Neuroscience
Les inhibiteurs en neurosciences sont des composés conçus pour moduler l'activité de protéines, d'enzymes ou de récepteurs spécifiques au sein du système nerveux. Ces inhibiteurs sont cruciaux pour étudier les mécanismes moléculaires sous-jacents au fonctionnement neuronal, à la transmission synaptique et aux maladies neurodégénératives. En ciblant les récepteurs des neurotransmetteurs, les canaux ioniques et les voies de signalisation, les inhibiteurs en neurosciences facilitent l'exploration du fonctionnement cérébral et le développement de stratégies thérapeutiques pour des troubles neurologiques tels que la maladie d'Alzheimer, de Parkinson et l'épilepsie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs en neurosciences de haute qualité pour soutenir vos recherches en neurobiologie, neuropharmacologie et sciences cognitives.
Sous-catégories appartenant à la catégorie "Neuroscience"
- récepteur 5-HT(1.025 produits)
- ACK(1 produits)
- AChR(648 produits)
- ATP Citrate Lyase(17 produits)
- Récepteur adrénergique(3.028 produits)
- BACE(37 produits)
- Bêta-amyloïde(231 produits)
- CaMK(73 produits)
- COX(602 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur GABA(372 produits)
- Gamma-sécrétase(63 produits)
- GluR(265 produits)
- GlyT(26 produits)
- Récepteur de l'histamine(385 produits)
- LRRK2(42 produits)
- Récepteur de la mélatonine(26 produits)
- NMDAR(10 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(327 produits)
Affichez 12 plus de sous-catégories
5637 produits trouvés pour "Neuroscience"
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Lafadofensine
CAS :Lafadofensine, a monoamine reuptake inhibitor, exhibits significant effects upon short-term administration.Formule :C16H16F2N2Couleur et forme :SolidMasse moléculaire :274.315SLAFVDVLN
SLAFVDVLN is a peptide molecule that functions as a BACE-1 inhibitor, exhibiting a Ki value of 94 nM. Additionally, SLAFVDVLN is capable of reducing the production of Aβ42.Formule :C45H72N10O14Couleur et forme :SolidMasse moléculaire :977.11SPL-707
CAS :SPL-707 is an effective and selective signal peptide peptidase-like 2a inhibitor (IC50: 80 nM).Formule :C27H28FN5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :505.54Monoamine oxidase
CAS :Enzyme that breaks down amines in the brain and body, affecting mood and brain function.Couleur et forme :SolidFurosemide sodium
CAS :Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.Formule :C12H10ClN2NaO5SDegré de pureté :99.52% - >99.99%Couleur et forme :SolidMasse moléculaire :352.73Substance P(1-4) Acetate
Substance P(1-4) Acetate is a neurokinin receptor (NK-R) antagonist, inhibiting the formation of PV EEC.Formule :C24H44N8O7Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :556.66Bencycloquidium Bromide
CAS :Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.Formule :C21H32BrNO2Couleur et forme :SolidMasse moléculaire :410.395-HT1AR agonist 2
5-HT1AR Agonist 2 (Compound 4f) is a potent agonist of the 5-HT1A receptor with a Ki value of 10.0 nM. It also binds to SERT, D2, and 5-HT6 receptors with Ki values of 2.8 nM, 23 nM, and 192 nM, respectively. Furthermore, this compound demonstrates stability in microsomes and induces hypothermia in mice.Formule :C31H31N5O3Couleur et forme :SolidMasse moléculaire :521.61AChE/BuChE-IN-6
AChE/BuChE-IN-6 (Compound 11f) is an inhibitor of AChE and BuChE, with IC50 values of 1.24 and 1.85 μg/mL, respectively. It exhibits strong DPPH radical scavenging activity (IC50 = 3.15 μg/mL). In vivo toxicity studies demonstrate that AChE/BuChE-IN-6 is safe, showing no significant differences in blood and biochemical parameters compared to controls, and no abnormalities in liver and kidney tissues. This compound shows potential for Alzheimer's disease research.Formule :C24H20ClN3O3Couleur et forme :SolidMasse moléculaire :433.887(S)-Vamicamide
