg349,00€200mg512,00€1mL*10mM (DMSO)59,00€Tiagabine
CAS :Tiagabine (NO050328) is an Anti-epileptic Agent.Formule :C20H25NO2S2Degré de pureté :99.25% - 99.67%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :375.55Gaboxadol hydrochloride
CAS :Gaboxadol (hydrochloride) is a GABAA receptor agonist.Formule :C6H9ClN2O2Degré de pureté :99.39%Masse moléculaire :176.601SKF89976A HCl
CAS :SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formule :C22H25NO2Couleur et forme :SolidMasse moléculaire :335.44Gabazine
CAS :Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formule :C15H18BrN3O3Degré de pureté :98.51% - 99.24%Couleur et forme :SolidMasse moléculaire :368.236-(4-Methoxyphenyl)-3-pyridazinamine
CAS :6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormule :C11H11N3ODegré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :201.22L-838417 D9
CAS :L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].Formule :C19H10D9F2N7ODegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :408.45Ref: TM-T22301
2mg34,00€5mg52,00€10mg71,00€25mg128,00€50mg200,00€100mg323,00€200mg447,00€1mL*10mM (DMSO)58,00€2'-O-Methylisoliquiritigenin
CAS :2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formule :C16H14O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :270.28Baclofen hydrochloride
CAS :Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formule :C10H13Cl2NO2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :250.1226-Methylflavone
CAS :6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formule :C16H12O2Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :236.27DL-Menthol
CAS :DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Formule :C10H20ODegré de pureté :99.74%Couleur et forme :White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Masse moléculaire :156.27Saclofen
CAS :Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Formule :C9H12ClNO3SDegré de pureté :99.17%Couleur et forme :White Crystalline SolidMasse moléculaire :249.71Ref: TM-T4440
1mg52,00€5mg113,00€10mg177,00€25mg340,00€50mg550,00€100mg860,00€200mg1.161,00€1mL*10mM (DMSO)108,00€Imepitoin
CAS :Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.Formule :C13H14ClN3O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :279.72U93631
CAS :GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formule :C17H21N3O2Degré de pureté :99.65% - 99.76%Couleur et forme :SolidMasse moléculaire :299.37Fluralaner
CAS :Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formule :C22H17Cl2F6N3O3Degré de pureté :99.72% - 99.99%Couleur et forme :Solid PowderMasse moléculaire :556.29Ginsenoside Rc
CAS :Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.
Formule :C53H90O22Degré de pureté :98.83% - 99.56%Couleur et forme :White PowderMasse moléculaire :1079.27NS11394
CAS :NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formule :C23H19N3ODegré de pureté :99.44% - 99.86%Couleur et forme :SolidMasse moléculaire :353.42Ref: TM-T2067
2mg34,00€5mg50,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€1mL*10mM (DMSO)58,00€ONO-8590580
CAS :ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.Formule :C21H21FN6Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :376.43Ref: TM-TQ0040
1mg57,00€5mg119,00€10mg166,00€25mg356,00€50mg532,00€100mg760,00€1mL*10mM (DMSO)133,00€Jujuboside A
CAS :Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formule :C58H94O26Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :1207.35Suritozole
CAS :Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptorFormule :C10H10FN3SDegré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :223.27Ref: TM-T8568
1mg58,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€1mL*10mM (DMSO)104,00€Basmisanil
CAS :Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFormule :C21H20FN3O5SDegré de pureté :99.21% - 99.42%Couleur et forme :SolidMasse moléculaire :445.46Ref: TM-T7165
2mg35,00€5mg52,00€10mg74,00€25mg116,00€50mg187,00€100mg356,00€500mg802,00€1mL*10mM (DMSO)49,00€Dihydroergotoxine mesylate
CAS :Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formule :C20H29N3O5SDegré de pureté :99.39% - ≥95%Couleur et forme :SolidMasse moléculaire :423.53Bicuculline
CAS :Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Formule :C20H17NO6Degré de pureté :98% - 99.99%Couleur et forme :Light Yellow PowderMasse moléculaire :367.35Loreclezole
CAS :Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Formule :C10H6Cl3N3Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :274.53Afloqualone
CAS :Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Formule :C16H14FN3ODegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :283.3Darigabat
CAS :Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formule :C22H21FN4O3SDegré de pureté :98.42% - 99.29%Couleur et forme :SolidMasse moléculaire :440.49Riluzole
CAS :Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.
Formule :C8H5F3N2OSDegré de pureté :99.71% - 99.88%Couleur et forme :PowderMasse moléculaire :234.2GABAA receptor agent 5
CAS :Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.Formule :C21H25N3O2SDegré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :383.51ABP-700
CAS :ABP-700 is a positive allosteric modulator of the GABAA receptor.Formule :C17H18N2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :314.34RO 4938581
CAS :RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).Formule :C13H8BrF2N5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.14DAA-1097
CAS :DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.Formule :C24H24ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :409.91(S)-3-Carboxy-4-hydroxyphenylglycine
CAS :group I metabotropic glutamate receptor antagonist and group II mGlu agonistFormule :C9H9NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :211.17BGT1-IN-9
CAS :BGT1-IN-9 is an M1 muscarinic agonist.Formule :C5H10ClN3O2Couleur et forme :SolidMasse moléculaire :179.605PNU-107484A
CAS :PNU-107484A is a unique GABA(A) receptor ligand.Formule :C18H23ClN6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :358.87CGP 46381
CAS :CGP 46381 is a GABAB receptor antagonist.Formule :C10H22NO2PDegré de pureté :98%Couleur et forme :White SolidMasse moléculaire :219.26PF-0713
CAS :PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.Formule :C14H22ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :206.32GS 39783
CAS :GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement andFormule :C15H23N5O2SDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :337.44Ro 41-3290
CAS :Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.Formule :C24H21ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :420.89SCH 50911
CAS :SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.Formule :C8H15NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :173.21Anxiolytic/nonsedative agent-1
CAS :TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formule :C18H15N3O4Degré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :337.33Ref: TM-T23445
1mg64,00€2mg96,00€5mg115,00€10mg150,00€25mg330,00€50mg472,00€100mg655,00€500mg1.293,00€CP-409092 hydrochloride
CAS :CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.Formule :C17H20ClN3O2Couleur et forme :SolidMasse moléculaire :333.81Ciclotizolam
CAS :Ciclotizolam, a thienotriazolodiazepine derivative and partial GABAA receptor agonist, has low efficacy but similar affinity as brotizolam.Formule :C20H18BrClN4SCouleur et forme :SolidMasse moléculaire :461.81Arbaclofen placarbil
CAS :Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.Formule :C19H26ClNO6Couleur et forme :SolidMasse moléculaire :399.87SH-053-S-CH3-2'F
CAS :SH-053-S-CH3-2'F is a potent and selective agonist of GABAA receptors.Formule :C23H18FN3O2Couleur et forme :SolidMasse moléculaire :387.41Ethyl dirazepate
CAS :Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.Formule :C18H14Cl2N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.22
