
récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
940 produits trouvés pour "récepteur 5-HT"
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TG6-10-1
CAS :<p>TG6-10-1 is an EP2 antagonist.</p>Formule :C23H23F3N2O4Degré de pureté :99.66% - ≥95%Couleur et forme :SolidMasse moléculaire :448.43Puerarin
CAS :<p>Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.</p>Formule :C21H20O9Degré de pureté :98.90% - 99.21%Couleur et forme :Yellow Brown Fine PowderMasse moléculaire :416.38Rotigotine Hydrochloride
CAS :<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Formule :C19H26ClNOSDegré de pureté :99.53% - 99.56%Couleur et forme :Almost White To White Crystalline PowderMasse moléculaire :351.93Rotigotine-
CAS :<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Formule :C19H25NOSDegré de pureté :98.08% - 99.59%Couleur et forme :SolidMasse moléculaire :315.47MK 212 hydrochloride
CAS :<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Formule :C8H11ClN4·HClDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :235.12Metadoxine
CAS :<p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>Formule :C8H11NO3·C5H7NO3Degré de pureté :99.19%Couleur et forme :Off-White PowderMasse moléculaire :298.29Intepirdine
CAS :<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Formule :C19H19N3O2SDegré de pureté :98% - 98.63%Couleur et forme :SolidMasse moléculaire :353.44Mosapride Citrate
CAS :<p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>Formule :C21H25ClFN3O3·C6H8O7Degré de pureté :99.70%Couleur et forme :White PowderMasse moléculaire :614.02GSK163090
CAS :<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Formule :C25H29N5ODegré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :415.53Tianeptine
CAS :<p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Formule :C21H25ClN2O4SDegré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :436.95Niaprazine
CAS :<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formule :C20H25FN4ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :356.44BRL-15572 dihydrochloride
CAS :<p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>Formule :C25H27ClN2O·2HClDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :479.87Dolasetron Mesylate hydrate
CAS :<p>Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.</p>Formule :C20H26N2O7SDegré de pureté :99.86% - 99.9%Couleur et forme :SolidMasse moléculaire :438.49PRX-08066
CAS :<p>PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.</p>Formule :C19H17ClFN5SDegré de pureté :97.79% - 98.07%Couleur et forme :SolidMasse moléculaire :401.89Ipsapirone hydrochloride
CAS :<p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>Formule :C19H24ClN5O3SCouleur et forme :SolidMasse moléculaire :437.94Donitriptan Mesylate
CAS :<p>Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.</p>Formule :C24H29N5O5SCouleur et forme :SolidMasse moléculaire :499.58Melitracen
CAS :<p>Melitracen is a tricyclic antidepressant.</p>Formule :C21H25NCouleur et forme :SolidMasse moléculaire :291.43Abaperidone Hydrochloride
CAS :<p>Abaperidone Hydrochloride is an atypical antipsychotic, potently binging to5-HT2 receptors and D2 receptors.</p>Formule :C25H26ClFN2O5Couleur et forme :SolidMasse moléculaire :488.94Melperone
CAS :<p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>Formule :C16H22FNODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :263.35Cannabigerol
CAS :<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Formule :C21H32O2Degré de pureté :99.59% - 99.92%Couleur et forme :SolidMasse moléculaire :316.48Temanogrel
CAS :<p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>Formule :C24H28N4O4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :436.52'-O-Methylisoliquiritigenin
CAS :<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formule :C16H14O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :270.28Alprenolol hydrochloride
CAS :<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Formule :C15H24ClNO2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :285.81idalopirdine
CAS :<p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>Formule :C20H19F5N2ODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :398.37Nuciferine
CAS :<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Formule :C19H21NO2Degré de pureté :98.76% - 99.79%Couleur et forme :SolidMasse moléculaire :295.38Naratriptan
CAS :<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Formule :C17H25N3O2SDegré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :335.47Methiothepin mesylate
CAS :<p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>Formule :C21H28N2O3S3Degré de pureté :98% - 99.92%Couleur et forme :SolidMasse moléculaire :452.65Rotundine
