Neuroscience
Les inhibiteurs en neurosciences sont des composés conçus pour moduler l'activité de protéines, d'enzymes ou de récepteurs spécifiques au sein du système nerveux. Ces inhibiteurs sont cruciaux pour étudier les mécanismes moléculaires sous-jacents au fonctionnement neuronal, à la transmission synaptique et aux maladies neurodégénératives. En ciblant les récepteurs des neurotransmetteurs, les canaux ioniques et les voies de signalisation, les inhibiteurs en neurosciences facilitent l'exploration du fonctionnement cérébral et le développement de stratégies thérapeutiques pour des troubles neurologiques tels que la maladie d'Alzheimer, de Parkinson et l'épilepsie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs en neurosciences de haute qualité pour soutenir vos recherches en neurobiologie, neuropharmacologie et sciences cognitives.
Sous-catégories appartenant à la catégorie "Neuroscience"
- récepteur 5-HT(1.025 produits)
- ACK(1 produits)
- AChR(647 produits)
- ATP Citrate Lyase(17 produits)
- Récepteur adrénergique(3.027 produits)
- BACE(37 produits)
- Bêta-amyloïde(230 produits)
- CaMK(73 produits)
- COX(602 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur GABA(373 produits)
- Gamma-sécrétase(62 produits)
- GluR(265 produits)
- GlyT(26 produits)
- Récepteur de l'histamine(385 produits)
- LRRK2(43 produits)
- Récepteur de la mélatonine(26 produits)
- NMDAR(10 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
Affichez 12 plus de sous-catégories
5639 produits trouvés pour "Neuroscience"
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Imagabalin
CAS :Imagabalin is an active compound used in the study of neurological diseases.Formule :C9H19NO2Couleur et forme :SolidMasse moléculaire :173.25SB236057
CAS :SB236057: potent selective inverse agonist at 5-HT autoreceptors; increases brain 5-HT; teratogen causing musculoskeletal defects in rodents.Formule :C33H34N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :534.655-HT1AR agonist 2
5-HT1AR Agonist 2 (Compound 4f) is a potent agonist of the 5-HT1A receptor with a Ki value of 10.0 nM. It also binds to SERT, D2, and 5-HT6 receptors with Ki values of 2.8 nM, 23 nM, and 192 nM, respectively. Furthermore, this compound demonstrates stability in microsomes and induces hypothermia in mice.Formule :C31H31N5O3Couleur et forme :SolidMasse moléculaire :521.615α-Androst-16-en-3α-ol
CAS :5α-Androst-16-en-3α-ol is a steroid pheromone that has been found in boar testes and human male axillary sweat and has diverse biological activities.1,2ItFormule :C19H30OCouleur et forme :SolidMasse moléculaire :274.448Guvacine hydrobromide
CAS :Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake.Formule :C6H10BrNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :208.05AChE/MAO-B-IN-7
AChE/MAO-B-IN-7 (VAV-8) is a compound that acts as a dual inhibitor of acetylcholinesterase (AChE) and MAO-B, with the ability to cross the blood-brain barrier. It also inhibits the aggregation of Aβ42, making it a valuable compound for Alzheimer's disease (AD) research.
Formule :C22H21N3O3Couleur et forme :SolidMasse moléculaire :375.42MAO-B-IN-4
MAO-B-IN-4 (Compound 26) is a reversible monoamine oxidase B (MAO-B) inhibitor with potent in vitro activity, characterized by an IC50 value of 9 nM.Formule :C23H20ClF2N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.87MAO-B-IN-37
CAS :MAO-B-IN-37 (Compound 37) is a derivative of TT01001 and acts as a selective inhibitor of monoamine oxidase B (MAO-B), with an IC50 of 270 nM. It exhibits good metabolic stability in mouse microsomes and shows strong affinity for human serum albumin.Formule :C14H12FN3O3Couleur et forme :SolidMasse moléculaire :289.26Methamnetamine hydrochloride
CAS :Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.Formule :C14H18ClNCouleur et forme :SolidMasse moléculaire :235.75Lysyl hydroxylase 2-IN-1
"Lysyl Hydroxylase 2-IN-1 (compound 12) is a selective inhibitor of lysyl hydroxylase 2 (LH2) with an IC50 of approximately 300 nM and demonstrates specificityFormule :C18H18N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.35MmTx2 toxin
MmTx2 toxin, extracted from the venom of the coral snake, serves as a modulator of the GABA A receptor, increasing its responsiveness to agonists.Formule :C295H450N94O97S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7185.95Lysyl hydroxylase 2-IN-2
Lysyl Hydroxylase 2-IN-2 (compound 13) is a potent inhibitor of Lysyl Hydroxylase 2 (LH2), exhibiting an IC50 of approximately 500 nM.Formule :C19H21N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.39(±)-Acetylcarnitine chloride
CAS :(±)-Acetylcarnitine chloride (Acetyl dl-carnitine chloride) is a weak cholinergic agonist with neuroprotective properties and can be used in studies of neuritis.
