Neuroscience
Les inhibiteurs en neurosciences sont des composés conçus pour moduler l'activité de protéines, d'enzymes ou de récepteurs spécifiques au sein du système nerveux. Ces inhibiteurs sont cruciaux pour étudier les mécanismes moléculaires sous-jacents au fonctionnement neuronal, à la transmission synaptique et aux maladies neurodégénératives. En ciblant les récepteurs des neurotransmetteurs, les canaux ioniques et les voies de signalisation, les inhibiteurs en neurosciences facilitent l'exploration du fonctionnement cérébral et le développement de stratégies thérapeutiques pour des troubles neurologiques tels que la maladie d'Alzheimer, de Parkinson et l'épilepsie. Chez CymitQuimica, nous offrons une gamme complète d'inhibiteurs en neurosciences de haute qualité pour soutenir vos recherches en neurobiologie, neuropharmacologie et sciences cognitives.
Sous-catégories appartenant à la catégorie "Neuroscience"
- récepteur 5-HT(940 produits)
- ACK(1 produits)
- AChR(574 produits)
- ATP Citrate Lyase(16 produits)
- Récepteur adrénergique(2.943 produits)
- BACE(36 produits)
- Bêta-amyloïde(204 produits)
- CaMK(68 produits)
- COX(561 produits)
- Récepteur de la dopamine(407 produits)
- Récepteur GABA(336 produits)
- Gamma-sécrétase(59 produits)
- GluR(255 produits)
- GlyT(24 produits)
- Récepteur de l'histamine(358 produits)
- LRRK2(33 produits)
- Récepteur de la mélatonine(24 produits)
- NMDAR(28 produits)
- Récepteur OX(40 produits)
- Récepteur opioïde(297 produits)
Affichez 12 plus de sous-catégories
5398 produits trouvés pour "Neuroscience"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
BSBM6
CAS :<p>BSBM6 is an inhibitor of Aβ aggregation and neuronal toxicity that acts by reversing the aggregation and toxicity of amyloid-β peptides.</p>Formule :C23H29N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :427.49Ebiratide TFA
<p>Ebiratide (HOE-427) TFA is a derivative of ACTH4-9 that exerts its effect directly on the central nervous system, enhancing memory. Ebiratide TFA also promotes the metabolism of acetylcholine (ACh) in the rat brain.</p>Formule :C48H73N11O10S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :996.23 (free base)HTR2A antagonist 1
<p>HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.</p>Formule :C35H43Cl2F2N5O4Couleur et forme :SolidMasse moléculaire :706.65Lu AE51090
CAS :<p>Lu AE51090 is a selective muscarinic M1 receptor agonist with minimal off-target effects, receptor function and selective pharmacological modulation.</p>Formule :C24H29N3O3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :407.51Binospirone
CAS :<p>Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study of movement disorders associated with neurologic dysfunction.</p>Formule :C20H26N2O4Degré de pureté :97.57% - 98.96%Couleur et forme :SoildMasse moléculaire :358.43Pomaglumetad methionil anhydrous
CAS :<p>LY2140023, potential schizophrenia treatment, is an oral prodrug of LY404039, a selective mGlu2/3 agonist.</p>Formule :C12H18N2O7S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :366.41OXA(17-33) TFA
<p>OXA(17-33) TFA: Potent OX1 agonist, ~23x more selective for OX1 (EC50=8.29nM) than OX2 (187nM).</p>Formule :C81H126F3N23O24Couleur et forme :SolidMasse moléculaire :18633-Chloroamphetamine hydrochloride
CAS :<p>3-Chloroamphetamine hydrochloride is a derivative of amphetamine that acts as a central nervous system stimulant by releasing serotonin and dopamine.</p>Formule :C9H13Cl2NCouleur et forme :SolidMasse moléculaire :206.115-HT2A receptor agonist-6
CAS :<p>5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.</p>Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.364-Hydroxy MPT
CAS :<p>4-Hydroxy MPT (4-OH-MPT) is a serotonin-active compound that acts as an agonist for 5-HT2A and 5-HT2B receptors, with EC50 values of 3.82 nM and 3.4 nM, respectively.</p>Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.32Dalidnetug
CAS :<p>Dalidnetug is a humanized monoclonal antibody that targets human β-amyloid precursor protein (APP). By specifically binding to APP, Dalidnetug reduces the production of β-amyloid (Aβ), thereby demonstrating activity in clearing β-amyloid. This compound holds potential for research in Alzheimer's disease.</p>Couleur et forme :Liquid(-)-2-Phenylpropylamine
