Neuroscience
Les inhibiteurs en neurosciences sont des composés conçus pour moduler l'activité de protéines, d'enzymes ou de récepteurs spécifiques au sein du système nerveux. Ces inhibiteurs sont cruciaux pour étudier les mécanismes moléculaires sous-jacents au fonctionnement neuronal, à la transmission synaptique et aux maladies neurodégénératives. En ciblant les récepteurs des neurotransmetteurs, les canaux ioniques et les voies de signalisation, les inhibiteurs en neurosciences facilitent l'exploration du fonctionnement cérébral et le développement de stratégies thérapeutiques pour des troubles neurologiques tels que la maladie d'Alzheimer, de Parkinson et l'épilepsie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs en neurosciences de haute qualité pour soutenir vos recherches en neurobiologie, neuropharmacologie et sciences cognitives.
Sous-catégories appartenant à la catégorie "Neuroscience"
- récepteur 5-HT(1.025 produits)
- ACK(1 produits)
- AChR(647 produits)
- ATP Citrate Lyase(17 produits)
- Récepteur adrénergique(3.028 produits)
- BACE(37 produits)
- Bêta-amyloïde(231 produits)
- CaMK(73 produits)
- COX(602 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur GABA(373 produits)
- Gamma-sécrétase(62 produits)
- GluR(265 produits)
- GlyT(26 produits)
- Récepteur de l'histamine(385 produits)
- LRRK2(42 produits)
- Récepteur de la mélatonine(26 produits)
- NMDAR(10 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
Affichez 12 plus de sous-catégories
5638 produits trouvés pour "Neuroscience"
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Imidafenacin Metabolite M4
CAS :Imidafenacin M4 is a CYP3A4-formed metabolite of the muscarinic antagonist imidafenacin.Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.368N-desmethyl Zolmitriptan
CAS :DZT, an active metabolite of zolmitriptan, agonizes 5-HT1B/D receptors; contracts human cerebral arteries (EC50=100nM).Formule :C15H19N3O2Couleur et forme :SolidMasse moléculaire :273.33β-Amyloid (33-40)
CAS :β-Amyloid (33-40) is a peptide comprising amino acids 33 to 40 of the beta-amyloid protein.Formule :C32H58N8O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :730.92CNS-Penetrant Compound Library
A unique collection of 509 CNS-Penetrant compounds for high throughput screening (HTS) and high content screening (HCS);Couleur et forme :Odour SolidRef: TM-L5900
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demanderBiperiden Hydrochloride
CAS :Biperiden HCl is an anti-Parkinson's drug, blocks M1 receptors, manages all Parkinson's types, and is FDA-approved. Non-toxic at 0.11 mg/kg to rats' cognition.Formule :C21H30ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :347.92SCH-900229
CAS :SCH-900229, a potent presenilin 1 selective γ-secretase inhibitor, used to treat Alzheimer’s Disease.Formule :C21H21ClF2O6S2Couleur et forme :SolidMasse moléculaire :506.97Dalidnetug
CAS :Dalidnetug is a humanized monoclonal antibody that targets human β-amyloid precursor protein (APP). By specifically binding to APP, Dalidnetug reduces the production of β-amyloid (Aβ), thereby demonstrating activity in clearing β-amyloid. This compound holds potential for research in Alzheimer's disease.Couleur et forme :LiquidLanuginosine
CAS :Lanuginosine, an aporphine alkaloid, exhibits cytotoxicity against U251.Formule :C18H11NO4Couleur et forme :SolidMasse moléculaire :305.28C2-8
CAS :C2-8 inhibits polyQ aggregation, IC50=25 μM (HDQ51), 0.05 μM (PC12 cells), reduces neurodegeneration in Huntington's models.Formule :C19H14Br2N2O3SCouleur et forme :SolidMasse moléculaire :510.2Trivalent GalNAc-DBCO