CAS :(S)-Vamicamide is an anti-anticholinergic compound.Formule :C18H23N3ODegré de pureté :99.48% - 99.65%Couleur et forme :SoildMasse moléculaire :297.39I2-IRs ligand-1
I2-IRs ligand-1 (Compound 12d) is an orally active compound capable of crossing the blood-brain barrier. It exhibits high affinity for imidazoline I2 receptors (I2-IRs) with a pKi of 9.98. This compound can enhance cognitive deficits in aging mice and possesses analgesic, anti-inflammatory, and neuroprotective properties. I2-IRs ligand-1 is applicable for research in Alzheimer's disease and related pain disorders.Formule :C21H23ClFN2O4PCouleur et forme :SolidMasse moléculaire :452.84Inaperisone
CAS :Inaperisone: a novel muscle relaxant that indirectly inhibits voiding reflex via brainstem GABAB receptors.Formule :C16H23NODegré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :245.36hAChE/hBuChE-IN-1
hAChE/hBuChE-IN-1 (compound C2) acts as a dual inhibitor of cholinesterases, exhibiting IC50 values of 514 nM for hAChE and 358 nM for hBuChE. It is orally active and capable of enhancing cognitive function and spatial memory.Formule :C30H31FN2O3Couleur et forme :SolidMasse moléculaire :486.577β-Amyloid (29-40)
CAS :β-Amyloid (29-40) is a fragment of Amyloid-β peptide.Alzheimer's beta amyloid peptide (29-40/42) C-terminal fragments have physical and chemical propertiesFormule :C49H88N12O13SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1085.36Paynantheine
CAS :Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.Formule :C23H28N2O4Couleur et forme :SolidMasse moléculaire :396.485-HT5AR/5-HT6R ligand-1
5-HT5AR/5-HT6R ligand-1 (Compound PP10) is a ligand for serotonin receptors, exhibiting high affinity for the 5-HT5A and 5-HT6 receptors with Ki values of 59 nM and 96 nM, respectively. It possesses some antiproliferative activity against tumor cells and can be utilized in cancer research.Formule :C25H30N4O2SCouleur et forme :SolidMasse moléculaire :450.6Lu AE51090
CAS :Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.Formule :C24H29N3O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :407.51α-Conotoxin EI
CAS :Selective antagonist of neuromuscular nicotinic receptors α1β1γδFormule :C83H125N27O27S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2093.37Iloperidone metabolite P95
CAS :Iloperidone metabolite P95, a non-brain penetrating compound, binds 5-HT2A, α1-, α2B-, α2C-receptors with Ki of 7.08-83.18 nM.Formule :C23H25FN2O5Couleur et forme :SolidMasse moléculaire :428.46Asenapine citrate
CAS :Asenapine citrate: atypical antipsychotic for schizophrenia, bipolar disorder; targets serotonin, adrenoceptors, dopamine, histamine (pKi: 8.2-10.5).Formule :C23H24ClNO8Couleur et forme :SolidMasse moléculaire :477.89(R)-(+)-Anatabine
CAS :(R)-(+)-Anatabine is an less active R-enantiomer of Anatabine. Anatabine is a potent agonist of α4β2 nAChR.Formule :C10H12N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :160.22Rovalpituzumab MMAE
Rovalpituzumab-MMAE (Anti-DLL3 Reference Antibody), produced in CHO cells, consists of a huIgG1 heavy chain and a hukappa light chain. The molecular weight of this antibody is predicted to be 145.02 kDa.Couleur et forme :LiquidMasse moléculaire :145 kDaPseudocoptisine acetate
CAS :Pseudocoptisine acetate is a quaternary alkaloid isolated from the tubers of Corydalis turtschaninovii,with anti-inflammatory properties.Formule :C21H17NO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :379.36Fasciculic acid A
CAS :Fasciculic acid A is a calmodulin antagonist isolated from mushroom Naematoloma fasciculare.Formule :C36H60O8Couleur et forme :SolidMasse moléculaire :620.868AChE-IN-37
AChE-IN-37 (compound A2) is an acetylcholinesterase inhibitor with an inhibitory concentration (IC50) of 0.23 µM.Formule :C21H12ClNO7SCouleur et forme :SolidMasse moléculaire :457.84[Ala11,D-Leu15]-Orexin B(human)
CAS :OX2 receptor agonist with 400x selectivity vs OX1. EC50: 0.13 nM (OX2), 52 nM (OX1).Formule :C120H206N44O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2857.285-HT6R antagonist 6