Formule :C9H18ClNO4Degré de pureté :99.98%Couleur et forme :White Crystalline PowderMasse moléculaire :239.75-(2-Aminopropyl)indole
CAS :5-(2-Aminopropyl)indole is an orally active psychoactive substance that inhibits monoamine oxidase (MAO) and exhibits long-lasting stimulant effects.Formule :C11H14N2Couleur et forme :SolidMasse moléculaire :174.24NMDA receptor antagonist 6
NMDA Receptor Antagonist 6 (Compound 13b) functions as an antagonist at the glycine-binding site of the NMDA receptor and demonstrates cytoneuroprotectiveFormule :C25H23NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.465-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formule :C24H26N4O2SCouleur et forme :SolidMasse moléculaire :434.55CALP2 TFA
CALP2 TFA, a CaM antagonist with 7.9 µM Kd, blocks CaM-dependent enzymes, boosts Ca2+ levels, and activates macrophages.Formule :C70H105F3N14O15SCouleur et forme :SolidMasse moléculaire :1471.72Dalidnetug
CAS :Dalidnetug is a humanized monoclonal antibody that targets human β-amyloid precursor protein (APP). By specifically binding to APP, Dalidnetug reduces the production of β-amyloid (Aβ), thereby demonstrating activity in clearing β-amyloid. This compound holds potential for research in Alzheimer's disease.Couleur et forme :LiquidArotinolol hydrochloride
CAS :Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.Formule :C15H22ClN3O2S3Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :408Kynuramine
CAS :Kynuramine is an aromatic ketone containing the aniline structure.
Formule :C9H12N2OCouleur et forme :SolidMasse moléculaire :164.20C18 L-erythro Ceramide (d18:1/18:0)
CAS :C18 L-erythro Ceramide, a natural stereoisomer, inhibits rat brain mt-CDase with IC50 of 8.8 μM.Formule :C36H71NO3Couleur et forme :SolidMasse moléculaire :565.95γ-Acetylenic GABA hydrochloride
CAS :γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.Formule :C6H10ClNO2Degré de pureté :97.83% - 99.44%Couleur et forme :SolidMasse moléculaire :163.6KGP-25
KGP-25 is an inhibitor of the voltage-gated sodium channel 1.8 (Nav1.8), utilized for analgesia by targeting the peripheral nervous system (PNS). Additionally, it targets the γ-aminobutyric acid subtype A receptor (GABAA) in the central nervous system (CNS) for use as a general anesthetic.Couleur et forme :Odour Solid4-Methylamphetamine hydrochloride
CAS :4-Methylamphetamine hydrochloride is a 5-HT1A receptor agonist that induces a decrease in body temperature in rats by binding to the 5-HT1A receptor. Additionally, it increases the extracellular levels of neurotransmitters norepinephrine (NE), dopamine (DA), and serotonin (5-HT) by affecting their transporters. 4-Methylamphetamine hydrochloride is applicable in the study of neurological disorders.Formule :C10H16ClNCouleur et forme :SolidMasse moléculaire :185.69Antidepressant agent 10
CAS :Compound PDK0386, with CAS No. 87691-87-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0386 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C11H13N3SMasse moléculaire :219.306Hydroxytacrine maleate
CAS :Hydroxytacrine maleate (Velnacrine maleate) is a cholinesterase inhibitor used in the study of Alzheimer's type dementia (SDAT).Formule :C17H18N2O5Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :330.34Substance P(1-4) Acetate
Substance P(1-4) Acetate is a neurokinin receptor (NK-R) antagonist, inhibiting the formation of PV EEC.Formule :C24H44N8O7Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :556.665-methoxy-α-Ethyltryptamine
CAS :5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects.
