récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
1025 produits trouvés pour "récepteur 5-HT"
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AVN-322
CAS :AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Formule :C17H20ClN5O2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :393.89MS 245 oxalate
CAS :MS 245 oxalate is a 5-HT6 antagonist.Formule :C21H24N2O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.49LY 334370 hydrochloride
CAS :5-HT1F receptor agonistFormule :C21H23ClFN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :387.88Methiothepin maleate
CAS :Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.Formule :C24H28N2O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :472.62Irindalone
CAS :IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.Formule :C24H29FN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.51EGIS-7625
CAS :EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.Formule :C18H24Cl2N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :399.32Glemanserin
CAS :Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Formule :C20H25NODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :295.42Ref: TM-T22964
1mg38,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg119,00€25mg259,00€50mg409,00€100mg605,00€500mg1.288,00€DV 7028 hydrochloride
CAS :DV 7028 hydrochloride is a 5-HT2A receptor antagonist.Formule :C21H26ClFN4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :436.91Org37684
CAS :5-HT2 receptors agonistFormule :C14H20ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :269.77L-775,606
CAS :L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.Formule :C25H29FN6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :432.54AR-A 2
CAS :AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).Formule :C27H36N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.6PNU-282987 S enantiomer hydrochloride
CAS :(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.Formule :C14H18Cl2N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :301.21Donitriptan
CAS :Donitriptan 是一种 5-HT 受体激动剂，对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。
Formule :C23H25N5O2Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :403.48Quinupramine
CAS :Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formule :C21H24N2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :304.43PNU-282987 free base
CAS :PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.
Formule :C14H17ClN2ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :264.75Masupirdine free base
CAS :Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formule :C21H24BrN3O3SDegré de pureté :98.36% - 99.65%Couleur et forme :SolidMasse moléculaire :478.4(Z)-Thiothixene
CAS :(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.
Formule :C23H29N3O2S2Degré de pureté :99.21%Couleur et forme :Yellow To Yellow With A Tan Cast PowderMasse moléculaire :443.63Teniloxazine
CAS :Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.Formule :C16H19NO2SDegré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :289.39R 59-022 hydrochloride
CAS :R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.
Formule :C27H27ClFN3OSDegré de pureté :97.7%Couleur et forme :SolidMasse moléculaire :496.04RS 42358-197
CAS :RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formule :C19H23ClN2ODegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :330.85Ref: TM-T20739
1mg158,00€1mL*10mM (DMSO)349,00€5mg351,00€10mg527,00€25mg783,00€50mg1.054,00€100mg1.414,00€200mg1.908,00€Lecozotan HCl
CAS :Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.
Formule :C28H30ClN5O3Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :520.02DA-6886
CAS :DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formule :C19H28Cl2N6O2Degré de pureté :99.91% - 99.99%Couleur et forme :SolidMasse moléculaire :443.37Adoprazine
CAS :Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.
Formule :C24H24FN3O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :405.46Femoxetine hydrochloride
CAS :Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formule :C20H26ClNO2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :347.88Goxalapladib
CAS :Goxalapladib（GSK 677116） is a small molecule compound that can be used to treat cardiovascular risks associated with atherosclerosis.Formule :C40H39F5N4O3Degré de pureté :99.64% - 99.93%Couleur et forme :SolidMasse moléculaire :718.75Cyamemazine
CAS :Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formule :C19H21N3SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :323.46Tedatioxetine
CAS :Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formule :C18H21NSDegré de pureté :99.76% - >99.99%Couleur et forme :SolidMasse moléculaire :283.43Landipirdine
CAS :Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Formule :C18H19FN2O3SDegré de pureté :97.61% - 99.99%Couleur et forme :SolidMasse moléculaire :362.42Faxeladol
CAS :Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Formule :C15H23NODegré de pureté :98.77% - 99.67%Couleur et forme :SolidMasse moléculaire :233.35Cianopramine
CAS :Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.Formule :C20H23N3Degré de pureté :99.92% - 99.92%Couleur et forme :SolidMasse moléculaire :305.42BL-1020 Mesylate
CAS :BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formule :C28H45ClN4O11S4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :777.39Viloxazine
CAS :Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormule :C13H19NO3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :237.29CP 96021
CAS :"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."