CAS :<p>(-)-2-Phenylpropylamine ((S)-2-Phenylpropylamine) (compound 3b) functions as an inhibitor for both MAO-A and MAO-B, with Ki values of 584 μM and 156 μM, respectively.</p>Formule :C9H13NCouleur et forme :SolidMasse moléculaire :135.21NNC 11-1607
CAS :<p>NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.</p>Formule :C30H32N6O2S2Couleur et forme :SolidMasse moléculaire :572.74Methyllycaconitine citrate
CAS :<p>Methyllycaconitine citrate (MLA) is an α7 neuronal nicotinic acetylcholine receptor (α7nAChR) antagonist that crosses the blood-brain barrier.</p>Formule :C43H58N2O17Degré de pureté :98.03% - 98.91%Couleur et forme :SolidMasse moléculaire :874.92Timegadine hydrochloride
CAS :<p>Timegadine hydrochloride (SR1368 hydrochloride) is the hydrochloride salt form of Timegadine. It is an orally active inhibitor of COX and lipo-oxygenase, effectively suppressing COX in rabbit platelets and rat brain with IC50 values of 5 nM and 20 μM, respectively, and inhibiting lipo-oxygenase in horse and rabbit platelets with an IC50 of 100 μM. Timegadine hydrochloride also exhibits anti-arthritis activity.</p>Formule :C20H24ClN5SCouleur et forme :SolidMasse moléculaire :401.96Malaoxon
CAS :<p>Malaoxon is used as an insecticide.</p>Formule :C10H19O7PSCouleur et forme :SolidMasse moléculaire :314.29(Rac)-Sabcomeline
CAS :<p>(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.</p>Formule :C10H15N3ODegré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :193.25Pridinol hydrochloride
CAS :<p>Pridinolhydrochloride is the hydrochloride form of Pridinol. Pridinol hydrochloride is an orally active anticholinergic agent, which can also be used as a muscle relaxant.</p>Formule :C20H26ClNOCouleur et forme :SolidMasse moléculaire :331.88γ-DGG TFA
CAS :<p>Gamma-DGG TFA is an antagonist of excitatory amino acids that can inhibit depolarization induced by NMDA, Kainate, and Quisqualate. In addition, it counteracts excitatory postsynaptic potentials (e.p.s.p.) in rat hippocampal slices.</p>Formule :C9H13F3N2O7Couleur et forme :SolidMasse moléculaire :318.2Salvianolic acid H
CAS :<p>Salvianolic acid H is a strong inhibitor of acetylcholinesterase (AChE) [1].</p>Formule :C27H22O12Couleur et forme :SolidMasse moléculaire :538.462-APB hydrochloride
CAS :<p>2-APB is an analog of 6-APB and falls under the category of benzofuran derivatives, known for its psychoactive properties. Certain benzofuran derivatives also exhibit monoamine oxidase-A (MAO-A) inhibitory activity.</p>Formule :C11H14ClNOCouleur et forme :SolidMasse moléculaire :211.69R 50595
CAS :<p>R 50595 is a selective non-competitive cisapride antagonist.</p>Formule :C30H35Cl2F2N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.52Methalthiazide
CAS :<p>Methalthiazide enhances the activity of natural agonists of AMPA receptors and can be utilized in schizophrenia research.</p>Formule :C12H16ClN3O4S3Couleur et forme :SolidMasse moléculaire :397.92Minaprine
CAS :<p>Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.</p>Formule :C17H22N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.38N-Desmethyl Pimavanserin
CAS :<p>N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment of insomnia and other sleep disorders.</p>Formule :C24H32FN3O2Degré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :413.53COX-2-IN-33
<p>COX-2-IN-33 (compound 5f) is a selective COX-2 inhibitor with an IC50 value of 45.5 nM and exhibits potential as an anti-inflammatory agent.</p>Formule :C20H13ClF3N5O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :479.8Endosulfan I
CAS :<p>Endosulfan I is one of the two major stereoisomers of the broad-spectrum insecticide Endosulfan inhibi the GABA/benzodiazepine/picrotoxin complex</p>Formule :C9H6Cl6O3SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :406.93RS 56812
CAS :<p>RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.</p>Formule :C18H21N3O2Degré de pureté :99.38%Couleur et forme :SoildMasse moléculaire :311.38Withasomniferolide B
CAS :<p>Withasomniferolide B, a withanolide from Withania somnifera root, activates GABAA receptors.</p>Formule :C28H36O4Couleur et forme :SolidMasse moléculaire :436.58Calmodulin Kinase IINtide, Myristoylated