5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.Formule :C24H26N4O2SCouleur et forme :SolidMasse moléculaire :434.55Fasciculic acid B
CAS :Fasciculic acid B: ester of fasciculol B, 3-hydroxy-methylglutaric acid; a calmodulin antagonist from Naematoloma fasciculare.Formule :C36H60O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :636.86Br-PBTC
CAS :Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.Formule :C14H15BrN2OSCouleur et forme :SolidMasse moléculaire :339.25Orexin B, human
CAS :Orexin B, human agonizes Orexin receptors (OX1 Ki=420 nM, OX2 Ki=36 nM), promotes feeding in rats, and is a neuropeptide.Formule :C123H212N44O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2899.34CAY10787
CAS :CAY10787, an oxysterol, inhibits GABAA receptors (IC50s: 1-1.5μM) and lessens GABA responses in mouse DRG neurons.Formule :C27H42OCouleur et forme :SolidMasse moléculaire :382.632Orexin A (human, rat, mouse)
CAS :Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.Formule :C152H243N47O44S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3561.1PD24
PD24 serves as an inhibitor of both acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE), with inhibitory concentrations (IC50) of 1.72 μM for humanFormule :C24H22N2O6Couleur et forme :SolidMasse moléculaire :434.44GABAA receptor modulator-4
GABAA receptor modulator-4 (Compound 4) acts as a negative allosteric modulator of the GABAA receptor. It inhibits the peak and steady-state currents mediated by the α1β3γ2 GABAA receptors, with an IC50 of 10 μM for both.Formule :C15H17BrO4SCouleur et forme :SolidMasse moléculaire :373.26Naratriptan D3 Hydrochloride
CAS :Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.Formule :C17H26ClN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.94LY86057
CAS :LY86057 is a bioactive chemical.Formule :C20H26N2O3Couleur et forme :SolidMasse moléculaire :342.439(Rac)-Sabcomeline
CAS :(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.Formule :C10H15N3ODegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :193.25Ref: TM-T68135L1
1mg109,00€2mg160,00€5mg261,00€10mg374,00€25mg583,00€50mg803,00€100mg1.063,00€200mg1.431,00€TRV-7019
CAS :TRV-7019: BBB-permeable radioligand for brain imaging, used in diagnosing amyloid diseases, MS, and brain tumors.Formule :C14H12INO3Couleur et forme :SolidMasse moléculaire :369.15[Ala11,D-Leu15]-Orexin B acetate
[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).Formule :C122H210N44O37SDegré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :2917.31SB 216641
CAS :SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety disorders and depression.Formule :C28H30N4O4Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :486.56Trivalent GalNAc-DBCO
CAS :Trivalent GalNAc-DBCO is a synthetic ligand composed of three GalNAc units linked to DBCO. Trivalent GalNAc-DBCO undergoes strain-promoted alkyne–azide cycloaddition (SPAAC) reactions with azide-containing molecules without the need for copper catalysis. Trivalent GalNAc-DBCO binds specifically to the asialoglycoprotein receptor (ASGPR), thereby directing conjugated molecules into hepatocytes for lysosomal degradation through receptor-mediated endocytosis. Trivalent GalNAc-DBCO is extensively applied in studies of liver-targeted drug delivery, targeted degradation strategies, and hepatocyte-specific molecular engineering.Formule :C91H144N12O34Degré de pureté :96.33%Masse moléculaire :1950.18VU6028418
CAS :VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).Formule :C23H27F3N4OCouleur et forme :SolidMasse moléculaire :432.491JF-NP-26
Releases pain-blocking raseglurant under 405 nm light. Inhibits Quisqualate. Analgesic in vivo. Quantum yield: 0.18.Couleur et forme :SolidLY 293284
CAS :LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.Formule :C19H26N2OCouleur et forme :SolidMasse moléculaire :298.42β-Amyloid (1-15)