CAS :<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Formule :C21H25NO4Degré de pureté :99.8% - 99.91%Couleur et forme :Off-White SolidMasse moléculaire :355.43BMY 7378 dihydrochloride
CAS :<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42F-15599
CAS :<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Formule :C19H21ClF2N4ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :394.85Pirenperone
CAS :<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Formule :C23H24FN3O2Degré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :393.457-Amino-4-(trifluoromethyl)coumarin
CAS :<p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>Formule :C10H6F3NO2Degré de pureté :97.31% - 97.84%Couleur et forme :Yellow PowderMasse moléculaire :229.16Cariprazine
CAS :<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formule :C21H32Cl2N4ODegré de pureté :99.68% - 99.87%Couleur et forme :SolidMasse moléculaire :427.41Almotriptan Malate
CAS :<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Formule :C17H25N3O2S·C4H6O5Degré de pureté :99.95%Couleur et forme :Pale Yellow SolidMasse moléculaire :469.55Escitalopram Oxalate
CAS :<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Formule :C22H23FN2O5Degré de pureté :97.39% - 99.73%Couleur et forme :White SolidMasse moléculaire :414.43Serotonin hydrochloride
CAS :<p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>Formule :C10H13ClN2ODegré de pureté :98.05% - 99.93%Couleur et forme :White To Cream PowderMasse moléculaire :212.676Azaphen
CAS :<p>Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.</p>Formule :C16H21Cl2N5ODegré de pureté :97.62%Couleur et forme :SolidMasse moléculaire :370.28Piboserod
CAS :<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Formule :C22H31N3O2Degré de pureté :97.21% - 99.49%Couleur et forme :SolidMasse moléculaire :369.5Perospirone
CAS :<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Formule :C23H30N4O2SDegré de pureté :99.23%Couleur et forme :White PowderMasse moléculaire :426.57SB399885
CAS :<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formule :C18H21Cl2N3O4SDegré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :446.35LY334370
CAS :<p>LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM</p>Formule :C21H22FN3ODegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :351.42Sevoflurane
CAS :<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Formule :C4H3F7ODegré de pureté :98%Couleur et forme :Less Oil Colorless OilMasse moléculaire :200.05Geissoschizine methyl ether
CAS :<p>Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.</p>Formule :C22H26N2O3Degré de pureté :99.24% - 99.68%Couleur et forme :SolidMasse moléculaire :366.45Ansofaxine hydrochloride
CAS :<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97Tropisetron
CAS :<p>Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.</p>Formule :C17H20N2O2Degré de pureté :99.68%Couleur et forme :White SolidMasse moléculaire :284.35Nelotanserin
CAS :<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Formule :C18H15BrF2N4O2Degré de pureté :98.42% - 99.88%Couleur et forme :SolidMasse moléculaire :437.24Amitriptyline
CAS :<p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>Formule :C20H23NDegré de pureté :98.24% - 99.64%Couleur et forme :Crystals SolidMasse moléculaire :277.4Brexpiprazole HCl
CAS :<p>Brexpiprazole HCl (OPC 34712 dihydrochloride) is a new antipsychotic drug.</p>Formule :C25H27N3O2S·xHClDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :433.6Sarpogrelate hydrochloride
CAS :<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Formule :C24H32ClNO6Degré de pureté :99.73%Couleur et forme :Colorless LiquidMasse moléculaire :465.97Lurasidone hydrochloride
CAS :<p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.</p>Formule :C28H36N4O2S·HClDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :529.14PRX-07034 hydrochloride
CAS :<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Formule :C21H29Cl2N3O4SDegré de pureté :98.5%Couleur et forme :SolidMasse moléculaire :490.44Clozapine N-Oxide
CAS :<p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>Formule :C18H19ClN4ODegré de pureté :98.43% - 99.94%Couleur et forme :SolidMasse moléculaire :342.82Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Formule :C35H47FN10O8Degré de pureté :97.97%Couleur et forme :SolidMasse moléculaire :754.85Cinitapride
CAS :<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Formule :C21H30N4O4Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :402.49Pergolide mesylate
CAS :<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Formule :C20H30N2O3S2Degré de pureté :99.70%Couleur et forme :White To Off-White SolidMasse moléculaire :410.59Dasotraline hydrochloride