<p>Myristoylated Calmodulin Kinase IINtide (Myr-CaMKIINtide) serves as a selective and noncompetitive inhibitor of CaMKII [1].</p>Formule :C156H275N47O43Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3497.14C175-0062
CAS :<p>C175-0062, a monoamine oxidase B (MAO-B) inhibitor, is applicable in research focused on neurodegenerative disorders such as Parkinson's disease (PD), Alzheimer's disease (AD), and amyotrophic lateral sclerosis (ALS) [1].</p>Formule :C21H18N2O5Couleur et forme :SolidMasse moléculaire :378.38Anti-inflammatory agent 52
<p>Anti-inflammatory agent 52 (compound 7j) is an orally active, selective COX-2 inhibitor with the capability to induce G2/M phase arrest and exhibit anti-HT29</p>Formule :C24H21ClN2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :452.95AChE-IN-70
<p>AChE-IN-70 (compound 4) is an acetylcholinesterase inhibitor. It exhibits larvicidal activity against mosquito larvae (Culex pipiens L.), making it useful for mosquito control research.</p>Couleur et forme :Odour SolidBSB
CAS :<p>BSB is a Congo red-derived fluorescent probe, an amyloid protein imaging agent, interacting with amyloid fibrils formed by Aβ (1-40) peptides in rodents.</p>Formule :C24H17BrO6Degré de pureté :95.53%Couleur et forme :SolidMasse moléculaire :481.29Vortioxetine D8
CAS :<p>Vortioxetine D8 is a deuterium-labeled antidepressant inhibiting 5-HT1A/B, 5-HT3A, 5-HT7 receptors & SERT (Ki: 15-1.6 nM).</p>Formule :C18H22N2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.5(S)-3,4-DCPG HCl
<p>(S)-3,4-DCPG HCl is a selective mGluR8a agonist, impacting AV12-664 cells with an EC50 of 31 nM.</p>Formule :C10H10ClNO6Degré de pureté :99.53% - 99.9%Couleur et forme :SoildMasse moléculaire :275.64Lupanine hydrochloride
CAS :<p>Lupanine hydrochloride, a Sparteine derivative, binds to nAChR with a Ki of 500 nM and has ganglioplegic properties.</p>Formule :C15H25ClN2OCouleur et forme :SolidMasse moléculaire :284.83COX-2-IN-31
<p>COX-2-IN-31 (compound 7b) is an orally active dual inhibitor targeting COX-2 (IC50=60 nM) and 5-LOX (IC50=1.9 μM).</p>Formule :C17H16N6O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :400.41Methamnetamine hydrochloride
CAS :<p>Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.</p>Formule :C14H18ClNCouleur et forme :SolidMasse moléculaire :235.75PZ-1922
<p>PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R and 5-HT3R with K i values of 17 nM and 0.45 nM, respectively.</p>Degré de pureté :98%Couleur et forme :Odour SolidGluN2B receptor modulator-1
CAS :<p>GluN2B receptor modulator-1 is a selective negative allosteric modulator of NMDA receptor GluN2B subunits (IC50 31 nM), valuable for neuropharmacology studies.</p>Formule :C17H15F3N4O2SDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :396.39MAO-B-IN-3
<p>MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a Ki</p>Formule :C24H25N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.47β-Amyloid (1-9)
CAS :<p>This is an N-terminal fragment of beta amyloid.</p>Formule :C42H60N14O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1033.01MAO-B-IN-18
<p>MAO-B-IN-18 is a potent, selective inhibitor of MAO B, demonstrating IC50 values of 52 nM for hMAO B and 14 μM for hMAO A.</p>Formule :C25H22N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :458.47NT 13 acetate
<p>NT 13 acetate is a partial agonist of NMDA receptor and can be used for research on depression, anxiety, and other related diseases.</p>Formule :C20H34N4O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :474.515-AAM-2-CP
CAS :<p>5-AAM-2-CP is one of the major metabolites of Acetamiprid. Acetamiprid, a nAChR agonist, is a neonicotinoid insecticide used worldwide.</p>Formule :C8H9ClN2ODegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :184.62Octamylamine
CAS :<p>Octamylamine is a bioactive chemical.</p>Formule :C13H29NCouleur et forme :SolidMasse moléculaire :199.3761(Iso)-Landipirdine
CAS :<p>(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.</p>Formule :C18H19FN2O3SDegré de pureté :98.50%Couleur et forme :SoildMasse moléculaire :362.42Antidepressant agent 3
<p>Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.</p>Formule :C17H30ClN5O2SCouleur et forme :SolidMasse moléculaire :403.974-hydroxy DiPT hydrochloride
CAS :<p>4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.</p>Formule :C16H25ClN2OCouleur et forme :SolidMasse moléculaire :296.84