CAS :Trivalent GalNAc-DBCO is a synthetic ligand composed of three GalNAc units linked to DBCO. Trivalent GalNAc-DBCO undergoes strain-promoted alkyne–azide cycloaddition (SPAAC) reactions with azide-containing molecules without the need for copper catalysis. Trivalent GalNAc-DBCO binds specifically to the asialoglycoprotein receptor (ASGPR), thereby directing conjugated molecules into hepatocytes for lysosomal degradation through receptor-mediated endocytosis. Trivalent GalNAc-DBCO is extensively applied in studies of liver-targeted drug delivery, targeted degradation strategies, and hepatocyte-specific molecular engineering.Formule :C91H144N12O34Degré de pureté :96.33%Masse moléculaire :1950.18Neural Regeneration Compound Library
A unique collection of 149 neuroregeneration related compounds for high throughput and high content screening;Couleur et forme :Odour SolidRef: TM-L7700
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demanderGABAA receptor modulator-4
GABAA receptor modulator-4 (Compound 4) acts as a negative allosteric modulator of the GABAA receptor. It inhibits the peak and steady-state currents mediated by the α1β3γ2 GABAA receptors, with an IC50 of 10 μM for both.Formule :C15H17BrO4SCouleur et forme :SolidMasse moléculaire :373.26LY86057
CAS :LY86057 is a bioactive chemical.Formule :C20H26N2O3Couleur et forme :SolidMasse moléculaire :342.439Apoptosis Compound Library
A unique collection of 1760 apoptosis-related compounds for apoptosis research, research in tumorigenesis, and anti-cancer drug screening;Couleur et forme :Odour SolidRef: TM-L9000
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demanderSKF-83566 hydrochloride
CAS :SKF-83566 hydrochloride is a D1-like dopamine receptor antagonist, inhibiting dopamine transporters and mitigating GBP-induced CPP.Formule :C17H19BrClNODegré de pureté :99.27%Couleur et forme :SoildMasse moléculaire :368.69Minesapride
CAS :Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.
Formule :C21H31ClN4O5Degré de pureté :99.85% - 99.88%Couleur et forme :SolidMasse moléculaire :454.955-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formule :C24H26N4O2SCouleur et forme :SolidMasse moléculaire :434.55Fabesetron
CAS :Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.Formule :C18H19N3OCouleur et forme :SolidMasse moléculaire :293.37Iloperidone metabolite P95
CAS :Iloperidone metabolite P95, a non-brain penetrating compound, binds 5-HT2A, α1-, α2B-, α2C-receptors with Ki of 7.08-83.18 nM.Formule :C23H25FN2O5Couleur et forme :SolidMasse moléculaire :428.465-HT5AR/5-HT6R ligand-1
5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.Formule :C25H30N4O2SCouleur et forme :SolidMasse moléculaire :450.6Xaliproden
CAS :Xaliproden is a biochemical.Formule :C24H22F3NCouleur et forme :SolidMasse moléculaire :381.43I2-IRs ligand-1
I2-IRs ligand-1 (Compound 12d) is an orally active compound capable of crossing the blood-brain barrier. It exhibits high affinity for imidazoline I2 receptors (I2-IRs) with a pKi of 9.98. This compound can enhance cognitive deficits in aging mice and possesses analgesic, anti-inflammatory, and neuroprotective properties. I2-IRs ligand-1 is applicable for research in Alzheimer's disease and related pain disorders.Formule :C21H23ClFN2O4PCouleur et forme :SolidMasse moléculaire :452.84(+)-OSU 6162
CAS :(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Formule :C15H23NO2SDegré de pureté :98.19%Couleur et forme :SoildMasse moléculaire :281.41Ref: TM-T60027
1mg73,00€5mg146,00€1mL*10mM (DMSO)155,00€10mg208,00€25mg319,00€50mg447,00€100mg600,00€200mg808,00€ACG548B
CAS :ACG548B inhibits AChE/BChE with IC50s of 1.78/0.496 μM; favors AChE over BChE/ChoK.Formule :C38H34Br2Cl2N4Couleur et forme :SolidMasse moléculaire :777.43Anticonvulsant agent 2
CAS :Anticonvulsant agent 2 is a potent orally active anticonvulsant that has shown antiepileptic activity in a model of drug-resistant epilepsy.Formule :C21H17ClN2Degré de pureté :99.77%Couleur et forme :SoildMasse moléculaire :332.83Small Cardioactive Peptide B (SCPB)
