récepteur 5-HT
Les récepteurs 5-HT, également connus sous le nom de récepteurs de la sérotonine, sont un groupe de récepteurs couplés aux protéines G (GPCR) qui médiatisent les effets de la sérotonine, un neurotransmetteur impliqué dans la régulation de l'humeur, l'anxiété, le sommeil, l'appétit et d'autres processus physiologiques. Ces récepteurs sont divisés en plusieurs sous-types, chacun ayant des fonctions et des propriétés pharmacologiques distinctes. Les modulateurs des récepteurs 5-HT sont largement étudiés pour leurs rôles dans le traitement de la dépression, des troubles anxieux et d'autres affections neuropsychiatriques. Chez CymitQuimica, nous offrons une gamme de modulateurs des récepteurs 5-HT de haute qualité pour soutenir vos recherches en neuropharmacologie, troubles de l'humeur et signalisation GPCR.
1025 produits trouvés pour "récepteur 5-HT"
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Alverine citrate
CAS :Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.Formule :C26H35NO7Degré de pureté :98.53% - 99.43%Couleur et forme :CoaMasse moléculaire :473.57Gevotroline
CAS :Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a 5-HT2 receptor antagonist that can be used to study behavioral disorders.Formule :C19H20FN3Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :309.38Loxapine succinate
CAS :Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.Formule :C22H24ClN3O5Degré de pureté :99.69%Couleur et forme :White To Of-White SolidMasse moléculaire :445.9p-MPPI hydrochloride
CAS :p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.Formule :C25H28ClIN4O2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :578.87Ref: TM-T16421
2mg38,00€5mg56,00€10mg88,00€25mg138,00€50mg222,00€100mg351,00€200mg522,00€1mL*10mM (DMSO)94,00€Fluoxetine
CAS :Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.Formule :C17H18F3NODegré de pureté :99.07% - 99.28%Couleur et forme :SolidMasse moléculaire :309.33Ziprasidone hydrochloride
CAS :Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFormule :C21H22CL2N4OSDegré de pureté :97.97% - 99.82%Couleur et forme :SolidMasse moléculaire :449.4Zolmitriptan
CAS :Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.Formule :C16H21N3O2Degré de pureté :99.69% - 99.91%Couleur et forme :White Or Kind Of White PowderMasse moléculaire :287.36Blonanserin
CAS :Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.Formule :C23H30FN3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :367.50Olanzapine
CAS :Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formule :C17H20N4SDegré de pureté :99.86% - ≥95%Couleur et forme :Yellowish Crystalline PowderMasse moléculaire :312.43Ketanserin
CAS :Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formule :C22H22FN3O3Degré de pureté :99.19% - 99.73%Couleur et forme :SolidMasse moléculaire :395.43Azatadine dimaleate
CAS :Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.
Formule :C28H30N2O8Degré de pureté :99.7% - >99.99%Couleur et forme :PowderMasse moléculaire :522.55Eletriptan hydrobromide
CAS :Eletriptan hydrobromide (Eletriptan HBr) is an orally active agonist with specific affinity for the 5-hydroxytriptamine1B/1D receptor.Formule :C22H27BrN2O2SDegré de pureté :99.69% - 99.85%Couleur et forme :Tan SolidMasse moléculaire :463.43Ref: TM-T0216
2mg37,00€5mg54,00€10mg66,00€25mg127,00€50mg205,00€100mg341,00€200mg504,00€1mL*10mM (DMSO)59,00€Aripiprazole
CAS :Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formule :C23H27Cl2N3O2Degré de pureté :99.43% - 99.62%Couleur et forme :Colourless Flake Crystalline SolidMasse moléculaire :448.39CP-809101 hydrochloride
CAS :CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formule :C15H18Cl2N4ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :341.24Protriptyline hydrochloride
CAS :Protriptyline HCl: a tricyclic antidepressant that increases norepinephrine and serotonin levels and has anticholinergic effects.Formule :C19H21N·HClDegré de pureté :98.54% - 99.98%Couleur et forme :SolidMasse moléculaire :299.84Trazodone hydrochloride
CAS :Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.Formule :C19H23Cl2N5ODegré de pureté :99.5% - 99.52%Couleur et forme :SolidMasse moléculaire :408.33Naluzotan hydrochloride
CAS :Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.