Formule :C13H18N2ODegré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :218.29(D-Asp1)-Amyloid β-Protein (1-42)
CAS :(D-Asp1)-Amyloid β-Protein (1-42), a peptide fragment of amyloid β-protein (Aβ), serves as the primary constituent of vascular and parenchymal amyloid depositsFormule :C203H311N55O60SCouleur et forme :SolidMasse moléculaire :4514.04(S)-UFR2709 hydrochloride
CAS :(S)-UFR2709 HCl: competitive nAChR blocker, prefers α4β2 over α7, lessens anxiety & alcohol intake in rats, studies nicotine addiction.Formule :C13H18ClNO2Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :255.74Ebiratide TFA
Ebiratide (HOE-427) TFA is a derivative of ACTH4-9 that exerts its effect directly on the central nervous system, enhancing memory. Ebiratide TFA also promotes the metabolism of acetylcholine (ACh) in the rat brain.Formule :C48H73N11O10S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :996.23 (free base)SB 258585
CAS :SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.Formule :C18H22IN3O3SDegré de pureté :99.77%Couleur et forme :SoildMasse moléculaire :487.36MAO-B-IN-25
MAO-B-IN-25 (compound 92) is a selective inhibitor of monoamine oxidase B (MAO-B), exhibiting inhibitory half-maximal inhibitory concentrations (IC50) of 240 nMFormule :C16H13BrO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.18(Rac)-Sabcomeline
CAS :(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.Formule :C10H15N3ODegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :193.25Ref: TM-T68135L1
1mg109,00€2mg160,00€5mg261,00€10mg374,00€25mg583,00€50mg803,00€100mg1.063,00€200mg1.431,00€AChE-IN-60
AChE-IN-60 (compound 6k) is a potent inhibitor of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), with IC50 values of 27 nM and 43 nM, respectively. It also inhibits monoamine oxidase MAO-A and MAO-B, with IC50 values of 353 nM and 716 nM, respectively.Formule :C24H29N3O4S3Masse moléculaire :519.13202(Rac)-5-Carboxy tolterodine
CAS :(Rac)-5-Carboxy tolterodine is an inactive metabolite of Tolterodine, which acts as a muscarinic acetylcholine receptor antagonist.Formule :C22H29NO3Couleur et forme :SolidMasse moléculaire :355.47COX-2-IN-33
COX-2-IN-33 (compound 5f) is a selective COX-2 inhibitor with an IC50 value of 45.5 nM and exhibits potential as an anti-inflammatory agent.Formule :C20H13ClF3N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.8Methyl piperate
CAS :Methylpiperic acid, a piperine alkaloid, exhibits potent inhibitory activity on monoamine oxidase (MAO), with differing efficacy on isoforms: greater inhibitionFormule :C13H12O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :232.23PZ-1922
PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.Degré de pureté :98%Couleur et forme :Odour SolidACHE Inhibitor 12
CAS :ACHE Inhibitor 12 inhibited acetylcholinesterase with an IC50 value of 0.38 µM.Formule :C11H12ODegré de pureté :97.07%Couleur et forme :SolidMasse moléculaire :160.21MRS7925
MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosisFormule :C20H26IN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :511.36PSEM 308 hydrochloride
PSAM agonist targeting PSAML141F-GlyR and related ion channels in mice; ideal concentration ≤5 mg/kg; plasmids at Addgene.Couleur et forme :SolidMetixene
CAS :Metixene is an anticholinergic drug. It was developed as a treatment against Parkinson's disease.Formule :C20H23NSCouleur et forme :LiquidMasse moléculaire :309.47AChE/BChE-IN-25
AChE/BChE-IN-25 (Compound 6e) is an orally active inhibitor of hAChE and eqBChE, with IC50 values of 7.9 nM and 0.79 nM, respectively. This compound exhibits antioxidant activity, effective in scavenging free radicals with an IC50 of 22.91 μM. AChE/BChE-IN-25 demonstrates neuroprotective effects by reducing mitochondrial and cellular oxidative stress in a Drosophila Alzheimer's model and improves spatial and cognitive memory impairments induced by Scopolamine in mouse models.Formule :C21H24ClN3O2Couleur et forme :SolidMasse moléculaire :385.89BRD9 ligand-6
