Neuroscience
Les inhibiteurs en neurosciences sont des composés conçus pour moduler l'activité de protéines, d'enzymes ou de récepteurs spécifiques au sein du système nerveux. Ces inhibiteurs sont cruciaux pour étudier les mécanismes moléculaires sous-jacents au fonctionnement neuronal, à la transmission synaptique et aux maladies neurodégénératives. En ciblant les récepteurs des neurotransmetteurs, les canaux ioniques et les voies de signalisation, les inhibiteurs en neurosciences facilitent l'exploration du fonctionnement cérébral et le développement de stratégies thérapeutiques pour des troubles neurologiques tels que la maladie d'Alzheimer, de Parkinson et l'épilepsie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs en neurosciences de haute qualité pour soutenir vos recherches en neurobiologie, neuropharmacologie et sciences cognitives.
Sous-catégories appartenant à la catégorie "Neuroscience"
- récepteur 5-HT(1.025 produits)
- ACK(1 produits)
- AChR(648 produits)
- ATP Citrate Lyase(17 produits)
- Récepteur adrénergique(3.028 produits)
- BACE(37 produits)
- Bêta-amyloïde(231 produits)
- CaMK(73 produits)
- COX(602 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur GABA(372 produits)
- Gamma-sécrétase(63 produits)
- GluR(265 produits)
- GlyT(26 produits)
- Récepteur de l'histamine(385 produits)
- LRRK2(42 produits)
- Récepteur de la mélatonine(26 produits)
- NMDAR(10 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(327 produits)
Affichez 12 plus de sous-catégories
5637 produits trouvés pour "Neuroscience"
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Naratriptan D3 Hydrochloride
CAS :Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.Formule :C17H26ClN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.94AChE-IN-4
AChE-IN-4 is an acetylcholine esterase inhibitor (AChEI) with an IC50 value of 24.1 μM.Formule :C32H25BrN6O4SCouleur et forme :SolidMasse moléculaire :669.55LY3027788
CAS :LY3027788, potent oral prodrug of LY3020371, is a strong mGlu2/3 antagonist with notable antidepressant effects.Formule :C25H31F2NO11SCouleur et forme :SolidMasse moléculaire :591.58MAO-B-IN-20
MAO-B-IN-20, potent with 0.037 μM IC50, is stable and BBB permeable, useful for Parkinson's research.Formule :C20H18F2N2O2Couleur et forme :SolidMasse moléculaire :356.37SIB 1553A
CAS :SIB 1553A is an agonist of nAChRs, a cognitive enhancer that can be used to study diseases associated with neurodegeneration.Formule :C13H19NOSDegré de pureté :99.79%Couleur et forme :SoildMasse moléculaire :237.36Emraclidine
CAS :Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.Formule :C20H21F3N4ODegré de pureté :99.63% - 99.96%Couleur et forme :SolidMasse moléculaire :390.4Ref: TM-T9694
1mg120,00€2mg170,00€5mg289,00€1mL*10mM (DMSO)319,00€10mg467,00€25mg835,00€50mg1.134,00€100mg1.504,00€γ-Secretase Modulators
CAS :gamma-Secretase Modulators serves as a useful treatment for Alzheimer's disease by inhibiting the production of Amyloid-β.Formule :C26H24F3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :483.48Guanylyl Imidodiphosphate (lithium salt)
CAS :Guanylyl Imidodiphosphate (lithium salt) is a non-hydrolyzable GTP analog that increases adenylate cyclase activity.Formule :C10H13Li4N6O13P3Couleur et forme :SolidMasse moléculaire :545.93BU 226 hydrochloride
CAS :BU 226 hydrochloride demonstrates affinity for imidazoline (I) receptors, in particular the I2 binding site with a Ki of 1.4 nM.Formule :C12H12ClN3Degré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :233.7mGluR5 modulator 1
CAS :mGluR5 modulator 1 is a positive modulator for mGluR5, used in schizophrenia and cognitive research.Formule :C18H19ClFN3O2Couleur et forme :SolidMasse moléculaire :363.82SB 258585
CAS :SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.Formule :C18H22IN3O3SDegré de pureté :99.77%Couleur et forme :SoildMasse moléculaire :487.36sabcomeline
CAS :Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.Formule :C10H15N3OCouleur et forme :SolidMasse moléculaire :193.25LU-32-176B
CAS :LU32-176B is a bioactive chemical.Formule :C23H24F2N2O2Couleur et forme :SolidMasse moléculaire :398.45Feralolide
CAS :Feralolide, a dihydroisocoumarin from the methanolic extract of aloe vera resin, functions as a dual inhibitor of acetylcholinesterase (AChE) andFormule :C18H16O7Couleur et forme :SolidMasse moléculaire :344.32AChE-IN-36
AChE-IN-36 (compound A4) is an acetylcholinesterase inhibitor with an IC50 of 0.04 μM, influencing ROS levels and modulating the gene expression of NRF2 [1].Formule :C25H21ClO5SCouleur et forme :SolidMasse moléculaire :468.95Tabernanthalog
CAS :TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.Formule :C14H18N2ODegré de pureté :99.82% - 99.89%Couleur et forme :SoildMasse moléculaire :230.31Ref: TM-T60221
1mg175,00€2mg264,00€1mL*10mM (DMSO)344,00€5mg404,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€3-Aminopropylphosphinic acid
CAS :3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).
