Neuroscience
Les inhibiteurs en neurosciences sont des composés conçus pour moduler l'activité de protéines, d'enzymes ou de récepteurs spécifiques au sein du système nerveux. Ces inhibiteurs sont cruciaux pour étudier les mécanismes moléculaires sous-jacents au fonctionnement neuronal, à la transmission synaptique et aux maladies neurodégénératives. En ciblant les récepteurs des neurotransmetteurs, les canaux ioniques et les voies de signalisation, les inhibiteurs en neurosciences facilitent l'exploration du fonctionnement cérébral et le développement de stratégies thérapeutiques pour des troubles neurologiques tels que la maladie d'Alzheimer, de Parkinson et l'épilepsie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs en neurosciences de haute qualité pour soutenir vos recherches en neurobiologie, neuropharmacologie et sciences cognitives.
Sous-catégories appartenant à la catégorie "Neuroscience"
- récepteur 5-HT(1.025 produits)
- ACK(1 produits)
- AChR(648 produits)
- ATP Citrate Lyase(17 produits)
- Récepteur adrénergique(3.028 produits)
- BACE(37 produits)
- Bêta-amyloïde(231 produits)
- CaMK(73 produits)
- COX(602 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur GABA(372 produits)
- Gamma-sécrétase(63 produits)
- GluR(265 produits)
- GlyT(26 produits)
- Récepteur de l'histamine(385 produits)
- LRRK2(42 produits)
- Récepteur de la mélatonine(26 produits)
- NMDAR(10 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(327 produits)
Affichez 12 plus de sous-catégories
5637 produits trouvés pour "Neuroscience"
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VU10010
CAS :VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.
Formule :C17H16ClN3OSDegré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :345.85Anpirtoline free base
CAS :Anpirtoline: potent 5-HT1B agonist; lowers serotonin synthesis; reduces aggression; 5-HT3 antagonist; crosses blood-brain barrier.Formule :C10H13ClN2SCouleur et forme :SolidMasse moléculaire :228.74Pempidine
CAS :Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Formule :C10H21NDegré de pureté :98.18% - 99.28%Couleur et forme :Colorless - Light Yellow Clear LiquidMasse moléculaire :155.28Oxotremorine sesquifumarate
CAS :Oxotremorine sesquifumarate is a muscarinic agonist.
Formule :C12H18N2OC4H4O4Degré de pureté :97.94%Couleur et forme :SolidMasse moléculaire :380.39SKF89976A HCl
CAS :SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formule :C22H25NO2Couleur et forme :SolidMasse moléculaire :335.44Hemicholinium 3
CAS :Hemicholinium 3 is a potent and selective choline uptake blocker.Formule :C24H34Br2N2O4Degré de pureté :98% - 99.95%Couleur et forme :SolidMasse moléculaire :574.35Escitalopram Oxalate
CAS :Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formule :C22H23FN2O5Degré de pureté :97.39% - 99.73%Couleur et forme :White SolidMasse moléculaire :414.43Ref: TM-T6493
10mg37,00€1mL*10mM (DMSO)42,00€25mg52,00€50mg63,00€100mg86,00€200mg118,00€500mg187,00€1g268,00€Dinotefuran
CAS :Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formule :C7H14N4O3Degré de pureté :99.89%Couleur et forme :White Crystalline PowderMasse moléculaire :202.21Sofpironium bromide
CAS :Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Formule :C22H32BrNO5Degré de pureté :98.85%Couleur et forme :SolidMasse moléculaire :470.4Ref: TM-T28827
1mg74,00€5mg160,00€1mL*10mM (DMSO)165,00€10mg250,00€25mg452,00€50mg680,00€100mg1.008,00€200mg1.349,00€Revefenacin
CAS :Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formule :C35H43N5O4Degré de pureté :98.12%Couleur et forme :SolidMasse moléculaire :597.75SKF89976A hydrochloride
CAS :SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormule :C22H26ClNO2Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :371.9Ref: TM-T12930
1mg34,00€5mg65,00€1mL*10mM (DMSO)71,00€10mg89,00€25mg167,00€50mg264,00€100mg409,00€200mg590,00€Miltirone
CAS :Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formule :C19H22O2Degré de pureté :99.22% - 99.66%Couleur et forme :SolidMasse moléculaire :282.38PNU-282987 S enantiomer free base
CAS :PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).Formule :C14H17ClN2ODegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :264.75Ref: TM-T7695
1mg71,00€5mg161,00€1mL*10mM (DMSO)180,00€10mg219,00€25mg338,00€50mg460,00€100mg623,00€200mg837,00€Org 25543 hydrochloride
CAS :Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 = 16 nM for hGlyT2).Formule :C24H33ClN2O4Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :448.983Autocamtide 2 TFA(129198-88-5 free base)
Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.Formule :C67H119F3N22O22Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1641.79Prucalopride Succinate
CAS :Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formule :C18H26ClN3O3·C4H6O4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :485.96CCMI
CAS :CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.Formule :C19H15Cl2N3O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :388.25L-838417 D9
CAS :L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].Formule :C19H10D9F2N7ODegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :408.45Ref: TM-T22301
2mg34,00€5mg52,00€1mL*10mM (DMSO)58,00€10mg71,00€25mg128,00€50mg200,00€100mg323,00€200mg447,00€Amitriptyline
CAS :Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.Formule :C20H23NDegré de pureté :98.24% - 99.64%Couleur et forme :Crystals SolidMasse moléculaire :277.4Phenibut (hydrochloride)
CAS :Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formule :C10H14ClNO2Degré de pureté :99.93%Couleur et forme :White Crystalline PowderMasse moléculaire :215.68Jagged-1 (188-204) TFA(219127-21-6 free base)
Jagged-1 (188-204) TFA, a JAG-1 skin protein fragment, induces epidermal maturation and keratinocyte stratification.Formule :C95H128F3N25O28S3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :2221.37W-84 dibromide
CAS :W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Formule :C32H44Br2N4O4Degré de pureté :95.56%Couleur et forme :SolidMasse moléculaire :708.52Opiranserin hydrochloride
CAS :Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormule :C21H35ClN2O5Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T9833
1mg90,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€AC-90179 HCl
CAS :AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formule :C23H31ClN2O2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :402.96CFMTI
CAS :CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.Formule :C19H16FN5ODegré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :349.36Ref: TM-T3482
1mg57,00€2mg82,00€5mg120,00€1mL*10mM (DMSO)133,00€10mg170,00€25mg304,00€50mg432,00€100mg602,00€Avagacestat
CAS :Avagacestat (BMS-708163) (BMS-708163) is a potent, selective, orally bioavailable γ-secretase inhibitor of Aβ40 and Aβ42 with IC50 of 0.3 nM and 0.27 nM,Formule :C20H17ClF4N4O4SDegré de pureté :98.87% - 99.73%Couleur et forme :SolidMasse moléculaire :520.89Ref: TM-T6249
1mg38,00€5mg77,00€1mL*10mM (DMSO)88,00€10mg116,00€25mg215,00€50mg310,00€100mg450,00€200mg605,00€4-Acetamidobutanoic acid
CAS :4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formule :C6H11NO3Degré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :145.16VUF 10166
CAS :VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Formule :C13H15ClN4Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :262.74Lurasidone
CAS :Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formule :C28H36N4O2SDegré de pureté :99.78% - 99.91%Couleur et forme :SolidMasse moléculaire :492.683,5-Bis(4-nitrophenoxy)benzoic acid
CAS :3,5-Bis(4-nitrophenoxy)benzoic acid (Compound W) is an inhibitor of γ-secretase. It decreases the released levels of Aβ42 and notch-1 Aβ-like peptide 25.Formule :C19H12N2O8Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :396.31Amyloid β-Protein 10-20 acetate
Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) is a fragment of Amyloid-β peptide, maybe used in the research ofFormule :C73H103N17O18Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :1506.65YO-01027
CAS :YO-01027 (DBZ) is a potent γ-secretase inhibitor.Formule :C26H23F2N3O3Degré de pureté :97.21% - 99.58%Couleur et forme :SolidMasse moléculaire :463.48Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formule :C35H47FN10O8Degré de pureté :97.97%Couleur et forme :SolidMasse moléculaire :754.85Neurotensin TFA
Neurotensin TFA (39379-15-2) is a 13-amino acid neuropeptide with opioid-independent pain relief, acting in the CNS and gut, linked to numerous disorders.Formule :C80H122F3N21O22Degré de pureté :99.41%Couleur et forme :SolidMasse moléculaire :1786.98Dasotraline hydrochloride
CAS :Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formule :C16H16Cl3NDegré de pureté :98.92% - 99.6%Couleur et forme :SolidMasse moléculaire :328.66N-Desmethylclozapine
CAS :N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.8Ref: TM-T5158
2mg34,00€5mg48,00€1mL*10mM (DMSO)58,00€10mg79,00€25mg152,00€50mg235,00€100mg344,00€200mg490,00€TBPB
CAS :TBPB is an allosteric M1 mAChR agonist.