CAS :<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Formule :C16H16Cl3NDegré de pureté :98.92% - 99.6%Couleur et forme :SolidMasse moléculaire :328.66L-745870 trihydrochloride
CAS :<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.215-Benzyloxygramine
CAS :<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Formule :C18H20N2ODegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :280.36N-Desmethylclozapine
CAS :<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.8NGB 2904
CAS :<p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>Formule :C28H29Cl2N3ODegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :494.46Chlorprothixene
CAS :<p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>Formule :C18H18ClNSDegré de pureté :98.77% - 99.756%Couleur et forme :Pale Yellow Crystals SolidMasse moléculaire :315.86Piperacetazine
CAS :<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57Loxapine
CAS :<p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>Formule :C18H18ClN3ODegré de pureté :99.88%Couleur et forme :Pale Yellowish Crystals From Petroleum Ether SolidMasse moléculaire :327.81Brexpiprazole
CAS :<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57Jatrorrhizine
CAS :<p>Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.</p>Formule :C20H20NO4Degré de pureté :97.18% - 99.06%Couleur et forme :SolidMasse moléculaire :338.38Urapidil
CAS :<p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>Formule :C20H29N5O3Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :387.48RS-127445 hydrochloride
CAS :<p>RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).</p>Formule :C17H17ClFN3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :317.79Zacopride hydrochloride
CAS :<p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>Formule :C15H20ClN3O2·HClDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :346.268-Hydroxy-DPAT hydrobromide
CAS :<p>8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.</p>Formule :C16H26BrNODegré de pureté :98.90% - 99.09%Couleur et forme :SolidMasse moléculaire :328.29SB-203186 hydrochloride
CAS :<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Formule :C16H20N2O2·HClDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :308.81Myristicin
CAS :<p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>Formule :C11H12O3Degré de pureté :99.828%Couleur et forme :LiquidMasse moléculaire :192.21Hypidone hydrochloride
CAS :<p>Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor</p>Formule :C18H23ClN2O2Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :334.84Vortioxetine
CAS :<p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>Formule :C18H22N2SDegré de pureté :99.34% - 99.34%Couleur et forme :SolidMasse moléculaire :298.45BRL 54443
CAS :<p>BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).</p>Formule :C14H18N2ODegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :230.316-fluoro-DL-Tryptophan
CAS :<p>6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.</p>Formule :C11H11FN2O2Degré de pureté :99.25%Couleur et forme :Off-White PowderMasse moléculaire :222.22Serotonin
CAS :<p>Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!</p>Formule :C10H12N2ODegré de pureté :97.47% - 99.92%Couleur et forme :SolidMasse moléculaire :176.22NAN-190 hydrobromide
CAS :<p>NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.</p>Formule :C23H28BrN3O3Degré de pureté :95.20%Couleur et forme :SolidMasse moléculaire :474.39Perospirone hydrochloride
CAS :<p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :4633-AQC
CAS :<p>3-AQC is a competitive antagonist of 5-HT3.</p>Formule :C20H21N5O4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :395.41AVN-101
CAS :<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Formule :C21H25ClN2Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :340.89SCH-23390 hydrochloride
CAS :<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Formule :C17H19Cl2NODegré de pureté :98% - 99.83%Couleur et forme :SolidMasse moléculaire :324.24Mosapride
CAS :<p>Mosapride (AS-4370) is a selective 5HT4 agonist</p>Formule :C21H25ClFN3O3Degré de pureté :99.56%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :421.89Tianeptine sodium salt
CAS :<p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>Formule :C21H24ClN2NaO4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :458.93Vilazodone Hydrochloride
CAS :<p>Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of the</p>Formule :C26H27N5O2·HClDegré de pureté :99.56% - >99.99%Couleur et forme :SolidMasse moléculaire :477.99Xaliproden hydrochloride
CAS :<p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89lumateperone Tosylate
CAS :<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Formule :C31H36FN3O4SDegré de pureté :95.83% - 99.95%Couleur et forme :SolidMasse moléculaire :565.7Cerlapirdine