CAS :BRD9 ligand-6 serves as a ligand for the target protein in PROTAC applications. It is utilized in the synthesis of FHD-609.Formule :C21H21N3O4Couleur et forme :SolidMasse moléculaire :379.41Dihydrochalcone
CAS :Compound PDK0018, with CAS No. 1083-30-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0018 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C15H14OCouleur et forme :SolidMasse moléculaire :210.27[Ala2,8,9,11,19,22,24,25,27,28]-VIP
CAS :[Ala2,8,9,11,19,22,24,25,27,28]-VIP can be used for related research in the field of life sciences. Its product number is T36637 and CAS number is 866552-34-3.Formule :C131H219N41O33SCouleur et forme :SolidMasse moléculaire :2928.51BU 226 hydrochloride
CAS :BU 226 hydrochloride demonstrates affinity for imidazoline (I) receptors, in particular the I2 binding site with a Ki of 1.4 nM.Formule :C12H12ClN3Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :233.74-hydroxy DiPT hydrochloride
CAS :4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.Formule :C16H25ClN2OCouleur et forme :SolidMasse moléculaire :296.84Pridinol hydrochloride
CAS :Pridinolhydrochloride is the hydrochloride form of Pridinol. Pridinol hydrochloride is an orally active anticholinergic agent, which can also be used as a muscle relaxant.Formule :C20H26ClNOCouleur et forme :SolidMasse moléculaire :331.883-Hydroxy desalkylflurazepam
CAS :3-Hydroxy desalkylflurazepam is a benzodiazepine compound with potential sedative and anxiolytic effects.Formule :C15H10ClFN2O2Couleur et forme :SolidMasse moléculaire :304.7GABA-IN-1
GABA-IN-1 (Compound 6), a GABA inhibitor, exhibits larvicidal and insecticidal properties, achieving a mortality rate of 93% at a concentration of 50 mg/L [1].Couleur et forme :Odour SolidBrexanolone caprilcerbate
CAS :Brexanolone caprilcerbate is an effective positive allosteric modulator of the GABAA receptor.Formule :C48H78O12Couleur et forme :SolidMasse moléculaire :847.13AChE/BChE-IN-22
AChE/BChE-IN-22 (compound 7) exhibits competitive inhibition against both AChE and BChE enzymes, with inhibition constants of 28.18 μM and 41.74 μM respectively.Formule :C14H11F3N2O4SCouleur et forme :SolidMasse moléculaire :360.316,9-Dichloro-1,2,3,4-tetrahydroacridine
CAS :6,9-Dichloro-1,2,3,4-tetrahydroacridine is a synthetic intermediate in the synthesis of tacrine-based acetylcholinesterase (AChE) inhibitors.1It is also anFormule :C13H11Cl2NCouleur et forme :SolidMasse moléculaire :252.139Merinetug
CAS :Merinetug is a humanized IgG1κ antibody that targets Amyloid Beta (Aβ). Its corresponding isotype control is Human IgG1 kappa, Isotype Control.Couleur et forme :LiquidAChE-IN-41
AChE-IN-41 (Compound 2), a Galantamine-Memantine hybrid, possesses cholinesterase inhibitory capabilities.Couleur et forme :Odour Solid(+)-Coclaurine hydrochloride
CAS :(+)-Coclaurine hydrochloride, also known as (+)-(R)-Coclaurine, is a benzyltetrahydroisoquinoline alkaloid extracted from multiple plant species.Formule :C17H20ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.8AAK1-IN-11
AAK1-IN-11 is an inhibitor of AAK1 (adaptor associated kinase 1) with an IC50 of 2 nM, and it exhibits antiviral activity.Couleur et forme :Odour Solid(-)-2-Phenylpropylamine
CAS :(-)-2-Phenylpropylamine ((S)-2-Phenylpropylamine) (compound 3b) functions as an inhibitor for both MAO-A and MAO-B, with Ki values of 584 μM and 156 μM, respectively.Formule :C9H13NCouleur et forme :SolidMasse moléculaire :135.21HTR2A antagonist 1
HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.Formule :C35H43Cl2F2N5O4Couleur et forme :SolidMasse moléculaire :706.65Aβ1-14-εK-KKK-MvF5 Th
Aβ1-14-εK-KKK-MvF5 Th (UB311 immunogen I) is a biologically active peptide and one of the Aβ1–14 targeting peptides (B-cell epitope) used in UB-311.