Formule :C3H10NO2PCouleur et forme :SolidMasse moléculaire :123.092Org 13011
CAS :Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Formule :C18H25F3N4ODegré de pureté :98.02%Couleur et forme :SoildMasse moléculaire :370.41Ref: TM-T28258L
1mg109,00€5mg261,00€1mL*10mM (DMSO)266,00€10mg374,00€25mg583,00€50mg803,00€100mg1.063,00€200mg1.431,00€Cyclodrine
CAS :Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.Formule :C19H29NO3Degré de pureté :97.62%Couleur et forme :SoildMasse moléculaire :319.44Ref: TM-T10914L
1mg73,00€1mL*10mM (DMSO)148,00€5mg149,00€10mg212,00€25mg319,00€50mg447,00€100mg610,00€200mg822,00€β-Amyloid (1-28)
CAS :β-Amyloid (1-28) is a β-Amyloid protein fragment involved in metal binding.Formule :C145H209N41O46Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3262.51Alosetron-d3
CAS :Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Formule :C17H18N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :297.37TAT-CN21 (scrambled)
TAT-CN21(scrambled) is a control peptide lacking specific targeting activity and serves as a negative control for TatCN21. TatCN21 is an effective and selective inhibitory peptide for calcium/calmodulin-dependent protein kinase II (CaMKII).Couleur et forme :Odour Solidβ-Secretase Inhibitor II
CAS :β-Secretase Inhibitor II is a tripeptide aldehyde compound that acts as an inhibitor of β-Secretase.Formule :C25H39N3O5Couleur et forme :SolidMasse moléculaire :461.59LE 300
CAS :LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Formule :C20H22N2Degré de pureté :97.91% - 98.79%Couleur et forme :SolidMasse moléculaire :290.4XL01126
XL01126 degrades LRRK2 (DC50: 14 nM G2019S, 32 nM WT), crosses the blood-brain barrier, aiding Parkinson's studies.Formule :C50H64ClFN10O6S2Couleur et forme :SolidMasse moléculaire :1019.69R-(+)-Cotinine
CAS :R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.Formule :C10H12N2OCouleur et forme :SolidMasse moléculaire :176.22(S)-3,4-DCPG HCl
(S)-3,4-DCPG HCl is a selective mGluR8a agonist, impacting AV12-664 cells with an EC50 of 31 nM.Formule :C10H10ClNO6Degré de pureté :99.53% - 99.86%Couleur et forme :SoildMasse moléculaire :275.64Ref: TM-T23288L
1mg173,00€1mL*10mM (DMSO)394,00€5mg437,00€10mg625,00€25mg982,00€50mg1.341,00€100mg1.773,00€500mg3.565,00€α-Conotoxin PIA
CAS :Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nMFormule :C79H125N27O25S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1981.3Epiboxidine hydrochloride
CAS :Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.Formule :C10H15ClN2OCouleur et forme :SolidMasse moléculaire :214.69Tropicamide
CAS :Tropicamide (Ro 1-7683), a synthetic atropine-like muscarinic antagonist, dilates pupils and paralyzes eye muscles for diagnostic use.Formule :C17H20N2O2Degré de pureté :99.78% - 99.94%Couleur et forme :White PowderMasse moléculaire :284.35Atracurium
CAS :Atracurium (BW-33A) is a competitive AChR antagonist and non-depolarizing muscle relaxant that may cause bronchoconstriction.Formule :C53H72N2O122Couleur et forme :SolidMasse moléculaire :929.14FRM-024
CAS :FRM-024 is a powerful gamma secretase modulator with the ability to penetrate the central nervous system (CNS), designed specifically for the treatment ofFormule :C22H22ClN5O2Couleur et forme :SolidMasse moléculaire :423.9Zanapezil free base
CAS :Zanapezil (TAK-147): potent, selective AChE inhibitor; reversible; IC50=51.2 nM; moderate M1/M2 inhibition; AD research potential.Formule :C25H32N2OCouleur et forme :SolidMasse moléculaire :376.544p-HTAA
CAS :Pentamer Hydrogen Thiophene Acetic Acid (p-HTAA) is a compound that specifically targets and labels amyloid-beta (Aβ) deposits in the brains of living mice [1].Formule :C24H16O4S5Couleur et forme :SolidMasse moléculaire :528.71Sintamil
CAS :Sintamil is a useful organic compound for research related to life sciences. The catalog number is T71697 and the CAS number is 16398-39-3.Formule :C18H20ClN3O4Couleur et forme :SolidMasse moléculaire :377.822-Methyl-1-indanone