CAS :<p>Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.</p>Formule :C22H23N3O3SDegré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :409.5Cariprazine hydrochloride
CAS :<p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>Formule :C21H33Cl3N4ODegré de pureté :99.78% - >99.99%Couleur et forme :SolidMasse moléculaire :463.87Lerisetron
CAS :<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Formule :C18H20N4Degré de pureté :99.15% - 99.82%Couleur et forme :SolidMasse moléculaire :292.38Indophagolin
CAS :<p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>Formule :C19H15BrClF3N2O3SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :523.75Amperozide
CAS :<p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>Formule :C23H29F2N3ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :401.49Metoclopramide hydrochloride hydrate
CAS :<p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>Formule :C14H25Cl2N3O3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :354.27Eltoprazine hydrochloride
CAS :<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Vortioxetine hydrobromide
CAS :<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Formule :C18H22N2S·HBrDegré de pureté :98.85% - 99.98%Couleur et forme :SolidMasse moléculaire :379.36Azaphen dihydrochloride monohydrate
CAS :<p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>Formule :C16H23Cl2N5O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :388.29RS-67333
CAS :<p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>Formule :C19H29ClN2O2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :352.9SB 243213
CAS :<p>SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.</p>Formule :C22H19F3N4O2Degré de pureté :98.78% - 99.86%Couleur et forme :SolidMasse moléculaire :428.41(S)-Mirtazapine
CAS :<p>(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.</p>Formule :C17H19N3Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :265.35Renzapride
CAS :<p>Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.</p>Formule :C16H22ClN3O2Degré de pureté :98.97% - 99.09%Couleur et forme :SolidMasse moléculaire :323.82Ketanserin tartrate
CAS :<p>Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.</p>Formule :C26H28FN3O9Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :545.51Tandospirone
CAS :<p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>Formule :C21H29N5O2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :383.49Setiptiline
CAS :<p>Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.</p>Formule :C19H19NDegré de pureté :98.05% - 98.07%Couleur et forme :SolidMasse moléculaire :261.36Latrepirdine dihydrochloride
CAS :<p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>Formule :C21H25N3·2HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :392.37Rizatriptan
CAS :<p>Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.</p>Formule :C15H19N5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :269.35(R)-Mirtazapine
CAS :<p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>Formule :C17H19N3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :265.35Rotigotine
CAS :<p>Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.</p>Formule :C19H25NOSDegré de pureté :99.04% - 99.88%Couleur et forme :SolidMasse moléculaire :315.47LP-533401 hydrochloride
CAS :<p>LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.</p>Formule :C27H23ClF4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.94Citalopram
CAS :<p>Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.</p>Formule :C20H21FN2ODegré de pureté :99.78% - 99.89%Couleur et forme :SolidMasse moléculaire :324.39WAY-100635 maleate
CAS :<p>WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).</p>Formule :C25H34N4O2·xC4H4O4Degré de pureté :>99.99%Couleur et forme :White SolidMasse moléculaire :538.645Jatrorrhizine chloride
CAS :<p>Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.</p>Formule :C20H20ClNO4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :373.8S1RA
CAS :<p>S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2</p>Formule :C20H23N3O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :337.42Syk Inhibitor II
CAS :<p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>Formule :C14H15F3N6ODegré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :340.3R 59-022
CAS :<p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>Formule :C27H26FN3OSDegré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :459.58Cyproheptadine hydrochloride
CAS :<p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>Formule :C21H21N·HClDegré de pureté :99.88% - 99.97%Couleur et forme :SolidMasse moléculaire :323.86Risperidone Mesylate
CAS :<p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>Formule :C24H31FN4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.59Escitalopram
