récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
1025 produits trouvés pour "récepteur 5-HT"
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Jatrorrhizine
CAS :Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.Formule :C20H20NO4Degré de pureté :97.18% - 99.06%Couleur et forme :SolidMasse moléculaire :338.38Urapidil
CAS :Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formule :C20H29N5O3Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :387.48RS-127445 hydrochloride
CAS :RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formule :C17H17ClFN3Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :317.79Zacopride hydrochloride
CAS :Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formule :C15H20ClN3O2·HClDegré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :346.26Ref: TM-T5336
1mg34,00€5mg71,00€1mL*10mM (DMSO)79,00€10mg99,00€25mg212,00€50mg385,00€100mg618,00€200mg859,00€8-Hydroxy-DPAT hydrobromide
CAS :8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.Formule :C16H26BrNODegré de pureté :98.90% - 99.99%Couleur et forme :SolidMasse moléculaire :328.29SB-203186 hydrochloride
CAS :SB 203186 hydrochloride is a potent 5-HT4 receptor antagonistFormule :C16H20N2O2·HClDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :308.81Myristicin
CAS :Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formule :C11H12O3Degré de pureté :99.828%Couleur et forme :LiquidMasse moléculaire :192.21Hypidone hydrochloride
CAS :Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitorFormule :C18H23ClN2O2Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :334.84Vortioxetine
CAS :Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formule :C18H22N2SDegré de pureté :99.34% - 99.34%Couleur et forme :SolidMasse moléculaire :298.45Ref: TM-T2395
1mL*10mM (DMSO)46,00€10mg48,00€25mg65,00€50mg90,00€100mg117,00€200mg203,00€500mg333,00€1g477,00€BRL 54443
CAS :BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formule :C14H18N2ODegré de pureté :98.07%Couleur et forme :SolidMasse moléculaire :230.316-fluoro-DL-Tryptophan
CAS :6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formule :C11H11FN2O2Degré de pureté :99.25%Couleur et forme :Off-White PowderMasse moléculaire :222.22Serotonin
CAS :Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Formule :C10H12N2ODegré de pureté :97.47% - 99.92%Couleur et forme :SolidMasse moléculaire :176.22Ref: TM-TN2437
2mg34,00€1mL*10mM (DMSO)46,00€5mg52,00€10mg85,00€25mg157,00€50mg250,00€100mg404,00€200mg585,00€NAN-190 hydrobromide
CAS :NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formule :C23H28BrN3O3Degré de pureté :95.20%Couleur et forme :SolidMasse moléculaire :474.39Perospirone hydrochloride
CAS :Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :4633-AQC
CAS :3-AQC is a competitive antagonist of 5-HT3.Formule :C20H21N5O4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :395.41AVN-101
CAS :AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formule :C21H25ClN2Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :340.89Ref: TM-T26690
1mg34,00€5mg75,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg205,00€50mg334,00€100mg557,00€200mg790,00€SCH-23390 hydrochloride
CAS :SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formule :C17H19Cl2NODegré de pureté :98% - 99.83%Couleur et forme :SolidMasse moléculaire :324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€1mL*10mM (DMSO)78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€Mosapride
CAS :Mosapride (AS-4370) is a selective 5HT4 agonistFormule :C21H25ClFN3O3Degré de pureté :99.56%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :421.89Tianeptine sodium salt
CAS :Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formule :C21H24ClN2NaO4SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :458.93Vilazodone Hydrochloride
CAS :Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormule :C26H27N5O2·HClDegré de pureté :99.56% - >99.99%Couleur et forme :SolidMasse moléculaire :477.99Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg38,00€5mg80,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg222,00€50mg356,00€100mg512,00€200mg735,00€lumateperone Tosylate
CAS :lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formule :C31H36FN3O4SDegré de pureté :95.83% - 99.95%Couleur et forme :SolidMasse moléculaire :565.7Cerlapirdine
CAS :Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Formule :C22H23N3O3SDegré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :409.5Ref: TM-T30798
1mg81,00€5mg170,00€1mL*10mM (DMSO)198,00€10mg274,00€25mg543,00€50mg780,00€100mg1.074,00€Cariprazine hydrochloride
CAS :Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formule :C21H33Cl3N4ODegré de pureté :99.78% - >99.99%Couleur et forme :SolidMasse moléculaire :463.87Lerisetron