CAS :2-Methyl-1-indanone is an acetylcholinesterase inhibitor and can be used for biochemical experiments and drug synthesis.Formule :C10H10ODegré de pureté :96.6%Couleur et forme :SolidMasse moléculaire :146.19M 8218
CAS :M 8218 is a bioactive chemical.Formule :C20H29NO2Couleur et forme :SolidMasse moléculaire :315.45β-Amyloid (11-22)
CAS :β-Amyloid (11-22) is a peptide fragment of β-Amyloid.Beta-amyloid peptide (Abeta), the major constituent of amyloid plaques in the brains of Alzheimer’sFormule :C70H102N18O18Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1483.67Arisugacin G
CAS :Arisugacin G, a microbial metabolite, is a structural analogue of Arisugacin A. Unlike its analogue, Arisugacin G does not exhibit activity against AChE (acetylcholinesterase).Formule :C27H32O5Couleur et forme :SolidMasse moléculaire :436.54BuChE-IN-21
BuChE-IN-21 (compound SXF3) is a potent and selective inhibitor of BuChE, demonstrating inhibitory effects on eqBuChE and hBuChE with IC50 values of 0.05 and 0.04 μM, respectively. Additionally, BuChE-IN-21 exhibits significant anti-inflammatory activity.Formule :C16H23NO2Couleur et forme :SolidMasse moléculaire :261.17288MGS0028
CAS :MGS0028 is a selective agonist of metabotropic glutamate 2/3 receptor, it could reverse abnormal behaviors in mice induced by isolation rearing.Formule :C8H8FNO5Couleur et forme :SolidMasse moléculaire :217.15Suntinorexton
CAS :Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.Formule :C23H28F2N2O4SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :466.54Ref: TM-T39807
1mg171,00€5mg418,00€1mL*10mM (DMSO)428,00€10mg666,00€25mg1.017,00€50mg1.372,00€100mg1.793,00€200mg2.405,00€BRD9 ligand-6
CAS :BRD9 ligand-6 serves as a ligand for the target protein in PROTAC applications. It is utilized in the synthesis of FHD-609.Formule :C21H21N3O4Couleur et forme :SolidMasse moléculaire :379.41β-Amyloid (1-17)
CAS :This synthetic peptide consists of amino acids 1 to 17 of beta amyloid protein. This peptide can be employed in beta amyloid solubility studies.Formule :C90H130N28O29Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2068.2β-Amyloid (12-20)
CAS :β-Amyloid (12-20) is a peptide fragment of β-Amyloid.Thsis peptide contain the amino acid residues VFF at position (18-20), suggesting that this triad hasFormule :C57H83N15O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1154.368-Aminoadenine
CAS :8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.Formule :C5H6N6Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :150.14Duloxetine D3 hydrochloride
CAS :Duloxetine D3 HCl is a deuterium-labeled SNRI, treats depression/GAD, Ki 4.6 nM.Formule :C18H20ClNOSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.89Pep63
CAS :Pep63, a neuroprotective peptide (VFQVRARTVA), enhances synaptic plasticity and memory. It competitively binds with Aβ1-42 oligomers, thereby inhibiting the formation of Aβ fibrils. Pep63 is employed in research focused on Alzheimer's disease (AD).Formule :C51H87N17O13Couleur et forme :SolidMasse moléculaire :1146.34VVZ-149
VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.Couleur et forme :Solid4,4-Difluorobenzhydrol
CAS :Compound PDK0200, with CAS No. 365-24-2, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0200 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C13H10F2OCouleur et forme :Off-White CrystalsMasse moléculaire :220.21α-Conotoxin imi
CAS :alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.Formule :C52H78N20O15S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1351.56UCM 549
CAS :UCM 549 is a bioactive chemical.Formule :C19H21NO2Couleur et forme :SolidMasse moléculaire :295.381-(2-Methoxyphenyl)piperazine hydrochloride
CAS :Compound PDK0265, with CAS No. 5464-78-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0265 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C11H16N2OMasse moléculaire :192.25GABOB (β-hydroxy-GABA)