Formule :C25H32N4ODegré de pureté :97.87% - 99.9%Couleur et forme :SolidMasse moléculaire :404.55L-745870 trihydrochloride
CAS :L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.21FITM
CAS :FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).Formule :C18H18FN5OSDegré de pureté :97.25% - 99.23%Couleur et forme :SolidMasse moléculaire :371.43Ref: TM-T7292
1mg34,00€2mg44,00€1mL*10mM (DMSO)62,00€5mg66,00€10mg92,00€25mg177,00€50mg268,00€100mg394,00€Chlorprothixene
CAS :Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formule :C18H18ClNSDegré de pureté :98.77% - 99.756%Couleur et forme :Pale Yellow Crystals SolidMasse moléculaire :315.86NGB 2904
CAS :NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Formule :C28H29Cl2N3ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :494.46Ref: TM-T28167
500mgÀ demander2mg38,00€5mg55,00€1mL*10mM (DMSO)72,00€10mg86,00€25mg155,00€50mg264,00€100mg374,00€Piperacetazine
CAS :Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formule :C128H219N45O36SDegré de pureté :94.61%Couleur et forme :SolidMasse moléculaire :2996.45OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formule :C79H125N23O22Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :1748.98Almotriptan
CAS :Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formule :C17H25N3O2SDegré de pureté :99.85%Couleur et forme :Light Yellow Or White PowerMasse moléculaire :335.46VU0467154
CAS :VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.Formule :C17H15F3N4O3S2Degré de pureté :99.51% - 99.53%Couleur et forme :SolidMasse moléculaire :444.45Ref: TM-T17244
1mg47,00€2mg63,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg126,00€25mg236,00€50mg400,00€100mg695,00€200mg945,00€S26131
CAS :S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki ofFormule :C31H34N2O4Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :498.61Bitopertin
CAS :Bitopertin (Paliflutine) (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki of 8.1 nM for human hGlyT1b and IC50 of 22-25 nMFormule :C21H20F7N3O4SDegré de pureté :98.57% - 98.71%Couleur et forme :SolidMasse moléculaire :543.46PU02
CAS :PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.Formule :C16H12N4SDegré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :292.36Rizatriptan benzoate
CAS :Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormule :C22H25N5O2Degré de pureté :99% - 99.79%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :391.47Ref: TM-T1512
10mg44,00€1mL*10mM (DMSO)48,00€25mg74,00€50mg119,00€100mg173,00€200mg259,00€500mg437,00€Trazodone
CAS :Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formule :C19H22ClN5ODegré de pureté :99.79% - 99.92%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :371.86Ramosetron hydrochloride
CAS :Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.Formule :C17H18ClN3ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :315.8Idalopirdine Hydrochloride
CAS :Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.Formule :C20H20ClF5N2ODegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :434.83p-Hydroxybenzaldehyde
CAS :1.Formule :C7H6O2Degré de pureté :99.05% - 99.86%Couleur et forme :SolidMasse moléculaire :122.12TG6-10-1
CAS :TG6-10-1 is an EP2 antagonist.Formule :C23H23F3N2O4Degré de pureté :99.66% - ≥95%Couleur et forme :SolidMasse moléculaire :448.43Tacrine hydrochloride (hydrate)
CAS :Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.Formule :C13H14N2·XHCl·XH2ODegré de pureté :99.01% - 99.89%Couleur et forme :SolidMasse moléculaire :234.72JLK6
CAS :JLK6 was a gamma-secretase inhibitor that does not interfere with Notch signallingFormule :C10H8ClNO3Degré de pureté :96.50%Couleur et forme :SolidMasse moléculaire :225.63Ref: TM-T21890
1mg84,00€5mg152,00€1mL*10mM (DMSO)160,00€10mg212,00€25mg354,00€50mg504,00€100mg685,00€200mg888,00€AMN082 free base
CAS :AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.Formule :C28H28N2Degré de pureté :97.75% - 97.79%Couleur et forme :SolidMasse moléculaire :392.54Ref: TM-T21935L
5mg50,00€1mL*10mM (DMSO)52,00€10mg74,00€25mg135,00€50mg212,00€100mg340,00€200mg475,00€MCI-225