CAS :SCPB: neurally active peptide, boosts adenylate cyclase in heart/gills, EC50s: 0.1 μM (heart), 1.0 μM (gills).Formule :C52H80N14O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1141.41Sandaracopimaric acid
CAS :Sandaracopimaric acid, an anti-inflammatory diterpene, relaxes pulmonary arteries with an EC50 of 43.93 μM.Formule :C20H30O2Couleur et forme :SolidMasse moléculaire :302.456,9-Dichloro-1,2,3,4-tetrahydroacridine
CAS :6,9-Dichloro-1,2,3,4-tetrahydroacridine is a synthetic intermediate in the synthesis of tacrine-based acetylcholinesterase (AChE) inhibitors.1It is also anFormule :C13H11Cl2NCouleur et forme :SolidMasse moléculaire :252.1391H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)-
CAS :1H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)- is a low activity isomer of S 18986.Formule :C10H12N2O2SDegré de pureté :99.96%Couleur et forme :SoildMasse moléculaire :224.28Aducanumab
CAS :Aducanumab (BIIB037) is an IgG1 antibody targeting amyloid beta to treat Alzheimer's; it's brain-permeable.Degré de pureté :95% - 97.10%Couleur et forme :LiquidMasse moléculaire :145.93 kDaDAA-1106
CAS :DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.Formule :C23H22FNO4Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :395.42Crenezumab
CAS :Crenezumab (MABT 5102A) is a fully humanized anti-amyloid-beta antibody that binds to multiple forms of amyloid-beta (Aβ) for the study of Alzheimer's disease.Degré de pureté :97.5% (SDS-PAGE); 95.3% (SEC-HPLC) - 97.5% (SDS-PAGE); 95.3% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :143.32 kDaLY-426965 hydrochloride
CAS :LY-426965 hydrochloride is a bioactive chemical.Formule :C28H39ClN2O2Couleur et forme :SolidMasse moléculaire :471.07DISC-0974
DISC-0974 is a humanized antibody targeting RGMC/HFE2, which can be used to study urogenital system diseases.Couleur et forme :LiquidMasse moléculaire :145.66 kDaPolyglutamine binding peptide 1
CAS :Polyglutamine binding peptide 1 (QBP1) is a peptide inhibitor of polyglutamine (polyQ). It effectively inhibits polyQ protein aggregation in vitro and prevents polyQ-induced cell death in cell cultures.Formule :C72H90N16O16Couleur et forme :SolidMasse moléculaire :1435.583-Aminopropylphosphonic Acid
CAS :3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding
Formule :C3H10NO3PDegré de pureté :99.84%Couleur et forme :Light Yellow LiquidMasse moléculaire :139.09Aceclidine (hydrochloride)
CAS :agonist of muscarinic receptorsFormule :C9H16ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :205.68Neuronal Signaling Compound Library
A unique collection of xnum compounds targeting CNS signaling for high throughput screening (HTS) and high content screening (HCS) for new drugs;Couleur et forme :Odour SolidRef: TM-L2600
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demanderCDD0102 HCl
CAS :CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.Formule :C8H13ClN4ODegré de pureté :99.7%Couleur et forme :SoildMasse moléculaire :216.67(Iso)-Landipirdine
CAS :(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Formule :C18H19FN2O3SDegré de pureté :98.94%Couleur et forme :SoildMasse moléculaire :362.42Coumarinic acid
CAS :Coumarinic acid serves as a brain-penetrating inhibitor of AChE (acetylcholinesterase) and β-amyloid, with applications in anti-Alzheimer's drug research [1].Formule :C9H8O3Couleur et forme :SolidMasse moléculaire :164.16AL 34662
CAS :AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also aFormule :C10H13N3ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :191.23Flupyradifurone
CAS :Flupyradifurone (flupyradifurone) is a systemic insecticide and nicotinic acetylcholine receptor (nAChR) agonist interfer nervous system of insects.Formule :C12H11ClF2N2O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :288.68Methoxy-X04
CAS :Methoxy-X04, a derivative of Congo red and Chrysamine-G, is a brain-permeable fluorescent probe for amyloid-β (Aβ).