CAS :GABOB, an epilepsy treatment, is GABA's analogue and may act as a neurotransmitter.Formule :C4H9NO3Couleur et forme :White To Light Yellow Crystal PowderMasse moléculaire :119.125H-Pyrido[4,3-b]indole
CAS :5H-Pyrido[4,3-b]indole is a potential AchE/ChE inhibitor with potential antiviral activity for the study of neurodegenerative diseases.Formule :C11H8N2Degré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :168.2Dihydrochalcone
CAS :Compound PDK0018, with CAS No. 1083-30-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0018 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C15H14OCouleur et forme :SolidMasse moléculaire :210.27(S)-AMPA HCl
(S)-AMPA HCl (L-AMPA HCl) is a selective AMPA receptor agonist with potential antidepressant activity. It can be used in research on Parkinson's disease.Formule :C7H11ClN2O4Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :222.63SD-254
CAS :SD-254 is a deuterium analog of Effexor, with fewer side effects and a longer half-life.Formule :C17H27NO2Masse moléculaire :286.46M4 mAChR agonist-1
CAS :M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).Formule :C14H18N4OSDegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :290.38Atagabalin
CAS :Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.Formule :C10H19NO2Couleur et forme :SolidMasse moléculaire :185.26Hydroxytacrine maleate
CAS :Hydroxytacrine maleate (Velnacrine maleate) is a cholinesterase inhibitor used in the study of Alzheimer's type dementia (SDAT).Formule :C17H18N2O5Degré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :330.34Eletriptan
CAS :Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.Formule :C22H26N2O2SCouleur et forme :SolidMasse moléculaire :382.52Sulamserod
CAS :Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular relatedFormule :C19H28ClN3O5SDegré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :445.96RA306
RA306 is an orally active CAMK2 inhibitor that effectively disrupts the PEAK1/CAMK2 signaling pathway. It demonstrates anti-tumor activity by inhibiting proliferation, migration, and invasion of breast cancer cells. Additionally, RA306 shows potential in cardiac disease research, as it improves dilated cardiomyopathy in mice.Couleur et forme :Odour SolidOXA(17-33)
CAS :Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.Formule :C79H125N23O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1749(S)-Vamicamide
CAS :(S)-Vamicamide is an anti-anticholinergic compound.Formule :C18H23N3ODegré de pureté :99.48% - 99.65%Couleur et forme :SoildMasse moléculaire :297.39Flupyradifurone
CAS :Flupyradifurone (flupyradifurone) is a systemic insecticide and nicotinic acetylcholine receptor (nAChR) agonist interfer nervous system of insects.Formule :C12H11ClF2N2O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :288.68N-Ethyl-N-(3-pyridylmethyl)amine
CAS :N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.Formule :C8H12N2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :136.19Rasagiline 13C3 mesylate racemic
CAS :Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible monoamine oxidase inhibitor.Formule :C13H17NO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :270.32Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formule :C15H11N5OCouleur et forme :SolidMasse moléculaire :277.28AChE-IN-76
AChE-IN-76 (compound 6) is an acetylcholinesterase inhibitor with an IC50 of 7.6 nM.Couleur et forme :Odour Solidα5-GABAA receptor modulator 1
α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.Formule :C21H20FN3O4Couleur et forme :SolidMasse moléculaire :397.4AL 34662
CAS :AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also aFormule :C10H13N3ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :191.23K1833
K1833 is an inhibitor and reactivator of human acetylcholinesterase (hrAChE), exhibiting an inhibition concentration (IC50) of 58$.Couleur et forme :Odour SolidBuChE-IN-16
