Récepteur GABA
Les récepteurs GABA sont les principaux récepteurs de neurotransmetteurs inhibiteurs du système nerveux central, jouant un rôle crucial dans la régulation de l'excitabilité neuronale et le maintien de l'équilibre entre excitation et inhibition. La dysfonction des récepteurs GABA est impliquée dans divers troubles neurologiques et psychiatriques, notamment l'épilepsie, l'anxiété et la dépression. Chez CymitQuimica, nous proposons une gamme complète de modulateurs des récepteurs GABA pour soutenir vos recherches en neurobiologie, santé mentale et développement thérapeutique.
371 produits trouvés pour "Récepteur GABA"
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Broflanilide
CAS :Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.Formule :C25H14BrF11N2O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :663.29Ref: TM-T10618
1mg52,00€2mg74,00€5mg111,00€10mg180,00€25mg358,00€50mg588,00€100mg835,00€1mL*10mM (DMSO)131,00€Afoxolaner
CAS :Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.Formule :C26H17ClF9N3O3Degré de pureté :99.1% - 99.38%Couleur et forme :SolidMasse moléculaire :625.87GABAA receptor agent 1
CAS :GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.Formule :C13H8ClN3O2Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :273.67Ref: TM-T11349
1mg35,00€5mg79,00€10mg111,00€25mg215,00€50mg323,00€100mg469,00€200mg647,00€1mL*10mM (DMSO)86,00€Bemegride
CAS :Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Formule :C8H13NO2Degré de pureté :99.89%Couleur et forme :Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Masse moléculaire :155.19Phenelzine sulfate
CAS :Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Formule :C8H14N2O4SDegré de pureté :98.38% - 99.83%Couleur et forme :SolidMasse moléculaire :234.27Fluxametamide
CAS :Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Formule :C20H16Cl2F3N3O3Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :474.26Lotilaner
CAS :Lotilaner is a parasiticide.Formule :C20H14Cl3F6N3O3SDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :596.76Ref: TM-T15775
1mg44,00€2mg58,00€5mg94,00€10mg144,00€25mg335,00€50mg550,00€100mg882,00€200mg1.188,00€1mL*10mM (DMSO)111,00€Isoguvacine hydrochloride
CAS :Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.Formule :C6H10ClNO2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :163.6Pentetrazol
CAS :Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.Formule :C6H10N4Degré de pureté :99.67% - 99.90%Couleur et forme :Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Masse moléculaire :138.17Flumazenil
CAS :Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormule :C15H14FN3O3Degré de pureté :99.72% - 99.98%Couleur et forme :Less Crystals Colourless CrystalsMasse moléculaire :303.29γ-Aminobutyric acid
CAS :γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Formule :C4H9NO2Degré de pureté :99.95%Couleur et forme :White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderMasse moléculaire :103.12Phenibut
CAS :Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Formule :C10H13NO2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :179.22Domperidone EP Impurity A
CAS :Domperidone EP Impurity A is used as pharmaceutical intermediates.Formule :C12H14ClN3ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :251.71Baclofen
CAS :Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formule :C10H12ClNO2Degré de pureté :98% - >99.99%Couleur et forme :1992)Masse moléculaire :213.66GET73
CAS :GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.Formule :C13H16F3NO2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :275.27Ref: TM-T11393
5mg39,00€10mg56,00€25mg104,00€50mg158,00€100mg230,00€200mg340,00€1mL*10mM (DMSO)44,00€UK-124114
CAS :Selamectin, a derivative of ivermectin, is a macrocyclic lactone that enhances chloride channels in nematodes, inhibiting H. contortus larval growth.Formule :C43H63NO11Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :769.96Etifoxine hydrochloride
CAS :Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.Formule :C17H18Cl2N2ODegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :337.24FG 7142
CAS :FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.Formule :C13H11N3ODegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :225.25Ref: TM-T11277
2mg33,00€5mg60,00€10mg92,00€25mg149,00€50mg213,00€100mg318,00€200mg442,00€1mL*10mM (DMSO)39,00€Topiramate
CAS :Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.Formule :C12H21NO8SDegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :339.36Nikethamide
CAS :Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of endFormule :C10H14N2ODegré de pureté :99.42%Couleur et forme :Followed By A Faint Sensation Of The Warmth (Ntp 1992)Masse moléculaire :178.23Nefiracetam