CAS :β-Amyloid (1-15) (Amyloid β-Protein (1-15)) is a fragment of β-amyloid protein used in the study of Alzheimer's disease.Formule :C78H107N25O27Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :1826.84LU-32-176B
CAS :LU32-176B is a bioactive chemical.Formule :C23H24F2N2O2Couleur et forme :SolidMasse moléculaire :398.45Feralolide
CAS :Feralolide, a dihydroisocoumarin from the methanolic extract of aloe vera resin, functions as a dual inhibitor of acetylcholinesterase (AChE) andFormule :C18H16O7Couleur et forme :SolidMasse moléculaire :344.32Zicronapine fumarate
CAS :Zicronapine fumarate, an antipsychotic, targets D1/D2 & 5-HT2A receptors; may treat neuropsychiatric conditions.Formule :C26H31ClN2O4Couleur et forme :SolidMasse moléculaire :470.99AChE-IN-36
AChE-IN-36 (compound A4) is an acetylcholinesterase inhibitor with an IC50 of 0.04 μM, influencing ROS levels and modulating the gene expression of NRF2 [1].Formule :C25H21ClO5SCouleur et forme :SolidMasse moléculaire :468.95Tabernanthalog
CAS :TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.Formule :C14H18N2ODegré de pureté :99.82% - 99.89%Couleur et forme :SoildMasse moléculaire :230.31Ref: TM-T60221
1mg175,00€2mg264,00€1mL*10mM (DMSO)344,00€5mg404,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€Orexin A (human, rat, mouse) acetate
Orexin A (human, rat, mouse) acetate (Hypocretin-1 (human, rat, mouse) acetate) is an excitatory neuropeptide with analgesic properties.Formule :C154H247N47O46S4Couleur et forme :SolidMasse moléculaire :3621.153-Aminopropylphosphinic acid
CAS :3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).
Formule :C3H10NO2PCouleur et forme :SolidMasse moléculaire :123.092C2-8
CAS :C2-8 inhibits polyQ aggregation, IC50=25 μM (HDQ51), 0.05 μM (PC12 cells), reduces neurodegeneration in Huntington's models.Formule :C19H14Br2N2O3SCouleur et forme :SolidMasse moléculaire :510.2Cyclodrine
CAS :Cyclodrine (Cyclopent) is a cholinergic (muscarinic, nicotinic) (mAChR and nAChR) receptor antagonist.Formule :C19H29NO3Degré de pureté :97.62%Couleur et forme :SoildMasse moléculaire :319.44Ref: TM-T10914L
1mg73,00€1mL*10mM (DMSO)148,00€5mg149,00€10mg212,00€25mg319,00€50mg447,00€100mg610,00€200mg822,00€TIM-098a
TIM-098a is a selective AAK1 inhibitor with an IC50 of 0.24 µM. It does not inhibit CaMKK isoforms. By inhibiting AAK1 kinase activity, TIM-098a disrupts AAK1-regulated endocytosis.
Formule :C18H11N3O2Masse moléculaire :301.08513Amyloid β Peptide (42-1)(human) acetate
Amyloid β Peptide (42-1)(human) acetate is the inactive form of Amyloid β Peptide (1-42).Degré de pureté :95.20%Couleur et forme :SoildBlestrin D
CAS :Blestrin D: BChE mixed-type inhibitor, IC50=8.1μM, from Bletilla striata, for AD research.Formule :C30H24O6Couleur et forme :SolidMasse moléculaire :480.51XL01126
XL01126 degrades LRRK2 (DC50: 14 nM G2019S, 32 nM WT), crosses the blood-brain barrier, aiding Parkinson's studies.Formule :C50H64ClFN10O6S2Couleur et forme :SolidMasse moléculaire :1019.69Nardoguaianone J
CAS :Nardoguaianone J, a guaiane-type compound isolated from the roots of Nardostachys chinensis, has been shown to enhance SERT activity [1][2].Formule :C15H22O2Couleur et forme :SolidMasse moléculaire :234.33SCH-900229
CAS :SCH-900229, a potent presenilin 1 selective γ-secretase inhibitor, used to treat Alzheimer’s Disease.Formule :C21H21ClF2O6S2Couleur et forme :SolidMasse moléculaire :506.97SB656104
CAS :SB656104 is a bioactive chemical.Formule :C25H30ClN3O3SCouleur et forme :SolidMasse moléculaire :488.04α-Conotoxin PIA
CAS :Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nMFormule :C79H125N27O25S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1981.3AChE-IN-49
AChE-IN-49 (Compd (S)-7g) is an acetylcholinesterase (AChE) inhibitor with an IC50 value of 0.0003 μM.Formule :C31H28BrClN2O3Masse moléculaire :590.09718epi-Aszonalenin A