CAS :<p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>Formule :C20H21FN2ODegré de pureté :99.82%Couleur et forme :White Or White Crystalline PowderMasse moléculaire :324.39N-Methyl amisulpride
CAS :<p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>Formule :C18H29N3O4SCouleur et forme :SolidMasse moléculaire :383.51Keto Ziprasidone
CAS :<p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>Formule :C21H19ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.92Arazasetron HCl
CAS :<p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>Formule :C17H20ClN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.81Brexpiprazole-d8
CAS :<p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>Formule :C25H27N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :441.62Amitriptyline-d6 Hydrochloride
CAS :<p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>Formule :C20H18D6ClNCouleur et forme :SolidMasse moléculaire :319.90Mirtazapine D3
CAS :<p>Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .</p>Formule :C17H19N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :268.375-Methyltryptamine hydrochloride
CAS :<p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>Formule :C11H15ClN2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :210.703Penbutolol sulfate
CAS :<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Formule :C18H29NO2H2O4SDegré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :340.47Ketanserinol
CAS :<p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>Formule :C22H24FN3O3Couleur et forme :SolidMasse moléculaire :397.447-Desmethyl-3-hydroxyagomelatine
CAS :<p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>Formule :C14H15NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :245.27Diclofensine
CAS :<p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>Formule :C17H17Cl2NODegré de pureté :97.01% - 98.13%Couleur et forme :SolidMasse moléculaire :322.23Hydroxy ziprasidone
CAS :<p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>Formule :C21H21ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.94Pardoprunox
CAS :<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Formule :C12H15N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.27SB 271046 hydrochloride
CAS :<p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.</p>Formule :C20H22ClN3O3S2·HClDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :488.45Paroxetine hydrochloride hemihydrate
CAS :<p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>Formule :C38H44Cl2F2N2O7Degré de pureté :99.949%Couleur et forme :SolidMasse moléculaire :749.67Dolasetron Mesylate
CAS :<p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>Formule :C20H24N2O6SDegré de pureté :99.05%Couleur et forme :White PowderMasse moléculaire :420.48LY 344864
CAS :<p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>Formule :C21H22FN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.42Ampreloxetine
CAS :<p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>Formule :C18H18F3NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :321.342-Methyl-5-HT maleate
CAS :<p>2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.</p>Formule :C15H18N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :306.31Ro 04-6790
CAS :<p>Ro 04-6790 is a 5-HT6 receptor antagonist.</p>Formule :C12H16N6O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :308.36ST1936
CAS :<p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>Formule :C13H17ClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :236.74Org37684
CAS :<p>5-HT2 receptors agonist</p>Formule :C14H20ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :269.77Donitriptan
CAS :<p>Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。</p>Formule :C23H25N5O2Degré de pureté :98.76%Couleur et forme :SolidMasse moléculaire :403.48AR-A 2
CAS :<p>AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).</p>Formule :C27H36N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :448.6AVN-322
CAS :<p>AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.</p>Formule :C17H20ClN5O2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :393.89Alniditan dihydrochloride
CAS :<p>Alniditan dihydrochloride is a potent 5-HT1D agonist and migraine-abortive agent.</p>Formule :C17H28Cl2N4OCouleur et forme :SolidMasse moléculaire :375.34Methiothepin maleate
CAS :<p>Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.</p>Formule :C24H28N2O4S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :472.62RS 56812 hydrochloride
CAS :<p>5-HT3 partial agonist</p>Formule :C18H22ClN3O2Degré de pureté :98.62%Couleur et forme :SolidMasse moléculaire :347.84AL-37350A