Formule :C199H318N56O55Masse moléculaire :4372.38081LP-20
CAS :LP-20 is a bioactive chemical.Formule :C17H20N2OCouleur et forme :SolidMasse moléculaire :268.35Iloperidone metabolite P95
CAS :Iloperidone metabolite P95, a non-brain penetrating compound, binds 5-HT2A, α1-, α2B-, α2C-receptors with Ki of 7.08-83.18 nM.Formule :C23H25FN2O5Couleur et forme :SolidMasse moléculaire :428.46Lu AE51090
CAS :Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.Formule :C24H29N3O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :407.51Tampramine
CAS :Tampramine: a TCA and selective norepinephrine inhibitor, with low affinity for other receptors, potential treatment for FST depression.
Formule :C23H24N4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :356.46Imipramine N-oxide
CAS :Imipramine N-oxide is a tricyclic antidepressant (TCA) and imipramine analogue used to treat depression.Formule :C19H24N2ODegré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :296.41Ref: TM-T74205
1mg72,00€5mg157,00€1mL*10mM (DMSO)167,00€10mg241,00€25mg409,00€50mg565,00€100mg794,00€Trivalent GalNAc-DBCO
CAS :Trivalent GalNAc-DBCO is a synthetic ligand composed of three GalNAc units linked to DBCO. Trivalent GalNAc-DBCO undergoes strain-promoted alkyne–azide cycloaddition (SPAAC) reactions with azide-containing molecules without the need for copper catalysis. Trivalent GalNAc-DBCO binds specifically to the asialoglycoprotein receptor (ASGPR), thereby directing conjugated molecules into hepatocytes for lysosomal degradation through receptor-mediated endocytosis. Trivalent GalNAc-DBCO is extensively applied in studies of liver-targeted drug delivery, targeted degradation strategies, and hepatocyte-specific molecular engineering.Formule :C91H144N12O34Degré de pureté :96.33%Masse moléculaire :1950.18FGIN-1-43
CAS :FGIN-1-43 is a potent and specific ligand for the mitochondrial DBI receptor.Formule :C28H36Cl2N2ODegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :487.5Pyrazolam
CAS :Pyrazolam is a psychoactive benzodiazepine compound serving as a central nervous system depressant. [Pyrazolam] can lead to psychomotor impairment.Formule :C16H12BrN5Couleur et forme :SolidMasse moléculaire :354.22,6-DMA hydrochloride
CAS :2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.Formule :C11H18ClNO2Couleur et forme :SolidMasse moléculaire :231.725-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFormule :C17H22Cl2N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.37BSBM6
CAS :BSBM6 is an inhibitor of Aβ aggregation and neuronal toxicity that acts by reversing the aggregation and toxicity of amyloid-β peptides.Formule :C23H29N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :427.49Adatanserin hydrochloride
CAS :Adatanserin hydrochloride (WY50324 hydrochloride) is a 5-HT(1A)/5-HT(2) receptor ligand that is neuroprotective and may be used in the study of depression.Formule :C21H32ClN5ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :405.96(Iso)-Atagabalin HCl
CAS :(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.Formule :C10H20ClNO2Degré de pureté :99.88% - >99.99%Couleur et forme :SoildMasse moléculaire :221.72Calmodulin-Dependent Protein Kinase II 290-309 acetate
Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM).Formule :C105H189N31O26SDegré de pureté :96.7%Couleur et forme :SolidMasse moléculaire :2333.88TB-11
CAS :TB-11 is an inhibitor of Cathepsin D with IC50 values of 0.126 nM (Cathepsin D), 1.92 nM (Cathepsin E), and 48.8 nM (BACE1). It is primarily utilized in oncological research.Formule :C52H78N8O12Couleur et forme :SolidMasse moléculaire :1007.22LOX-IN-4
CAS :LOX-IN-4 (Compound 112) is an inhibitor of lysyl oxidase (LOX). It holds potential for use in cancer research.Formule :C20H24Cl2FN3O2SCouleur et forme :SolidMasse moléculaire :460.39BIMU 8
CAS :BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.Formule :C19H27ClN4O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :378.9Ref: TM-T21946
1mg85,00€5mg168,00€1mL*10mM (DMSO)175,00€10mg235,00€25mg394,00€50mg582,00€100mg827,00€500mg1.674,00€Tiquizium
CAS :Tiquizium has effective Antimuscarinic effect, and causes significant bronchodilation in patients with chronic obstructive pulmonary disease.