BuChE-IN-16 (Compound 6a) is an orally active, blood-brain barrier-permeable, and selective BuChE inhibitor with an IC50 of 0.33 μM. It exhibits anti-inflammatory and neuroprotective effects, improves cognitive function in Alzheimer's disease (AD) zebrafish models, and alleviates scopolamine-induced memory impairment in mice. BuChE-IN-16 is applicable for Alzheimer's disease research.Formule :C16H22N2O3Couleur et forme :SolidMasse moléculaire :290.36Tampramine
CAS :Tampramine: a TCA and selective norepinephrine inhibitor, with low affinity for other receptors, potential treatment for FST depression.
Formule :C23H24N4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :356.46PSEN1-IN-1
PSEN1-IN-1 (Compound (+)-13b) functions as an inhibitor of PSEN1, displaying potent inhibition of the PSEN1-APH1A and PSEN1-APH1B complexes with respective IC50Formule :C20H19ClF3NO3SCouleur et forme :SolidMasse moléculaire :445.882'-O-Succinyl-cAMP
CAS :2'-O-Monosuccinyladenosine-3',5'-cyclic monophosphate is an immunogenic derivative of cAMP that has been used to generate anti-cAMP antisera and antibodies.1,2Formule :C14H16N5O9PCouleur et forme :SolidMasse moléculaire :429.282(Iso)-Landipirdine
CAS :(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.Formule :C18H19FN2O3SDegré de pureté :98.94%Couleur et forme :SoildMasse moléculaire :362.42CDD0102 HCl
CAS :CDD0102 HCl is a selective and potent M1 muscarinic receptor agonist for the treatment of Alzheimer's disease.Formule :C8H13ClN4ODegré de pureté :99.7%Couleur et forme :SoildMasse moléculaire :216.67mHTT-IN-1
CAS :mHTT-IN-1 is a potent inhibitor of toxic mHTT, linked to Huntington's disease, with an EC50 of 46 nM.Formule :C18H19N7OSCouleur et forme :SolidMasse moléculaire :381.455-HT2A receptor agonist-5
CAS :5-HT2A receptor agonist-5 (compound I-3) is a potent 5-HT2A agonist with a Ki value of 0.017 µM and exhibits antidepressant activity.Formule :C23H29N3OCouleur et forme :SolidMasse moléculaire :363.5Davunetide acetate
Davunetide acetate is derived from activity-dependent neuroprotective protein existing in the mammalian CNS.
Formule :C38H64N10O14Degré de pureté :99.52% - 99.78%Couleur et forme :SolidMasse moléculaire :884.97Xanthohumol I
Xanthohumol I is a natural product that can be used as a reference standard.Formule :C21H22O6Couleur et forme :SolidMasse moléculaire :370.401Polyglutamine binding peptide 1
CAS :Polyglutamine binding peptide 1 (QBP1) is a peptide inhibitor of polyglutamine (polyQ). It effectively inhibits polyQ protein aggregation in vitro and prevents polyQ-induced cell death in cell cultures.Formule :C72H90N16O16Couleur et forme :SolidMasse moléculaire :1435.58β-Amyloid (1-15)
CAS :β-Amyloid (1-15) (Amyloid β-Protein (1-15)) is a fragment of β-amyloid protein used in the study of Alzheimer's disease.Formule :C78H107N25O27Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :1826.84CAY10787
CAS :CAY10787, an oxysterol, inhibits GABAA receptors (IC50s: 1-1.5μM) and lessens GABA responses in mouse DRG neurons.Formule :C27H42OCouleur et forme :SolidMasse moléculaire :382.632Notch 1 TFA
Notch 1 TFA encodes a member of the NOTCH family of proteins.Formule :C64H98N15F3O25S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1614.81AChE/BChE-IN-15
AChE/BChE-IN-15 (Compound 6d) serves as an inhibitor for both acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), presenting inhibition constants (Formule :C29H30N6O3Couleur et forme :SolidMasse moléculaire :510.59BChE-IN-21
BChE-IN-21, a potent inhibitor of butyrylcholinesterase (BChE), exhibits an inhibition constant (IC50) of 0.14 ± 0.02 μM, indicating promise for research inCouleur et forme :Odour Solid(Rac)-5-Hydroxymethyl Tolterodine hydrochloride
CAS :(Rac)-5-Hydroxymethyl Tolterodine HCl, or (Rac)-Desfesoterodine HCl, is a potent mAChR blocker researched for overactive bladder.