CAS :<p>AL-37350A is a 5-HT2 receptor-selective agonist with ocular hypotensive activity.</p>Formule :C14H18N2OCouleur et forme :SolidMasse moléculaire :230.31CUMI-101
CAS :<p>CUMI-101 is an agonist of 5-HT1A receptor.</p>Formule :C19H27N5O3Couleur et forme :SolidMasse moléculaire :373.45Ifoxetine sulfate
CAS :<p>Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.</p>Formule :C13H19NO2H2O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :270.34WAY 629 hydrochloride
CAS :<p>5-HT2C agonist</p>Formule :C15H19ClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :262.78E55888
CAS :<p>E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.</p>Formule :C16H23N3Couleur et forme :SolidMasse moléculaire :257.37Etoperidone hydrochloride
CAS :<p>Etoperidone hydrochloride is an antidepressant agent.</p>Formule :C19H29Cl2N5OCouleur et forme :SolidMasse moléculaire :414.37LEK 8841
CAS :<p>LEK 8841 is an ergoline derivative that is a potential antipsychotic.</p>Formule :C21H24BrN3O4SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :494.4Clovoxamine
CAS :<p>Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.</p>Formule :C14H21ClN2O2Degré de pureté :99.44% - 99.75%Couleur et forme :SolidMasse moléculaire :284.78Lofepramine hydrochloride
CAS :<p>Lofepramine is a serotonin and norepinephrine reuptake inhibitor. Lofepramine is also a psychotropic IMIPRAMINE derivative.</p>Formule :C26H28Cl2N2ODegré de pureté :98%Couleur et forme :Off-White SolidMasse moléculaire :455.42Alosetron ((Z)-2-butenedioate)
CAS :<p>Alosetron (GR 68755) (Z)-2-butenedioate is a Serotonin 5HT3-receptor antagonist that is used in the treatment of irritable bowel syndrome.</p>Formule :C21H22N4O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.425-Carboxamidotryptamine maleate
CAS :<p>5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.</p>Formule :C15H17N3O5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :319.31SB-221284
CAS :<p>5-HT2C/2B receptor antagonist</p>Formule :C16H14F3N3OSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :353.36PF-3246799
CAS :<p>PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.</p>Formule :C15H17N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :239.32SB 272183
CAS :<p>SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.</p>Formule :C29H28ClN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :498.02Amitriptylinoxide
CAS :<p>Amitriptylinoxide is an antidepressant.</p>Formule :C20H23NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.4GW-876167
CAS :<p>GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.</p>Formule :C16H21N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.37BGC 20-761
CAS :<p>BGC20-761: selective 5-HT6/Dopamine antagonist; enhances memory, potential antipsychotic. K i - 5-HT6: 20 nM, 5-HT2A: 69 nM, D2: 140 nM.</p>Formule :C19H22N2OCouleur et forme :SolidMasse moléculaire :294.39EMDT
CAS :<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Formule :C15H22N2ODegré de pureté :97.66% - 99.78%Couleur et forme :SolidMasse moléculaire :246.35Captodiame
CAS :<p>Captodiame is an antihistamine agent.</p>Formule :C21H29NS2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :359.59S(-)-8-Hydroxy-DPAT hydrobromide
CAS :<p>S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.</p>Formule :C16H26BrNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.29SB-737050A
CAS :<p>SB-737050A, a 5-HT antagonist, is used potentially for the treatment of schizophrenia.</p>Formule :C22H23ClN2O3S2Couleur et forme :SolidMasse moléculaire :463.01GSK-215083
CAS :<p>GSK-215083: a PET quinoline-based 5-HT6 antagonist radioligand, binds 5HT6 in striatum and 5HT2A in frontal cortex.</p>Formule :C20H20FN3O2SCouleur et forme :SolidMasse moléculaire :385.46Adatanserin
CAS :<p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>Formule :C21H31N5ODegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :369.5EMD 386088 hydrochloride
CAS :<p>EMD 386088 hydrochloride is a 5-HT6 receptor agonist.</p>Formule :C14H16Cl2N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :283.2SB-269970
CAS :<p>SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).</p>Formule :C18H28N2O3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.49p-MPPF dihydrochloride
CAS :<p>p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.</p>Formule :C25H29Cl2FN4O2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :507.43QF0301B
CAS :<p>QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.</p>Formule :C23H28N2O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :364.48(4E)-SUN9221
CAS :<p>(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in</p>Formule :C25H31FN4O3Degré de pureté :97.79%Couleur et forme :SolidMasse moléculaire :454.54Mirisetron