Formule :C19H24NS2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :330.53Dual AChE-MAO B-IN-3
Compound C10 is a potent dual AChE/MAO-B inhibitor with IC50s of 0.58μM (AChE) and 0.41μM (MAO-B), useful in Alzheimer's research.Formule :C30H26F3NO3Couleur et forme :SolidMasse moléculaire :505.53MAO-B-IN-20
MAO-B-IN-20, potent with 0.037 μM IC50, is stable and BBB permeable, useful for Parkinson's research.Formule :C20H18F2N2O2Couleur et forme :SolidMasse moléculaire :356.37Dicloromezotiaz
CAS :Dicloromezotiaz: Potent insecticide targeting nAChRs, controls various lepidoptera.Formule :C19H12Cl3N3O2SCouleur et forme :SolidMasse moléculaire :452.74RA306
RA306 is an orally active CAMK2 inhibitor that effectively disrupts the PEAK1/CAMK2 signaling pathway. It demonstrates anti-tumor activity by inhibiting proliferation, migration, and invasion of breast cancer cells. Additionally, RA306 shows potential in cardiac disease research, as it improves dilated cardiomyopathy in mice.Couleur et forme :Odour SolidSKF-83566 hydrochloride
CAS :SKF-83566 hydrochloride is a D1-like dopamine receptor antagonist, inhibiting dopamine transporters and mitigating GBP-induced CPP.Formule :C17H19BrClNODegré de pureté :99.27%Couleur et forme :SoildMasse moléculaire :368.69VVZ-149
VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.Couleur et forme :SolidMonoamine oxidase
CAS :Enzyme that breaks down amines in the brain and body, affecting mood and brain function.Couleur et forme :Solidβ-Amyloid (29-40)
CAS :β-Amyloid (29-40) is a fragment of Amyloid-β peptide.Alzheimer's beta amyloid peptide (29-40/42) C-terminal fragments have physical and chemical propertiesFormule :C49H88N12O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1085.36OXA(17-33)
CAS :Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.Formule :C79H125N23O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1749β-Amyloid (1-16)
CAS :β-Amyloid (1-16) is an amyloidogenic protein fragment with a sequence derived from β-amyloid.Formule :C84H119N27O28Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1955.04SPL-707
CAS :SPL-707 is an effective and selective signal peptide peptidase-like 2a inhibitor (IC50: 80 nM).Formule :C27H28FN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :505.54AChE/BChE-IN-14
AChE/BChE-IN-14 (compound 13), a benzylisoquinoline alkaloid extracted from Fissistigma polyanthum roots, demonstrates inhibitory effects on bothFormule :C19H23NO3Couleur et forme :SolidMasse moléculaire :313.39Cianopramine hydrochloride
CAS :Cianopramine hydrochloride is a bio-active chemical.Formule :C20H24ClN3Couleur et forme :SolidMasse moléculaire :341.88Pirimiphos-ethyl
CAS :Pirimiphos-ethyl is used as an organophosphorus pesticide.Formule :C13H24N3O3PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.39BChE-IN-12
CAS :BChE-IN-12, non-competitive BChE inhibitor from Bletilla striata, IC50=2.3μM; potential Alzheimer’s research.Formule :C31H30O5Couleur et forme :SolidMasse moléculaire :482.57N-Ethyl-N-(3-pyridylmethyl)amine
CAS :N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.Formule :C8H12N2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :136.19Rasagiline 13C3 mesylate racemic
CAS :Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible monoamine oxidase inhibitor.Formule :C13H17NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :270.32Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formule :C15H11N5OCouleur et forme :SolidMasse moléculaire :277.28Orexin A (human, rat, mouse) (TFA)
Endogenous orexin receptor agonist with Ki of 20 nM (OX1) and 38 nM (OX2), promotes feeding, may regulate sleep-wake cycle.Formule :C154H244N47F3O46S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3675.12LY3027788
CAS :LY3027788, potent oral prodrug of LY3020371, is a strong mGlu2/3 antagonist with notable antidepressant effects.Formule :C25H31F2NO11SCouleur et forme :SolidMasse moléculaire :591.58
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