Formule :C29H21FN4OSDegré de pureté :97.81% - 99.62%Couleur et forme :SoildMasse moléculaire :492.57Cilansetron
CAS :Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.Formule :C20H21N3ODegré de pureté :99.82% - 99.98%Couleur et forme :SolidMasse moléculaire :319.4E6801
CAS :E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formule :C17H18ClN5O2S2Degré de pureté :96.32% - 97.24%Couleur et forme :SolidMasse moléculaire :423.94Ticalopride
CAS :Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formule :C14H20ClN3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :313.78SPD-473 citrate
CAS :SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Formule :C23H31Cl2NO8SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :552.47Roxindole
CAS :Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formule :C23H26N2ODegré de pureté :98.03% - 98.93%Couleur et forme :SolidMasse moléculaire :346.47Aplindore Fumarate
CAS :Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formule :C22H22N2O7Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :426.42Nexopamil
CAS :Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.
Formule :C24H40N2O3Degré de pureté :97.87% - >99.99%Couleur et forme :SolidMasse moléculaire :404.59ATC 0175
CAS :ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.Formule :C23H26ClF2N5ODegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :461.93Perphenazine dihydrochloride
CAS :Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formule :C21H28Cl3N3OSDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :476.89Liafensine
CAS :Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Formule :C24H22N4Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :366.46Piromelatine
CAS :Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity withFormule :C17H16N2O4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :312.32Ref: TM-T34081
1mg60,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg178,00€25mg334,00€50mg522,00€100mg713,00€Lensiprazine
CAS :Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFormule :C24H27FN4O2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :422.5H-9 dihydrochloride
CAS :H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formule :C11H15Cl2N3O2SDegré de pureté :97.3%Couleur et forme :SolidMasse moléculaire :324.235-HT6/7 antagonist 1
CAS :5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.
Formule :C22H20FN3O3Degré de pureté :98.78% - 99.26%Couleur et forme :SolidMasse moléculaire :393.41Litoxetine
CAS :Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Formule :C16H19NODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :241.33Ref: TM-T67956
1mg92,00€1mL*10mM (DMSO)178,00€5mg207,00€10mg309,00€25mg527,00€50mg755,00€100mg1.044,00€500mg2.088,00€BMY-14802 hydrochloride
CAS :BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formule :C18H23ClF2N4ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :384.85Tiospirone
CAS :Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.Formule :C24H32N4O2SDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :440.6Ref: TM-T24885
1mg123,00€5mg293,00€1mL*10mM (DMSO)354,00€10mg537,00€25mg863,00€50mg1.161,00€100mg1.558,00€5-HT1A modulator 1
CAS :5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formule :C21H25N3O2SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :383.51Pimethixene maleate
CAS :Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.Formule :C23H23NO4SDegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :409.5Ecopipam
CAS :Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.Formule :C19H20ClNODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :313.82Ricasetron
CAS :Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formule :C19H27N3ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :313.44Anpirtoline hydrochloride
CAS :Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formule :C10H14Cl2N2SDegré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :265.20Rilapine
CAS :Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Formule :C22H20ClN3Degré de pureté :97.76% - 99.20%Couleur et forme :SolidMasse moléculaire :361.87Sarizotan HCl
CAS :Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Formule :C22H22ClFN2ODegré de pureté :96%Couleur et forme :SolidMasse moléculaire :384.87Agomelatine hydrochloride
CAS :Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).Formule :C15H18ClNO2Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :279.76Fananserin
CAS :Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formule :C23H24FN3O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :425.52Ref: TM-T15270
2mg39,00€5mg52,00€1mL*10mM (DMSO)58,00€10mg77,00€25mg110,00€50mg166,00€100mg236,00€200mg349,00€cis-Urocanic acid
CAS :cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formule :C6H6N2O2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :138.12Repinotan
CAS :Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.Formule :C21H24N2O4SDegré de pureté :99%Couleur et forme :SolidMasse moléculaire :400.49Ensaculin
CAS :Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.Formule :C26H32N2O5Degré de pureté :99.56% - 99.81%Couleur et forme :SolidMasse moléculaire :452.54LY 272015 hydrochloride
CAS :LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formule :C21H25ClN2O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :372.89ML 10302 hydrochloride
CAS :ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Formule :C15H22Cl2N2O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :349.25LY266097 hydrochloride
CAS :LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.