CAS :Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formule :C14H18N2O2Degré de pureté :97.37%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :246.3Clomethiazole
CAS :Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.Formule :C6H8ClNSDegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :161.65L-Cycloserine
CAS :L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formule :C3H6N2O2Degré de pureté :99.75% - 99.99%Couleur et forme :Crystals White PowderMasse moléculaire :102.09Chlormezanone
CAS :Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.Formule :C11H12ClNO3SDegré de pureté :99.86% - >99.99%Couleur et forme :Crystals SolidMasse moléculaire :273.743,4,5-Trimethoxycinnamic acid
CAS :3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFormule :C12H14O5Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :238.24Pivagabine
CAS :Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.Formule :C9H17NO3Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :187.24LAU159
CAS :LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).Formule :C17H12ClN3O2Degré de pureté :98.7% - 99.38%Couleur et forme :SolidMasse moléculaire :325.75Ref: TM-T11822
1mg110,00€2mg160,00€5mg219,00€10mg395,00€25mg653,00€50mg888,00€100mg1.243,00€500mg2.493,00€NEO 376
CAS :NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Formule :C20H24ClN3ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :357.88Ref: TM-T12207
1mg74,00€5mg140,00€10mg215,00€25mg373,00€50mg522,00€100mg702,00€200mg944,00€1mL*10mM (DMSO)156,00€Emamectin Benzoate
CAS :Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFormule :C56H81NO15Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :1008.256Oxiracetam
CAS :Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.
Formule :C6H10N2O3Degré de pureté :99.67%Couleur et forme :White Crystalline PowderMasse moléculaire :158.16α5-GABAA receptor modulator 1
α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.Formule :C21H20FN3O4Couleur et forme :SolidMasse moléculaire :397.4α-Casozepine
CAS :α-Casozepine,Bioactive peptide from milk α-S1 casein. Binds GABA receptors. Anti-anxiety effects.Formule :C60H94N14O16Couleur et forme :SolidMasse moléculaire :1267.47RuBi-GABA
CAS :Ruthenium-bipyridine-triphenylphosphine caged GABAFormule :C42H39F6N5O2P2RuDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :922.8DAA-1106
CAS :DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.Formule :C23H22FNO4Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :395.42Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formule :C15H11N5OCouleur et forme :SolidMasse moléculaire :277.28Nipecotic acid
CAS :Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.
Formule :C6H11NO2Couleur et forme :Off-White To Pale Yellow-Beige PowderMasse moléculaire :129.16Fipronil sulfone
CAS :Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.Formule :C12H4Cl2F6N4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :453.14Chrodrimanin B
CAS :Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.Formule :C27H32O8Couleur et forme :SolidMasse moléculaire :484.545Imagabalin
CAS :Imagabalin is an active compound used in the study of neurological diseases.Formule :C9H19NO2Couleur et forme :SolidMasse moléculaire :173.25Lesogaberan napadisylate
CAS :Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Formule :C13H17FNO5PSCouleur et forme :SolidMasse moléculaire :349.31Furosemide sodium
CAS :Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.Formule :C12H10ClN2NaO5SDegré de pureté :99.52% - >99.99%Couleur et forme :SolidMasse moléculaire :352.73Azocarnil
Azocarnil is a GABAergic agonist-enhancer used in neurological system research.Couleur et forme :Odour Solid6,7-dimethylisatin
CAS :6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.Formule :C10H9NO2Degré de pureté :98.98%Couleur et forme :SolidMasse moléculaire :175.18Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Formule :C19H38ClN5O2SCouleur et forme :SolidMasse moléculaire :436.06Nitrazolam
CAS :Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.Formule :C17H13N5O2Couleur et forme :SolidMasse moléculaire :319.32epi-Aszonalenin A
CAS :epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.Formule :C25H25N3O3Couleur et forme :SolidMasse moléculaire :415.48CGP 35348
CAS :CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。Formule :C8H20NO4PDegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :225.22Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Couleur et forme :Odour SolidAHN-683
CAS :AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.Formule :C42H32FN3O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :709.72Ion Channel Targeted Library
A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;
Couleur et forme :Odour Solid