Formule :C23H20O3Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :344.4Tiflucarbine
CAS :Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity of solubleFormule :C16H17FN2SDegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :288.38Pep63
CAS :Pep63, a neuroprotective peptide (VFQVRARTVA), enhances synaptic plasticity and memory. It competitively binds with Aβ1-42 oligomers, thereby inhibiting the formation of Aβ fibrils. Pep63 is employed in research focused on Alzheimer's disease (AD).Formule :C51H87N17O13Couleur et forme :SolidMasse moléculaire :1146.34Suntinorexton
CAS :Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.Formule :C23H28F2N2O4SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :466.54Ref: TM-T39807
1mg171,00€5mg418,00€1mL*10mM (DMSO)428,00€10mg666,00€25mg1.017,00€50mg1.372,00€100mg1.793,00€200mg2.405,00€Sodium Channel Targeted Library
A unique collection of xnum sodium channel blockers and agonists for high throughput and high content screening;Couleur et forme :Odour SolidRef: TM-L7400
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demanderTMPH
CAS :TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.Formule :C16H31NO2Degré de pureté :99.78%Couleur et forme :SoildMasse moléculaire :269.42Ref: TM-T60080
2mg35,00€1mL*10mM (DMSO)54,00€5mg55,00€10mg84,00€25mg133,00€50mg205,00€100mg301,00€200mg425,00€α-Conotoxin AuIB
CAS :Selective antagonist of α3β4 nicotinic acetylcholine receptors.Formule :C65H89N17O21S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1572.76isomer-Cilansetron
CAS :isomer-Cilansetron is an isomer of Cilansetron.Formule :C20H21N3ODegré de pureté :99.92% - 99.96%Couleur et forme :SoildMasse moléculaire :319.4COX-2-IN-33
COX-2-IN-33 (compound 5f) is a selective COX-2 inhibitor with an IC50 value of 45.5 nM and exhibits potential as an anti-inflammatory agent.Formule :C20H13ClF3N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.8[D-Trp7,9,10]-Substance P
CAS :Substance P analog that inhibits activation of Gq/11 by M1 muscarinic ACh receptors. Does not inhibit Gi/o activation by M2 ACh receptors.Formule :C79H105N21O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1588.89CaMKIIα-PHOTAC
CaMKIIα-PHOTAC is a photochemically targeted chimera (PHOTAC) that specifically targets Ca2+/calmodulin-dependent protein kinase II α (CaMKIIα).Formule :C54H58Cl2N10O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1094Xylamidine
CAS :Xylamidine is a biochemical.Formule :C19H24N2O2Couleur et forme :SolidMasse moléculaire :312.41MmTx1 toxin
Micrurotoxin 1 (MmTx1 toxin) acts as an allosteric modulator of GABA A receptors, enhancing the receptor's sensitivity to its agonist [1].Formule :C295H455N95O97S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7205(Iso)-Atagabalin HCl
CAS :(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.Formule :C10H20ClNO2Degré de pureté :99.88% - >99.99%Couleur et forme :SoildMasse moléculaire :221.72FGIN-1-43
CAS :FGIN-1-43 is a potent and specific ligand for the mitochondrial DBI receptor.Formule :C28H36Cl2N2ODegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :487.5(+)-Coclaurine hydrochloride
CAS :(+)-Coclaurine hydrochloride, also known as (+)-(R)-Coclaurine, is a benzyltetrahydroisoquinoline alkaloid extracted from multiple plant species.Formule :C17H20ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.8Antidepressant agent 5
CAS :Antidepressant agent 5 is a 7-substituted tetrahydroisoquinoline derivative with antidepressant activity.Antidepressant agent 5 acts similarly to magnoflorine
Formule :C20H25NO3Degré de pureté :99.34%Couleur et forme :SoildMasse moléculaire :327.42Guvacine hydrobromide
CAS :Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake.Formule :C6H10BrNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :208.05Imagabalin
CAS :Imagabalin is an active compound used in the study of neurological diseases.Formule :C9H19NO2Couleur et forme :SolidMasse moléculaire :173.25Methyl piperate