CAS :epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.Formule :C25H25N3O3Couleur et forme :SolidMasse moléculaire :415.48Methyllycaconitine citrate
CAS :Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.Formule :C43H58N2O17Degré de pureté :98.03% - 98.91%Couleur et forme :SolidMasse moléculaire :874.92FRM-024
CAS :FRM-024 is a powerful gamma secretase modulator with the ability to penetrate the central nervous system (CNS), designed specifically for the treatment ofFormule :C22H22ClN5O2Couleur et forme :SolidMasse moléculaire :423.9SSAO inhibitor-1
CAS :SSAO Inhibitor-1 blocks SSAO, has anti-inflammatory effects, used in liver disease research.Formule :C17H24FN5O2Couleur et forme :SolidMasse moléculaire :349.41AChE-IN-60
AChE-IN-60 (compound 6k) is a potent inhibitor of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE), with IC50 values of 27 nM and 43 nM, respectively. It also inhibits monoamine oxidase MAO-A and MAO-B, with IC50 values of 353 nM and 716 nM, respectively.Formule :C24H29N3O4S3Masse moléculaire :519.13202p-HTAA
CAS :Pentamer Hydrogen Thiophene Acetic Acid (p-HTAA) is a compound that specifically targets and labels amyloid-beta (Aβ) deposits in the brains of living mice [1].Formule :C24H16O4S5Couleur et forme :SolidMasse moléculaire :528.71Sintamil
CAS :Sintamil is a useful organic compound for research related to life sciences. The catalog number is T71697 and the CAS number is 16398-39-3.Formule :C18H20ClN3O4Couleur et forme :SolidMasse moléculaire :377.82N-desmethyl Zolmitriptan
CAS :DZT, an active metabolite of zolmitriptan, agonizes 5-HT1B/D receptors; contracts human cerebral arteries (EC50=100nM).Formule :C15H19N3O2Couleur et forme :SolidMasse moléculaire :273.332-Methyl-1-indanone
CAS :2-Methyl-1-indanone is an acetylcholinesterase inhibitor and can be used for biochemical experiments and drug synthesis.Formule :C10H10ODegré de pureté :96.6%Couleur et forme :SolidMasse moléculaire :146.19M 8218
CAS :M 8218 is a bioactive chemical.Formule :C20H29NO2Couleur et forme :SolidMasse moléculaire :315.45β-Amyloid (11-22)
CAS :β-Amyloid (11-22) is a peptide fragment of β-Amyloid.Beta-amyloid peptide (Abeta), the major constituent of amyloid plaques in the brains of Alzheimer’sFormule :C70H102N18O18Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1483.67CPN-351
CAS :CPN-351 (compound 9a) is a pentapeptide that acts as a selective antagonist for human NMUR1, with a pA2 value of 7.35. It exhibits ten times greater antagonistic activity toward human NMUR1 compared to NMUR2. CPN-351 is applicable in inflammation research.Formule :C45H61N13O6SMasse moléculaire :912.11BuChE-IN-21
BuChE-IN-21 (compound SXF3) is a potent and selective inhibitor of BuChE, demonstrating inhibitory effects on eqBuChE and hBuChE with IC50 values of 0.05 and 0.04 μM, respectively. Additionally, BuChE-IN-21 exhibits significant anti-inflammatory activity.Formule :C16H23NO2Couleur et forme :SolidMasse moléculaire :261.17288Imidafenacin Metabolite M4
CAS :Imidafenacin M4 is a CYP3A4-formed metabolite of the muscarinic antagonist imidafenacin.Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.368MGS0028
CAS :MGS0028 is a selective agonist of metabotropic glutamate 2/3 receptor, it could reverse abnormal behaviors in mice induced by isolation rearing.Formule :C8H8FNO5Couleur et forme :SolidMasse moléculaire :217.15Vortioxetine D8
CAS :Vortioxetine D8 is a deuterium-labeled antidepressant inhibiting 5-HT1A/B, 5-HT3A, 5-HT7 receptors & SERT (Ki: 15-1.6 nM).Formule :C18H22N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.5Brexpiprazole S-oxide D8
CAS :Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled metabolite of Brexpiprazole, a partial agonist at 5-HT1A and dopamine receptors.Formule :C25H19D8N3O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :457.61β-Amyloid (35-42)