Formule :C23H39ClN4O3SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :487.1Tropanserin
CAS :Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.Formule :C17H23NO2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :273.37Terfenadine
CAS :Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.Formule :C32H41NO2Degré de pureté :98.76% - 99.75%Couleur et forme :SolidMasse moléculaire :471.67Asenapine Maleate
CAS :Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Formule :C21H20ClNO5Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :401.84Ondansetron hydrochloride dihydrate
CAS :Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.Formule :C18H19N3O·HCl·2H2ODegré de pureté :99.92%Couleur et forme :White Crystal PowderMasse moléculaire :365.862-Bromo-6-methoxynaphthalene
CAS :2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.Formule :C11H9BrODegré de pureté :98.51%Couleur et forme :White To Off-White PowderMasse moléculaire :237.09Frovatriptan succinate hydrate
CAS :Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.Formule :C18H25N3O6Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :379.41Trimipramine maleate
CAS :Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Formule :C24H30N2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :410.51Talipexole dihydrochloride
CAS :Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical andFormule :C10H17Cl2N3SDegré de pureté :99.89%Couleur et forme :Light Yellow SolidMasse moléculaire :282.23Ref: TM-T14490
2mg34,00€5mg49,00€10mg75,00€25mg137,00€50mg212,00€100mg340,00€200mg504,00€1mL*10mM (DMSO)50,00€Pizotifen
CAS :Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available in the USA.Formule :C19H21NSDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :295.44Lofepramine
CAS :Lofepramine (Leo 640) is a potent tricyclic antidepressant that is extensively metabolized to desipramine.Formule :C26H27ClN2ODegré de pureté :98.38%Couleur et forme :Crystals From Methanol Or Acetone SolidMasse moléculaire :418.96Ref: TM-T15773
1mg34,00€2mg46,00€5mg66,00€10mg93,00€25mg167,00€50mg245,00€100mg356,00€200mg530,00€1mL*10mM (DMSO)73,00€Iloperidone
CAS :Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formule :C24H27FN2O4Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :426.48PF-04995274
CAS :PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formule :C23H32N2O6Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :432.51Tenilapine
CAS :Tenilapine is a neuroleptic compound that can be used to study atypical antipsychotics.Formule :C17H16N4S2Degré de pureté :99.58% - >99.99%Couleur et forme :SoildMasse moléculaire :340.47Fluvoxamine maleate
CAS :Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxietyFormule :C19H25F3N2O6Degré de pureté :99.92% - 99.94%Couleur et forme :White Crystalline PowderMasse moléculaire :434.41Ref: TM-T1077
10mg51,00€25mg69,00€50mg85,00€100mg115,00€200mg170,00€500mg278,00€1mL*10mM (DMSO)52,00€Mianserin hydrochloride
CAS :Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.Formule :C18H21ClN2Degré de pureté :99.63% - 99.82%Couleur et forme :White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedMasse moléculaire :300.83JNJ-18038683
CAS :JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.Formule :C26H28ClN3O7Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :529.97Ref: TM-T11720
2mg34,00€5mg52,00€10mg86,00€25mg161,00€50mg245,00€100mg363,00€200mg515,00€1mL*10mM (DMSO)52,00€Mebhydrolin napadisylate
CAS :Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFormule :C19H20N2C10H8O6S2Degré de pureté :99.35% - 99.96%Couleur et forme :White Or Almost White CrystallineMasse moléculaire :420.52Cyproheptadine hydrochloride sesquihydrate
CAS :Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formule :C21H24ClNODegré de pureté :99.77% - >99.99%Couleur et forme :White To Slightly Yellowish Crystalline SolidMasse moléculaire :341.88Bufotenidine hydrochloride(487-91-2 Free base)
CAS :Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.Formule :C13H19ClN2ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :254.76Promazine hydrochloride
CAS :Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.Formule :C17H21ClN2SDegré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :320.88Naftidrofuryl oxalate
CAS :Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.Formule :C26H35NO7Degré de pureté :97.12% - 98.38%Couleur et forme :SolidMasse moléculaire :473.56Perphenazine
CAS :Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Formule :C21H26ClN3OSDegré de pureté :99.3% - 99.99%Couleur et forme :SolidMasse moléculaire :403.97Vilazodone
CAS :Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.Formule :C26H27N5O2Degré de pureté :99.61%Couleur et forme :Light Yellow SolidMasse moléculaire :441.52Quetiapine
CAS :Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.Formule :C21H25N3O2SDegré de pureté :99.14% - 99.63%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :383.51Desipramine hydrochloride
CAS :Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.Formule :C18H23ClN2Degré de pureté :99.58% - 99.96%Couleur et forme :White To Off-White PowderMasse moléculaire :302.84Dexchlorpheniramine Maleate
CAS :Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formule :C20H23ClN2O4Degré de pureté :99.58%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :390.86NEO 376
CAS :NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Formule :C20H24ClN3ODegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :357.88Ref: TM-T12207
1mg71,00€5mg133,00€10mg205,00€25mg353,00€50mg495,00€100mg665,00€200mg893,00€1mL*10mM (DMSO)147,00€Granisetron hydrochloride
CAS :Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapyFormule :C18H25ClN4ODegré de pureté :99.88% - 99.93%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :348.87Alosetron hydrochloride
CAS :Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.Formule :C17H19ClN4ODegré de pureté :99.90%Couleur et forme :Off-White PowderMasse moléculaire :330.81Lamotrigine
CAS :Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Formule :C9H7Cl2N5Degré de pureté :99.76% - 99.95%Couleur et forme :White To Pale Cream-Colored Powder Crystals From Isopropanol SolidMasse moléculaire :256.09Palonosetron hydrochloride
CAS :Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.Formule :C19H24N2O·HClDegré de pureté :99.84% - 99.92%Couleur et forme :White SolidMasse moléculaire :332.87Amisulpride
CAS :Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formule :C17H27N3O4SDegré de pureté :99.97% - 99.99%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :369.48Sertraline hydrochloride
CAS :Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.Formule :C17H18Cl3NDegré de pureté :99.12% - 99.99%Couleur et forme :Solid PowderMasse moléculaire :342.69Ref: TM-T0482
5mg49,00€10mg59,00€25mg98,00€50mg170,00€100mg222,00€200mg289,00€500mg487,00€1mL*10mM (DMSO)54,00€