CAS :Methylpiperic acid, a piperine alkaloid, exhibits potent inhibitory activity on monoamine oxidase (MAO), with differing efficacy on isoforms: greater inhibitionFormule :C13H12O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :232.23COX-1/2-IN-5
COX-1/2-IN-5 (compound 2a) functions as a dual inhibitor of COX1/2, demonstrating inhibitory concentrations (IC50) of 2.650 μM and 0.958 μM, respectively, and
Formule :C21H22N2O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :414.47Proadrenomedullin (1-20), human
CAS :Endogenous peptide; agonist of MRGPRX2 (EC50=251 nM); noncompetitive inhibitor of nicotinic receptors; reduces catecholamine secretion; antihypertensive.Formule :C112H178N36O27Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2460.84Mirtazapine N-oxide
CAS :Mirtazapine N-oxide, a mirtazapine metabolite, is produced by CYP1A2 and CYP3A4 in human liver.Formule :C17H19N3OCouleur et forme :SolidMasse moléculaire :281.359Lysyl hydroxylase 2-IN-1
"Lysyl Hydroxylase 2-IN-1 (compound 12) is a selective inhibitor of lysyl hydroxylase 2 (LH2) with an IC50 of approximately 300 nM and demonstrates specificityFormule :C18H18N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :310.35BChE-IN-16
BChE-IN-16 (compound 87) is a potent inhibitor of human butyrylcholinesterase (hBChE) exhibiting an inhibition concentration half-maximum (IC50) of 3.8 nM.Formule :C28H32FNO2Couleur et forme :SolidMasse moléculaire :433.56Fentonium bromide
CAS :Fentonium bromide is a biochemical.Formule :C31H34BrNO4Couleur et forme :SolidMasse moléculaire :564.515-methoxy-α-Ethyltryptamine
CAS :5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects.
Formule :C13H18N2ODegré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :218.29Glycerophosphorylethanolamine (sodium salt)
CAS :Glycerophosphorylethanolamine, a phosphatidylethanolamine metabolite, elevates in Alzheimer's and promotes Aβ40 aggregation.Formule :C5H13NNaO6PCouleur et forme :SolidMasse moléculaire :237.12Methylatropine (nitrate)
CAS :Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.Formule :C18H26N2O6Couleur et forme :SolidMasse moléculaire :366.414Calmodulin Kinase IINtide, Myristoylated
Myristoylated Calmodulin Kinase IINtide (Myr-CaMKIINtide) serves as a selective and noncompetitive inhibitor of CaMKII [1].Formule :C156H275N47O43Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3497.14MAO-B-IN-4
MAO-B-IN-4 (Compound 26) is a reversible monoamine oxidase B (MAO-B) inhibitor with potent in vitro activity, characterized by an IC50 value of 9 nM.Formule :C23H20ClF2N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :411.87LOX-IN-4
CAS :LOX-IN-4 (Compound 112) is an inhibitor of lysyl oxidase (LOX). It holds potential for use in cancer research.Formule :C20H24Cl2FN3O2SCouleur et forme :SolidMasse moléculaire :460.39Desmethyl Mirtazapine (hydrochloride)
CAS :Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Formule :C16H18ClN3Couleur et forme :SolidMasse moléculaire :287.79IHC3
IHC3 is a competitive and reversible monoamine oxidase B (MAO-B) inhibitor with an IC50 of 1.672 μM, which targets Cys172 within the enzyme's active site.Formule :C17H12FN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.3PZ-1922
PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.Degré de pureté :98%Couleur et forme :Odour SolidOxotremorine
CAS :Oxotremorine acts as an agonist of mAChR, specifically activating the M1 and M3 acetylcholine receptors. In drug discrimination experiments with macaques, it exhibits effects similar to nicotine.Formule :C12H18N2OCouleur et forme :SolidMasse moléculaire :206.28E3 ligase Ligand 41
CAS :E3 Ligase Ligand 41 (Compound SI-13) serves as a ligand for the E3 ubiquitin ligase DCAF16. It is designed to connect with SLF through a linker, enabling the formation of KB03-SLF.Formule :C13H12ClF3N2O4Couleur et forme :SolidMasse moléculaire :352.69Biphenyl-3′,3,4,4′-tetrol