CAS :Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formule :C18H20N4Degré de pureté :99.15% - 99.82%Couleur et forme :SolidMasse moléculaire :292.38Indophagolin
CAS :Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formule :C19H15BrClF3N2O3SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :523.75Amperozide
CAS :Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formule :C23H29F2N3ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :401.49Ref: TM-T23733
1mg87,00€5mg178,00€10mg295,00€1mL*10mM (DMSO)321,00€25mg497,00€50mg708,00€100mg964,00€500mg1.918,00€Metoclopramide hydrochloride hydrate
CAS :Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formule :C14H25Cl2N3O3Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :354.27Eltoprazine hydrochloride
CAS :Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Vortioxetine hydrobromide
CAS :Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formule :C18H22N2S·HBrDegré de pureté :98.85% - 99.98%Couleur et forme :SolidMasse moléculaire :379.36Azaphen dihydrochloride monohydrate
CAS :Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Formule :C16H23Cl2N5O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :388.29RS-67333
CAS :RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.Formule :C19H29ClN2O2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :352.9SB 243213
CAS :SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formule :C22H19F3N4O2Degré de pureté :98.78% - 99.86%Couleur et forme :SolidMasse moléculaire :428.41Jatrorrhizine chloride
CAS :Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Formule :C20H20ClNO4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :373.8Ketanserin tartrate
CAS :Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formule :C26H28FN3O9Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :545.51Latrepirdine dihydrochloride
CAS :Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formule :C21H25N3·2HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :392.37LP-533401 hydrochloride
CAS :LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formule :C27H23ClF4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.94Rizatriptan
CAS :Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formule :C15H19N5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :269.35Setiptiline
CAS :Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formule :C19H19NDegré de pureté :98.05% - 98.07%Couleur et forme :SolidMasse moléculaire :261.36Citalopram
CAS :Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formule :C20H21FN2ODegré de pureté :99.78% - 99.89%Couleur et forme :SolidMasse moléculaire :324.39(S)-Mirtazapine
CAS :(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formule :C17H19N3Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :265.35Rotigotine
CAS :Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formule :C19H25NOSDegré de pureté :99.04% - 99.88%Couleur et forme :SolidMasse moléculaire :315.47Tandospirone
CAS :Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formule :C21H29N5O2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :383.49Ref: TM-TQ0315
2mg37,00€5mg54,00€1mL*10mM (DMSO)59,00€10mg87,00€25mg141,00€50mg193,00€100mg308,00€200mg441,00€Renzapride
CAS :Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formule :C16H22ClN3O2Degré de pureté :98.97% - 99.09%Couleur et forme :SolidMasse moléculaire :323.82Ref: TM-T38507
1mg93,00€2mg124,00€5mg200,00€10mg359,00€25mg692,00€50mg945,00€100mg1.279,00€200mg1.701,00€WAY-100635 maleate
CAS :WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formule :C25H34N4O2·xC4H4O4Degré de pureté :99.96%Couleur et forme :White SolidMasse moléculaire :538.645Ref: TM-T3453
2mg43,00€5mg63,00€1mL*10mM (DMSO)74,00€10mg89,00€25mg150,00€50mg215,00€100mg316,00€500mg765,00€(R)-Mirtazapine
CAS :(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formule :C17H19N3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :265.35S1RA
CAS :S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formule :C20H23N3O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :337.42Syk Inhibitor II
CAS :Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formule :C14H15F3N6ODegré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :340.3R 59-022
CAS :R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formule :C27H26FN3OSDegré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :459.58Ref: TM-T16709
1mg35,00€5mg74,00€1mL*10mM (DMSO)75,00€10mg119,00€25mg269,00€50mg447,00€100mg733,00€200mg973,00€Cyproheptadine hydrochloride
CAS :Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
Formule :C21H21N·HClDegré de pureté :99.88% - 99.97%Couleur et forme :SolidMasse moléculaire :323.86