CAS :MCI-225 is a selective inhibitor of NA reuptake with 5-HT3 receptor antagonism.Formule :C17H17FN4SDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :328.4NS3861
CAS :NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based receptors.Formule :C12H14BrNSDegré de pureté :99.853%Couleur et forme :SolidMasse moléculaire :284.224F 4PP oxalate
CAS :4F 4PP oxalate is a 5-HT2A antagonist.Formule :C22H26FNO·C2H2O4Degré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :429.49Tasimelteon
CAS :Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formule :C15H19NO2Degré de pureté :98.93% - 99.93%Couleur et forme :SolidMasse moléculaire :245.32ARN2966
CAS :ARN2966 is an inhibitor of amyloid precursor protein (APP)and amyloid-β (Aβ) secretion.Formule :C12H12N2ODegré de pureté :99.52% - 99.86%Couleur et forme :SolidMasse moléculaire :200.24Ref: TM-T7490
1mg34,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg113,00€25mg222,00€50mg358,00€100mg530,00€500mg1.153,00€AZD3839 free base
CAS :AZD3839 free base is a potent and selective BACE1 inhibitor with Ki of 26.1 nM, about 14-fold selectivity over BACE2. Phase 1.Formule :C24H16F3N5Degré de pureté :99.93% - 99.96%Couleur et forme :SolidMasse moléculaire :431.41Serotonin
CAS :Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Formule :C10H12N2ODegré de pureté :97.47% - 99.92%Couleur et forme :SolidMasse moléculaire :176.22(2-Chloropyridin-4-yl)MethanaMine Hydrochloride
CAS :(2-Chloropyridin-4-yl)methanamine hydrochloride is a selective LOXL2 inhibitor(IC50 : 126 nM).Formule :C6H8Cl2N2Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :179.05NS11394
CAS :NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(Formule :C23H19N3ODegré de pureté :99.44% - 99.86%Couleur et forme :SolidMasse moléculaire :353.42Ref: TM-T2067
2mg34,00€5mg50,00€1mL*10mM (DMSO)58,00€10mg80,00€25mg131,00€50mg212,00€100mg321,00€200mg460,00€PHA 568487 free base
CAS :PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.Formule :C16H20N2O3Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :288.34NAN-190 hydrobromide
CAS :NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formule :C23H28BrN3O3Degré de pureté :95.20%Couleur et forme :SolidMasse moléculaire :474.39ACH-000143
CAS :ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formule :C13H16ClN3O3Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :297.74Ref: TM-T9193
1mg50,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg172,00€25mg304,00€50mg424,00€100mg583,00€200mg785,00€3-AQC
CAS :3-AQC is a competitive antagonist of 5-HT3.Formule :C20H21N5O4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :395.41VU 0238429
CAS :VU 0238429 (SCR-1481B1) is positive allosteric modulator of muscarinic acetylcholine receptor subtype 5 (mAChR5 or M5)( EC50 : 1.16 μM).Formule :C17H12F3NO4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :351.28Ref: TM-T8007
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg81,00€25mg137,00€50mg215,00€100mg340,00€500mg795,00€Ipratropium Bromide
CAS :Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.Formule :C20H30BrNO3Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :412.37Mosapride
CAS :Mosapride (AS-4370) is a selective 5HT4 agonistFormule :C21H25ClFN3O3Degré de pureté :99.56%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :421.89Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg38,00€5mg80,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg222,00€50mg356,00€100mg512,00€200mg735,00€GNE-7915
CAS :GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.Formule :C19H21F4N5O3Degré de pureté :98% - ≥95%Couleur et forme :SolidMasse moléculaire :443.4Ref: TM-T1945
5mg44,00€1mL*10mM (DMSO)48,00€10mg58,00€25mg108,00€50mg177,00€100mg299,00€200mg389,00€500mg645,00€MK-0752
CAS :MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).Formule :C21H21ClF2O4SDegré de pureté :98% - 99.55%Couleur et forme :SolidMasse moléculaire :442.9Tianeptine sodium salt
CAS :Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formule :C21H24ClN2NaO4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :458.93JHU37160