Formule :C21H24Cl2N2O2Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :407.33ADR-851 free base
CAS :ADR-851 free base is an antagonist of the HT3 receptor.Formule :C14H18ClN3O2Degré de pureté :97.88% - 98.39%Couleur et forme :SolidMasse moléculaire :295.778-OH-Dpat
CAS :8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.Formule :C16H25NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.38SB 699551 dihydrochloride
CAS :SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.Formule :C34H47Cl2N3ODegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :584.66Ref: TM-T23325
1mg50,00€5mg105,00€1mL*10mM (DMSO)142,00€10mg170,00€25mg295,00€50mg424,00€100mg583,00€MM 77 dihydrochloride
CAS :MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.Formule :C19H29Cl2N3O3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :418.36Ref: TM-T23007
1mg86,00€5mg157,00€10mg215,00€1mL*10mM (DMSO)281,00€25mg472,00€50mg687,00€100mg938,00€500mg1.882,00€SB-215505
CAS :SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).Formule :C19H16ClN3ODegré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :337.85-HT2 antagonist 1
CAS :5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Formule :C22H29FN4O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :400.49Ref: TM-T12597
1mg642,00€5mg1.288,00€1mL*10mM (DMSO)1.521,00€10mg1.738,00€25mg2.583,00€50mg3.484,00€100mg4.708,00€SB228357
CAS :SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.Formule :C22H17F4N3O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :431.385HT6-ligand-1
CAS :5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).Formule :C20H22BrN3O2SDegré de pureté :99.24% - 99.93%Couleur et forme :SolidMasse moléculaire :448.38Itasetron
CAS :Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.
Formule :C16H20N4O2Degré de pureté :98.58% - 99.33%Couleur et forme :SolidMasse moléculaire :300.36RS 67333 hydrochloride
CAS :RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formule :C19H30Cl2N2O2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :389.36LY-2624803
CAS :LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formule :C22H25N3O3Degré de pureté :99.78% - 99.97%Couleur et forme :SolidMasse moléculaire :379.45GR 46611
CAS :GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formule :C23H27N3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :377.48Lesopitron
CAS :Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Formule :C15H21ClN6Degré de pureté :99.33% - 99.46%Couleur et forme :SolidMasse moléculaire :320.82Ref: TM-T25672
1mg133,00€1mL*10mM (DMSO)323,00€5mg324,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€500mg2.872,00€Felcisetrag
CAS :Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.Formule :C25H37N5O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :455.59Ref: TM-T28934
1mg87,00€5mg215,00€1mL*10mM (DMSO)235,00€10mg318,00€25mg510,00€50mg692,00€100mg928,00€200mg1.251,00€PZ-1190
CAS :PZ-1190, a multitarget ligand for serotonin and dopamine receptors, exhibits potential antipsychotic activity in rodents [1].Formule :C27H30N4O2S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.68NAS-181
CAS :NAS-181 is a potent and selective rat 5-hydroxytryptamine 1B (r5-HT1B) antagonist (Ki: 47 nM).NAS-181 enhances the accumulation of 5-HTP in rat brain regions.Formule :C20H30N2O7SCouleur et forme :SolidMasse moléculaire :442.53LY108742
CAS :LY108742 is an antagonist of 5-HT2.Formule :C21H28N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :356.46SDZ-216525