CAS :<p>Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.</p>Formule :C24H31N3O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :393.52CP-809101
CAS :<p>CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Formule :C15H17ClN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.77Eplivanserin
CAS :<p>Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.</p>Formule :C19H21FN2O2Degré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :328.38GR 113808
CAS :<p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>Formule :C19H27N3O4SDegré de pureté :98.16%Couleur et forme :SolidMasse moléculaire :393.5AS19
CAS :<p>AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).</p>Formule :C18H25N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :283.41PNU-282987 S enantiomer hydrochloride
CAS :<p>(S)-PNU-282987, selective α7 nAChR agonist; Ki=26 nM (rat), weak on other receptors except 5-HT3; Ki=930 nM.</p>Formule :C14H18Cl2N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :301.21L-694,247
CAS :<p>L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.</p>Formule :C20H21N5O3SDegré de pureté :98.36%Couleur et forme :White SolidMasse moléculaire :411.485-HT7 agonist 1
CAS :<p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>Formule :C19H20ClN3Degré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :325.84Ziprasidone mesylate trihydrate
CAS :<p>Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.</p>Formule :C22H31ClN4O7S2Couleur et forme :SolidMasse moléculaire :563.08Way 100289
CAS :<p>Way 100289 is a selective 5-HT3 receptor antagonist.</p>Formule :C20H27N3O3Couleur et forme :SolidMasse moléculaire :357.45Cinitapride Hydrogen Tartrate
CAS :<p>Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors</p>Formule :C25H36N4O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :552.581Zimelidine dihydrochloride
CAS :<p>5-HT re-uptake inhibitor</p>Formule :C16H18BrClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :353.69CP94253 hydrochloride
CAS :<p>CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).</p>Formule :C15H20ClN3ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :293.795-HT6/5-HT2A receptor ligand-1
CAS :<p>Compound 33 is a dual 5-HT6/5-HT2A antagonist with Ki values of 2 nM and 11 nM, respectively, useful in neuro/psychiatric research.</p>Formule :C21H19FN2O2Couleur et forme :SolidMasse moléculaire :350.39(Rac)-WAY-161503
CAS :<p>(Rac)-WAY-161503 is a selective and high-affinity agonist of the 5-HT2C receptor (Ki: 4 nM; EC50: 12 nM), with anti-obesity and antidepressant effects.</p>Formule :C11H11Cl2N3ODegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :272.13Irindalone
CAS :<p>IrindaloneIrindalone is a potent serotonin (5-HT2) antagonist.</p>Formule :C24H29FN4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :408.51Blonanserin HCl
CAS :<p>Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.</p>Formule :C23H32Cl2FN3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.42Usmarapride free base
CAS :<p>Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.</p>Formule :C21H29N5O2Degré de pureté :99.91% - 99.91%Couleur et forme :SolidMasse moléculaire :383.49Pruvanserin hydrochloride
CAS :<p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>Formule :C22H22ClFN4ODegré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :412.89PNU-142633
CAS :<p>PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.</p>Formule :C24H30N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :422.52RS 64459-193
CAS :<p>RS 64459-193 has a high affinity for the 5-HT1A binding site.</p>Formule :C26H36Cl2N2O2Couleur et forme :SolidMasse moléculaire :479.48MHP 133
CAS :<p>MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).</p>Formule :C17H20ClN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :377.83Repinotan HCl
CAS :<p>Repinotan HCl (Bay-x-3702) is a 5-HT1A receptor agonist with potent neuroprotective effects for the study of ischemic stroke and traumatic brain injury.</p>Formule :C21H25ClN2O4SDegré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :436.95Iloperidone hydrochloride
CAS :<p>Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.</p>Formule :C24H28ClFN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :462.95TMPPAA
CAS :<p>TMPPAA is an allosteric agonist of 5-HT3 receptor.</p>Formule :C15H21NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :247.33Bifeprunox
CAS :<p>Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.</p>Formule :C24H23N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :385.46CJ 033466
CAS :<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Formule :C19H28ClN5ODegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :377.91Isamoltane hemifumarate
CAS :<p>5-HT1B antagonist</p>Formule :C16H22N202C4H404Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :332.4