CAS :β-Amyloid (35-42) is a peptide derived from the beta-amyloid protein, encompassing amino acids 35 through 42.Formule :C33H60N8O9SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :744.948-Aminoadenine
CAS :8-Aminoadenine (7H-purine-6,8-diamine) is a ligand for Adenine Receptor with Ki of 0.0341 μM.Formule :C5H6N6Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :150.14Duloxetine D3 hydrochloride
CAS :Duloxetine D3 HCl is a deuterium-labeled SNRI, treats depression/GAD, Ki 4.6 nM.Formule :C18H20ClNOSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :336.89β-Amyloid (35-25)
CAS :β-Amyloid (35-25) is the reverse sequence of β-Amyloid (25-35).Formule :C45H81N13O14SMasse moléculaire :1060.27Vanutide cridificar
CAS :Vanutide cridificar (ACC-001) is an aminoterminal Aβ1-7 peptide conjugate, employed in Alzheimer’s disease (AD) research [1].Couleur et forme :LiquidFITC-β-Ala-Amyloid β-Protein (1-42)
CAS :FITC-β-Ala-Amyloid β-Protein (1-42) is a polypeptide identified through peptide screening. This screening method predominantly utilizes immunoassays to gather active polypeptides and is used in studying protein interactions, conducting functional analyses, and screening antigen epitopes, with particular application in the research and development of active molecules.Formule :C227H327N57O66S2Masse moléculaire :4971.34251Lupanine hydrochloride
CAS :Lupanine hydrochloride, a Sparteine derivative, binds to nAChR with a Ki of 500 nM and has ganglioplegic properties.Formule :C15H25ClN2OCouleur et forme :SolidMasse moléculaire :284.83α-Conotoxin imi
CAS :alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.Formule :C52H78N20O15S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1351.56UCM 549
CAS :UCM 549 is a bioactive chemical.Formule :C19H21NO2Couleur et forme :SolidMasse moléculaire :295.38Lesogaberan napadisylate
CAS :Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Formule :C13H17FNO5PSCouleur et forme :SolidMasse moléculaire :349.315H-Pyrido[4,3-b]indole
CAS :5H-Pyrido[4,3-b]indole is a potential AchE/ChE inhibitor with potential antiviral activity for the study of neurodegenerative diseases.Formule :C11H8N2Degré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :168.2Fluphenazine-N-2-chloroethane (hydrochloride)
CAS :Fluphenazine: antipsychotic, binds dopamine D2 (Ki=0.55nM), inhibits calmodulin. Its derivative adds irreversible D2 antagonism and anticancer potential.Formule :C22H27Cl3F3N3SCouleur et forme :SolidMasse moléculaire :528.89Minaprine
CAS :Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.Formule :C17H22N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.38MR33317
MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.Formule :C22H28ClN3O2Masse moléculaire :401.187Atagabalin
CAS :Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.Formule :C10H19NO2Couleur et forme :SolidMasse moléculaire :185.26Eletriptan
CAS :Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.Formule :C22H26N2O2SCouleur et forme :SolidMasse moléculaire :382.52Sulamserod
CAS :Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular relatedFormule :C19H28ClN3O5SDegré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :445.96RA306
RA306 is an orally active CAMK2 inhibitor that effectively disrupts the PEAK1/CAMK2 signaling pathway. It demonstrates anti-tumor activity by inhibiting proliferation, migration, and invasion of breast cancer cells. Additionally, RA306 shows potential in cardiac disease research, as it improves dilated cardiomyopathy in mice.Couleur et forme :Odour SolidOXA(17-33)
CAS :Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.Formule :C79H125N23O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :17495-HT2A receptor agonist-5
CAS :5-HT2A receptor agonist-5 (compound I-3) is a potent 5-HT2A agonist with a Ki value of 0.017 µM and exhibits antidepressant activity.Formule :C23H29N3OCouleur et forme :SolidMasse moléculaire :363.5
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