CAS :Biphenyl-3′,3,4,4′-tetrol (BPT) is a potent inhibitor of Aβ40 aggregation and can be utilized in research related to neurodegenerative diseases such as Alzheimer's.Formule :C12H10O4Couleur et forme :SolidMasse moléculaire :218.21Lon 954
CAS :Lon 954, also known as Harmine, is a fluorescent harmala alkaloid belonging to the beta-carboline family of compounds.Formule :C9H10Cl3N3OCouleur et forme :SolidMasse moléculaire :282.55GAD65(247-266) epitope TFA
GAD65(247-266) epitope TFA, a T cell epitope derived from islet antigens, exhibits competitive binding to the type I diabetes-associated molecule I-A g7, albeitFormule :C111H174F3N27O29S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2535.99MmTx2 toxin
MmTx2 toxin, extracted from the venom of the coral snake, serves as a modulator of the GABA A receptor, increasing its responsiveness to agonists.Formule :C295H450N94O97S10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7185.95CALP2
CAS :CALP2 is a CaM antagonist blocking EF-hand/Ca2+ site; inhibits CaM phosphodiesterase, raises Ca2+, and activates alveolar macrophages.Formule :C68H104N14O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1357.72Lysyl hydroxylase 2-IN-2
Lysyl Hydroxylase 2-IN-2 (compound 13) is a potent inhibitor of Lysyl Hydroxylase 2 (LH2), exhibiting an IC50 of approximately 500 nM.Formule :C19H21N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :323.39MAO-B-IN-18
MAO-B-IN-18 is a potent, selective inhibitor of MAO B, demonstrating IC50 values of 52 nM for hMAO B and 14 μM for hMAO A.Formule :C25H22N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :458.47Kynuramine
CAS :Kynuramine is an aromatic ketone containing the aniline structure.
Formule :C9H12N2OCouleur et forme :SolidMasse moléculaire :164.20Emamectin B1a
CAS :Emamectin B1a can be used in relevant research in the life sciences. Its product number is T37663 and CAS number is 121124-29-6.
Formule :C49H75NO13Couleur et forme :SolidMasse moléculaire :886.133MAO-B-IN-24
MAO-B-IN-24 (compound 11h) is a selective, reversible, competitive inhibitor of MAO-B with an IC50 value of 1.60 μM.Formule :C20H18N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.37Chrysophanol-1-O-β-gentiobioside
CAS :Chrysophanol-1-O-β-gentiobioside, an anthraquinone glycoside obtained from the seeds of Cassia obtusifolia, exhibits targeted inhibition of hMAO-A isozymeFormule :C27H30O14Couleur et forme :SolidMasse moléculaire :578.52NMDA receptor antagonist 6
NMDA Receptor Antagonist 6 (Compound 13b) functions as an antagonist at the glycine-binding site of the NMDA receptor and demonstrates cytoneuroprotectiveFormule :C25H23NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :369.46MAO-B-IN-3
MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a KiFormule :C24H25N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.47Anisatin
Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.Formule :C15H20O8Couleur et forme :SolidMasse moléculaire :328.3175-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFormule :C17H22Cl2N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.37Alverine hydrochloride
CAS :Alverine hydrochloride is a parasympatholytic.Formule :C20H28ClNCouleur et forme :SolidMasse moléculaire :317.9Tranylcypromine
CAS :Tranylcypromine (SKF 385), a potent monoamine oxidase (MAO) inhibitor [1], is used in medicinal applications.Formule :C9H11NDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :133.19AChE/BChE-IN-14
AChE/BChE-IN-14 (compound 13), a benzylisoquinoline alkaloid extracted from Fissistigma polyanthum roots, demonstrates inhibitory effects on bothFormule :C19H23NO3Couleur et forme :SolidMasse moléculaire :313.39MAO-B-IN-25
MAO-B-IN-25 (compound 92) is a selective inhibitor of monoamine oxidase B (MAO-B), exhibiting inhibitory half-maximal inhibitory concentrations (IC50) of 240 nMFormule :C16H13BrO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :333.18MRS7925
MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosisFormule :C20H26IN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :511.36
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