CAS :JHU37160 is a DREADD agonist with Ki of 1.9 nM for hM3Dq, 3.6 nM for hM4Di, and EC50 of 18.5 nM (hM3Dq), 0.2 nM (hM4Di) in HEK-293 cell assays.Formule :C19H20ClFN4Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :358.84RO4929097
CAS :RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).Formule :C22H20F5N3O3Degré de pureté :98.5% - 99.51%Couleur et forme :SolidMasse moléculaire :469.4Vilazodone Hydrochloride
CAS :Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormule :C26H27N5O2·HClDegré de pureté :99.56% - >99.99%Couleur et forme :SolidMasse moléculaire :477.99Cerlapirdine
CAS :Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Formule :C22H23N3O3SDegré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :409.5Ref: TM-T30798
1mg81,00€5mg170,00€1mL*10mM (DMSO)198,00€10mg274,00€25mg543,00€50mg780,00€100mg1.074,00€Suritozole
CAS :Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptorFormule :C10H10FN3SDegré de pureté :99.25%Couleur et forme :SolidMasse moléculaire :223.27Ref: TM-T8568
1mg58,00€1mL*10mM (DMSO)104,00€5mg116,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€CZC-25146
CAS :CZC-25146, a stable LRRK2 inhibitor, IC50: 4.76 nM (wild-type), 6.87 nM (G2019S).Formule :C22H25FN6O4SDegré de pureté :97.68%Couleur et forme :SolidMasse moléculaire :488.54DORA-22
CAS :DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memoryFormule :C23H22F2N4O2Degré de pureté :97.67%Couleur et forme :SolidMasse moléculaire :424.44Ref: TM-T5500
1mg124,00€2mg178,00€5mg269,00€1mL*10mM (DMSO)314,00€10mg408,00€25mg672,00€50mg945,00€100mg1.279,00€lumateperone Tosylate
CAS :lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formule :C31H36FN3O4SDegré de pureté :95.83% - 99.95%Couleur et forme :SolidMasse moléculaire :565.7Chelidamic acid
CAS :Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.Formule :C7H5NO5Degré de pureté :98.11%Couleur et forme :Pale Yellow PowderMasse moléculaire :183.12Tinoridine hydrochloride
CAS :Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.Formule :C17H21ClN2O2SDegré de pureté :97.49%Couleur et forme :SolidMasse moléculaire :352.88Varenicline dihydrochloride
CAS :Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.Formule :C13H15Cl2N3Degré de pureté :99.88% - 99.97%Couleur et forme :SolidMasse moléculaire :284.18PBD-150
CAS :PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)Formule :C15H20N4O2SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :320.41Venlafaxine
CAS :Venlafaxine (Wy 45030), an arylalkanolamine serotonin-norepinephrine reuptake inhibitor (SNRI), is used to treat major generalised anxiety disorder (GAD),Formule :C17H27NO2Degré de pureté :99.2%Couleur et forme :White Solid CrystallineMasse moléculaire :277.4Imidafenacin
CAS :Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Formule :C20H21N3ODegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :319.4Dihydroergotoxine mesylate
CAS :Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formule :C20H29N3O5SDegré de pureté :99.39% - ≥95%Couleur et forme :SolidMasse moléculaire :423.53Indophagolin
CAS :Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formule :C19H15BrClF3N2O3SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :523.75Atracurium besylate
CAS :Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.Formule :C65H82N2O18S2Degré de pureté :98.94% - 99.71%Couleur et forme :SolidMasse moléculaire :1243.49Bicuculline
CAS :Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.Formule :C20H17NO6Degré de pureté :98% - 99.99%Couleur et forme :Light Yellow PowderMasse moléculaire :367.35Loreclezole
CAS :Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Formule :C10H6Cl3N3Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :274.53Afloqualone
CAS :Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Formule :C16H14FN3ODegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :283.3Pozanicline dihydrochloride
CAS :Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)Formule :C11H18Cl2N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.18Azaphen dihydrochloride monohydrate
CAS :Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Formule :C16H23Cl2N5O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :388.29