Formule :C22H32ClNO2Couleur et forme :SolidMasse moléculaire :377.95AChE-IN-29
AChE-IN-29, a 3-OH pyrrolidine derivative, acts as a cholinesterase (ChE) inhibitor with potent activity against human acetylcholinesterase (hAChE), electricFormule :C18H19BrN2O2Couleur et forme :SolidMasse moléculaire :375.26LY-426965 hydrochloride
CAS :LY-426965 hydrochloride is a bioactive chemical.Formule :C28H39ClN2O2Couleur et forme :SolidMasse moléculaire :471.07Sodium Channel Targeted Library
A unique collection of xnum sodium channel blockers and agonists for high throughput and high content screening;Couleur et forme :Odour SolidRef: TM-L7400
1mgÀ demander30μL*10mM (DMSO)À demander50μL*10mM (DMSO)À demander100μL*10mM (DMSO)À demander250μL*10mM (DMSO)À demander5-HT1AR/5-HT6R ligand-1
5-HT1AR/5-HT6R ligand-1 (Compound PP13) functions as a ligand for the 5-HT receptor, demonstrating high affinity for 5-HT1AR, 5-HT6R, and 5-HT7R with Ki values of 19, 69, and 198 nM, respectively. In HEK293 cells, it inhibits cAMP production with EC50 values of 1535, 488, and 53 nM for these receptors. Additionally, 5-HT1AR/5-HT6R ligand-1 exhibits antiproliferative effects on several cancer cell lines, including 1321N1, U87MG, MCF7, and AsPC-1, with IC50 values of 9.6, 13.6, 19.3, and 14.6 μM, respectively. The compound also shows antagonistic activity towards the dopamine receptor D2R, with a Ki of 1903 nM.Formule :C25H29ClN4O2SCouleur et forme :SolidMasse moléculaire :485.04CUR-IPA
CUR-IPA is a cholinesterase inhibitor with IC50 values of 5.99 μM for eAChE (electric eel), 59.30 μM for hAChE (human), and 60.66 μM for hBChE (human). It has free radical scavenging and antioxidant activity and is useful for researching cognitive dysfunction.Formule :C43H38N2O8Couleur et forme :SolidMasse moléculaire :710.77LY3020371
CAS :LY3020371: potent, selective mGlu 2/3 receptor antagonist with Ki of 5.26 nM (hmGluR2) and 2.50 nM (hmGluR3); key in depression studies.Formule :C15H15F2NO5SCouleur et forme :SolidMasse moléculaire :359.34Anticonvulsant agent 9
Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.Formule :C22H24N4O2Couleur et forme :SolidMasse moléculaire :376.45(-)-Eseroline fumarate
CAS :(-)-Eseroline fumarate, a Physostigmine metabolite and AChE inhibitor, triggers cancer cell LDH release and neuronal cell death.Formule :C17H22N2O5Couleur et forme :SolidMasse moléculaire :334.376,9-Dichloro-1,2,3,4-tetrahydroacridine
CAS :6,9-Dichloro-1,2,3,4-tetrahydroacridine is a synthetic intermediate in the synthesis of tacrine-based acetylcholinesterase (AChE) inhibitors.1It is also anFormule :C13H11Cl2NCouleur et forme :SolidMasse moléculaire :252.139
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