CAS :SDZ-216525, a 5-HT1A receptor antagonist, inhibits the tracheal contractions induced both by NKA (10 nM-3 microM) and 5-HT (10 nM-10 microM) (n=4-10).Formule :C25H28N4O5SCouleur et forme :SolidMasse moléculaire :496.58Dothiepin
CAS :Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancingFormule :C19H21NSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :295.44Mesembrine
CAS :Mesembrine is an alkaloid, a 5-HT transporter inhibitor (K i 1.4 nM), and inhibits PDE4B (IC50 7.8 μM).Formule :C17H23NO3Couleur et forme :SolidMasse moléculaire :289.375-HT2C agonist-3 free base
CAS :5-HT2C agonist-3 ((+)-19) free base, a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM), exhibits antipsychotic drug-like activity and inhibits Amphetamine-Formule :C19H22FNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.38UNC9994 hydrochloride
CAS :UNC9994 hydrochloride is a selective β-arrestin-biased D2R agonist, Ki of 79 nM, that stimulates β-arrestin and modulates cAMP.Formule :C21H23Cl3N2OSCouleur et forme :SolidMasse moléculaire :457.84Flesinoxan
CAS :Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).Formule :C22H26FN3O4Couleur et forme :SolidMasse moléculaire :415.46FPPQ
CAS :FPPQ blocks 5-HT3 and 5-HT6 receptors (Ki: 0.9 & 3 nM) and may improve psychosis and cognition.Formule :C21H19FN4O2SCouleur et forme :SolidMasse moléculaire :410.46Capeserod HCl
CAS :Capeserod HCl, a 5-hydroxytriptamine 4 (5-HT4) receptor agonist, is used potentially for the treatment of Alzheimer's disease.Formule :C23H26Cl2N4O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :493.38Befiradol
CAS :Befiradol (NLX-112) is an agonist of 5-HT1A receptor.Formule :C20H22ClF2N3OCouleur et forme :SolidMasse moléculaire :393.86GYKI-46903 HCl
CAS :GYKI-46903 is a noncompetitive 5-HT3 receptor antagonist.Formule :C17H21ClFNO2Couleur et forme :SolidMasse moléculaire :325.81Gentisein
CAS :Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7Formule :C13H8O5Degré de pureté :96.89%Couleur et forme :SolidMasse moléculaire :244.2LY 53857
CAS :LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.Formule :C27H36N2O7Couleur et forme :SolidMasse moléculaire :500.592Gepirone
CAS :Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater selectivity for the 5-HT1A receptor than SSRIs.Formule :C19H29N5O2Degré de pureté :99.35% - 99.89%Couleur et forme :SolidMasse moléculaire :359.47Cyanopindolol fumarate
CAS :Cyanopindolol fumarate is a 5-HT receptor antagonist [1].Formule :C16H21N3O2C4H4O4Couleur et forme :SolidMasse moléculaire :345.4Des-4-fluorobenzyl Mosapride
CAS :Des-4-fluorobenzyl Mosapride, the main metabolite of mosapride, acts as a gastroprokinetic agent improving upper gastrointestinal (GI) motility by stimulating the serotonin receptor 4 (5-HT4; EC50= 74.2 nM, in guinea pig ileal longitudinal muscle myenteric plexus). It has been shown to increase colonic motility in dogs, horses, and guinea pigs in vivo. Mosapride, including this metabolite, is utilized in human and veterinary medicine to mitigate post-surgical and Parkinson's-induced constipation.Formule :C14H20ClN3O3Couleur et forme :SolidMasse moléculaire :313.785-HT2A antagonist 1
CAS :5-HT2A antagonist 1, from US5728835A & JP 1007727, may treat gastrointestinal and circulatory issues.Formule :C26H28N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.53LY-426965
CAS :LY-426965 is a selective, potent, orally bioavailable 5-HT1A antagonist.Formule :C28H38N2O2Couleur et forme :SolidMasse moléculaire :434.61DU-125530
CAS :DU-125530 is a 5-HT1A receptor antagonist.Formule :C23H26ClN3O5SCouleur et forme :SolidMasse moléculaire :491.99
